nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Antiangiogenic activity of terpenoids from Euphorbia neriifolia Linn
|
Qi, Wei-Yan |
|
|
96 |
C |
p. |
artikel |
2 |
Antibacterial sesquiterpenes from the stems and roots of Thuja sutchuenensis
|
Wang, Miaomiao |
|
|
96 |
C |
p. |
artikel |
3 |
Anti-inflammatory and anti-viral labdane diterpenoids from the fruits of Forsythia suspensa
|
Zhao, Lin |
|
|
96 |
C |
p. |
artikel |
4 |
Anti-inflammatory effects of an optimized PPAR-γ agonist via NF-κB pathway inhibition
|
Ju, Zhiran |
|
|
96 |
C |
p. |
artikel |
5 |
Antimicrobial screening and pharmacokinetic profiling of novel phenyl-[1,2,4]triazolo[4,3-a]quinoxaline analogues targeting DHFR and E. coli DNA gyrase B
|
Omar, Abdelsattar M. |
|
|
96 |
C |
p. |
artikel |
6 |
Arylidenes of Quinolin-2-one scaffold as Erlotinib analogues with activities against leukemia through inhibition of EGFR TK/ STAT-3 pathways
|
Elbastawesy, Mohammed A.I. |
|
|
96 |
C |
p. |
artikel |
7 |
Benzoxazole derivatives as new generation of anti-breast cancer agents
|
Omar, A.- Mohsen M.E. |
|
|
96 |
C |
p. |
artikel |
8 |
Binding patterns and structure–activity relationship of CDK8 inhibitors
|
Ma, Duo |
|
|
96 |
C |
p. |
artikel |
9 |
Cell active and functionally-relevant small-molecule agonists of calcitonin receptor
|
Zhao, Shuai |
|
|
96 |
C |
p. |
artikel |
10 |
Chemical constituents from Parrotia persica- Structural derivatization and their potential prolyl endopeptidase inhibition activity
|
Ali, Hassan |
|
|
96 |
C |
p. |
artikel |
11 |
Corrigendum to “Conjugates of tacrine and 1,2,4-thiadiazole derivatives as new potential multifunctional agents for Alzheimer's disease treatment: Synthesis, quantum-chemical characterization, molecular docking, and biological evaluation”. [Bioorg. Chem. 94C (2019)]
|
Makhaeva, Galina F. |
|
|
96 |
C |
p. |
artikel |
12 |
Corrigendum to “Synthesis of benzo[d]imidazo[2,1-b]thiazole-chalcone conjugates as microtubule targeting and apoptosis inducing agents” [Bioorg. Chem. 76 (2018) 1–12]
|
Sultana, Faria |
|
|
96 |
C |
p. |
artikel |
13 |
Corrigendum to “The modulating effect of lipid bilayer/p-coumaric acid interactions on electrical properties of model lipid membranes and human glioblastoma cells” [Bioorg. Chem. 92 (2019) 103242]
|
Naumowicz, Monika |
|
|
96 |
C |
p. |
artikel |
14 |
Design and novel synthetic approach supported with molecular docking and biological evidence for naphthoquinone-hydrazinotriazolothiadiazine analogs as potential anticancer inhibiting topoisomerase-IIB
|
Mohamady, Samy |
|
|
96 |
C |
p. |
artikel |
15 |
Design and synthesis of 3-benzylaminocoumarin-7-O-sulfamate derivatives as steroid sulfatase inhibitors
|
Hng, Yue |
|
|
96 |
C |
p. |
artikel |
16 |
Design of iodinated radioligands for SPECT imaging of central human 5-HT4R using a ligand lipophilicity efficiency approach
|
Babin, Victor |
|
|
96 |
C |
p. |
artikel |
17 |
Design, synthesis and ADMET prediction of bis-benzimidazole as anticancer agent
|
Rashid, Mohammad |
|
|
96 |
C |
p. |
artikel |
18 |
Design, synthesis and biological evaluation of betulin-3-yl 2-amino-2-deoxy-β-d-glycopyranosides
|
Myszka, Henryk |
|
|
96 |
C |
p. |
artikel |
19 |
Design, synthesis and biological evaluation of erythrina derivatives bearing a 1,2,3-triazole moiety as PARP-1 inhibitors
|
Li, Shuai |
|
|
96 |
C |
p. |
artikel |
20 |
Design, synthesis and evaluation of pyrazole bearing α-aminophosphonate derivatives as potential acetylcholinesterase inhibitors against Alzheimer’s disease
|
Shaikh, Sarfaraz |
