| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A FabG inhibitor targeting an allosteric binding site inhibits several orthologs from Gram-negative ESKAPE pathogens
|
Vella, Peter
|
|
|
30 |
C |
p.
|
artikel
|
| 2 |
Ancistrobrevidines A-C and related naphthylisoquinoline alkaloids with cytotoxic activities against HeLa and pancreatic cancer cells, from the liana Ancistrocladus abbreviatus
|
Fayez, Shaimaa
|
|
|
30 |
C |
p.
|
artikel
|
| 3 |
Assays for the identification and quantification of sialic acids: Challenges, opportunities and future perspectives
|
Cheeseman, Jack
|
|
|
30 |
C |
p.
|
artikel
|
| 4 |
A study of the structure-affinity relationship in SYA16263; is a D2 receptor interaction essential for inhibition of apormorphine-induced climbing behavior in mice?
|
Onyameh, Edem K.
|
|
|
30 |
C |
p.
|
artikel
|
| 5 |
Chemo-enzymatic synthesis of adenine substituted nicotinic acid adenine dinucleotide phosphate (NAADP) analogs
|
Su, Peiling
|
|
|
30 |
C |
p.
|
artikel
|
| 6 |
Design and synthesis of 14 and 15-membered macrocyclic scaffolds exhibiting inhibitory activities of hypoxia-inducible factor 1α
|
Shimizu, Takahiro
|
|
|
30 |
C |
p.
|
artikel
|
| 7 |
Design, synthesis and evaluation of PD-L1 peptide antagonists as new anticancer agents for immunotherapy
|
Orafaie, Ala
|
|
|
30 |
C |
p.
|
artikel
|
| 8 |
Discovery, development, chemical diversity and design of isoxazoline-based insecticides
|
Gonçalves, Itamar Luís
|
|
|
30 |
C |
p.
|
artikel
|
| 9 |
Discovery of a potent β-catenin destabilizer for overcoming the resistance of 5-fluorouracil in colorectal cancer
|
Ma, Kaiqing
|
|
|
30 |
C |
p.
|
artikel
|
| 10 |
Discovery of potent glycogen synthase kinase 3/cholinesterase inhibitors with neuroprotection as potential therapeutic agent for Alzheimer’s disease
|
Jiang, Xueyang
|
|
|
30 |
C |
p.
|
artikel
|
| 11 |
Editorial Board
|
|
|
|
30 |
C |
p.
|
artikel
|
| 12 |
Exploiting the antiproliferative potential of spiropyrazoline oxindoles in a human ovarian cancer cell line
|
Raposo, Luís R.
|
|
|
30 |
C |
p.
|
artikel
|
| 13 |
Graphical Abstract Contents Continued
|
|
|
|
30 |
C |
p.
|
artikel
|
| 14 |
Graphical abstract TOC
|
|
|
|
30 |
C |
p.
|
artikel
|
| 15 |
Graphical abstract TOC
|
|
|
|
30 |
C |
p.
|
artikel
|
| 16 |
Hit-to-lead optimization on aryloxybenzamide derivative virtual screening hit against SIRT
|
Yagci, Semih
|
|
|
30 |
C |
p.
|
artikel
|
| 17 |
Identification of N-acyl-N-indanyl-α-phenylglycinamides as selective TRPM8 antagonists designed to mitigate the risk of adverse effects
|
Kobayashi, Jun-ichi
|
|
|
30 |
C |
p.
|
artikel
|
| 18 |
In vitro and in vivo effects of inhibitors on actin and myosin
|
Richter, Sabine
|
|
|
30 |
C |
p.
|
artikel
|
| 19 |
JNK selective inhibitor, IQ-1S, protects the mice against lipopolysaccharides-induced sepsis
|
Nie, Zhelong
|
|
|
30 |
C |
p.
|
artikel
|
| 20 |
Lead optimization of 2-hydroxymethyl imidazoles as non-hydroxamate LpxC inhibitors: Discovery of TP0586532
|
Ushiyama, Fumihito
|
|
|
30 |
C |
p.
|
artikel
|
| 21 |
Lipophilic tail modifications of 2-(hydroxymethyl)pyrrolidine scaffold reveal dual sphingosine kinase 1 and 2 inhibitors
|
Li, Hao
|
|
|
30 |
C |
p.
|
artikel
|
| 22 |
MCC950, a NLRP3 inhibitor, ameliorates lipopolysaccharide-induced lung inflammation in mice
|
Wang, Lu
|
|
|
30 |
C |
p.
|
artikel
|
| 23 |
Methods to generate site-specific conjugates of antibody and protein
|
Park, Jisoo
|
|
|
30 |
C |
p.
