| no |
title |
author |
magazine |
year |
volume |
issue |
page(s) |
type |
| 1 |
2-Aminomethylthieno[3,2-d]pyrimidin-4(3H)-ones bearing 3-methylpyrazole hinge binding moiety: Highly potent, selective, and time-dependent inhibitors of Cdc7 kinase
|
Kurasawa, Osamu
|
|
2017
|
25 |
14 |
p. 3658-3670
13 p.
|
article
|
| 2 |
A novel serine racemase inhibitor suppresses neuronal over-activation in vivo
|
Mori, Hisashi
|
|
2017
|
25 |
14 |
p. 3736-3745
10 p.
|
article
|
| 3 |
Carboxylated aurone derivatives as potent inhibitors of xanthine oxidase
|
Muzychka, Oksana V.
|
|
2017
|
25 |
14 |
p. 3606-3613
8 p.
|
article
|
| 4 |
Click strategy using disodium salts of amino acids improves the water solubility of plinabulin and KPU-300
|
Yakushiji, Fumika
|
|
2017
|
25 |
14 |
p. 3623-3630
8 p.
|
article
|
| 5 |
Design, synthesis and evaluation of indole-2-carboxamides with pan anti-mycobacterial activity
|
Franz, Nicholas D.
|
|
2017
|
25 |
14 |
p. 3746-3755
10 p.
|
article
|
| 6 |
Development of novel N-3-bromoisoxazolin-5-yl substituted 2,3-benzodiazepines as noncompetitive AMPAR antagonists
|
Espahbodinia, Milad
|
|
2017
|
25 |
14 |
p. 3631-3637
7 p.
|
article
|
| 7 |
Development of WNK signaling inhibitors as a new class of antihypertensive drugs
|
Ishigami-Yuasa, Mari
|
|
2017
|
25 |
14 |
p. 3845-3852
8 p.
|
article
|
| 8 |
Discovery of BI 135585, an in vivo efficacious oxazinanone-based 11β hydroxysteroid dehydrogenase type 1 inhibitor
|
Zhuang, Linghang
|
|
2017
|
25 |
14 |
p. 3649-3657
9 p.
|
article
|
| 9 |
Discovery of Novel and Potent Stearoyl Coenzyme A Desaturase 1 (SCD1) Inhibitors as Anticancer Agents
|
Imamura, Keisuke
|
|
2017
|
25 |
14 |
p. 3768-3779
12 p.
|
article
|
| 10 |
Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1H-spiro(naphthalene-2,2′-piperidin)-1-ones as potassium-competitive acid blockers
|
Imaeda, Toshihiro
|
|
2017
|
25 |
14 |
p. 3719-3735
17 p.
|
article
|
| 11 |
Diverse size approach to incorporate and extend highly fluorescent unnatural nucleotides into DNA
|
Le, Binh Huy
|
|
2017
|
25 |
14 |
p. 3591-3596
6 p.
|
article
|
| 12 |
Editorial board
|
|
|
2017
|
25 |
14 |
p. IFC-
1 p.
|
article
|
| 13 |
Effect of the 3-halo substitution of the 2′-deoxy aminopyridinyl-pseudocytidine derivatives on the selectivity and stability of antiparallel triplex DNA with a CG inversion site
|
Wang, Lei
|
|
2017
|
25 |
14 |
p. 3853-3860
8 p.
|
article
|
| 14 |
18F-Labeled indole-based analogs as highly selective radioligands for imaging sigma-2 receptors in the brain
|
Wang, Liang
|
|
2017
|
25 |
14 |
p. 3792-3802
11 p.
|
article
|
| 15 |
Halogen-substituted catechol bisphosphates are potent and selective inhibitors of the transcription factor STAT5b
|
Elumalai, Nagarajan
|
|
2017
|
25 |
14 |
p. 3871-3882
12 p.
|
article
|
| 16 |
Identification and preliminary structure–activity relationships of 1-Indanone derivatives as novel indoleamine-2,3-dioxygenase 1 (IDO1) inhibitors
|
Gao, Dingding
|
|
2017
|
25 |
14 |
p. 3780-3791
12 p.
