| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Comparative analysis of the dual EGFR-DNA targeting and growth inhibitory properties of 6-mono-alkylamino- and 6,6-dialkylaminoquinazoline-based type II combi-molecules
|
Schmitt, Julie
|
|
|
192 |
C |
p.
|
artikel
|
| 2 |
Crystal structure of O-Acetylserine sulfhydralase (OASS) isoform 3 from Entamoeba histolytica: Pharmacophore-based virtual screening and validation of novel inhibitors
|
Dharavath, Sudhaker
|
|
|
192 |
C |
p.
|
artikel
|
| 3 |
Cyclometalated Ir(III)-8-oxychinolin complexes acting as red-colored probes for specific mitochondrial imaging and anticancer drugs
|
Meng, Ting
|
|
|
192 |
C |
p.
|
artikel
|
| 4 |
Design and synthesis of selective degraders of EGFRL858R/T790M mutant
|
Zhang, Xin
|
|
|
192 |
C |
p.
|
artikel
|
| 5 |
Design and synthesis of tripeptidyl furylketones as selective inhibitors against the β5 subunit of human 20S proteasome
|
Sun, Qi
|
|
|
192 |
C |
p.
|
artikel
|
| 6 |
Design, synthesis and biological evaluation of novel indazole-based derivatives as potent HDAC inhibitors via fragment-based virtual screening
|
Liu, Jian
|
|
|
192 |
C |
p.
|
artikel
|
| 7 |
Design, synthesis, and evaluation of new 2-(quinoline-4-yloxy)acetamide-based antituberculosis agents
|
Borsoi, Ana Flávia
|
|
|
192 |
C |
p.
|
artikel
|
| 8 |
Design, synthesis, and evaluation of N-phenyl-4-(2-phenylsulfonamido)-benzamides as microtubule-targeting agents in drug-resistant cancer cells, displaying HDAC inhibitory response
|
Wu, Wei-Cheng
|
|
|
192 |
C |
p.
|
artikel
|
| 9 |
Development of bivalent triarylalkene- and cyclofenil-derived dual estrogen receptor antagonists and downregulators
|
Knox, Alexandra
|
|
|
192 |
C |
p.
|
artikel
|
| 10 |
Diarylpentanoids with antitumor activity: A critical review of structure-activity relationship studies
|
Moreira, Joana
|
|
|
192 |
C |
p.
|
artikel
|
| 11 |
Discovery of a promising agent IQZ23 for the treatment of obesity and related metabolic disorders
|
Rao, Yong
|
|
|
192 |
C |
p.
|
artikel
|
| 12 |
Discovery of 1,6-naphthyridinone-based MET kinase inhibitor bearing quinoline moiety as promising antitumor drug candidate
|
Chen, Tao
|
|
|
192 |
C |
p.
|
artikel
|
| 13 |
Discovery of novel tertiary amide derivatives as NEDDylation pathway activators to inhibit the tumor progression in vitro and in vivo
|
Fu, Dong-Jun
|
|
|
192 |
C |
p.
|
artikel
|
| 14 |
Discovery of PROTAC BCL-XL degraders as potent anticancer agents with low on-target platelet toxicity
|
Zhang, Xuan
|
|
|
192 |
C |
p.
|
artikel
|
| 15 |
Discovery of pyrazole derivatives as cellular active inhibitors of histone lysine specific demethylase 5B (KDM5B/JARID1B)
|
Zhao, Bing
|
|
|
192 |
C |
p.
|
artikel
|
| 16 |
Discovery of pyridine tetrahydroisoquinoline thiohydantoin derivatives with low blood-brain barrier penetration as the androgen receptor antagonists
|
Xu, Xi
|
|
|
192 |
C |
p.
|
artikel
|
| 17 |
Editorial Board
|
|
|
|
192 |
C |
p.
|
artikel
|
| 18 |
Fluorinated derivatives of 2-phenyl-3-hydroxy-4(1H)-quinolinone as tubulin polymerization inhibitors
|
Řehulka, Jiří
|
|
|
192 |
C |
p.
|
artikel
|
| 19 |
Graphical abstract TOC
|
|
|
|
192 |
C |
p.
|
artikel
|
| 20 |
Graphical abstract TOC
|
|
|
|
192 |
C |
p.
|
artikel
|
| 21 |
Graphical abstract TOC continued
|
|
|
|
192 |
C |
p.
|
artikel
|
| 22 |
Histone deacetylase 3 (HDAC3) inhibitors as anticancer agents: A review
|
Sarkar, Rajat
|
|
|
192 |
C |
p.
|
artikel
|
| 23 |
Janus kinases (JAKs): The efficient therapeutic targets for autoimmune diseases and myeloproliferative disorders
|
Xu, Pengfei
|
|
|
192 |
C |
p.
|
artikel
|
| 24 |
Multi-target drug discovery: An opportunity for novel and repurposed bioactive compounds
|
Alcaro, Stefano
|
|
|
192 |
C |
p.
|
artikel
|
| 25 |
Non-polyphenolic natural inhibitors of amyloid aggregation
|
Ma, Liang
|
|
|
192 |
C |
p.
|
artikel
|
| 26 |
Novel androgen receptor antagonist identified by structure-based virtual screening, structural optimization, and biological evaluation
|
Tang, Qin
|
|
|
192 |
C |
p.
|
artikel
|
| 27 |
Overview of cannabidiol (CBD) and its analogues: Structures, biological activities, and neuroprotective mechanisms in epilepsy and Alzheimer’s disease
|
Li, Han
|
|
|
192 |
C |
p.
|
artikel
|
| 28 |
Repurposed drug candidates for antituberculosis therapy
|
An, Qi
|
|
|
192 |
C |
p.
|
artikel
|
| 29 |
Sensitive fluorogenic substrates for sirtuin deacylase inhibitor discovery
|
Yang, Ling-Ling
|
|
|
192 |
C |
p.
|
artikel
|
| 30 |
Structure-thermodynamics-relationships of hepatitis C viral NS3 protease inhibitors
|
Wypych, Rachel M.
|
|
|
192 |
C |
p.
|
artikel
|
| 31 |
Synthesis and biological evaluation of acridine-based histone deacetylase inhibitors as multitarget agents against Alzheimer’s disease
|
Tseng, Hui-Ju
|
|
|
192 |
C |
p.
|
artikel
|
| 32 |
Synthesis of antiplatelet ortho-carbonyl hydroquinones with differential action on platelet aggregation stimulated by collagen or TRAP-6
|
Méndez, Diego
|
|
|
192 |
C |
p.
|
artikel
|
| 33 |
Synthesis of multimeric pyrrolidine iminosugar inhibitors of human β-glucocerebrosidase and α-galactosidase A: First example of a multivalent enzyme activity enhancer for Fabry disease
|
Martínez-Bailén, Macarena
|
|
|
192 |
C |
p.
|
artikel
|
| 34 |
The development of advanced structural framework as multi-target-directed ligands for the treatment of Alzheimer’s disease
|
Sang, Zhipei
|
|
|
192 |
C |
p.
|
artikel
|
| 35 |
True or false? Challenges and recent highlights in the development of aspirin prodrugs
|
Willetts, Steffan
|
|
|
192 |
C |
p.
|
artikel
|
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