nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A dual-emission fluorescent probe for discriminating cysteine from homocysteine and glutathione in living cells and zebrafish models
|
Lu, Zhengliang |
|
|
92 |
C |
p. |
artikel |
2 |
A novel adaptive fluorescent probe for cell labelling
|
Coman, Anca G. |
|
|
92 |
C |
p. |
artikel |
3 |
Anti-cancer activity of the cell membrane-permeable phytic acid prodrug
|
Masunaga, Takuya |
|
|
92 |
C |
p. |
artikel |
4 |
Anti-inflammatory flavonoids from root bark of Broussonetia papyrifera in LPS-stimulated RAW264.7 cells
|
Ryu, Hyung Won |
|
|
92 |
C |
p. |
artikel |
5 |
Antiprotozoal activities of marine polyether triterpenoids
|
Díaz-Marrero, Ana R. |
|
|
92 |
C |
p. |
artikel |
6 |
Arylpropionic acid-derived NSAIDs: New insights on derivatization, anticancer activity and potential mechanism of action
|
Gouda, Ahmed M. |
|
|
92 |
C |
p. |
artikel |
7 |
Biflavones from Ginkgo biloba as inhibitors of human thrombin
|
Chen, Tian-Ran |
|
|
92 |
C |
p. |
artikel |
8 |
Bioactivity-based analysis and chemical characterization of hypoglycemic and antioxidant components from Artemisia argyi
|
Xiao, Jian-Qi |
|
|
92 |
C |
p. |
artikel |
9 |
Biscoumarin-1,2,3-triazole hybrids as novel anti-diabetic agents: Design, synthesis, in vitro α-glucosidase inhibition, kinetic, and docking studies
|
Asgari, Mohammad Sadegh |
|
|
92 |
C |
p. |
artikel |
10 |
Chemical constituents and synergistic anti-gout studies on Eurycoma longifolia and potential mechanisms evaluation based on systemic analysis approach
|
Liu, Ying |
|
|
92 |
C |
p. |
artikel |
11 |
Chemical constituents from Alismatis Rhizoma and their anti-inflammatory activities in vitro and in vivo
|
Liu, Shan-shan |
|
|
92 |
C |
p. |
artikel |
12 |
Chemical constituents from Lonicera japonica flower buds and their anti-hepatoma and anti-HBV activities
|
Ge, Lanlan |
|
|
92 |
C |
p. |
artikel |
13 |
Corrigendum to “Design, synthesis and biological evaluation of pyrazolopyrimidinone based potent and selective PDE5 inhibitors for treatment of erectile dysfunction” [Bioorg. Chem. 89 (2019) 103022]
|
Reddy, G. Lakshma |
|
|
92 |
C |
p. |
artikel |
14 |
Coumarin tethered cyclic imides as efficacious glucose uptake agents and investigation of hit candidate to probe its binding mechanism with human serum albumin
|
Reddy, Dinesh S. |
|
|
92 |
C |
p. |
artikel |
15 |
Curcumane C and (±)-curcumane D, an unusual seco-cadinane sesquiterpenoid and a pair of unusual nor-bisabolane enantiomers with significant vasorelaxant activity from Curcuma longa
|
Qiao, Ming-Ming |
|
|
92 |
C |
p. |
artikel |
16 |
Design and evaluation of non-carboxylate 5-arylidene-2-thioxo-4-imidazolidinones as novel non-competitive inhibitors of protein tyrosine phosphatase 1B
|
Ottanà, Rosaria |
|
|
92 |
C |
p. |
artikel |
17 |
Design and synthesis of fluorogenic substrate-based probes for detecting Cathepsin B activity
|
Wang, Shusheng |
|
|
92 |
C |
p. |
artikel |
18 |
Design and synthesis of novel pyridazinoquinazoline derivatives as potent VEGFR-2 inhibitors: In vitro and in vivo study
|
El-Gazzar, Marwa G. |
|
|
92 |
C |
p. |
artikel |
19 |
Design, synthesis and antifungal activity evaluation of isocryptolepine derivatives
|
Li, Jun-cai |
|
|
92 |
C |
p. |
artikel |
20 |
Design, synthesis, and biological activity of Plastoquinone analogs as a new class of anticancer agents
|
Bayrak, Nilüfer |
|
|
92 |
C |
p. |
artikel |
21 |
Design, synthesis, and biological evaluation of novel dual FFA1 (GPR40)/PPARδ agonists as potential anti-diabetic agents
|
Li, Zheng |
|
|
92 |
C |
p. |
artikel |
22 |
