BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
Titel:
BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
Auteur:
Jennings, Laura E. Schiedel, Matthias Hewings, David S. Picaud, Sarah Laurin, Corentine M.C. Bruno, Paul A. Bluck, Joseph P. Scorah, Amy R. See, Larissa Reynolds, Jessica K. Moroglu, Mustafa Mistry, Ishna N. Hicks, Amy Guzanov, Pavel Clayton, James Evans, Charles N.G. Stazi, Giulia Biggin, Philip C. Mapp, Anna K. Hammond, Ester M. Humphreys, Philip G. Filippakopoulos, Panagis Conway, Stuart J.