nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Acriflavine and proflavine hemisulfate as potential antivirals by targeting Mpro
|
Liang, Jing |
|
|
129 |
C |
p. |
artikel |
2 |
Allyl phenyl selenides as H2O2 acceptors to develop ROS-responsive theranostic prodrugs
|
Yang, Xue-Yan |
|
|
129 |
C |
p. |
artikel |
3 |
Anti-inflammatory butanolides and lignanoids from the root of Machilus zuihoensis var. mushaensis
|
Yang, Shuen-Shin |
|
|
129 |
C |
p. |
artikel |
4 |
Anti-proliferative tirucallane triterpenoids from gum resin of Boswellia sacra
|
Zhang, Bingyang |
|
|
129 |
C |
p. |
artikel |
5 |
Assessing p-tolyloxy-1,3,4-oxadiazole acetamides as lipoxygenase inhibitors assisted by in vitro and in silico studies
|
Bashir, Bushra |
|
|
129 |
C |
p. |
artikel |
6 |
Biosynthesis, characterization and biomedical potential of Arthrospira indica SOSA-4 mediated SeNPs
|
Afzal, Bushra |
|
|
129 |
C |
p. |
artikel |
7 |
Callicarpnoids A–C, structurally intriguing ent-Clerodane diterpenoid dimers with cytotoxicity against MCF-7 and HCT-116 cell lines from Callicarpa arborea Roxb
|
Cheng, Bin |
|
|
129 |
C |
p. |
artikel |
8 |
Cationic RGD peptidomimetic nanoconjugates as effective tumor targeting gene delivery vectors with antimicrobial potential
|
Ahmadi, Zeba |
|
|
129 |
C |
p. |
artikel |
9 |
CC1007, a small molecular compound, suppresses multiple myeloma via upregulation of Nur77
|
Zhu, Shicong |
|
|
129 |
C |
p. |
artikel |
10 |
Chemical synthesis of fluorinated and iodinated 17β-HSD3 inhibitors and evaluation for imaging prostate cancer tumors and tissue biodistribution
|
Poirier, Donald |
|
|
129 |
C |
p. |
artikel |
11 |
Construction of an in vivo NIR fluorescent probe for revealing the correlation between inflammation and mitochondrial hydrogen sulfide and viscosity
|
Cui, Yali |
|
|
129 |
C |
p. |
artikel |
12 |
Design and synthesis of N-(1-(6-(substituted phenyl)-pyridazin-3-yl)-piperidine-3-yl)-amine derivatives as JMJD6 inhibitors
|
Qian, Yuqing |
|
|
129 |
C |
p. |
artikel |
13 |
Design, synthesis and antitumor activity evaluation of novel indole acrylamide derivatives as IMPDH inhibitors
|
Jia, Hong-Wei |
|
|
129 |
C |
p. |
artikel |
14 |
Design, synthesis and biological evaluation of 2-aminopyridine derivatives as USP7 inhibitors
|
Xu, Xiaoming |
|
|
129 |
C |
p. |
artikel |
15 |
Design, synthesis and biological evaluation of dehydroabietic acid derivative as potent vasodilatory agents
|
Wu, Dan |
|
|
129 |
C |
p. |
artikel |
16 |
Design, synthesis, and biological evaluation of novel sulfamoylbenzamide derivatives as HBV capsid assembly modulators
|
Wang, Shuo |
|
|
129 |
C |
p. |
artikel |
17 |
Design, synthesis and biological evaluation of novel tumor hypoxia-activated EGFR tyrosine kinase inhibitors
|
Jia, Tingting |
|
|
129 |
C |
p. |
artikel |
18 |
Design, synthesis and biological evaluation of pyranocarbazole derivatives against Alzheimer’s disease, with antioxidant, neuroprotective and cognition enhancing properties
|
Zang, Yingda |
|
|
129 |
C |
p. |
artikel |
19 |
Design, synthesis, and in vitro evaluation of novel antifungal triazoles containing substituted 1,2,3-triazole-methoxyl side chains
|
Xie, Fei |
|
|
129 |
C |
p. |
artikel |
20 |
Design, synthesis, and molecular docking of novel pyrazole-chalcone analogs of lonazolac as 5-LOX, iNOS and tubulin polymerization inhibitors with potential anticancer and anti-inflammatory activities