Design, synthesis and biological evaluation of some tetrazole acetamide derivatives as novel non-carboxylic PTP1B inhibitors
|
Maheshwari, Neelesh |
|
|
92 |
C |
p. |
artikel |
23 |
Design, synthesis and biological evaluation of theophylline containing variant acetylene derivatives as α-amylase inhibitors
|
Ruddarraju, Radhakrishnam Raju |
|
|
92 |
C |
p. |
artikel |
24 |
Design, synthesis and molecular docking of benzophenone conjugated with oxadiazole sulphur bridge pyrazole pharmacophores as anti inflammatory and analgesic agents
|
Zabiulla, |
|
|
92 |
C |
p. |
artikel |
25 |
Design, synthesis and molecular docking of novel pyrazolo[1,5-a][1,3,5]triazine derivatives as CDK2 inhibitors
|
Oudah, Khulood H. |
|
|
92 |
C |
p. |
artikel |
26 |
Design, synthesis, and molecular docking study of new piperazine derivative as potential antimicrobial agents
|
Patil, Mahadev |
|
|
92 |
C |
p. |
artikel |
27 |
Design, synthesis, in-vitro evaluation and molecular docking studies of novel indole derivatives as inhibitors of SIRT1 and SIRT2
|
Manjula, Ramu |
|
|
92 |
C |
p. |
artikel |
28 |
Design, synthesis, in vitro evaluation, molecular docking and ADME properties studies of hybrid bis-coumarin with thiadiazole as a new inhibitor of Urease
|
Alomari, Munther |
|
|
92 |
C |
p. |
artikel |
29 |
Development of novel chromeno[4,3-c]pyrazol-4(2H)-one derivates containing piperazine as inhibitors of PI3Kα
|
Yin, Yong |
|
|
92 |
C |
p. |
artikel |
30 |
Dihydro-β-agarofuran sesquiterpenoid derivatives with anti-inflammatory activity from the leaves of Tripterygium wilfordii
|
He, Qing-Jun |
|
|
92 |
C |
p. |
artikel |
31 |
Discovery and optimization of 5,7-dihydro-6H-pyrrolo[2,3-d]pyrimidin-6-one derivatives as mTORC1/mTORC2 dual inhibitors
|
Hu, Shengquan |
|
|
92 |
C |
p. |
artikel |
32 |
Discovery, molecular dynamic simulation and biological evaluation of structurally diverse cholinesterase inhibitors with new scaffold through shape-based pharmacophore virtual screening
|
Yang, Hongyu |
|
|
92 |
C |
p. |
artikel |
33 |
Discovery of a series of selective and cell permeable beta-secretase (BACE1) inhibitors by fragment linking with the assistance of STD-NMR
|
Fang, Wei-Shuo |
|
|
92 |
C |
p. |
artikel |
34 |
Discovery of certain benzyl/phenethyl thiazolidinone-indole hybrids as potential anti-proliferative agents: Synthesis, molecular modeling and tubulin polymerization inhibition study
|
Sigalapalli, Dilep Kumar |
|
|
92 |
C |
p. |
artikel |
35 |
Discovery of diverse diterpenoid scaffolds from Euphorbia antiquorum and their activity against RANKL-induced osteoclastogenesis
|
Yin, Zhi-Yong |
|
|
92 |
C |
p. |
artikel |
36 |
Discovery of 2-ethoxy-4-(methoxymethyl)benzamide derivatives as potent and selective PTP1B inhibitors
|
Xie, Fangzhou |
|
|
92 |
C |
p. |
artikel |
37 |
Discovery of HWL-088: A highly potent FFA1/GPR40 agonist bearing a phenoxyacetic acid scaffold
|
Li, Zheng |
|
|
92 |
C |
p. |
artikel |
38 |
Discovery of indoline derivatives that inhibit esophageal squamous cell carcinoma growth by Noxa mediated apoptosis
|
Fu, Dong-Jun |
|
|
92 |
C |
p. |
artikel |
39 |
Disulfide bridge as a linker in nucleic acids’ bioconjugation. Part I: An overview of synthetic strategies
|
Stasińska, Anna R. |
|
|
92 |
C |
p. |
artikel |
40 |
Dual-targeting antitumor conjugates derived from platinum(IV) prodrugs and microtubule inhibitor CA-4 significantly exhibited potent ability to overcome cisplatin resistance
|
Huang, Xiaochao |
|
|
92 |
C |
p. |
artikel |
41 |
Dual VEGFR-2/PIM-1 kinase inhibition towards surmounting the resistance to antiangiogenic agents via hybrid pyridine and thienopyridine-based scaffolds: Design, synthesis and biological evaluation
