| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A calmodulin-derived peptide TI-16 inhibits Alzheimer's disease progression by decreasing Aβ burden and restoring calcium dyshomeostasis
|
Su, Jingyang
|
|
|
160 |
C |
p.
|
artikel
|
| 2 |
A comprehensive review on anti-inflammatory, antibacterial, anticancer and antifungal properties of several bivalent transition metal complexes
|
AlAli, Anas
|
|
|
160 |
C |
p.
|
artikel
|
| 3 |
A double-ionic macrocycle based on cyanostilbene: First organic fluorescence sensor based small molecular system for detecting cholesterol
|
Wu, Yunmei
|
|
|
160 |
C |
p.
|
artikel
|
| 4 |
A fluorometric and naked eye readable neuraminidase probe for influenza virus detection
|
Chang, Hao
|
|
|
160 |
C |
p.
|
artikel
|
| 5 |
A novel photoactivatable coumarin-based fluorescent “turn-on” probe: Synthesis and applications for H2S detection in living cells and zebrafish models
|
Sontisiri, Pakornsiri
|
|
|
160 |
C |
p.
|
artikel
|
| 6 |
A novel Quinazoline derivative exerts anti-tumor effects in non-small cell lung cancer through Wnt/β-catenin pathway inhibition
|
Zhao, Menglong
|
|
|
160 |
C |
p.
|
artikel
|
| 7 |
A rationale approach in developing proline based small peptide as U-shaped analogues of arachidonic acid: Dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase for developing anti-inflammatory agents
|
Vivesh, Vivesh
|
|
|
160 |
C |
p.
|
artikel
|
| 8 |
Benzimidazole derivatives protect pancreatic β-cells against cytokine-induced apoptosis
|
Hussain, Shafqat
|
|
|
160 |
C |
p.
|
artikel
|
| 9 |
Biosynthesis of the quinovosamycin nucleoside antibiotics diverges from that of tunicamycins by additional sugar processing genes
|
Sumang, Felaine Anne
|
|
|
160 |
C |
p.
|
artikel
|
| 10 |
Carvacrol/thymol derivatives as highly selective BuChE inhibitors with anti-inflammatory activities: Discovery and bio-evaluation
|
Zhang, Yuan-Lin
|
|
|
160 |
C |
p.
|
artikel
|
| 11 |
Computer aided design of CGA-N9 derived peptides based on oligopeptide transporters and their antifungal evaluations
|
Yan, Fu
|
|
|
160 |
C |
p.
|
artikel
|
| 12 |
Design, and synthesis of 2,4-thiazolidinedione substituted 1,3,5-triazine derivatives as anti-HIV agent via inhibition of reverse transcriptase along with anti-SARS CoV-2, antibacterial and antibiofilm activity
|
Singh, Saumya
|
|
|
160 |
C |
p.
|
artikel
|
| 13 |
Design, synthesis and bio-evaluation of 2,5-disubstituted thiazole derivatives for potential treatment of acute myeloid leukemia through targeting CDK9
|
Chen, Sumeng
|
|
|
160 |
C |
p.
|
artikel
|
| 14 |
Design, synthesis and biological evaluation of imine-containing inhibitors against the triple-mutant EGFR kinases based on the scaffold of osimertinib
|
Ding, Shi
|
|
|
160 |
C |
p.
|
artikel
|
| 15 |
Design, synthesis, and evaluation of 1,4-benzodioxane-hydrazone derivatives as potential therapeutics for skin cancer: In silico, in vitro, and in vivo studies
|
Akbar, Saleem
|
|
|
160 |
C |
p.
|
artikel
|
| 16 |
Design, synthesis and in vitro and in vivo biological evaluation of matrine derivatives as efficient anticancer agents with the characteristics of endoplasmic reticulum stress induction and apoptosis activation
|
Wang, Xingdong
|
|
|
160 |
C |
p.
|
artikel
|
| 17 |
Design, synthesis and in vitro evaluation of non-steroidal anti-inflammatory prodrugs for osteoarthritis
|
Voitovich, Iuliia
|
|
|
160 |
C |
p.
|
artikel
|
| 18 |
Development and evaluation of 18F-labeled novel radiopharmaceuticals for PET imaging of fibroblast activation protein expressing tumors
|
Zhang, Qingyu
|
|
|
160 |
C |
p.
|
artikel
|
| 19 |
Development of 2- and 3-prenylated quinolines and tetrahydroquinolines with PPAR activity: From hit to lead and a novel pan-PPAR agonist as a potential candidate for metabolic syndrome
|
Villarroel-Vicente, Carlos
|
|
|
160 |
C |
p.
|
artikel
|
| 20 |
Discovery of a novel Thiazole amide inhibitor of Inflammasome and Pyroptosis pathways
|
Dai, Zhen
|
|
|
160 |
C |
p.
|
artikel
|
| 21 |
Discovery of naturally inspired antimicrobial peptides using deep learning
|
Yang, Cai-Ling
|
|
|
160 |
C |
p.