|
Ahmed, Asmaa H.H. |
|
|
129 |
C |
p. |
artikel |
21 |
Design, synthesis and pharmacological evaluation of 2-arylurea-1,3,5-triazine derivative (XIN-9): A novel potent dual PI3K/mTOR inhibitor for cancer therapy
|
Sun, Xin |
|
|
129 |
C |
p. |
artikel |
22 |
Design, synthesis, spectroscopic characterization, in vitro tyrosinase inhibition, antioxidant evaluation, in silico and kinetic studies of substituted indole-carbohydrazides
|
Iraji, Aida |
|
|
129 |
C |
p. |
artikel |
23 |
Development of a nitroreductase-dependent theranostic payload for antibody-drug conjugate
|
Su, Zheng |
|
|
129 |
C |
p. |
artikel |
24 |
Development of fluorescent dual-FRET probe for simultaneous detection of caspase-8 and caspase-9 activities and their relative quantification
|
Porubský, Martin |
|
|
129 |
C |
p. |
artikel |
25 |
Development of novel cyanopyridines as PIM-1 kinase inhibitors with potent anti-prostate cancer activity: Synthesis, biological evaluation, nanoparticles formulation and molecular dynamics simulation
|
Ibrahim, Mona H. |
|
|
129 |
C |
p. |
artikel |
26 |
Development of novel nitric oxide-releasing quinolinedione/furoxan hybrids as NQO1 inhibitors for intervention of drug-resistanthepatocellular cancer
|
Zhang, Xiaoyan |
|
|
129 |
C |
p. |
artikel |
27 |
Discovery of a potent EGFR and ALK dual mutation inhibitor containing N-(3-((4-((2-(cyclopropylsulfinyl)phenyl)amino)pyrimidin-2-yl)amino) phenyl)acrylamide scaffold
|
Li, Wei |
|
|
129 |
C |
p. |
artikel |
28 |
Discovery of bicyclic polyprenylated acylphloroglucinols from Hypericum himalaicum with glucose transporter 4 translocation activity
|
Cheng, Haitao |
|
|
129 |
C |
p. |
artikel |
29 |
Discovery of novel β-carboline-1,2,3-triazole hybrids as AChE/GSK-3β dual inhibitors for Alzheimer's disease treatment
|
Liu, Wenjie |
|
|
129 |
C |
p. |
artikel |
30 |
Discovery of novel dihydropyrazole-stilbene derivatives for ameliorating heart failure through modulation of p38/NF-κB signaling pathway
|
Liu, Zhigang |
|
|
129 |
C |
p. |
artikel |
31 |
Discovery of novel heterocyclic derivatives as potential glycogen phosphorylase inhibitors with a cardioprotective effect
|
Yan, Zhiwei |
|
|
129 |
C |
p. |
artikel |
32 |
Discovery of novel 1,2,4-triazole derivatives as xanthine oxidoreductase inhibitors with hypouricemic effects
|
Yang, Yajun |
|
|
129 |
C |
p. |
artikel |
33 |
Discovery of 12β-oxygenated oleanolic acid alkyl esters as potent and selective FXR modulators exhibiting hyperglycemia amelioration in vivo
|
Wang, Shaorong |
|
|
129 |
C |
p. |
artikel |
34 |
Discovery of potent and selective dual cholinesterases and β-secretase inhibitors in pomegranate as a treatment for Alzheimer’s disease
|
Yousof Ali, Md. |
|
|
129 |
C |
p. |
artikel |
35 |
Discovery of selective HDAC6 inhibitors capped by flavonoid or flavonoid-analogous moieties as anti-cancer therapeutics simultaneously harboring anti-proliferative and immunomodulatory activities
|
He, Ge |
|
|
129 |
C |
p. |
artikel |
36 |
Discovery, optimization and evaluation of isothiazolo[5,4-b]pyridine derivatives as RIPK1 inhibitors with potent in vivo anti-SIRS activity
|
Hao, Yongjin |
|
|
129 |
C |
p. |
artikel |
37 |
Dual-modal polypeptide-containing contrast agents for magnetic resonance/fluorescence imaging
|
Zheng, Si-Yao |
|
|
129 |
C |
p. |
artikel |
38 |
Editorial Board
|
|
|
|
129 |
C |
p. |
artikel |
39 |
