| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Arylazolyl(azinyl)thioacetanilides. Part 16: Structure-based bioisosterism design, synthesis and biological evaluation of novel pyrimidinylthioacetanilides as potent HIV-1 inhibitors
|
Li, Xiao
|
|
2014
|
22 |
19 |
p. 5290-5297
8 p.
|
artikel
|
| 2 |
Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII
|
Riafrecha, Leonardo E.
|
|
2014
|
22 |
19 |
p. 5308-5314
7 p.
|
artikel
|
| 3 |
Design and discovery of 5-hydroxy-6-oxo-1,6-dihydropyrimidine-4-carboxamide inhibitors of HIV-1 integrase
|
Zhang, Daoguang
|
|
2014
|
22 |
19 |
p. 5446-5453
8 p.
|
artikel
|
| 4 |
Design, synthesis and biological evaluation of novel 6H-benzo[c]chromen-6-one, and 7,8,9,10-tetrahydro-benzo[c]chromen-6-one derivatives as potential cholinesterase inhibitors
|
Gulcan, Hayrettin Ozan
|
|
2014
|
22 |
19 |
p. 5141-5154
14 p.
|
artikel
|
| 5 |
Design, synthesis and evaluation of 2-aminothiazole derivatives as sphingosine kinase inhibitors
|
Vogt, Dominik
|
|
2014
|
22 |
19 |
p. 5354-5367
14 p.
|
artikel
|
| 6 |
Design, synthesis and in vitro pharmacology of GluK1 and GluK3 antagonists. Studies towards the design of subtype-selective antagonists through 2-carboxyethyl-phenylalanines with substituents interacting with non-conserved residues in the GluK binding sites
|
Sköld, Niklas
|
|
2014
|
22 |
19 |
p. 5368-5377
10 p.
|
artikel
|
| 7 |
Design, synthesis and SAR exploration of tri-substituted 1,2,4-triazoles as inhibitors of the annexin A2–S100A10 protein interaction
|
Reddy, Tummala R.K.
|
|
2014
|
22 |
19 |
p. 5378-5391
14 p.
|
artikel
|
| 8 |
Development of p-carborane-based nonsteroidal progesterone receptor antagonists
|
Fujii, Shinya
|
|
2014
|
22 |
19 |
p. 5329-5337
9 p.
|
artikel
|
| 9 |
Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
|
Hasui, Tomoaki
|
|
2014
|
22 |
19 |
p. 5428-5445
18 p.
|
artikel
|
| 10 |
Editorial board
|
|
|
2014
|
22 |
19 |
p. IFC-
1 p.
|
artikel
|
| 11 |
Flexible, polymer-supported synthesis of sphingosine derivatives provides ceramides with enhanced biological activity
|
El-Dahshan, Adeeb
|
|
2014
|
22 |
19 |
p. 5506-5512
7 p.
|
artikel
|
| 12 |
From human immunodeficiency virus non-nucleoside reverse transcriptase inhibitors to potent and selective antitrypanosomal compounds
|
Venkatraj, Muthusamy
|
|
2014
|
22 |
19 |
p. 5241-5248
8 p.
|
artikel
|
| 13 |
Graphical contents list
|
|
|
2014
|
22 |
19 |
p. 5123-5132
10 p.
|
artikel
|
| 14 |
Hepatocyte-targeting gene delivery using a lipoplex composed of galactose-modified aromatic lipid synthesized with click chemistry
|
Sakashita, Mizuha
|
|
2014
|
22 |
19 |
p. 5212-5219
8 p.
|
artikel
|
| 15 |
Incorporation of triphenylphosphonium functionality improves the inhibitory properties of phenothiazine derivatives in Mycobacterium tuberculosis
|
Dunn, Elyse A.
|
|
2014
|
22 |
19 |
p. 5320-5328
9 p.
|
artikel
|
| 16 |
Love–Hate ligands for high resolution analysis of strain in ultra-stable protein/small molecule interaction
|
Fairhead, Michael
|
|
2014
|
22 |
19 |
p. 5476-5486
11 p.
|
artikel
|
| 17 |
Novel chromogenic aminopeptidase substrates for the detection and identification of clinically important microorganisms
|
Cellier, Marie
|
|
2014
|
22 |
19 |
p. 5249-5269
21 p.
|
artikel
|
| 18 |
Novel fluorinated pyrrolo[1,2-a]pyrazine-2,6-dione derivatives: Synthesis and anticonvulsant evaluation in animal models of epilepsy
|
Dawidowski, Maciej
|
|
2014
|
22 |
19 |
p. 5410-5427
18 p.
|
artikel
|
| 19 |
Optimization of physicochemical properties and safety profile of novel bacterial topoisomerase type II inhibitors (NBTIs) with activity against Pseudomonas aeruginosa
|
Reck, Folkert
|
|
2014
|
22 |
19 |
p. 5392-5409
18 p.
