| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibition
|
Igawa, Hideyuki
|
|
2016
|
24 |
11 |
p. 2486-2503
18 p.
|
artikel
|
| 2 |
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel non-basic 1-(2H-indazole-5-yl)pyridin-2(1H)-one derivatives and mitigation of mutagenicity in Ames test
|
Igawa, Hideyuki
|
|
2016
|
24 |
11 |
p. 2504-2518
15 p.
|
artikel
|
| 3 |
Antiplasmodial phloroglucinol derivatives from Syncarpia glomulifera
|
Su, Qingxi
|
|
2016
|
24 |
11 |
p. 2544-2548
5 p.
|
artikel
|
| 4 |
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists
|
Vergelli, Claudia
|
|
2016
|
24 |
11 |
p. 2530-2543
14 p.
|
artikel
|
| 5 |
1,6-Bis[(benzyloxy)methyl]uracil derivatives—Novel antivirals with activity against HIV-1 and influenza H1N1 virus
|
Geisman, Alexander N.
|
|
2016
|
24 |
11 |
p. 2476-2485
10 p.
|
artikel
|
| 6 |
Cytoprotective small molecule modulators of endoplasmic reticulum stress
|
Munshi, Soumyabrata
|
|
2016
|
24 |
11 |
p. 2382-2388
7 p.
|
artikel
|
| 7 |
Design, discovery, modelling, synthesis, and biological evaluation of novel and small, low toxicity s-triazine derivatives as HIV-1 non-nucleoside reverse transcriptase inhibitors
|
Viira, Birgit
|
|
2016
|
24 |
11 |
p. 2519-2529
11 p.
|
artikel
|
| 8 |
Design, synthesis and biological evaluation of benzyloxyphenyl-methylaminophenol derivatives as STAT3 signaling pathway inhibitors
|
Gao, Dingding
|
|
2016
|
24 |
11 |
p. 2549-2558
10 p.
|
artikel
|
| 9 |
Design, synthesis and in vitro evaluation studies of sulfonyl-amino-acetamides as small molecule BACE-1 inhibitors
|
Jain, Priti
|
|
2016
|
24 |
11 |
p. 2567-2575
9 p.
|
artikel
|
| 10 |
Discovery and optimization of 1,7-disubstituted-2,2-dimethyl-2,3-dihydroquinazolin-4(1H)-ones as potent and selective PKCθ inhibitors
|
Katoh, Taisuke
|
|
2016
|
24 |
11 |
p. 2466-2475
10 p.
|
artikel
|
| 11 |
3D-QSAR-aided design, synthesis, in vitro and in vivo evaluation of dipeptidyl boronic acid proteasome inhibitors and mechanism studies
|
Lei, Meng
|
|
2016
|
24 |
11 |
p. 2576-2588
13 p.
|
artikel
|
| 12 |
Editorial board
|
|
|
2016
|
24 |
11 |
p. IFC-
1 p.
|
artikel
|
| 13 |
Exploration of 3-methylisoquinoline-4-carbonitriles as protein kinase A inhibitors of Plasmodium falciparum
|
Buskes, Melissa J.
|
|
2016
|
24 |
11 |
p. 2389-2396
8 p.
|
artikel
|
| 14 |
Highly efficient method for 125I-radiolabeling of biomolecules using inverse-electron-demand Diels–Alder reaction
|
Choi, Mi Hee
|
|
2016
|
24 |
11 |
p. 2589-2594
6 p.
|
artikel
|
| 15 |
New imidazoquinoxaline derivatives: Synthesis, biological evaluation on melanoma, effect on tubulin polymerization and structure–activity relationships
|
Zghaib, Zahraa
|
|
2016
|
24 |
11 |
p. 2433-2440
8 p.
|
artikel
|
| 16 |
Quinazolines and quinazolinones as ubiquitous structural fragments in medicinal chemistry: An update on the development of synthetic methods and pharmacological diversification
|
Khan, Imtiaz
|
|
2016
|
24 |
11 |
p. 2361-2381
21 p.
|
artikel
|
| 17 |
Substituted quinolines as noncovalent proteasome inhibitors
|
McDaniel, Tanner J.
|
|
2016
|
24 |
11 |
p. 2441-2450
10 p.
|
artikel
|
| 18 |
Synergistic reduction of HIV-1 infectivity by 5-azacytidine and inhibitors of ribonucleotide reductase
|
Rawson, Jonathan M.O.
|
|
2016
|
24 |
11 |
p. 2410-2422
13 p.
|
artikel
|
| 19 |
Synthesis and biological evaluation of sialyl-oligonucleotide conjugates targeting leukocyte B trans-membranal receptor CD22 as delivery agents for nucleic acid drugs
|
St-Pierre, Gabrielle
|
|
2016
|
24 |
11 |
p. 2397-2409
13 p.
|
artikel
|
| 20 |
Synthesis and evaluation of 4-(2-hydroxypropyl)piperazin-1-yl) derivatives as Hsp90 inhibitors
|
Cherfaoui, Bahidja
|
|
2016
|
24 |
11 |
p. 2423-2432
10 p.
|
artikel
|
| 21 |
Synthesis of novel amide and urea derivatives of thiazol-2-ethylamines and their activity against Trypanosoma brucei rhodesiense
|
Patrick, Donald A.
|
|
2016
|
24 |
11 |
p. 2451-2465
15 p.
|
artikel
|
| 22 |
Synthesis of 24(S)-hydroxycholesterol esters responsible for the induction of neuronal cell death
|
Shibuya, Kimiyuki
|
|
2016
|
24 |
11 |
p. 2559-2566
8 p.
|
artikel
|
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