nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A bifunctional fluorescence probe for dual-channel detecting of mitochondrial viscosity and endogenous/exogenous peroxynitrite
|
Li, Minglu |
|
|
119 |
C |
p. |
artikel |
2 |
A coumarin-based fluorescent probe for specific detection of cysteine in the lysosome of living cells
|
Lu, Guowei |
|
|
119 |
C |
p. |
artikel |
3 |
An abiotic fluorescent probe for the detection and quantification of carcinoembryonic antigen
|
Lee, Jung-Seop |
|
|
119 |
C |
p. |
artikel |
4 |
A near-infrared, colorimetric and ratiometric fluorescent sensor with high sensitivity to hydrogen peroxide and viscosity for solutions detection and imaging living cells
|
Liu, Daili |
|
|
119 |
C |
p. |
artikel |
5 |
A novel Cereblon E3 ligase modulator with antitumor activity in gastrointestinal cancer
|
Lier, Svenja |
|
|
119 |
C |
p. |
artikel |
6 |
Antibacterial, antibiofilm, anti-inflammatory, and wound healing effects of nanoscale multifunctional cationic alternating copolymers
|
Hooshmand, Seyyed Emad |
|
|
119 |
C |
p. |
artikel |
7 |
Anti-inflammatory, ulcerogenic and platelet activation evaluation of novel 1,4-diaryl-1,2,3-triazole neolignan-celecoxib hybrids
|
Felipe, Josyelen L. |
|
|
119 |
C |
p. |
artikel |
8 |
Baicalin ameliorates 2,4-dinitrochlorobenzene-induced atopic dermatitis-like skin lesions in mice through modulating skin barrier function, gut microbiota and JAK/STAT pathway
|
Wang, Lan |
|
|
119 |
C |
p. |
artikel |
9 |
Biocatalytic one pot three component approach: Facile synthesis, characterization, molecular modelling and hypoglycemic studies of new thiazolidinedione festooned quinoline analogues catalyzed by alkaline protease from Aspergillus niger
|
Angajala, Gangadhara |
|
|
119 |
C |
p. |
artikel |
10 |
Chamaejasmenin E from Stellera chamaejasme induces apoptosis of hepatocellular carcinoma cells by targeting c-Met in vitro and in vivo
|
Yu, Xiao-Qi |
|
|
119 |
C |
p. |
artikel |
11 |
Click ferrocenyl-erlotinib conjugates active against erlotinib-resistant non-small cell lung cancer cells in vitro
|
Biegański, Przemysław |
|
|
119 |
C |
p. |
artikel |
12 |
Construction of synergistic pH/H2O2-responsive prodrug for prolonging blood circulation and accelerating cellular internalization
|
Liu, Jun |
|
|
119 |
C |
p. |
artikel |
13 |
Corrigendum to “Daphnegiravone D from Daphne giraldii induces cell death by targeting ATR in Hep3B cells” [Bioorg. Chem. 110 (2021) 104802]
|
Shang, Xin-Yue |
|
|
119 |
C |
p. |
artikel |
14 |
C6-structural optimizations of 2-aryl-1H-pyrazole-S-DABOs: From anti-HIV to anti-DENV activity
|
Rui, Ruo-Mei |
|
|
119 |
C |
p. |
artikel |
15 |
Cyclometalated Ru(II)-isoquinoline complexes overcome cisplatin resistance of A549/DDP cells by downregulation of Nrf2 via Akt/GSK-3β/Fyn pathway
|
Chen, Lanmei |
|
|
119 |
C |
p. |
artikel |
16 |
Degrading FLT3-ITD protein by proteolysis targeting chimera (PROTAC)
|
Chen, Yong |
|
|
119 |
C |
p. |
artikel |
17 |
Design and synthesis of epigallocatechin (EGC) analogs selective to inhibit α-amylase over α-glucosidases via the incorporation of caffeine acid and its derivatives
|
Chen, Wenming |
|
|
119 |
C |
p. |
artikel |
18 |
Design and synthesis of fluorinated peptides for analysis of fluorous effects on the interconversion of polyproline helices
|
Li, Meng-Che |
|
|
119 |
C |
p. |
artikel |
19 |
Design and synthesis of ibuprofen-quinoline conjugates as potential anti-inflammatory and analgesic drug candidates
|
Ghanim, Amany M. |
|
|
119 |
C |
p. |
artikel |
