Discovery of BI 135585, an in vivo efficacious oxazinanone-based 11β hydroxysteroid dehydrogenase type 1 inhibitor
Titel:
Discovery of BI 135585, an in vivo efficacious oxazinanone-based 11β hydroxysteroid dehydrogenase type 1 inhibitor
Auteur:
Zhuang, Linghang Tice, Colin M. Xu, Zhenrong Zhao, Wei Cacatian, Salvacion Ye, Yuan-Jie Singh, Suresh B. Lindblom, Peter McKeever, Brian M. Krosky, Paula M. Zhao, Yi Lala, Deepak Kruk, Barbara A. Meng, Shi Howard, Lamont Johnson, Judith A. Bukhtiyarov, Yuri Panemangalore, Reshma Guo, Joan Guo, Rong Himmelsbach, Frank Hamilton, Bradford Schuler-Metz, Annette Schauerte, Heike Gregg, Richard McGeehan, Gerard M. Leftheris, Katerina Claremon, David A.