|
artikel
|
| 20 |
Oxadiazoles and thiadiazoles: Novel α-glucosidase inhibitors
|
Kashtoh, Hamdy
|
|
2014
|
22 |
19 |
p. 5454-5465
12 p.
|
artikel
|
| 21 |
Prodrug oncrasin-266 improves the stability, pharmacokinetics, and safety of NSC-743380
|
Wu, Shuhong
|
|
2014
|
22 |
19 |
p. 5234-5240
7 p.
|
artikel
|
| 22 |
Pyrazolone–quinazolone hybrids: A novel class of human 4-hydroxyphenylpyruvate dioxygenase inhibitors
|
Xu, Yu-Ling
|
|
2014
|
22 |
19 |
p. 5194-5211
18 p.
|
artikel
|
| 23 |
Quinazoline–sulfonamides with potent inhibitory activity against the α-carbonic anhydrase from Vibrio cholerae
|
Alafeefy, Ahmed M.
|
|
2014
|
22 |
19 |
p. 5133-5140
8 p.
|
artikel
|
| 24 |
Semi-synthesis of biologically active nisin hybrids composed of the native lanthionine ABC-fragment and a cross-stapled synthetic DE-fragment
|
Slootweg, Jack C.
|
|
2014
|
22 |
19 |
p. 5345-5353
9 p.
|
artikel
|
| 25 |
Shogaol–huprine hybrids: Dual antioxidant and anticholinesterase agents with β-amyloid and tau anti-aggregating properties
|
Pérez-Areales, F. Javier
|
|
2014
|
22 |
19 |
p. 5298-5307
10 p.
|
artikel
|
| 26 |
Synthesis and biological evaluation of podophyllotoxin congeners as tubulin polymerization inhibitors
|
Kamal, Ahmed
|
|
2014
|
22 |
19 |
p. 5466-5475
10 p.
|
artikel
|
| 27 |
Synthesis and biological evaluation of 1,2,3-triazole linked aminocombretastatin conjugates as mitochondrial mediated apoptosis inducers
|
Kamal, Ahmed
|
|
2014
|
22 |
19 |
p. 5155-5167
13 p.
|
artikel
|
| 28 |
Synthesis and evaluation of a 18F-labeled spirocyclic piperidine derivative as promising σ1 receptor imaging agent
|
Chen, Yuan-Yuan
|
|
2014
|
22 |
19 |
p. 5270-5278
9 p.
|
artikel
|
| 29 |
Synthesis and structure–activity relationships of novel, potent, orally active hypoxia-inducible factor-1 inhibitors
|
Nagao, Satoshi
|
|
2014
|
22 |
19 |
p. 5513-5529
17 p.
|
artikel
|
| 30 |
Synthesis, anti-cancer and anti-inflammatory activity of novel 2-substituted isoflavenes
|
Eiffe, Eleanor
|
|
2014
|
22 |
19 |
p. 5182-5193
12 p.
|
artikel
|
| 31 |
Synthesis of fluorinated analogues of sphingosine-1-phosphate antagonists as potential radiotracers for molecular imaging using positron emission tomography
|
Prasad, Vysakh Pushpa
|
|
2014
|
22 |
19 |
p. 5168-5181
14 p.
|
artikel
|
| 32 |
Synthesis of α-l-rhamnosyl ceramide and evaluation of its binding with anti-rhamnose antibodies
|
Long, David E.
|
|
2014
|
22 |
19 |
p. 5279-5289
11 p.
|
artikel
|
| 33 |
Synthesis of non-prenyl analogues of baccharin as selective and potent inhibitors for aldo-keto reductase 1C3
|
Endo, Satoshi
|
|
2014
|
22 |
19 |
p. 5220-5233
14 p.
|
artikel
|
| 34 |
Synthetic (+)-terrein suppresses interleukin-6/soluble interleukin-6 receptor induced-secretion of vascular endothelial growth factor in human gingival fibroblasts
|
Mandai, Hiroki
|
|
2014
|
22 |
19 |
p. 5338-5344
7 p.
|
artikel
|
| 35 |
The enantiomers of the 1′,6′-isomer of neplanocin A: Synthesis and antiviral properties
|
Ye, Wei
|
|
2014
|
22 |
19 |
p. 5315-5319
5 p.
|
artikel
|
| 36 |
Thieno[2,3-d]pyrimidine-2-carboxamides bearing a carboxybenzene group at 5-position: Highly potent, selective, and orally available MMP-13 inhibitors interacting with the S1″ binding site
|
Nara, Hiroshi
|
|
2014
|
22 |
19 |
p. 5487-5505
19 p.
|
artikel
|
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