|
Rizk, Ola H. |
|
|
92 |
C |
p. |
artikel |
42 |
Editorial Board
|
|
|
|
92 |
C |
p. |
artikel |
43 |
Effects of Picrasma quassioides and its active constituents on Alzheimer's disease in vitro and in vivo
|
Guo, Eryan |
|
|
92 |
C |
p. |
artikel |
44 |
Exploring antidiabetic potential of adamantyl-thiosemicarbazones via aldose reductase (ALR2) inhibition
|
Shehzad, Muhammad Tariq |
|
|
92 |
C |
p. |
artikel |
45 |
First example of Azo-Sulfa conjugated chromene moieties: Synthesis, characterization, antimicrobial assessment, docking simulation as potent class I histone deacetylase inhibitors and antitumor agents
|
Okasha, Rawda M. |
|
|
92 |
C |
p. |
artikel |
46 |
Geranylated carbazole alkaloids with potential neuroprotective activities from the stems and leaves of Clausena lansium
|
Liu, Yan-Ping |
|
|
92 |
C |
p. |
artikel |
47 |
Germacrane-type sesquiterpenoids with cytotoxic activity from Sigesbeckia orientalis
|
Liu, Na |
|
|
92 |
C |
p. |
artikel |
48 |
Identification of novel small-molecule inhibitors of α-methylacyl-CoA racemase (AMACR; P504S) and structure-activity relationships
|
Petrova, Yoana D. |
|
|
92 |
C |
p. |
artikel |
49 |
Identification of potential inflammatory inhibitors from Aster tataricus
|
Su, Xiang Dong |
|
|
92 |
C |
p. |
artikel |
50 |
Immunomodulatory activities of zinc(II)phthalocyanine on the mammalian macrophages through p38 pathway: Potential ex vivo immunomodulatory PDT reagents
|
Yüzer, Abdulcelil |
|
|
92 |
C |
p. |
artikel |
51 |
In vitro assessment of 3-alkoxy-5-nitroindazole-derived ethylamines and related compounds as potential antileishmanial drugs
|
Martín-Montes, Álvaro |
|
|
92 |
C |
p. |
artikel |
52 |
Issue TOC
|
|
|
|
92 |
C |
p. |
artikel |
53 |
Juniperanol: First total synthesis and evaluation in Type 2 Diabetes disease
|
Carrër, A. |
|
|
92 |
C |
p. |
artikel |
54 |
Molecular interaction of manganese based carbon monoxide releasing molecule (MnCORM) with human serum albumin (HSA)
|
Vidhyapriya, Pitchavel |
|
|
92 |
C |
p. |
artikel |
55 |
New A2A adenosine receptor antagonists: a structure-based upside-down interaction in the receptor cavity
|
Lambertucci, Catia |
|
|
92 |
C |
p. |
artikel |
56 |
New carboxamides bearing benzenesulphonamides: Synthesis, molecular docking and pharmacological properties
|
Eze, Florence Uchenna |
|
|
92 |
C |
p. |
artikel |
57 |
New cytotoxic tricycloalternarenes from fungus Alternaria brassicicola
|
Li, Fengli |
|
|
92 |
C |
p. |
artikel |
58 |
New pyrimidine-benzoxazole/benzimidazole hybrids: Synthesis, antioxidant, cytotoxic activity, in vitro cyclooxygenase and phospholipase A2-V inhibition
|
Abdelgawad, Mohamed A. |
|
|
92 |
C |
p. |
artikel |
59 |
New series of fused pyrazolopyridines: Synthesis, molecular modeling, antimicrobial, antiquorum-sensing and antitumor activities
|
El-Gohary, N.S. |
|
|
92 |
C |
p. |
artikel |
60 |
New triazinoindole bearing thiazole/oxazole analogues: Synthesis, α-amylase inhibitory potential and molecular docking study
|
Rahim, Fazal |
|
|
92 |
C |
p. |
artikel |
61 |
NO inhibitory diterpenoids as potential anti-inflammatory agents from Euphorbia antiquorum
|
An, Lijun |
|
|
92 |
C |
p. |
artikel |
62 |
Novel 2-arylthiopropanoyl-CoA inhibitors of α-methylacyl-CoA racemase 1A (AMACR; P504S) as potential anti-prostate cancer agents
|
Yevglevskis, Maksims |
|
|
92 |
C |
p. |
artikel |
63 |
Novel conjugates with dual suppression of glutathione S-transferases and tryptophan-2,3-dioxygenase activities for improving hepatocellular carcinoma therapy
|
Hua, Shixian |
|
|
92 |
C |
p. |
artikel |
64 |
Novel 3,4-dihydro-4-oxoquinazoline-based acetohydrazides: Design, synthesis and evaluation of antitumor cytotoxicity and caspase activation activity