|
|
96 |
C |
p. |
artikel |
21 |
Design, synthesis, in vitro antimicrobial evaluation and molecular docking studies of indol-2-one tagged with morpholinosulfonyl moiety as DNA gyrase inhibitors
|
Salem, Mohamed A. |
|
|
96 |
C |
p. |
artikel |
22 |
Dihydropyridines as potential α-amylase and α-glucosidase inhibitors: Synthesis, in vitro and in silico studies
|
Yousuf, Hina |
|
|
96 |
C |
p. |
artikel |
23 |
Discovery of novel glyceraldehyde-3-phosphate dehydrogenase inhibitor via docking-based virtual screening
|
Li, Ting |
|
|
96 |
C |
p. |
artikel |
24 |
Editorial Board
|
|
|
|
96 |
C |
p. |
artikel |
25 |
Efficient synthesis of NIR emitting bis[2-(2′-hydroxylphenyl)benzoxazole] derivative and its potential for imaging applications
|
Wang, Junfeng |
|
|
96 |
C |
p. |
artikel |
26 |
Engineered β-hairpin scaffolds from human prion protein regions: Structural and functional investigations of aggregates
|
Di Natale, Concetta |
|
|
96 |
C |
p. |
artikel |
27 |
Enhanced antitumor potential induced by chloroacetate-loaded benzophenones acting as fused tubulin-pyruvate dehydrogenase kinase 1 (PDHK1) ligands
|
Ghinet, Alina |
|
|
96 |
C |
p. |
artikel |
28 |
Enzymatic studies with 3-oxa n-3 DPA
|
Pangopoulos, Maria K. |
|
|
96 |
C |
p. |
artikel |
29 |
Flavan derivative enantiomers and drimane sesquiterpene lactones from the Inonotus obliquus with neuroprotective effects
|
Zou, Chun-Xin |
|
|
96 |
C |
p. |
artikel |
30 |
Four pairs of alkaloid enantiomers from Isatis indigotica Fortune Ex Land with neuroprotective effects against H2O2-induced SH-SY5Y cell injury
|
Xi, Yu-Fei |
|
|
96 |
C |
p. |
artikel |
31 |
Identification, in vitro evaluation and modeling studies of the constituents from the roots of Arnebia euchroma for antitumor activity and STAT3 inhibition
|
Cao, Huihui |
|
|
96 |
C |
p. |
artikel |
32 |
Isolation and characterization of cytotoxic withanolides from the calyx of Physalis alkekengi L. var franchetii
|
Sun, Yi |
|
|
96 |
C |
p. |
artikel |
33 |
Isoxazole-containing 5′ mRNA cap analogues as inhibitors of the translation initiation process
|
Piecyk, Karolina |
|
|
96 |
C |
p. |
artikel |
34 |
Issue TOC
|
|
|
|
96 |
C |
p. |
artikel |
35 |
Lanostane triterpene glycosides from the flowers of Lyonia ovalifolia var. hebecarpa and their antiproliferative activities
|
Zhang, Hanqi |
|
|
96 |
C |
p. |
artikel |
36 |
Molecular hybrid design, synthesis, in vitro and in vivo anticancer evaluation, and mechanism of action of N-acylhydrazone linked, heterobivalent β-carbolines
|
Guo, Liang |
|
|
96 |
C |
p. |
artikel |
37 |
Morpholine as ubiquitous pharmacophore in medicinal chemistry: Deep insight into the structure-activity relationship (SAR)
|
Kumari, Archana |
|
|
96 |
C |
p. |
artikel |
38 |
Mulberry anthocyanins exert anti-AGEs effects by selectively trapping glyoxal and structural-dependently blocking the lysyl residues of β-lactoglobulins
|
Khalifa, Ibrahim |
|
|
96 |
C |
p. |
artikel |
39 |
Network pharmacology based investigation into the bioactive compounds and molecular mechanisms of Schisandrae Chinensis Fructus against drug-induced liver injury
|
Li, Xiankuan |
|
|
96 |
C |
p. |
artikel |
40 |
New approach in the characterization of bioactive compounds isolated from Calycotome spinosa (L.) Link leaves by the use of negative electrospray ionization LITMS n , LC-ESI-MS/MS, as well as NMR analysis
|
Cherfia, Radia |
|
|
96 |
C |
p. |
artikel |
41 |
New benzenesulfonamide scaffold-based cytotoxic agents: Design, synthesis, cell viability, apoptotic activity and radioactive tracing studies