|
article
|
| 17 |
Novel sulfonamide-containing 2-indolinones that selectively inhibit tumor-associated alpha carbonic anhydrases
|
Karalı, Nilgün
|
|
2017
|
25 |
14 |
p. 3714-3718
5 p.
|
article
|
| 18 |
Optimization and biological evaluation of 2-aminobenzothiazole derivatives as Aurora B kinase inhibitors
|
Lee, Eun
|
|
2017
|
25 |
14 |
p. 3614-3622
9 p.
|
article
|
| 19 |
Screening for bioactive natural products from a 67-compound library of Glycyrrhiza inflata
|
Lin, Yan
|
|
2017
|
25 |
14 |
p. 3706-3713
8 p.
|
article
|
| 20 |
Searching for novel N1-substituted benzimidazol-2-ones as non-nucleoside HIV-1 RT inhibitors
|
Ferro, Stefania
|
|
2017
|
25 |
14 |
p. 3861-3870
10 p.
|
article
|
| 21 |
Site-specific conjugation of fibroblast growth factor 2 (FGF2) based on incorporation of alkyne-reactive unnatural amino acid
|
Swiderska, K.W.
|
|
2017
|
25 |
14 |
p. 3685-3693
9 p.
|
article
|
| 22 |
Structure-activity relationships for flavone interactions with amyloid β reveal a novel anti-aggregatory and neuroprotective effect of 2′,3′,4′-trihydroxyflavone (2-D08)
|
Marsh, Dylan T.
|
|
2017
|
25 |
14 |
p. 3827-3834
8 p.
|
article
|
| 23 |
Succinamide derivatives of melampomagnolide B and their anti-cancer activities
|
Janganati, Venumadhav
|
|
2017
|
25 |
14 |
p. 3694-3705
12 p.
|
article
|
| 24 |
Synthesis and anticancer activity of novel aza-artemisinin derivatives
|
Jana, Sampad
|
|
2017
|
25 |
14 |
p. 3671-3676
6 p.
|
article
|
| 25 |
Synthesis and evaluation of c-di-4′-thioAMP as an artificial ligand for c-di-AMP riboswitch
|
Shiraishi, Kazuto
|
|
2017
|
25 |
14 |
p. 3883-3889
7 p.
|
article
|
| 26 |
Synthesis and evaluation of novel dual BRD4/HDAC inhibitors
|
Amemiya, Seika
|
|
2017
|
25 |
14 |
p. 3677-3684
8 p.
|
article
|
| 27 |
Synthesis and pharmacological evaluation of novel chromone derivatives as balanced multifunctional agents against Alzheimer's disease
|
Li, Fan
|
|
2017
|
25 |
14 |
p. 3815-3826
12 p.
|
article
|
| 28 |
Synthesis and preliminary biological evaluation of radiolabeled 5-BDBD analogs as new candidate PET radioligands for P2X4 receptor
|
Wang, Min
|
|
2017
|
25 |
14 |
p. 3835-3844
10 p.
|
article
|
| 29 |
Synthesis of nοvel artemisinin dimers with polyamine linkers and evaluation of their potential as anticancer agents
|
Magoulas, George E.
|
|
2017
|
25 |
14 |
p. 3756-3767
12 p.
|
article
|
| 30 |
Synthesis of oligonucleotides containing novel G-clamp analogue with C8-tethered group in phenoxazine ring: Implication to qPCR detection of the low-copy Kemerovo virus dsRNA
|
Varizhuk, Anna M.
|
|
2017
|
25 |
14 |
p. 3597-3605
9 p.
|
article
|
| 31 |
Synthesis, spectroscopic characterization and biological evaluation of unsymmetrical aminosquarylium cyanine dyes
|
Friães, Sofia
|
|
2017
|
25 |
14 |
p. 3803-3814
12 p.
|
article
|
| 32 |
The impact of the halogen bonding on D2 and 5-HT1A/5-HT7 receptor activity of azinesulfonamides of 4-[(2-ethyl)piperidinyl-1-yl]phenylpiperazines with antipsychotic and antidepressant properties
|
Partyka, Anna
|
|
2017
|
25 |
14 |
p. 3638-3648
11 p.
|
article
|
Journal description