Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
Title:
Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
Author:
Hasui, Tomoaki Ohyabu, Norio Ohra, Taiichi Fuji, Koji Sugimoto, Takahiro Fujimoto, Jun Asano, Kouhei Oosawa, Masato Shiotani, Sachiko Nishigaki, Nobuhiro Kusumoto, Keiji Matsui, Hideki Mizukami, Atsushi Habuka, Noriyuki Sogabe, Satoshi Endo, Satoshi Ono, Midori Siedem, Christopher S. Tang, Tony P. Gauthier, Cassandra De Meese, Lisa A. Boyd, Steven A. Fukumoto, Shoji