|
Nissan, Yassin M. |
|
|
96 |
C |
p. |
artikel |
42 |
New cassane-type diterpenoids from kernels of Caesalpinia bonduc (Linn.) Roxb. and their inhibitory activities on phosphodiesterase (PDE) and nuclear factor-kappa B (NF-κB) expression
|
Liu, Ting |
|
|
96 |
C |
p. |
artikel |
43 |
New obovatol trimeric neolignans with NO inhibitory activity from the leaves of Magnolia officinalis var. biloba
|
Vu, Van-Tuan |
|
|
96 |
C |
p. |
artikel |
44 |
New polyazamacrocyclic 3-hydroxy-4-pyridinone based ligands for iron depletion antitumor activity
|
Liu, Xiaoguang |
|
|
96 |
C |
p. |
artikel |
45 |
Novel pyrazine based anti-tubercular agents: Design, synthesis, biological evaluation and in silico studies
|
Hassan, Nayera W. |
|
|
96 |
C |
p. |
artikel |
46 |
Pegylated triarylmethanes: Synthesis, antimicrobial activity, anti-proliferative behavior and in silico studies
|
Ricco, Christophe |
|
|
96 |
C |
p. |
artikel |
47 |
Pharmacophore-fusing design of pyrimidine sulfonylacetanilides as potent non-nucleoside inhibitors of HIV-1 reverse transcriptase
|
Sang, Yali |
|
|
96 |
C |
p. |
artikel |
48 |
Preparative scale application of Mucor circinelloides ene–reductase and alcohol dehydrogenase activity for the asymmetric bioreduction of α,β-unsaturated γ-ketophosphonates
|
Janicki, Ignacy |
|
|
96 |
C |
p. |
artikel |
49 |
Protein tyrosine phosphatase 1B (PTP1B) inhibitorsfrom the deep-sea fungus Penicillium chrysogenum SCSIO 07007
|
Han, Wenrong |
|
|
96 |
C |
p. |
artikel |
50 |
Protostane-type triterpenoids as natural soluble epoxide hydrolase inhibitors: Inhibition potentials and molecular dynamics
|
Sun, Cheng-Peng |
|
|
96 |
C |
p. |
artikel |
51 |
Ruthenium derivatives attenuate LPS-induced inflammatory responses and liver injury via suppressing NF-κB signaling and free radical production
|
Jayakumar, Thanasekaran |
|
|
96 |
C |
p. |
artikel |
52 |
Search for non-acidic ALR2 inhibitors: Evaluation of flavones as targeted agents for the management of diabetic complications
|
Vyas, Bhawna |
|
|
96 |
C |
p. |
artikel |
53 |
Serratane triterpenoids isolated from Lycopodium clavatum by bioactivity-guided fractionation attenuate the production of inflammatory mediators
|
Jo, Ara |
|
|
96 |
C |
p. |
artikel |
54 |
Single-step synthesis and in vitro anti-mycobacterial activity of novel nitrofurantoin analogues
|
Zuma, Nonkululeko H. |
|
|
96 |
C |
p. |
artikel |
55 |
S-seco-porphyrazine as a new member of the seco-porphyrazine family – Synthesis, characterization and photocytotoxicity against cancer cells
|
Mlynarczyk, Dariusz T. |
|
|
96 |
C |
p. |
artikel |
56 |
Stephalagine, an aporphine alkaloid from Annona crassiflora fruit peel, induces antinociceptive effects by TRPA1 and TRPV1 channels modulation in mice
|
Justino, Allisson Benatti |
|
|
96 |
C |
p. |
artikel |
57 |
Structural characterization, neuroprotective and hepatoprotective activities of flavonoids from the bulbs of Heleocharis dulcis
|
Ma, Qinge |
|
|
96 |
C |
p. |
artikel |
58 |
Structure-based design and optimization of pyrimidine- and 1,2,4-triazolo[4,3-a]pyrimidine-based matrix metalloproteinase-10/13 inhibitors via Dimroth rearrangement towards targeted polypharmacology
|
El Ashry, El Sayed Helmy |
|
|
96 |
C |
p. |
artikel |
59 |
Structure based discovery of novel hexokinase 2 inhibitors
|
Liu, Yang |
|
|
96 |
C |
p. |
artikel |
60 |
Synthesis and biological evaluation of myricetin-pentadienone hybrids as potential anti-inflammatory agents in vitro and in vivo
|
Liu, Chao |
|
|
96 |
C |
p. |
artikel |
61 |