Ethyl-4-(aryl)-6-methyl-2-(oxo/thio)-3,4-dihydro-1H-pyrimidine-5-carboxylates: Silica supported bismuth(III)triflate catalyzed synthesis and antioxidant activity
|
Gajjala, Raghavendra Reddy |
|
|
129 |
C |
p. |
artikel |
40 |
Eucarbwenstols A–H, eight novel compounds from Eucalyptus robusta prevents MPC-5 injury via ROS modulation and regulation of mitochondrial membrane potential
|
Chen, Ting |
|
|
129 |
C |
p. |
artikel |
41 |
Exploring the anti-influenza virus activity of novel triptolide derivatives targeting nucleoproteins
|
Jiang, Na |
|
|
129 |
C |
p. |
artikel |
42 |
Fragment-based discovery of orphan nuclear receptor Nur77/NGFI-B ligands
|
Arifi, Silvia |
|
|
129 |
C |
p. |
artikel |
43 |
Guaiane-type sesquiterpenoids with various ring skeletons from Daphne bholua uncovered by molecular networking and structural revisions of previously reported analogues
|
Dong, Shu-Hui |
|
|
129 |
C |
p. |
artikel |
44 |
HDAC/JAK dual target inhibitors of cancer-related targets: The success of nonclearable linked pharmacophore mode
|
Zhao, Liyun |
|
|
129 |
C |
p. |
artikel |
45 |
Hemicyanine-based pH-responsive probes for rapid hypoxia detection in cancer cells
|
Wangngae, Sirilak |
|
|
129 |
C |
p. |
artikel |
46 |
Human dihydrofolate reductase inhibition effect of 1-Phenylpyrazolo[3,4–d]pyrimidines: Synthesis, antitumor evaluation and molecular modeling study
|
Salem, Ibrahim M. |
|
|
129 |
C |
p. |
artikel |
47 |
Hydantoin based dual inhibitors of ALR2 and PARP-1: Design, synthesis, in-vitro and in-vivo evaluation
|
Kumar, Manoj |
|
|
129 |
C |
p. |
artikel |
48 |
Identification of a novel nitroflavone-based scaffold for designing mutant-selective EGFR tyrosine kinase inhibitors targeting T790M and C797S resistance in advanced NSCLC
|
Minnelli, Cristina |
|
|
129 |
C |
p. |
artikel |
49 |
Identification of thienopyrimidine glycinates as selective inhibitors for h-NTPDases
|
Begum, Zahra |
|
|
129 |
C |
p. |
artikel |
50 |
Isolation and synthesis of rocaglaol derivatives by inhibiting Wnt/β-catenin and MAPK signaling pathways against colorectal cancer
|
Li, Yanan |
|
|
129 |
C |
p. |
artikel |
51 |
1,2-Isoselenazol-3(2H)-one derivatives as NDM-1 inhibitors displaying synergistic antimicrobial effects with meropenem on NDM-1 producing clinical isolates
|
Yue, Kairui |
|
|
129 |
C |
p. |
artikel |
52 |
Issue TOC
|
|
|
|
129 |
C |
p. |
artikel |
53 |
Lactate dehydrogenase A inhibitors with a 2,8-dioxabicyclo[3.3.1]nonane scaffold: A contribution to molecular therapies for primary hyperoxalurias
|
Alejo-Armijo, Alfonso |
|
|
129 |
C |
p. |
artikel |
54 |
Mahanimbine isolated from Murraya koenigii inhibits P-glycoprotein involved in lung cancer chemoresistance
|
Mondal, Priya |
|
|
129 |
C |
p. |
artikel |
55 |
Mesenchymal stem cells-derived HIF-1α-overexpressed extracellular vesicles ameliorate hypoxia-induced pancreatic β cell apoptosis and senescence through activating YTHDF1-mediated protective autophagy
|
Fang, Jiali |
|
|
129 |
C |
p. |
artikel |
56 |
Mitochondria targeted dual-fluorescent probe for bio-imaging viscosity and F− with different fluorescence signals
|
Dhiman, Sukhvinder |
|
|
129 |
C |
p. |
artikel |
57 |
Natural carbazole alkaloid murrayafoline A displays potent anti-neuroinflammatory effect by directly targeting transcription factor Sp1 in LPS-induced microglial cells
|
Li, Chao-Hua |
|
|
129 |
C |
p. |
artikel |
58 |
