| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A Cell-Based Renilla Luminescence Reporter Plasmid Assay for High-Throughput Screening to Identify Novel FDA-Approved Drug Inhibitors of HPV-16 Infection
|
Walhart, Tara
|
|
|
|
1 |
p. 79-86
|
artikel
|
| 2 |
A Fluorescence-Based High-Throughput Assay for the Identification of Anticancer Reagents Targeting Fructose-1,6-Bisphosphate Aldolase
|
Cho, Eun Jeong
|
|
2018
|
|
1 |
p. 1-10
|
artikel
|
| 3 |
A High-Throughput Dose-Response Cellular Thermal Shift Assay for Rapid Screening of Drug Target Engagement in Living Cells, Exemplified Using SMYD3 and IDO1
|
McNulty, Dean E.
|
|
2018
|
|
1 |
p. 34-46
|
artikel
|
| 4 |
A high-throughput MALDI-TOF MS biochemical screen for small molecule inhibitors of the antigen aminopeptidase ERAP1
|
Müller, Leonie
|
|
|
|
1 |
p. 3-11
|
artikel
|
| 5 |
A High-Throughput Screening Strategy to Identify Inhibitors of SSB Protein–Protein Interactions in an Academic Screening Facility
|
Voter, Andrew F.
|
|
2018
|
|
1 |
p. 94-101
|
artikel
|
| 6 |
A High-Throughput Screening Triage Workflow to Authenticate a Novel Series of PFKFB3 Inhibitors
|
St-Gallay, Stephen A.
|
|
2018
|
|
1 |
p. 11-22
|
artikel
|
| 7 |
Amoxapine Demonstrates Incomplete Inhibition of β-Glucuronidase Activity from Human Gut Microbiota
|
Yang, Wei
|
|
2018
|
|
1 |
p. 76-83
|
artikel
|
| 8 |
Aqueous Solubility Enhancement for Bioassays of Insoluble Inhibitors and QSPR Analysis: A TNF-α Study
|
Mettou, Anthi
|
|
2018
|
|
1 |
p. 84-93
|
artikel
|
| 9 |
A Rapid Phenotypic Whole-Cell Screening Approach for the Identification of Small-Molecule Inhibitors That Counter β-Lactamase Resistance in Pseudomonas aeruginosa
|
Collia, Deanna
|
|
2018
|
|
1 |
p. 55-64
|
artikel
|
| 10 |
A Sensitive and Selective Immunoassay for the Quantitation of Serum Latent Myostatin after In Vivo Administration of SRK-015, a Selective Inhibitor of Myostatin Activation
|
Cote, Shaun M.
|
|
|
|
1 |
p. 95-103
|
artikel
|
| 11 |
Characterization and comparison of hypoxia inducing factors on tumor growth and metastasis between two- and three-dimensional cancer models
|
Chan, Leo Li-Ying
|
|
|
|
1 |
p. 59-65
|
artikel
|
| 12 |
Consideration of vendor-related differences in hepatic metabolic stability data to optimize early ADME screening in drug discovery
|
Shah, Pranav
|
|
|
|
1 |
p. 34-39
|
artikel
|
| 13 |
Corrigendum to DNA methylation-induced ablation of miR-133a accelerates cancer aggressiveness in glioma through upregulating peroxisome proliferator-activated receptor γ [SLAS Discov. 2022 Sep 5;S2472-5552(22)13691-9. doi: 10.1016/j.slasd.2022.08.004.]
|
Liu, Liang
|
|
|
|
1 |
p. 48
|
artikel
|
| 14 |
Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening
|
Lee, Olivia W.
|
|
|
|
1 |
p. 9-20
|
artikel
|
| 15 |
Deep Learning Image Analysis of High-Throughput Toxicology Assay Images
|
Tandon, Arpit
|
|
|
|
1 |
p. 29-38
|
artikel
|
| 16 |
Detection and impact of hypoxic regions in multicellular tumor spheroid cultures formed by head and neck squamous cell carcinoma cells lines
|
Close, David A.
|
|
|
|
1 |
p. 39-54
|
artikel
|
| 17 |
Development and Implementation of an HTS-Compatible Assay for the Discovery of Selective Small-Molecule Ligands for Pre-microRNAs
|
Lorenz, Daniel A.