Synthesis and biological evaluation of novel 5,6,7-trimethoxy flavonoid salicylate derivatives as potential anti-tumor agents
|
Liu, Renbo |
|
|
96 |
C |
p. |
artikel |
62 |
Synthesis and biological evaluations of N′-substituted methylene-4-(quinoline-4-amino) benzoylhydrazides as potential anti-hepatoma agents
|
Li, Baicun |
|
|
96 |
C |
p. |
artikel |
63 |
Synthesis and characterization of novel 99mTc-DGC nano-complexes for improvement of heart diagnostic
|
Ardestani, Mehdi Shafiee |
|
|
96 |
C |
p. |
artikel |
64 |
Synthesis and evaluation of novel S-benzyl- and S-alkylphthalimide- oxadiazole -benzenesulfonamide hybrids as inhibitors of dengue virus protease
|
Hamdani, Syeda Shamila |
|
|
96 |
C |
p. |
artikel |
65 |
Synthesis and in vitro investigation of novel cytotoxic pyrimidine and pyrazolopyrimidne derivatives showing apoptotic effect
|
Ragab, Fatma A. |
|
|
96 |
C |
p. |
artikel |
66 |
Synthesis, in vitro, and in vivo (Zebra fish) antitubercular activity of 7,8-dihydroquinolin-5(6H)-ylidenehydrazinecarbothioamides
|
Marvadi, Sandeep kumar |
|
|
96 |
C |
p. |
artikel |
67 |
Synthesis, molecular docking and antimicrobial activity of new fused pyrimidine and pyridine derivatives
|
Radwan, Mohamed A.A. |
|
|
96 |
C |
p. |
artikel |
68 |
Synthesis of a 1,2,3-bistriazole derivative of embelin and evaluation of its effect on high-fat diet fed-streptozotocin-induced type 2 diabetes in rats and molecular docking studies
|
Stalin, Antony |
|
|
96 |
C |
p. |
artikel |
69 |
Synthesis of a novel series of (Z)-3,5-disubstituted thiazolidine-2,4-diones as promising anti-breast cancer agents
|
El-Kashef, Hussein |
|
|
96 |
C |
p. |
artikel |
70 |
Synthesis of flavonoids nitrogen mustard derivatives and study on their antitumor activity in vitro
|
Yan, Xi |
|
|
96 |
C |
p. |
artikel |
71 |
Synthesis of naphthalimide-phenanthro[9,10-d]imidazole derivatives: In vitro evaluation, binding interaction with DNA and topoisomerase inhibition
|
Singh, Iqubal |
|
|
96 |
C |
p. |
artikel |
72 |
Synthesis of some N-aroyl-2-oxindole benzenesulfonamide conjugates with carbonic anhydrase inhibitory activity
|
George, Riham F. |
|
|
96 |
C |
p. |
artikel |
73 |
Synthesis of sulpha drug based hydroxytriazene derivatives: Anti-diabetic, antioxidant, anti-inflammatory activity and their molecular docking studies
|
Sharma, Poonam |
|
|
96 |
C |
p. |
artikel |
74 |
Synthesis, structure elucidation, and in vitro pharmacological evaluation of novel polyfluoro substituted pyrazoline type sulfonamides as multi-target agents for inhibition of acetylcholinesterase and carbonic anhydrase I and II enzymes
|
Yamali, Cem |
|
|
96 |
C |
p. |
artikel |
75 |
Synthetic routes to nanoconjugates of anthracyclines
|
Piorecka, Kinga |
|
|
96 |
C |
p. |
artikel |
76 |
Tacrine-xanomeline and tacrine-iperoxo hybrid ligands: Synthesis and biological evaluation at acetylcholinesterase and M1 muscarinic acetylcholine receptors
|
Maspero, Marco |
|
|
96 |
C |
p. |
artikel |
77 |
Tsaokopyranols A–M, 2,6-epoxydiarylheptanoids from Amomum tsao-ko and their α-glucosidase inhibitory activity
|
He, Xiao-Feng |
|
|
96 |
C |
p. |
artikel |
78 |
Uncommon nornardosinane, seconeolemnane and related sesquiterpenoids from Xisha soft coral Litophyton nigrum
|
Yang, Fan |
|
|
96 |
C |
p. |
artikel |
79 |
Unexpected CK2β-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2
|
Pietsch, Markus |
|
|
96 |
C |
p. |
artikel |
80 |
Young apple polyphenols as natural α-glucosidase inhibitors: In vitro and in silico studies
|
Gong, Tian |
|
|
96 |
C |
p. |
artikel |