Natural phenylethanoid glycosides diuretics derived from Lagopsis supina: Biological activity, mechanism, molecular docking, and structure-activity relationship
|
Yang, Li |
|
|
129 |
C |
p. |
artikel |
59 |
New anti-inflammatory and non-cytotoxic metabolites of methylstenbolone obtained by microbial transformation
|
Aamer, Muhammad |
|
|
129 |
C |
p. |
artikel |
60 |
New polyphenolic glycosides from the stems of Caesalpinia cucullata and their inhibitory effect on methicillin-resistant Staphylococcus aureus with different ways
|
Jing, Wenhua |
|
|
129 |
C |
p. |
artikel |
61 |
Nicotinonitrile-derived apoptotic inducers: Design, synthesis, X-ray crystal structure and Pim kinase inhibition
|
Aboukhatwa, Shaimaa M. |
|
|
129 |
C |
p. |
artikel |
62 |
Nitroreductase-induced bioorthogonal ligation for prodrug activation: A traceless strategy for cancer-specific imaging and therapy
|
Hu, Liangkui |
|
|
129 |
C |
p. |
artikel |
63 |
Novel chiral Schiff base Palladium(II), Nickel(II), Copper(II) and Iron(II) complexes: Synthesis, characterization, anticancer activity and molecular docking studies
|
Basaran, Eyüp |
|
|
129 |
C |
p. |
artikel |
64 |
Novel diaryl ether derivatives as InhA inhibitors: Design, synthesis and antimycobacterial activity
|
Abdelaziz, Ola A. |
|
|
129 |
C |
p. |
artikel |
65 |
Novel 1,3-diaryl pyrazole derivatives bearing methylsulfonyl moiety: Design, synthesis, molecular docking and dynamics, with dual activities as anti-inflammatory and anticancer agents through selectively targeting COX-2
|
Shaker, Ahmed M.M. |
|
|
129 |
C |
p. |
artikel |
66 |
Novel 5,6-diphenyl-1,2,4-triazine-3-thiol derivatives as dual COX-2/5-LOX inhibitors devoid of cardiotoxicity
|
Saraf, Poorvi |
|
|
129 |
C |
p. |
artikel |
67 |
Novel spirooxindole based benzimidazole scaffold: In vitro, nanoformulation and in vivo studies on anticancer and antimetastatic activity of breast adenocarcinoma
|
Barakat, Assem |
|
|
129 |
C |
p. |
artikel |
68 |
Novel synthesis naringenin-benzyl piperazine derivatives prevent glioblastoma invasion by inhibiting the hypoxia-induced IL6/JAK2/STAT3 axis and activating caspase-dependent apoptosis
|
Zaim, Ömer |
|
|
129 |
C |
p. |
artikel |
69 |
Optimization of a cell surface vimentin binding peptoid to extract antagonist effect on lung cancer cells
|
Zhang, Haowen |
|
|
129 |
C |
p. |
artikel |
70 |
Peptide inhibitors of angiotensin-I converting enzyme based on angiotensin (1–7) with selectivity for the C-terminal domain
|
da Silva, Rogerio L. |
|
|
129 |
C |
p. |
artikel |
71 |
Photodynamic antitumor activity of Gallium(III) and Phosphorus(V) complexes of trimethoxyl A2B triaryl corrole
|
Yang, Wu |
|
|
129 |
C |
p. |
artikel |
72 |
Prospect of ULK1 modulators in targeting regulatory T cells
|
Park, Youngjun |
|
|
129 |
C |
p. |
artikel |
73 |
Pseudoamaolides A-O, anti-inflammatory triterpene spiroketal lactones from seeds of Pseudolarix amabilis
|
Zhu, Yuxun |
|
|
129 |
C |
p. |
artikel |
74 |
Rational development of an ESIPT-based fluorescent probe with large Stokes shift for imaging of hydrogen sulfide in live cells
|
Du, Yuting |
|
|
129 |
C |
p. |
artikel |
75 |
Recent advances in transition metal-catalyzed reactions of chloroquinoxalines: Applications in bioorganic chemistry
|
Sujeevan Reddy, Gangireddy |
|
|
129 |
C |
p. |
artikel |
76 |
Repurposing N-hydroxy thienopyrimidine-2,4-diones (HtPD) as inhibitors of human cytomegalovirus pUL89 endonuclease: Synthesis and biological characterization
