| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Aminobenzosuberone derivatives as PfA-M1 inhibitors: Molecular recognition and antiplasmodial evaluation
|
Salomon, Emmanuel
|
|
|
98 |
C |
p.
|
artikel
|
| 2 |
Anti-influenza virus activity of benzo[d]thiazoles that target heat shock protein 90
|
Lamut, Andraž
|
|
|
98 |
C |
p.
|
artikel
|
| 3 |
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors
|
Moi, Davide
|
|
|
98 |
C |
p.
|
artikel
|
| 4 |
Application of carbamyl in structural optimization
|
Wang, Kuanglei
|
|
|
98 |
C |
p.
|
artikel
|
| 5 |
Benzo[a]phenoxazinium chlorides: Synthesis, antifungal activity, in silico studies and evaluation as fluorescent probes
|
Leitão, Maria Inês P.S.
|
|
|
98 |
C |
p.
|
artikel
|
| 6 |
Bioactive bisbenzylisoquinoline alkaloids from the roots of Stephania tetrandra
|
Wang, Renzhong
|
|
|
98 |
C |
p.
|
artikel
|
| 7 |
Caseahomopene A, a ring-expanded homotriterpenoid from Casearia kurzii showing anti-inflammatory activities in vitro and in vivo
|
An, Lijun
|
|
|
98 |
C |
p.
|
artikel
|
| 8 |
Corrigendum to “Synthesis of novel 2-aminobenzothiazole derivatives as potential antimicrobial agents with dual DNA gyrase/topoisomerase IV inhibition” [Bioorg. Chem. 94 (2020) 103437]
|
Ismail, Magda M.F.
|
|
|
98 |
C |
p.
|
artikel
|
| 9 |
Design and characterization of a novel structural class of Kv1.3 inhibitors
|
Hendrickx, Louise Antonia
|
|
|
98 |
C |
p.
|
artikel
|
| 10 |
Design and Synthesis of some new 2,4,6-trisubstituted quinazoline EGFR inhibitors as targeted anticancer agents
|
Allam, Heba Abdelrasheed
|
|
|
98 |
C |
p.
|
artikel
|
| 11 |
Design, synthesis and anti-HBV activity evaluation of new substituted imidazo[4,5-b]pyridines
|
Gerasi, Maria
|
|
|
98 |
C |
p.
|
artikel
|
| 12 |
Design, synthesis and biological evaluation of coumarin linked 1,2,4-oxadiazoles as selective carbonic anhydrase IX and XII inhibitors
|
Thacker, Pavitra S.
|
|
|
98 |
C |
p.
|
artikel
|
| 13 |
Design, synthesis and biological evaluation of novel 5,6,7-trimethoxy-N-aryl-2-styrylquinolin-4-amines as potential anticancer agents and tubulin polymerization inhibitors
|
Mirzaei, Salimeh
|
|
|
98 |
C |
p.
|
artikel
|
| 14 |
Design, synthesis and docking studies of novel benzopyrone derivatives as anticonvulsants
|
Abd-Allah, Walaa Hamada
|
|
|
98 |
C |
p.
|
artikel
|
| 15 |
Design, synthesis and evaluation of targeted hypoxia-activated prodrugs applied to chondrosarcoma chemotherapy
|
Gerard, Yvain
|
|
|
98 |
C |
p.
|
artikel
|
| 16 |
Design, synthesis and evaluation of wound healing activity for β-sitosterols derivatives as potent Na+/K+-ATPase inhibitors
|
Cui, Shaoyu
|
|
|
98 |
C |
p.
|
artikel
|
| 17 |
Design, synthesis, antitumor activity and theoretical calculation of novel PI3Ka inhibitors
|
Jin, Ru-Yi
|
|
|
98 |
C |
p.
|
artikel
|
| 18 |
Development of a classification model for the antigenotoxic activity of flavonoids
|
Tuenter, Emmy
|
|
|
98 |
C |
p.
|
artikel
|
| 19 |
Discovery of thiazole-based-chalcones and 4-hetarylthiazoles as potent anticancer agents: Synthesis, docking study and anticancer activity
|
Farghaly, Thoraya A.
|
|
|
98 |
C |
p.
|
artikel
|
| 20 |
Diterpenoids from the leaves of Casearia kurzii showing cytotoxic activities
|
Liang, Yue
|
|
|
98 |
C |
p.
|
artikel
|
| 21 |
Drug-like property optimization: Discovery of orally bioavailable quinazoline-based multi-targeted kinase inhibitors
|
Lin, Shu-Yu
|
|
|
98 |
C |
p.