|
artikel
|
| 22 |
Discovery of new 1,2,3,4-tetrahydro-β-carboline derivatives decorated with 3-N-substituted propionyl moiety flexibly bridged-chain as reactive oxygen species inducer for efficient antibacterial treatment
|
Yang, Yike
|
|
|
160 |
C |
p.
|
artikel
|
| 23 |
Discovery of small molecule ACC inhibitors: Potential treatment for excessive sebum secretion
|
Feng, Xilong
|
|
|
160 |
C |
p.
|
artikel
|
| 24 |
Diterpenes as nitric oxide secretion inhibitors from Kaempferia koratensis rhizomes
|
Kongwaen, Patcharin
|
|
|
160 |
C |
p.
|
artikel
|
| 25 |
Drug repurposing of 6-AZA-UTP and itraconazole reveals novel B3GALT5 inhibitors for pancreatic cancer
|
Botcha, Lavanya
|
|
|
160 |
C |
p.
|
artikel
|
| 26 |
Editorial Board
|
|
|
|
160 |
C |
p.
|
artikel
|
| 27 |
Efficient extraction of Licochalcone a with deep eutectic solvent: A promising drug for the treatment of dermatophytosis
|
Sun, Chunlan
|
|
|
160 |
C |
p.
|
artikel
|
| 28 |
Engaging an engineered PARP-2 catalytic domain mutant to solve the complex structures harboring approved drugs for structure analyses
|
Wang, Xiaoyu
|
|
|
160 |
C |
p.
|
artikel
|
| 29 |
Genome-guided discovery of coublibactins from Nocardia coubleae and their gallium complexes with potent antileukemic activity
|
Tao, Qiaoqiao
|
|
|
160 |
C |
p.
|
artikel
|
| 30 |
Ginsenoside Rd and chrysophanol: Modulating the serine-glycine-one-carbon pathway to enhance neuroprotection in intracerebral hemorrhage
|
Zhao, Xingping
|
|
|
160 |
C |
p.
|
artikel
|
| 31 |
Green synthesis of selenium nanoparticles, and its conjugation with antibacterial proteins for enhancing their antibacterial activity
|
Mourad, Amany N.
|
|
|
160 |
C |
p.
|
artikel
|
| 32 |
Hybride nanoparticles composed of SN38-modified [12]aneN3 and biotinylated lipids for targeted and synergistic lung Cancer therapy
|
Xu, De-Zhong
|
|
|
160 |
C |
p.
|
artikel
|
| 33 |
Identification of novel AURKA inhibitors against neuroblastoma using a virtual screening approach
|
Yin, Hongli
|
|
|
160 |
C |
p.
|
artikel
|
| 34 |
Inhibition of FLT3-induced signalling in refractory acute myeloid leukaemia
|
Yang, Jingmei
|
|
|
160 |
C |
p.
|
artikel
|
| 35 |
Interaction mechanisms between α-glucosidase and procyanidin dimers with different galloyl moiety: Multi-spectral analysis and molecular dynamics simulation
|
Wang, Mengting
|
|
|
160 |
C |
p.
|
artikel
|
| 36 |
Investigation of binding mechanisms between bovine serum albumin and flutamide using multispectral techniques and molecular dynamics simulations
|
Li, Ning
|
|
|
160 |
C |
p.
|
artikel
|
| 37 |
Issue TOC
|
|
|
|
160 |
C |
p.
|
artikel
|
| 38 |
2β-methoxy-2-deethoxyphantomolin synergistically enhances epirubicin effect against triple-negative breast cancer via targeted inhibition of AKT and HR pathways
|
Gu, Jianyi
|
|
|
160 |
C |
p.
|
artikel
|
| 39 |
Neuroprotective triterpenoids from Astragalus membranaceus stems and leaves: Anti-inflammatory and anti-apoptotic mechanisms for memory improvement via in vivo and in vitro models
|
Cheng, Yan-Gang
|
|
|
160 |
C |
p.
|
artikel
|
| 40 |
New acetamide-sulfonamide scaffolds with potential renal radiomodulatory effects: Insights into NF-κB pathway interactions
|
Ghorab, Mostafa M.
|
|
|
160 |
C |
p.
|
artikel
|
| 41 |
New alkanesulfonate-based quinazolinone-acetohydrazide scaffolds: Rational design, synthesis, molecular docking, anticancer properties and potential EGFR and its T790M/L858R mutants inhibitors
|
Morsy, Nagy A.
|
|
|
160 |
C |
p.
|
artikel
|
| 42 |
New steroidal saponins from Physochlainae Radix: Structures and anti-inflammatory efficacy
|
Tan, Jin-Yan
|
|
|
160 |
C |
p.
|
artikel
|
| 43 |
Novel ALK inhibitors containing DAAP fragments: Rational drug design and anti-tumor activity research
|
Wang, Ran
|
|
|
160 |
C |
p.
|
artikel
|
| 44 |
Novel benzofuran-conjugated indolin-2-ones as anticancer agents; design, synthesis, biological assessments, and molecular modeling insights
|
Eldehna, Wagdy M.
|
|
|
160 |
C |
p.