20 |
Design, synthesis and biological evaluation studies of novel small molecule ENPP1 inhibitors for cancer immunotherapy
|
Gangar, Mukesh |
|
|
119 |
C |
p. |
artikel |
21 |
Design, synthesis, and evaluation of novel pyridone derivatives as potent BRD4 inhibitors for the potential treatment of prostate cancer
|
Jiang, Wenhua |
|
|
119 |
C |
p. |
artikel |
22 |
Design, synthesis and SAR study of Fluorine-containing 3rd-generation taxoids
|
Wang, Changwei |
|
|
119 |
C |
p. |
artikel |
23 |
Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new anti-vitiligo compounds
|
Yang, Bi-juan |
|
|
119 |
C |
p. |
artikel |
24 |
Design, synthesis, biological screening and molecular docking studies of novel multifunctional 1,4-di (aryl/heteroaryl) substituted piperazine derivatives as potential antitubercular and antimicrobial agents
|
Mekonnen Sanka, Bruktawit |
|
|
119 |
C |
p. |
artikel |
25 |
Design, synthesis, in vitro antiproliferative evaluation and GSK-3β kinase inhibition of a new series of pyrimidin-4-one based amide conjugates
|
Khan, Imran |
|
|
119 |
C |
p. |
artikel |
26 |
Development of novel indolin-2-one derivative incorporating thiazole moiety as DHFR and quorum sensing inhibitors: Synthesis, antimicrobial, and antibiofilm activities with molecular modelling study
|
Alzahrani, Abdullah Y. |
|
|
119 |
C |
p. |
artikel |
27 |
Discovery of 7-alkyloxy- [1,2,4] triazolo[1,5-a] pyrimidine derivatives as selective positive modulators of GABAA1 and GABAA4 receptors with potent antiepileptic activity
|
Wu, Jun |
|
|
119 |
C |
p. |
artikel |
28 |
Discovery of linear unnatural peptides as potent mutant isocitrate dehydrogenase 1 inhibitors by Ugi reaction
|
Zhou, Xuechen |
|
|
119 |
C |
p. |
artikel |
29 |
Discovery of N-(2-benzyl-4-oxochroman-7-yl)-2-(5-(ethylsulfonyl) pyridin-2-yl) acetamide (b12) as a potent, selective, and orally available novel retinoic acid receptor-related orphan receptor γt inverse agonist
|
Chen, Lei |
|
|
119 |
C |
p. |
artikel |
30 |
Discovery of N-(1,3,4-thiadiazol-2-yl)benzamide derivatives containing a 6,7-methoxyquinoline structure as novel EGFR/HER-2 dual-target inhibitors against cancer growth and angiogenesis
|
Li, Xin-yang |
|
|
119 |
C |
p. |
artikel |
31 |
Discovery of pyrido[3,4-b]indol-1-one derivatives as novel non-covalent Bruton’s tyrosine kinase (BTK) inhibitors
|
Dou, Dou |
|
|
119 |
C |
p. |
artikel |
32 |
Discovery of urease inhibitory effect of sulfamate derivatives: Biological and computational studies
|
Zaib, Sumera |
|
|
119 |
C |
p. |
artikel |
33 |
Diterpenoids from Euphorbia helioscopia and their enhancement of NK cell-mediated killing of NSCLC cells
|
Mu, Hong-yan |
|
|
119 |
C |
p. |
artikel |
34 |
Downsizing antibodies: Towards complementarity-determining region (CDR)-based peptide mimetics
|
Van holsbeeck, Kevin |
|
|
119 |
C |
p. |
artikel |
35 |
Editorial Board
|
|
|
|
119 |
C |
p. |
artikel |
36 |
Euphoesulatin A prevents osteoclast differentiation and bone loss via inhibiting RANKL-induced ROS production and NF-κB and MAPK signal pathways
|
Zhang, Yu-ting |
|
|
119 |
C |
p. |
artikel |
37 |
Exploring the binding mode of ester-based cationic gemini surfactants with calf thymus DNA: A detailed physicochemical, spectroscopic and theoretical study
|
Akram, Mohd |
|
|
119 |
C |
p. |
artikel |
38 |
Hollongdione arylidene derivatives induce antiproliferative activity against melanoma and breast cancer through pro-apoptotic and antiangiogenic mechanisms
|
Smirnova, Irina |
|
|
119 |
C |
p. |
artikel |
39 |