|
Huan, Le Cong |
|
|
92 |
C |
p. |
artikel |
65 |
Novel inhibitors of leukocyte transendothelial migration
|
Getter, Tamar |
|
|
92 |
C |
p. |
artikel |
66 |
Novel N-benzylpyridinium moiety linked to arylisoxazole derivatives as selective butyrylcholinesterase inhibitors: Synthesis, biological evaluation, and docking study
|
Vafadarnejad, Fahimeh |
|
|
92 |
C |
p. |
artikel |
67 |
Novel pyridazinone derivatives as butyrylcholinesterase inhibitors
|
Dundar, Yasemin |
|
|
92 |
C |
p. |
artikel |
68 |
Novel [1,2,4]triazolo[1,5-a]pyrimidine derivatives as potent antitubulin agents: Design, multicomponent synthesis and antiproliferative activities
|
Yang, Fang |
|
|
92 |
C |
p. |
artikel |
69 |
Nusbiarylins, a new class of antimicrobial agents: Rational design of bacterial transcription inhibitors targeting the interaction between the NusB and NusE proteins
|
Qiu, Yangyi |
|
|
92 |
C |
p. |
artikel |
70 |
Optimization study towards more potent thiazolidine-2,4-dione IKK-β modulator: Synthesis, biological evaluation and in silico docking simulation
|
Elkamhawy, Ahmed |
|
|
92 |
C |
p. |
artikel |
71 |
Physapubescin I from husk tomato suppresses SW1990 cancer cell growth by targeting kidney-type glutaminase
|
Yang, Kai-Yin |
|
|
92 |
C |
p. |
artikel |
72 |
Promising antibacterial agents against multidrug resistant Staphylococcus aureus
|
Gatadi, Srikanth |
|
|
92 |
C |
p. |
artikel |
73 |
Pyrazole[3,4-d]pyridazine derivatives: Molecular docking and explore of acetylcholinesterase and carbonic anhydrase enzymes inhibitors as anticholinergics potentials
|
Taslimi, Parham |
|
|
92 |
C |
p. |
artikel |
74 |
Rational design of some substituted phenyl azanediyl (bis) methylene phosphonic acid derivatives as potential anticancer agents and imaging probes: Computational inputs, chemical synthesis, radiolabeling, biodistribution and gamma scintigraphy
|
Khedr, Mohammed A. |
|
|
92 |
C |
p. |
artikel |
75 |
Recent advances in the synthetic and medicinal perspective of quinolones: A review
|
Dhiman, Prashant |
|
|
92 |
C |
p. |
artikel |
76 |
Spirocyclic sulfonamides with carbonic anhydrase inhibitory and anti-neuropathic pain activity
|
Kalisha Vali, Y. |
|
|
92 |
C |
p. |
artikel |
77 |
2-Styrylchromone derivatives as potent and selective monoamine oxidase B inhibitors
|
Takao, Koichi |
|
|
92 |
C |
p. |
artikel |
78 |
Synthesis and biological evaluation of a novel series of curcumin-peptide derivatives as PepT1-mediated transport drugs
|
Zhang, Jiyun |
|
|
92 |
C |
p. |
artikel |
79 |
Synthesis and biological evaluation of tetrazole derivatives as TNF-α, IL-6 and COX-2 inhibitors with antimicrobial activity: Computational analysis, molecular modeling study and region-specific cyclization using 2D NMR tools
|
Lamie, Phoebe F. |
|
|
92 |
C |
p. |
artikel |
80 |
Synthesis and biological evaluation of thiazolidine-2,4-dione-pyrazole conjugates as antidiabetic, anti-inflammatory and antioxidant agents
|
Bansal, Garima |
|
|
92 |
C |
p. |
artikel |
81 |
Synthesis and comparative carbonic anhydrase inhibition of new Schiff’s bases incorporating benzenesulfonamide, methanesulfonamide, and methylsulfonylbenzene scaffolds
|
El-Azab, Adel S. |
|
|
92 |
C |
p. |
artikel |
82 |
Synthesis and investigation of inhibitory activities of imidazole derivatives against the metallo-β-lactamase IMP-1
|
Khalili Arjomandi, Omid |
|
|
92 |
C |
p. |
artikel |
83 |
Synthesis and investigation of polyhydroxylated pyrrolidine derivatives as novel chemotypes showing dual activity as glucosidase and aldose reductase inhibitors
|
Guazzelli, Lorenzo |
|
|
92 |