|
artikel
|
| 22 |
Editorial Board
|
|
|
|
98 |
C |
p.
|
artikel
|
| 23 |
Euphoresulanes A–M, structurally diverse jatrophane diterpenoids from Euphorbia esula
|
Xie, Xing-Lin
|
|
|
98 |
C |
p.
|
artikel
|
| 24 |
Expeditious and eco-friendly synthesis of new multifunctionalized pyrrole derivatives and evaluation of their antioxidant property
|
Kundu, Tania
|
|
|
98 |
C |
p.
|
artikel
|
| 25 |
Extending the use of tadalafil scaffold: Development of novel selective phosphodiesterase 5 inhibitors and histone deacetylase inhibitors
|
ElHady, Ahmed K.
|
|
|
98 |
C |
p.
|
artikel
|
| 26 |
Glucocerebrosidase (GCase) activity modulation by 2-alkyl trihydroxypiperidines: Inhibition and pharmacological chaperoning
|
Clemente, F.
|
|
|
98 |
C |
p.
|
artikel
|
| 27 |
Identification of natural products as selective PTP1B inhibitors via virtual screening
|
Yang, Ying
|
|
|
98 |
C |
p.
|
artikel
|
| 28 |
Incorporation of amino moiety to alepterolic acid improve activity against cancer cell lines: Synthesis and biological evaluation
|
Zhang, Sheng
|
|
|
98 |
C |
p.
|
artikel
|
| 29 |
Isolation of benzolactones, Ganodumones A–F from Ganoderma lucidum and their antibacterial activities
|
Lu, Shuang-Yang
|
|
|
98 |
C |
p.
|
artikel
|
| 30 |
Isoquinoline alkaloids from the roots of Zanthoxylum rigidum as multi-target inhibitors of cholinesterase, monoamine oxidase A and Aβ1-42 aggregation
|
Plazas, Erika
|
|
|
98 |
C |
p.
|
artikel
|
| 31 |
Issue TOC
|
|
|
|
98 |
C |
p.
|
artikel
|
| 32 |
Leucettamine B analogs and their carborane derivative as potential anti-cancer agents: Design, synthesis, and biological evaluation
|
Hsu, Ming-Hua
|
|
|
98 |
C |
p.
|
artikel
|
| 33 |
Methoxy-enriched cationic stilbenes as anticancer therapeutics
|
Yousuf, Md
|
|
|
98 |
C |
p.
|
artikel
|
| 34 |
Multifunctional isoxazolidine derivatives as α-amylase and α-glucosidase inhibitors
|
Ghabi, Ameni
|
|
|
98 |
C |
p.
|
artikel
|
| 35 |
New thymol and isothymol derivatives from Eupatorium fortunei and their cytotoxic effects
|
Yu, Yue
|
|
|
98 |
C |
p.
|
artikel
|
| 36 |
New 1,2,4-triazole/pyrazole hybrids linked to oxime moiety as nitric oxide donor celecoxib analogs: Synthesis, cyclooxygenase inhibition anti-inflammatory, ulcerogenicity, anti-proliferative activities, apoptosis, molecular modeling and nitric oxide release studies
|
Fadaly, Wael A.A.
|
|
|
98 |
C |
p.
|
artikel
|
| 37 |
NMR for screening and a biochemical assay: Identification of new FPPS inhibitors exerting anticancer activity
|
Grimaldi, Manuela
|
|
|
98 |
C |
p.
|
artikel
|
| 38 |
Novel 1H-pyrazolo[3,4-d]pyrimidin-6-amino derivatives as potent selective Janus kinase 3 (JAK3) inhibitors. Evaluation of their improved effect for the treatment of rheumatoid arthritis
|
Yin, Yuan
|
|
|
98 |
C |
p.
|
artikel
|
| 39 |
Novel paeonol derivatives: Design, synthesis and anti-inflammatory activity in vitro and in vivo
|
Hu, Yang Sheng
|
|
|
98 |
C |
p.
|
artikel
|
| 40 |
N-1,2,3-triazole-isatin derivatives for cholinesterase and β-amyloid aggregation inhibition: A comprehensive bioassay study
|
Marques, Carolina S.
|
|
|
98 |
C |
p.
|
artikel
|
| 41 |
Potent colchicine-site ligands with improved intrinsic solubility by replacement of the 3,4,5-trimethoxyphenyl ring with a 2-methylsulfanyl-6-methoxypyridine ring
|
Álvarez, Raquel
|
|
|
98 |
C |
p.