H2O2-Responsive amphiphilic polymer with aggregation-induced emission (AIE) for DOX delivery and tumor therapy
|
Liang, Ya-Xuan |
|
|
119 |
C |
p. |
artikel |
40 |
Identification and synthesis of selective cholesterol esterase inhibitor using dynamic combinatorial chemistry
|
Zhao, Shuang |
|
|
119 |
C |
p. |
artikel |
41 |
Identification of NLRP3 as a covalent target of 1,6-O,O-diacetylbritannilactone against neuroinflammation by quantitative thiol reactivity profiling (QTRP)
|
Wang, Min-Ran |
|
|
119 |
C |
p. |
artikel |
42 |
3-Imino derivative-sulfahydantoins: Synthesis, in vitro antibacterial and cytotoxic activities and their DNA interactions
|
Başkan, Ceren |
|
|
119 |
C |
p. |
artikel |
43 |
Indoles and 1-(3-(benzyloxy)benzyl)piperazines: Reversible and selective monoamine oxidase B inhibitors identified by screening an in-house compound library
|
Knez, Damijan |
|
|
119 |
C |
p. |
artikel |
44 |
Isolation, identification, and activity evaluation of antioxidant components from Inula viscosa: A bioguided approach
|
Zeouk, Ikrame |
|
|
119 |
C |
p. |
artikel |
45 |
Issue TOC
|
|
|
|
119 |
C |
p. |
artikel |
46 |
Membrane mechanism of temporin-1CEc, an antimicrobial peptide isolated from the skin secretions of Rana chensinensis, and its systemic analogs
|
Ji, Fangyu |
|
|
119 |
C |
p. |
artikel |
47 |
Multifunctional fluorescent probes for high-throughput characterization of hexosaminidase enzyme activity
|
Wang, Shaochi |
|
|
119 |
C |
p. |
artikel |
48 |
Natural-product-inspired design and synthesis of two series of compounds active against Trypanosoma cruzi: Insights into structure–activity relationship, toxicity, and mechanism of action
|
da Rosa, Rafael |
|
|
119 |
C |
p. |
artikel |
49 |
New aniline derivatives from the volva of Phallus rubrovolvatus and their anti-inflammatory activity
|
Lv, Jianhua |
|
|
119 |
C |
p. |
artikel |
50 |
New enantiomeric lignans and new meroterpenoids with nitric oxide release inhibitory activity from Piper puberulum
|
Zheng, Yuan-kun |
|
|
119 |
C |
p. |
artikel |
51 |
Novel synthesis of antibacterial pyrone derivatives using kinetics and mechanism of oxidation of azithromycin by alkaline permanganate
|
Ibrahim, Samia M. |
|
|
119 |
C |
p. |
artikel |
52 |
Novel thiophene Chalcones-Coumarin as acetylcholinesterase inhibitors: Design, synthesis, biological evaluation, molecular docking, ADMET prediction and molecular dynamics simulation
|
Hasan, Aso Hameed |
|
|
119 |
C |
p. |
artikel |
53 |
Ortho-hydroxy bioactive schiff base compounds: Design, comprehensive characterization, photophysical properties and elucidation of antimicrobial and mutagenic potentials
|
Nıbras Qader Qader, Israa |
|
|
119 |
C |
p. |
artikel |
54 |
Platinum(II) and Copper(II) complexes of asymmetric halogen-substituted [NNʹO] ligands: Synthesis, characterization, structural investigations and antiproliferative activity
|
Amiri Rudbari, Hadi |
|
|
119 |
C |
p. |
artikel |
55 |
Rational design and synthesis of Oreoch-2 analogues as efficient broad-spectrum antimicrobial peptides
|
Zhang, Na |
|
|
119 |
C |
p. |
artikel |
56 |
Recent advances in the synthesis of naturally occurring tetronic acids
|
Princiotto, Salvatore |
|
|
119 |
C |
p. |
artikel |
57 |
Structural optimizations and bioevaluation of N-substituted acridone derivatives as strong topoisomerase II inhibitors
|
Li, Zhi-Ying |
|
|
119 |
C |
p. |
artikel |
58 |
Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activity
|
Ragab, Mahmoud A. |
|
|
119 |
C |
p. |
artikel |
59 |