C |
p. |
artikel |
84 |
Synthesis, anticancer activity and molecular docking studies on 1,2-diarylbenzimidazole analogues as anti-tubulin agents
|
Zhang, Ya-Liang |
|
|
92 |
C |
p. |
artikel |
85 |
Synthesis, biological activity and molecular modeling of a new series of condensed 1,2,4-triazoles
|
El Bakri, Youness |
|
|
92 |
C |
p. |
artikel |
86 |
Synthesis, biological evaluation and in silico modelling studies of 1,3,5-trisubstituted pyrazoles carrying benzenesulfonamide as potential anticancer agents and selective cancer-associated hCA IX isoenzyme inhibitors
|
Yamali, Cem |
|
|
92 |
C |
p. |
artikel |
87 |
Synthesis, biological evaluation and molecular docking analysis of novel benzopyrimidinone derivatives as potential anti-tyrosinase agents
|
Chortani, Sarra |
|
|
92 |
C |
p. |
artikel |
88 |
Synthesis, in-vitro cholinesterase inhibition, in-vivo anticonvulsant activity and in-silico exploration of N-(4-methylpyridin-2-yl)thiophene-2-carboxamide analogs
|
Ahmad, Gulraiz |
|
|
92 |
C |
p. |
artikel |
89 |
Synthesis of d-desthiobiotin-AI-2 as a novel chemical probe for autoinducer-2 quorum sensing receptors
|
Miranda, Vanessa |
|
|
92 |
C |
p. |
artikel |
90 |
Synthesis of Mitomycin C and decarbamoylmitomycin C N 6 deoxyadenosine-adducts
|
Zheng, Maggie |
|
|
92 |
C |
p. |
artikel |
91 |
Synthesis, structural characterization and in vivo anti-diabetic evaluation of some new sulfonylurea derivatives in normal and silicate coated nanoparticle forms as anti-hyperglycemic agents
|
Sroor, Farid M. |
|
|
92 |
C |
p. |
artikel |
92 |
Targeted 8-hydroxyquinoline fragment based small molecule drug discovery against neglected botulinum neurotoxin type F
|
Chauhan, Ritika |
|
|
92 |
C |
p. |
artikel |
93 |
The application of safe for humans and the environment Polyversum antifungal agent containing living cells of Pythium oligandrum for biotransformation of prochiral ketones
|
Kołodziejska, Renata |
|
|
92 |
C |
p. |
artikel |
94 |
The modulating effect of lipid bilayer/p-coumaric acid interactions on electrical properties of model lipid membranes and human glioblastoma cells
|
Naumowicz, Monika |
|
|
92 |
C |
p. |
artikel |
95 |
The role of long noncoding RNA in major human disease
|
Zhang, Xiaoli |
|
|
92 |
C |
p. |
artikel |
96 |
Triazolopyridazine derivatives: Synthesis, cytotoxic evaluation, c-Met kinase activity and molecular docking
|
Ahmed, Eman M. |
|
|
92 |
C |
p. |
artikel |
97 |
Tyrosinase inhibitory effects of Vinca major and its secondary metabolites: Enzyme kinetics and in silico inhibition model of the metabolites validated by pharmacophore modelling
|
Sari, Suat |
|
|
92 |
C |
p. |
artikel |
98 |
Ultrasound mediated efficient synthesis of new 4-oxoquinazolin-3(4H)-yl)furan-2-carboxamides as potent tyrosinase inhibitors: Mechanistic approach through chemoinformatics and molecular docking studies
|
Dige, Nilam C. |
|
|
92 |
C |
p. |
artikel |
99 |
Umbelliferone derivatives exert neuroprotective effects by inhibiting monoamine oxidase A, self-amyloidβ aggregation, and lipid peroxidation
|
Seong, Su Hui |
|
|
92 |
C |
p. |
artikel |
100 |
Variedly connected 1,8-naphthalimide-7-chloroquinoline conjugates: Synthesis, anti-mycobacterial and cytotoxic evaluation
|
Shalini, |
|
|
92 |
C |
p. |
artikel |
101 |
Vernodalidimer L, a sesquiterpene lactone dimer from Vernonia extensa and anti-tumor effects of vernodalin, vernolepin, and vernolide on HepG2 liver cancer cells
|
Thongnest, Sanit |
|
|
92 |
C |
p. |
artikel |
102 |
Xanthones from the stems of Cudrania tricuspidata and their inhibitory effects on pancreatic lipase and fat accumulation
|
Jo, Yang Hee |
|
|
92 |
C |
p. |
artikel |