|
He, Tianyu |
|
|
129 |
C |
p. |
artikel |
77 |
SAR study of oxidative DIMs analogs targeting the Nur77-mediated apoptotic pathway of cancer cells
|
Chen, Xiaohui |
|
|
129 |
C |
p. |
artikel |
78 |
SAR study on Novel truxillic acid monoester-Based inhibitors of fatty acid binding proteins as Next-Generation antinociceptive agents
|
Wang, Hehe |
|
|
129 |
C |
p. |
artikel |
79 |
Sesquiterpene lactones from Elephantopus scaber exhibit cytotoxic effects on glioma cells by targeting GSTP1
|
Yan, Qiu-Lin |
|
|
129 |
C |
p. |
artikel |
80 |
Sonochemical synthesis and biological evaluation of isoquinolin-1(2H)-one/isoindolin-1-one derivatives: Discovery of a positive ago-allosteric modulator (PAAM) of 5HT2CR
|
Sandeep Kumar, Jetta |
|
|
129 |
C |
p. |
artikel |
81 |
Structure based design and synthesis of 3-(7-nitro-3-oxo-3,4-dihydroquinoxalin-2-yl)propanehydrazide derivatives as novel bacterial DNA-gyrase inhibitors: In-vitro, In-vivo, In-silico and SAR studies
|
Saleh, Marwa A. |
|
|
129 |
C |
p. |
artikel |
82 |
Structure-based screening and biological validation of the anti-thrombotic drug-dicoumarol as a novel and potent PPARγ-modulating ligand
|
Ma, Lei |
|
|
129 |
C |
p. |
artikel |
83 |
3-Substituted-2,3-Dihydrothiazole as a promising scaffold to design EGFR inhibitors
|
El-Haggar, Radwan |
|
|
129 |
C |
p. |
artikel |
84 |
Substituted phenethylamine-based β-lactam derivatives: Antimicrobial, anticancer, and β-lactamase inhibitory properties
|
Yildirim, Merve |
|
|
129 |
C |
p. |
artikel |
85 |
Synthesis and biological evaluation of novel dialkyl (4-amino-5H-chromeno[2,3-d]pyrimidin-5-yl)phosphonates
|
Sreelakshmi, Poola |
|
|
129 |
C |
p. |
artikel |
86 |
Synthesis and in vivo evaluation of new steviol derivatives that protect against cardiomyopathy by inhibiting ferroptosis
|
Xu, Chao |
|
|
129 |
C |
p. |
artikel |
87 |
Synthetic access to syn-functionalised chiral hydroxy pyrrolidines and pyrrolidones: Evaluation of α-glucosidase inhibition activity, docking studies and pharmacokinetics prediction
|
Mhaldar, Shashank N. |
|
|
129 |
C |
p. |
artikel |
88 |
Targeting neuronal calcium channels and GSK3β for Alzheimer’s disease with naturally-inspired Diels-Alder adducts
|
Bisi, Alessandra |
|
|
129 |
C |
p. |
artikel |
89 |
Targeting the kinetics mechanism of AMPA receptor inhibition by 2-oxo-3H-benzoxazole derivatives
|
Qneibi, Mohammad |
|
|
129 |
C |
p. |
artikel |
90 |
The Design, Structure–Activity, and kinetic studies of 3-Benzyl-5-oxa-1,2,3,4-Tetrahydro-2H-chromeno-(3,4-c)pyridin-8-yl sulfamates as Steroid sulfatase inhibitors
|
Chang, Chiao-Nien |
|
|
129 |
C |
p. |
artikel |
91 |
The multifaceted roles of peptides in “always-on” near-infrared fluorescent probes for tumor imaging
|
Xu, Haiwei |
|
|
129 |
C |
p. |
artikel |
92 |
Therapeutic potential of phospho-thiadiazole derivatives as anti-glioblastoma agents: synthesis, biological assessment and computational study
|
Gholivand, Khodayar |
|
|
129 |
C |
p. |
artikel |
93 |
Thiol-Michael addition based conjugate for glutathione activation and release
|
Liu, Zhengkun |
|
|
129 |
C |
p. |
artikel |
94 |
Versicotide G suppresses osteoclastogenesis and prevents osteolysis
|
Zhang, He |
|
|
129 |
C |
p. |
artikel |
95 |
Water-soluble dual lysosome/mitochondria-targeted fluorescent probe for detection of SO2 in water, food, herb, and live cells
|
Dong, Zhenming |
|
|
129 |
C |
p. |
artikel |