Discovery of N-(2-benzyl-4-oxochroman-7-yl)-2-(5-(ethylsulfonyl) pyridin-2-yl) acetamide (b12) as a potent, selective, and orally available novel retinoic acid receptor-related orphan receptor γt inverse agonist
Titel:
Discovery of N-(2-benzyl-4-oxochroman-7-yl)-2-(5-(ethylsulfonyl) pyridin-2-yl) acetamide (b12) as a potent, selective, and orally available novel retinoic acid receptor-related orphan receptor γt inverse agonist
Auteur:
Chen, Lei Su, Mei Jin, Qiu Wang, Chun-Gu Assani, Israa Wang, Mu-Xuan Zhao, Shi-Feng Lv, Shen-Min Wang, Jia-Wei Sun, Bo Li, Yan Liao, Zhi-Xin