|
artikel
|
| 45 |
Novel chloropyridazine sulfonamides as aromatase inhibitors and apoptotic inducers in breast cancer
|
Zahran, Sally S.
|
|
|
160 |
C |
p.
|
artikel
|
| 46 |
Optimization of Aminoindazole derivatives as highly selective covalent inhibitors for wild-type and mutant FGFR4
|
Guo, Jing
|
|
|
160 |
C |
p.
|
artikel
|
| 47 |
Peptidomimetics based on thiacalixarene with L-tyrosine moieties: Antibacterial activity against methicillin-resistant Staphylococcus aureus and degradation induced by binding to α-chymotrypsin
|
Terenteva, Olga
|
|
|
160 |
C |
p.
|
artikel
|
| 48 |
Photocaged fluorescent probes for spatiotemporally monitoring G-Quadruplex DNA in live cells
|
Zhao, Xuzi
|
|
|
160 |
C |
p.
|
artikel
|
| 49 |
Recent advances in PROTAC-based antiviral and antibacterial therapeutics
|
Zhou, Can
|
|
|
160 |
C |
p.
|
artikel
|
| 50 |
Redox dyshomeostasis-driven prodrug strategy for enhancing camptothecin-based chemotherapy: Selenization of SN38 as a case study
|
Xi, Junmin
|
|
|
160 |
C |
p.
|
artikel
|
| 51 |
S-adenosylmethionine inhibits non-small cell lung cancer and enhances chemosensitivity by targeting the P62/NF-κB axis and regulating autophagy and oxidative stress
|
Jin, Xuehang
|
|
|
160 |
C |
p.
|
artikel
|
| 52 |
Small molecule therapeutics for receptor-mediated targeting through liposomes in breast cancer treatment: A comprehensive review
|
Ghosh, Rashmi
|
|
|
160 |
C |
p.
|
artikel
|
| 53 |
Structure-activity relationship explorations of 2-(isoxazol-5-yl)phenyl-3,4-dihydroxybenzoate derivatives to develop potent Wnt/β-catenin pathway inhibitors for colorectal cancer treatment
|
Dong, Li
|
|
|
160 |
C |
p.
|
artikel
|
| 54 |
Synthesis and evaluation of novel amino pyrimidine derivatives containing sulfonamide and their application as EGFR inhibitors
|
Yao, Han
|
|
|
160 |
C |
p.
|
artikel
|
| 55 |
Synthesis of new selective agents with dual anti-inflammatory and SARS-CoV-2 Mpro inhibitory activity: Antipyrine-celecoxib hybrid analogues; COX-2, COVID-19 cytokine storm and replication inhibitory activities.
|
Abdelall, Eman K.A.
|
|
|
160 |
C |
p.
|
artikel
|
| 56 |
Synthesis of N-heterocyclic carbene‑selenium complexes modulating apoptosis and autophagy in cancer cells: Probing the interactions with biomolecules and enzymes
|
Ashraf, Rizwan
|
|
|
160 |
C |
p.
|
artikel
|
| 57 |
Synthesis, structure activity relationship and biological evaluation of indole sulfonohydrazide derivatives as antagonists of P2Y1 and P2Y6 receptors
|
Hameed, Abdul
|
|
|
160 |
C |
p.
|
artikel
|
| 58 |
Targeting Autotaxin with imidazole- and Triazolyl-based inhibitors: Biological insights from in vitro and in vivo studies in pulmonary fibrosis
|
Kim, Misu
|
|
|
160 |
C |
p.
|
artikel
|
| 59 |
The development of pyridazinone-based andrographolide derivatives as anti-cancer agents with the ability of inhibiting the TFAP4/Wnt/β-catenin signaling pathway
|
Zhang, Hang
|
|
|
160 |
C |
p.
|
artikel
|
| 60 |
The diphenylpyrimidine derivative as a novel HDAC6 inhibitor alleviates atopic dermatitis through anti-inflammatory effects facilitated via TLR4/MAPK, STAT3 and NF-κB pathways
|
Chen, Jin-Ting
|
|
|
160 |
C |
p.
|
artikel
|
| 61 |
Unlocking the potential of novel tetrahydro-β-carboline-based HDAC6 inhibitors for colorectal cancer therapy: Design, synthesis and biological evaluation
|
Hemida, Noreen
|
|
|
160 |
C |
p.
|
artikel
|
| 62 |
Unveiling a pyrroloindoline diketopiperazine biosynthetic pathway featuring a phytoene-synthase-like family prenyltransferase with distinct regioselectivity
|
Duan, He
|
|
|
160 |
C |
p.
|
artikel
|
| 63 |
Unveiling the potential of xanthines, discovery of potential 7-benzyl-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione derivatives with antifibrotic activity for liver injury
|
Mohamed, Abdalla R.
|
|
|
160 |
C |
p.
|
artikel
|
| 64 |
Whiteleg shrimp-derived Cryptides induce mitochondrial-mediated cytotoxicity in human breast Cancer
|
El-Aal, Amr Adel Ahmed Abd
|
|
|
160 |
C |
p.
|
artikel
|
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