| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A genetically selected cyclic peptide inhibitor of BCL6 homodimerization
|
Osher, Eliot L.
|
|
|
26 |
11 |
p. 3034-3038
|
artikel
|
| 2 |
A naphthalene diimide G-quadruplex ligand inhibits cell growth and down-regulates BCL-2 expression in an imatinib-resistant gastrointestinal cancer cell line
|
Gunaratnam, Mekala
|
|
|
26 |
11 |
p. 2958-2964
|
artikel
|
| 3 |
BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
|
Jennings, Laura E.
|
|
|
26 |
11 |
p. 2937-2957
|
artikel
|
| 4 |
Boronic acid inhibitors of the class A β-lactamase KPC-2
|
Zhou, Jingyuan
|
|
|
26 |
11 |
p. 2921-2927
|
artikel
|
| 5 |
Building bridges for highly selective, potent and stable oxytocin and vasopressin analogs
|
Beard, Rhiannon
|
|
|
26 |
11 |
p. 3039-3045
|
artikel
|
| 6 |
Design and synthesis of a fragment set based on twisted bicyclic lactams
|
Hassan, Haitham
|
|
|
26 |
11 |
p. 3030-3033
|
artikel
|
| 7 |
Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2
|
Moustakim, Moses
|
|
|
26 |
11 |
p. 2965-2972
|
artikel
|
| 8 |
Editorial
|
Fuchter, Matthew J.
|
|
|
26 |
11 |
p. 2919-2920
|
artikel
|
| 9 |
Editorial Board
|
|
|
|
26 |
11 |
p. ii
|
artikel
|
| 10 |
Graphical abstracts to be continued
|
|
|
|
26 |
11 |
p. I-III
|
artikel
|
| 11 |
Graphical abstract TOC
|
|
|
|
26 |
11 |
p. OBC
|
artikel
|
| 12 |
Graphical abstract TOC
|
|
|
|
26 |
11 |
p. IBC
|
artikel
|
| 13 |
Investigations on small molecule inhibitors targeting the histone H3K4 tri-methyllysine binding PHD-finger of JmjC histone demethylases
|
Bhushan, Bhaskar
|
|
|
26 |
11 |
p. 2984-2991
|
artikel
|
| 14 |
Novel non-ATP competitive small molecules targeting the CK2 α/β interface
|
Brear, Paul
|
|
|
26 |
11 |
p. 3016-3020
|
artikel
|
| 15 |
Practical application of ligand efficiency metrics in lead optimisation
|
Scott, James S.
|
|
|
26 |
11 |
p. 3006-3015
|
artikel
|
| 16 |
Site-selective installation of an electrophilic handle on proteins for bioconjugation
|
Lee, Bernadette
|
|
|
26 |
11 |
p. 3060-3064
|
artikel
|
| 17 |
Structure-activity relationships in a new class of non-substrate-like covalent inhibitors of the bacterial glycosyltransferase LgtC
|
Xu, Yong
|
|
|
26 |
11 |
p. 2973-2983
|
artikel
|
| 18 |
Structure activity relationship studies on rhodanines and derived enethiol inhibitors of metallo-β-lactamases
|
Zhang, Dong
|
|
|
26 |
11 |
p. 2928-2936
|
artikel
|
| 19 |
Synthesis and evaluation of aminobenzothiazoles as blockers of N- and T-type calcium channels
|
Sairaman, Anjali
|
|
|
26 |
11 |
p. 3046-3059
|
artikel
|
| 20 |
Synthesis and profiling of a 3-aminopyridin-2-one-based kinase targeted fragment library: Identification of 3-amino-5-(pyridin-4-yl)pyridin-2(1H)-one scaffold for monopolar spindle 1 (MPS1) and Aurora kinases inhibition
|
Fearon, Daren
|
|
|
26 |
11 |
p. 3021-3029
|
artikel
|
| 21 |
Synthesis and profiling of benzylmorpholine 1,2,4,5-tetraoxane analogue N205: Towards tetraoxane scaffolds with potential for single dose cure of malaria
|
O' Neill, Paul M.
|
|
|
26 |
11 |
p. 2996-3005
|
artikel
|
| 22 |
Thioamide substitution to probe the hydroxyproline recognition of VHL ligands
|
Soares, Pedro
|
|
|
26 |
11 |
p. 2992-2995
|
artikel
|
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