Digital Library
Close Browse articles from a journal
     Journal description
       All volumes of the corresponding journal
         All issues of the corresponding volume
                                       All articles of the corresponding issues
 
                             43 results found
no title author magazine year volume issue page(s) type
1 A FabG inhibitor targeting an allosteric binding site inhibits several orthologs from Gram-negative ESKAPE pathogens Vella, Peter

30 C p.
article
2 Ancistrobrevidines A-C and related naphthylisoquinoline alkaloids with cytotoxic activities against HeLa and pancreatic cancer cells, from the liana Ancistrocladus abbreviatus Fayez, Shaimaa

30 C p.
article
3 Assays for the identification and quantification of sialic acids: Challenges, opportunities and future perspectives Cheeseman, Jack

30 C p.
article
4 A study of the structure-affinity relationship in SYA16263; is a D2 receptor interaction essential for inhibition of apormorphine-induced climbing behavior in mice? Onyameh, Edem K.

30 C p.
article
5 Chemo-enzymatic synthesis of adenine substituted nicotinic acid adenine dinucleotide phosphate (NAADP) analogs Su, Peiling

30 C p.
article
6 Design and synthesis of 14 and 15-membered macrocyclic scaffolds exhibiting inhibitory activities of hypoxia-inducible factor 1α Shimizu, Takahiro

30 C p.
article
7 Design, synthesis and evaluation of PD-L1 peptide antagonists as new anticancer agents for immunotherapy Orafaie, Ala

30 C p.
article
8 Discovery, development, chemical diversity and design of isoxazoline-based insecticides Gonçalves, Itamar Luís

30 C p.
article
9 Discovery of a potent β-catenin destabilizer for overcoming the resistance of 5-fluorouracil in colorectal cancer Ma, Kaiqing

30 C p.
article
10 Discovery of potent glycogen synthase kinase 3/cholinesterase inhibitors with neuroprotection as potential therapeutic agent for Alzheimer’s disease Jiang, Xueyang

30 C p.
article
11 Editorial Board
30 C p.
article
12 Exploiting the antiproliferative potential of spiropyrazoline oxindoles in a human ovarian cancer cell line Raposo, Luís R.

30 C p.
article
13 Graphical Abstract Contents Continued
30 C p.
article
14 Graphical abstract TOC
30 C p.
article
15 Graphical abstract TOC
30 C p.
article
16 Hit-to-lead optimization on aryloxybenzamide derivative virtual screening hit against SIRT Yagci, Semih

30 C p.
article
17 Identification of N-acyl-N-indanyl-α-phenylglycinamides as selective TRPM8 antagonists designed to mitigate the risk of adverse effects Kobayashi, Jun-ichi

30 C p.
article
18 In vitro and in vivo effects of inhibitors on actin and myosin Richter, Sabine

30 C p.
article
19 JNK selective inhibitor, IQ-1S, protects the mice against lipopolysaccharides-induced sepsis Nie, Zhelong

30 C p.
article
20 Lead optimization of 2-hydroxymethyl imidazoles as non-hydroxamate LpxC inhibitors: Discovery of TP0586532 Ushiyama, Fumihito

30 C p.
article
21 Lipophilic tail modifications of 2-(hydroxymethyl)pyrrolidine scaffold reveal dual sphingosine kinase 1 and 2 inhibitors Li, Hao

30 C p.
article
22 MCC950, a NLRP3 inhibitor, ameliorates lipopolysaccharide-induced lung inflammation in mice Wang, Lu

30 C p.
article
23 Methods to generate site-specific conjugates of antibody and protein Park, Jisoo

30 C p.
article
24 Mitochondria-localizing curcumin-cryptolepine Zn(II) complexes and their antitumor activity Qin, Li-Qin

30 C p.
article
25 Mono- and bis-pyrazolophthalazines: Design, synthesis, cytotoxic activity, DNA/HSA binding and molecular docking studies Hamidinasab, Mahdia

30 C p.
article
26 Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181C Gao, Ping

30 C p.
article
27 Novel potent (dihydro)benzofuranyl piperazines as human histamine receptor ligands – Functional characterization and modeling studies on H3 and H4 receptors Corrêa, Michelle F.

30 C p.
article
28 Pegylated catalase as a potential alternative to treat vitiligo and UV induced skin damage Santos, João H.P.M.

30 C p.
article
29 Porphyrin and phthalocyanine photosensitizers designed for targeted photodynamic therapy of colorectal cancer Janas, Katarzyna

30 C p.
article
30 Potent leads based on CA-19L, an anti-HIV active HIV-1 capsid fragment Tsuji, Kohei

30 C p.
article
31 Profiling protein expression in Klebsiella pneumoniae with a carbohydrate-based covalent probe Metier, Camille C.

30 C p.
article
32 Quarternary α-cyanobenzylsulfonamides: A new subclass of CAA fungicides with excellent anti-Oomycetes activity Stierli, Daniel

30 C p.
article
33 Ratiometric nanoprobe for circulating tumor cell detection and intracellular hydrogen peroxide evaluation in colorectal cancer patients Pan, Ruijun

30 C p.
article
34 (S)-5′-C-Aminopropyl-2′-O-methyl nucleosides enhance antisense activity in cultured cells and binding affinity to complementary single-stranded RNA Kajino, Ryohei

30 C p.
article
35 (S)-Erypoegin K, an isoflavone isolated from Erythrina poeppigiana, is a novel inhibitor of topoisomerase IIα: Induction of G2 phase arrest in human gastric cancer cells Hikita, Kiyomi

30 C p.
article
36 Site-specific covalent labeling of His-tag fused proteins with N-acyl-N-alkyl sulfonamide reagent Thimaradka, Vikram

30 C p.
article
37 Soloxolone methyl, as a 18βH-glycyrrhetinic acid derivate, may result in endoplasmic reticulum stress to induce apoptosis in breast cancer cells Alper, Pinar

30 C p.
article
38 Synthesis and anticancer potential of novel 5,6-oxygenated and/or halogenated steroidal d-homo lactones Kuzminac, Ivana Z.

30 C p.
article
39 Synthesis and evaluation of tiaprofenic acid-derived UCHL5 deubiquitinase inhibitors Gurusingha Arachchige, Harshani S.

30 C p.
article
40 Synthesis, antitumor activity and structure-activity studies of novel pyridoxine-based bioisosteric analogs of estradiol Pugachev, Mikhail V.

30 C p.
article
41 Synthesis, characterization, in vitro SAR study, and preliminary in vivo toxicity evaluation of naphthylmethyl substituted bis-imidazolium salts Southerland, Marie R.

30 C p.
article
42 The 2′-caged-tethered-siRNA shows light-dependent temporal controlled RNAi activity for GFP gene into HEK293T cells Bollu, Amarnath

30 C p.
article
43 [1,2,4]Triazolo[4,3-c]quinazoline and bis([1,2,4]triazolo)[4,3-a:4′,3′-c]quinazoline derived DNA intercalators: Design, synthesis, in silico ADMET profile, molecular docking and anti-proliferative evaluation studies El-Adl, Khaled

30 C p.
article
                             43 results found
 
 Koninklijke Bibliotheek - National Library of the Netherlands