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Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibition |
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Titel: |
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibition |
Auteur: |
Igawa, Hideyuki Takahashi, Masashi Shirasaki, Mikio Kakegawa, Keiko Kina, Asato Ikoma, Minoru Aida, Jumpei Yasuma, Tsuneo Okuda, Shoki Kawata, Yayoi Noguchi, Toshihiro Yamamoto, Syunsuke Fujioka, Yasushi Kundu, Mrinalkanti Khamrai, Uttam Nakayama, Masaharu Nagisa, Yasutaka Kasai, Shizuo Maekawa, Tsuyoshi |
Verschenen in: |
Bioorganic & medicinal chemistry |
Paginering: |
Jaargang 24 (2016) nr. 11 pagina's 18 p. |
Jaar: |
2016 |
Inhoud: |
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Uitgever: |
Elsevier Ltd |
Bronbestand: |
Elektronische Wetenschappelijke Tijdschriften |
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