Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
Titel:
Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
Auteur:
Hasui, Tomoaki Ohyabu, Norio Ohra, Taiichi Fuji, Koji Sugimoto, Takahiro Fujimoto, Jun Asano, Kouhei Oosawa, Masato Shiotani, Sachiko Nishigaki, Nobuhiro Kusumoto, Keiji Matsui, Hideki Mizukami, Atsushi Habuka, Noriyuki Sogabe, Satoshi Endo, Satoshi Ono, Midori Siedem, Christopher S. Tang, Tony P. Gauthier, Cassandra De Meese, Lisa A. Boyd, Steven A. Fukumoto, Shoji