|
artikel
|
| 24 |
Mitochondria-localizing curcumin-cryptolepine Zn(II) complexes and their antitumor activity
|
Qin, Li-Qin
|
|
|
30 |
C |
p.
|
artikel
|
| 25 |
Mono- and bis-pyrazolophthalazines: Design, synthesis, cytotoxic activity, DNA/HSA binding and molecular docking studies
|
Hamidinasab, Mahdia
|
|
|
30 |
C |
p.
|
artikel
|
| 26 |
Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181C
|
Gao, Ping
|
|
|
30 |
C |
p.
|
artikel
|
| 27 |
Novel potent (dihydro)benzofuranyl piperazines as human histamine receptor ligands – Functional characterization and modeling studies on H3 and H4 receptors
|
Corrêa, Michelle F.
|
|
|
30 |
C |
p.
|
artikel
|
| 28 |
Pegylated catalase as a potential alternative to treat vitiligo and UV induced skin damage
|
Santos, João H.P.M.
|
|
|
30 |
C |
p.
|
artikel
|
| 29 |
Porphyrin and phthalocyanine photosensitizers designed for targeted photodynamic therapy of colorectal cancer
|
Janas, Katarzyna
|
|
|
30 |
C |
p.
|
artikel
|
| 30 |
Potent leads based on CA-19L, an anti-HIV active HIV-1 capsid fragment
|
Tsuji, Kohei
|
|
|
30 |
C |
p.
|
artikel
|
| 31 |
Profiling protein expression in Klebsiella pneumoniae with a carbohydrate-based covalent probe
|
Metier, Camille C.
|
|
|
30 |
C |
p.
|
artikel
|
| 32 |
Quarternary α-cyanobenzylsulfonamides: A new subclass of CAA fungicides with excellent anti-Oomycetes activity
|
Stierli, Daniel
|
|
|
30 |
C |
p.
|
artikel
|
| 33 |
Ratiometric nanoprobe for circulating tumor cell detection and intracellular hydrogen peroxide evaluation in colorectal cancer patients
|
Pan, Ruijun
|
|
|
30 |
C |
p.
|
artikel
|
| 34 |
(S)-5′-C-Aminopropyl-2′-O-methyl nucleosides enhance antisense activity in cultured cells and binding affinity to complementary single-stranded RNA
|
Kajino, Ryohei
|
|
|
30 |
C |
p.
|
artikel
|
| 35 |
(S)-Erypoegin K, an isoflavone isolated from Erythrina poeppigiana, is a novel inhibitor of topoisomerase IIα: Induction of G2 phase arrest in human gastric cancer cells
|
Hikita, Kiyomi
|
|
|
30 |
C |
p.
|
artikel
|
| 36 |
Site-specific covalent labeling of His-tag fused proteins with N-acyl-N-alkyl sulfonamide reagent
|
Thimaradka, Vikram
|
|
|
30 |
C |
p.
|
artikel
|
| 37 |
Soloxolone methyl, as a 18βH-glycyrrhetinic acid derivate, may result in endoplasmic reticulum stress to induce apoptosis in breast cancer cells
|
Alper, Pinar
|
|
|
30 |
C |
p.
|
artikel
|
| 38 |
Synthesis and anticancer potential of novel 5,6-oxygenated and/or halogenated steroidal d-homo lactones
|
Kuzminac, Ivana Z.
|
|
|
30 |
C |
p.
|
artikel
|
| 39 |
Synthesis and evaluation of tiaprofenic acid-derived UCHL5 deubiquitinase inhibitors
|
Gurusingha Arachchige, Harshani S.
|
|
|
30 |
C |
p.
|
artikel
|
| 40 |
Synthesis, antitumor activity and structure-activity studies of novel pyridoxine-based bioisosteric analogs of estradiol
|
Pugachev, Mikhail V.
|
|
|
30 |
C |
p.
|
artikel
|
| 41 |
Synthesis, characterization, in vitro SAR study, and preliminary in vivo toxicity evaluation of naphthylmethyl substituted bis-imidazolium salts
|
Southerland, Marie R.
|
|
|
30 |
C |
p.
|
artikel
|
| 42 |
The 2′-caged-tethered-siRNA shows light-dependent temporal controlled RNAi activity for GFP gene into HEK293T cells
|
Bollu, Amarnath
|
|
|
30 |
C |
p.
|
artikel
|
| 43 |
[1,2,4]Triazolo[4,3-c]quinazoline and bis([1,2,4]triazolo)[4,3-a:4′,3′-c]quinazoline derived DNA intercalators: Design, synthesis, in silico ADMET profile, molecular docking and anti-proliferative evaluation studies
|
El-Adl, Khaled
|
|
|
30 |
C |
p.
|
artikel
|
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