|
|
2018
|
|
1 |
p. 47-54
|
artikel
|
| 18 |
Development of a Bioluminescent High-Throughput Screening Assay for Nicotinamide Mononucleotide Adenylyltransferase (NMNAT)
|
Haubrich, Brad A.
|
|
|
|
1 |
p. 33-42
|
artikel
|
| 19 |
Development of a High-Throughput Fluorescence Polarization Assay to Detect Inhibitors of the FAK–Paxillin Interaction
|
Marlowe, Timothy
|
|
|
|
1 |
p. 21-32
|
artikel
|
| 20 |
Development of a high-throughput TR-FRET screening assay for a fast-cycling KRAS mutant
|
Larson, Jacob E.
|
|
|
|
1 |
p. 39-47
|
artikel
|
| 21 |
Development of a Screening Platform to Identify Small Molecules That Modify ELP1 Pre-mRNA Splicing in Familial Dysautonomia
|
Salani, Monica
|
|
2019
|
|
1 |
p. 57-67
|
artikel
|
| 22 |
Development of High-Throughput Screening Assays for Inhibitors of ETS Transcription Factors
|
Currie, Simon L.
|
|
2019
|
|
1 |
p. 77-85
|
artikel
|
| 23 |
DNA methylation-induced ablation of miR-133a accelerates cancer aggressiveness in glioma through upregulating peroxisome proliferator-activated receptor γ
|
Liu, Liang
|
|
|
|
1 |
p. 19-28
|
artikel
|
| 24 |
DNA Switch: Toehold-Mediated DNA Isothermal Amplification for Dengue Serotyping
|
Chan, Soo Khim
|
|
2019
|
|
1 |
p. 68-76
|
artikel
|
| 25 |
Erastin-Like Anti-Warburg Agents Prevent Mitochondrial Depolarization Induced by Free Tubulin and Decrease Lactate Formation in Cancer Cells
|
DeHart, David N.
|
|
2018
|
|
1 |
p. 23-33
|
artikel
|
| 26 |
Fragment-based screening: A new paradigm for ligand and target discovery
|
Knight, Sinéad
|
|
|
|
1 |
p. 3-7
|
artikel
|
| 27 |
Genome-scale functional genomics screening highlights genes impacting protein fucosylation in Chinese hamster ovary cells
|
Barlan, Kari
|
|
|
|
1 |
p. 52-58
|
artikel
|
| 28 |
High-throughput cell-based assays for identifying antagonists of multiple smoking-associated human nicotinic acetylcholine receptor subtypes
|
Kassner, Michelle
|
|
|
|
1 |
p. 68-76
|
artikel
|
| 29 |
High-Throughput cell-based immunofluorescence assays against influenza
|
Martinez-Gzegozewska, Yohanka
|
|
|
|
1 |
p. 66-76
|
artikel
|
| 30 |
High-throughput screening for identifying acetylcholinesterase inhibitors: Insights on novel inhibitors and the use of liver microsomes
|
Santillo, Michael F.
|
|
|
|
1 |
p. 65-67
|
artikel
|
| 31 |
Identification of Activators of Human Fumarate Hydratase by Quantitative High-Throughput Screening
|
Zhu, Hu
|
|
|
|
1 |
p. 43-56
|
artikel
|
| 32 |
Identification of Antimalarial Inhibitors Using Late-Stage Gametocytes in a Phenotypic Live/Dead Assay
|
Spicer, Timothy P.
|
|
2019
|
|
1 |
p. 38-46
|
artikel
|
| 33 |
Identification of Chemical Compounds That Inhibit the Function of Histidyl-tRNA Synthetase from Pseudomonas aeruginosa
|
Hu, Yanmei
|
|
2018
|
|
1 |
p. 65-75
|
artikel
|
| 34 |
Identification of positive modulators of TRPM5 channel from a high-throughput screen using a fluorescent membrane potential assay
|
Virginio, Caterina
|
|
|
|
1 |
p. 55-64
|
artikel
|
| 35 |
Identification of potent small molecule inhibitors of SARS-CoV-2 entry
|
Mediouni, Sonia
|
|
|
|
1 |
p. 8-19
|
artikel
|
| 36 |
Identification of Primary Natural Killer Cell Modulators by Chemical Library Screening with a Luciferase-Based Functional Assay
|
Hayek, Simon
|
|
2019
|
|
1 |
p. 25-37
|
artikel
|
| 37 |
Key aspects of modern GPCR drug discovery
|
Addis, Phil
|
|
|
|
1 |
p. 1-22
|
artikel
|
| 38 |
Lysyl-tRNA Synthetase from Pseudomonas aeruginosa: Characterization and Identification of Inhibitory Compounds
|
Balboa, Samantha
|
|
|
|
1 |
p. 57-69
|
artikel
|
| 39 |
Morphology-Based Analysis of Myoblasts for Prediction of Myotube Formation
|
Ishikawa, Kiyoshi
|
|
2019
|
|
1 |
p. 47-56
|
artikel
|
| 40 |
Multiplexed experimental strategies for fragment library screening against challenging drug targets using SPR biosensors
|
FitzGerald, Edward A.