|
artikel
|
| 42 |
S-benzyldithiocarbazate imine coordinated metal complexes kill Candida albicans by causing cellular apoptosis and necrosis
|
Malik, Manzoor Ahmad
|
|
|
98 |
C |
p.
|
artikel
|
| 43 |
Structural elucidation and in vivo anti-arthritic activity of β-amyrin and polpunonic acid isolated from the root bark of Ziziphus abyssinica HochstEx. A Rich (Rhamnaceae)
|
Henneh, Isaac T.
|
|
|
98 |
C |
p.
|
artikel
|
| 44 |
Structure-activity relationship and cardiac safety of 2-aryl-2-(pyridin-2-yl)acetamides as a new class of broad-spectrum anticonvulsants derived from Disopyramide
|
Dawidowski, Maciej
|
|
|
98 |
C |
p.
|
artikel
|
| 45 |
Synthesis and anti-inflammatory evaluation of new chalcone derivatives bearing bispiperazine linker as IL-1β inhibitors
|
Tang, Yan-Ling
|
|
|
98 |
C |
p.
|
artikel
|
| 46 |
Synthesis and biological evaluation of 2-epi-jaspine B analogs as selective sphingosine kinase 1 inhibitors
|
Yang, Haoran
|
|
|
98 |
C |
p.
|
artikel
|
| 47 |
Synthesis and biological evaluation of 6-phenylpurine linked hydroxamates as novel histone deacetylase inhibitors
|
Chen, Dizhong
|
|
|
98 |
C |
p.
|
artikel
|
| 48 |
Synthesis and evaluation of 18F-PTTCO-Cys40-Exendin-4 for PET imaging of ectopic insulinomas in rodents
|
Li, Junfeng
|
|
|
98 |
C |
p.
|
artikel
|
| 49 |
Synthesis and SAR studies of novel 1,2,4-oxadiazole-sulfonamide based compounds as potential anticancer agents for colorectal cancer therapy
|
Shamsi, Farheen
|
|
|
98 |
C |
p.
|
artikel
|
| 50 |
Synthesis, anticancer evaluation and molecular docking studies of new heterocycles linked to sulfonamide moiety as novel human topoisomerase types I and II poisons
|
Halawa, Ahmed H.
|
|
|
98 |
C |
p.
|
artikel
|
| 51 |
Synthesis, antimicrobial and chitinase inhibitory activities of 3-amidocoumarins
|
Sharma, Rajesh Kumar
|
|
|
98 |
C |
p.
|
artikel
|
| 52 |
Synthesis of indole based acetohydrazide analogs: Their in vitro and in silico thymidine phosphorylase studies
|
Taha, Muhammad
|
|
|
98 |
C |
p.
|
artikel
|
| 53 |
Synthesis of neocryptolepines and carbocycle-fused quinolines and evaluation of their anticancer and antiplasmodial activities
|
Akkachairin, Bhornrawin
|
|
|
98 |
C |
p.
|
artikel
|
| 54 |
Synthesis of novel 2-oxospiro[indoline-3,4′-[1,3]dithiine]-5′-carbonitrile derivatives by new spiro[indoline-3,4′-[1,3]dithiine]@Cu(NO3)2 supported on Fe3O4@gly@CE MNPs as efficient catalyst and evaluation of biological activity
|
Moghaddam-Manesh, Mohammadreza
|
|
|
98 |
C |
p.
|
artikel
|
| 55 |
Synthetic homoserine lactone analogues as antagonists of bacterial quorum sensing
|
Qin, Xiaofei
|
|
|
98 |
C |
p.
|
artikel
|
| 56 |
Tacrine-hydroxamate derivatives as multitarget-directed ligands for the treatment of Alzheimer’s disease: Design, synthesis, and biological evaluation
|
Xu, Ana
|
|
|
98 |
C |
p.
|
artikel
|
| 57 |
Technetium-99 m-PEGylated dendrimer-G2-(Dabcyle-Lys6,Phe7)-pHBSP: A novel Nano-Radiotracer for molecular and early detecting of cardiac ischemic region
|
Mohtavinejad, Naser
|
|
|
98 |
C |
p.
|
artikel
|
| 58 |
The insertion of functional groups in organic selenium compounds promote changes in mitochondrial parameters and raise the antibacterial activity
|
Stefanello, Sílvio Terra
|
|
|
98 |
C |
p.
|
artikel
|
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