Structure-Based design of Marine-derived Meridianin C derivatives as glycogen synthase kinase 3β inhibitors with improved oral bioavailability: From aminopyrimidyl-indoles to the sulfonyl analogues
|
Han, Shuwen |
|
|
119 |
C |
p. |
artikel |
60 |
Structure elucidation, biogenesis, and bioactivities of acylphloroglucinol-derived meroterpenoid enantiomers from Dryopteris crassirhizoma
|
Hai, Ping |
|
|
119 |
C |
p. |
artikel |
61 |
Synthesis and anti-inflammatory activities of glycyrrhetinic acid derivatives containing disulfide bond
|
Zhang, Qiuping |
|
|
119 |
C |
p. |
artikel |
62 |
Synthesis and biological evaluation of novel rhodanine-based structures with antiviral activity towards HHV-6 virus
|
Gentili, Valentina |
|
|
119 |
C |
p. |
artikel |
63 |
Synthesis and identification of a novel skeleton of N-(pyridin-3-yl) proline as a selective CDK4/6 inhibitor with anti-breast cancer activities
|
Liang, Jing-wei |
|
|
119 |
C |
p. |
artikel |
64 |
Synthesis and structure activity relationship of the first class of LXR inverse agonists
|
Elgendy, Bahaa |
|
|
119 |
C |
p. |
artikel |
65 |
Synthesis, anticancer evaluation and molecular docking of new benzothiazole scaffolds targeting FGFR-1
|
Abd El-Meguid, Eman A. |
|
|
119 |
C |
p. |
artikel |
66 |
Synthesis of N-aryl-2,6-diphenyl-2H-pyrazolo[4,3-c]pyridin-7-amines and their photodynamic properties in the human skin melanoma cell line G361
|
Razmienė, Beatričė |
|
|
119 |
C |
p. |
artikel |
67 |
Synthesis of new clioquinol derivatives as potent α-glucosidase inhibitors; molecular docking, kinetic and structure–activity relationship studies
|
Wali, Shoukat |
|
|
119 |
C |
p. |
artikel |
68 |
Synthesis of novel thiazolidinic-phthalimide derivatives evaluated as new multi-target antiepileptic agents
|
de Oliveira, Maria Cecilia V.A. |
|
|
119 |
C |
p. |
artikel |
69 |
Synthesis, structure, properties and antimicrobial activity of para trifluoromethyl phenylboronic derivatives
|
Adamczyk-Woźniak, Agnieszka |
|
|
119 |
C |
p. |
artikel |
70 |
Systemic pharmacological verification of Baixianfeng decoction regulating TNF-PI3K-Akt-NF-κB pathway in treating rheumatoid arthritis
|
Wei, Xin |
|
|
119 |
C |
p. |
artikel |
71 |
Tetrodecadazinone, a novel tetrodecamycin-pyridazinone hybrid with anti-liver fibrosis activity from Streptomyces sp. HU051
|
Liu, Ruo-Xi |
|
|
119 |
C |
p. |
artikel |
72 |
The C-terminal segment of Leishmania major HslU: Toward potential inhibitors of LmHslVU activity
|
Singh, Priyanka |
|
|
119 |
C |
p. |
artikel |
73 |
The molecular mechanism, targets, and novel molecules in the treatment of Alzheimer’s disease
|
Verma, Akash |
|
|
119 |
C |
p. |
artikel |
74 |
The role of remote flavin adenine dinucleotide pieces in the oxidative decarboxylation catalyzed by salicylate hydroxylase
|
Pereira, Mozart S. |
|
|
119 |
C |
p. |
artikel |
75 |
Total extract of Anemarrhenae Rhizoma attenuates bleomycin-induced pulmonary fibrosis in rats
|
Shen, Xue-Bin |
|
|
119 |
C |
p. |
artikel |
76 |
Utilization of cyanopyridine in design and synthesis of first-in-class anticancer dual acting PIM-1 kinase/HDAC inhibitors
|
Bass, Amr K.A. |
|
|
119 |
C |
p. |
artikel |
77 |
UV-guided isolation of enantiomeric polyacetylenes from Bupleurum scorzonerifolium Willd. with inhibitory effects against LPS-induced NO release in BV-2 microglial cells
|
Hong, Wei |
|
|
119 |
C |
p. |
artikel |
78 |
Virtual screening and in vitro validation of natural compound inhibitors against SARS-CoV-2 spike protein
|
Power, Helen |
|
|
119 |
C |
p. |
artikel |