|
|
|
|
1 |
p. 40-51
|
artikel
|
| 41 |
Novel Cell-Based Assay for Identification of LRRK2 Inhibitors Using Its Aberrant Regulation of a Pluripotency Gene
|
Ramonet, David
|
|
|
|
1 |
p. 104-112
|
artikel
|
| 42 |
Optimising cell-based bioassays via integrated design of experiments (ixDoE) - A practical guide
|
Solzin, J
|
|
|
|
1 |
p. 29-38
|
artikel
|
| 43 |
Rebuttal to Response to the Article “Enzyme–Inhibitor Interactions and a Simple, Rapid Method for Determining Inhibition Modality”
|
Copeland, Robert A.
|
|
|
|
1 |
p. 8
|
artikel
|
| 44 |
Reduced levels of serum EPA and DHA identified in patients with non-small-cell lung cancer using a new rapid validated LC-MS/MS method
|
Wang, Yi
|
|
|
|
1 |
p. 12-18
|
artikel
|
| 45 |
Response to the Article “Enzyme–Inhibitor Interactions and a Simple, Rapid Method for Determining Inhibition Modality”
|
Walsh, Ryan
|
|
|
|
1 |
p. 7
|
artikel
|
| 46 |
Screening of Antitubercular Compound Library Identifies Inhibitors of Mur Enzymes in Mycobacterium tuberculosis
|
Eniyan, Kandasamy
|
|
|
|
1 |
p. 70-78
|
artikel
|
| 47 |
Screening Strategies and Methods for Better Off-Target Liability Prediction and Identification of Small-Molecule Pharmaceuticals
|
Van Vleet, Terry R.
|
|
2019
|
|
1 |
p. 1-24
|
artikel
|
| 48 |
SLAS Discovery – The Next Generation of Research
|
Jump, Ally
|
|
|
|
1 |
p. 1-2
|
artikel
|
| 49 |
SLAS Discovery—What’s in a Name?
|
Campbell, Robert M.
|
|
|
|
1 |
p. 1
|
artikel
|
| 50 |
The National Cancer Institute’s Plated Compound Sets Can Be a Valuable Resource for Academic Researchers
|
Zweifach, Adam
|
|
|
|
1 |
p. 2-6
|
artikel
|
| 51 |
Therapeutic approaches for Type 1 Diabetes: Promising cell-based approaches to achieve ultimate success
|
Sepyani, Sahar
|
|
|
|
1 |
p. 23-33
|
artikel
|
| 52 |
The SLAS Discovery Editor's Top 10 for 2022
|
Campbell, Robert M.
|
|
|
|
1 |
p. 1-2
|
artikel
|
| 53 |
Three-Dimensional Control of Ion Channel Function through Optogenetics and Co-Culture
|
Agus, Viviana
|
|
2018
|
|
1 |
p. 102-108
|
artikel
|
| 54 |
Toward Label-Free SERS Detection of Proteins through Their Disulfide Bond Structure
|
Hassanain, Waleed A.
|
|
|
|
1 |
p. 87-94
|
artikel
|
| 55 |
Using measures of metabolic flux to align screening and clinical development: Avoiding pitfalls to enable translational studies
|
Satapati, Santhosh
|
|
|
|
1 |
p. 20-28
|
artikel
|
| 56 |
Virtual plates: Getting the best out of high content screens
|
Shapira Lots, Inbal
|
|
|
|
1 |
p. 77-85
|
artikel
|
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