nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A competent synthesis and efficient anti-inflammatory responses of isatinimino acridinedione moiety via suppression of in vivo NF-κB, COX-2 and iNOS signaling
|
Periyasami, Govindasami |
|
2019 |
90 |
C |
p. |
artikel |
2 |
Amino acids conjugated quinazolinone-Schiff’s bases as potential antimicrobial agents: Synthesis, SAR and molecular docking studies
|
Rakesh, K.P. |
|
2019 |
90 |
C |
p. |
artikel |
3 |
Antibacterial activity of 3,3′-dihydroxycurcumin (DHC) is associated with membrane perturbation
|
Polaquini, Carlos R. |
|
2019 |
90 |
C |
p. |
artikel |
4 |
Anticancer properties of N-alkyl-2, 4-diphenylimidazo [1, 2-a] quinoxalin-1-amine derivatives; kinase inhibitors
|
Rezaei, Zahra |
|
2019 |
90 |
C |
p. |
artikel |
5 |
Benzoxaboroles as dynamic covalent receptors for bioconjugation and transport of nucleosides and related drugs: Proof of action in HeLa cells
|
Samaniego Lopez, Cecilia |
|
2019 |
90 |
C |
p. |
artikel |
6 |
Bioactive aporphine alkaloids from the stems of Dasymaschalon rostratum
|
Yu, Zhangxin |
|
2019 |
90 |
C |
p. |
artikel |
7 |
Cytotoxic and neuroprotective activities of constituents from Alternaria alternate, a fungal endophyte of Psidium littorale
|
Xu, Jian |
|
2019 |
90 |
C |
p. |
artikel |
8 |
Cytotoxicity of oleanolic and ursolic acid derivatives toward hepatocellular carcinoma and evaluation of NF-κB involvement
|
Fontana, Gianfranco |
|
2019 |
90 |
C |
p. |
artikel |
9 |
Demethylbellidifolin isolated from Swertia bimaculate against human carboxylesterase 2: Kinetics and interaction mechanism merged with docking simulations
|
Liu, Tian-Tian |
|
2019 |
90 |
C |
p. |
artikel |
10 |
Design, synthesis and biological evaluation of novel thieno[3,2-d]pyrimidine and quinazoline derivatives as potent antitumor agents
|
Hu, Hao |
|
2019 |
90 |
C |
p. |
artikel |
11 |
Design, synthesis of celecoxib-tolmetin drug hybrids as selective and potent COX-2 inhibitors
|
Abdellatif, Khaled R.A. |
|
2019 |
90 |
C |
p. |
artikel |
12 |
Development of pyrazole and spiropyrazoline analogs as multifunctional agents for treatment of Alzheimer’s disease
|
Gutti, Gopichand |
|
2019 |
90 |
C |
p. |
artikel |
13 |
Dihydrofolate reductase inhibition effect of 5-substituted pyrido[2,3-d]pyrimidines: Synthesis, antitumor activity and molecular modeling study
|
Abdelaziz, Ola A. |
|
2019 |
90 |
C |
p. |
artikel |
14 |
Discovery of a novel DNA binding agent via design and synthesis of new thiazole hybrids and fused 1,2,4-triazines as potential antitumor agents: Computational, spectrometric and in silico studies
|
El-Wakil, Marwa H. |
|
2019 |
90 |
C |
p. |
artikel |
15 |
Discovery of aromatic amides with triazole-core as potent reversal agents against P-glycoprotein-mediated multidrug resistance
|
Qiu, Qianqian |
|
2019 |
90 |
C |
p. |
artikel |
16 |
Discovery of novel indole-based aroylhydrazones as anticonvulsants: Pharmacophore-based design
|
Angelova, Violina T. |
|
2019 |
90 |
C |
p. |
artikel |
17 |
DNA interaction and photodynamic antitumor activity of transition metal mono-hydroxyl corrole
|
Sun, Yan-Mei |
|
2019 |
90 |
C |
p. |
artikel |
18 |
Editorial Board
|
|
|
2019 |
90 |
C |
p. |
artikel |
19 |
Exploiting the 7-methylimidazo[1,5-a]pyrazin-8(7H)-one scaffold for the development of novel chemical inhibitors for Bromodomain and Extraterminal Domain (BET) family
|
Yang, Yifei |
|
2019 |
90 |
C |
p. |
artikel |
20 |
Extraction, isolation and in vitro evaluation of affinisine from Tabernaemontana catharinensis in human melanoma cells
|
Fagundes Rosales, Pauline |
|
2019 |
90 |
C |
p. |
artikel |
21 |
Facile synthesis and antimicrobial activity of CdS-Ag2S nanocomposites
|
Iqbal, Tahir |
|
2019 |
90 |
C |
p. |
artikel |
22 |
Green synthesis of selenium-N-heterocyclic carbene compounds: Evaluation of antimicrobial and anticancer potential
|
Kamal, Amna |
|
2019 |
90 |
C |
p. |
artikel |
23 |
Human neutrophil elastase (HNE) inhibitory polyprenylated acylphloroglucinols from the flowers of Hypericum ascyron
|
Li, Zuo Peng |
|
2019 |
90 |
C |
p. |
artikel |
24 |
Identification of chebulinic acid as a dual targeting inhibitor of protein tyrosine phosphatases relevant to insulin resistance
|
Yoon, Sun-Young |
|
2019 |
90 |
C |
p. |
artikel |
25 |
Identification of nicotinamide aminonaphthyridine compounds as potent RET kinase inhibitors and antitumor activities against RET rearranged lung adenocarcinoma
|
Wang, Modi |
|
2019 |
90 |
C |
p. |
artikel |
26 |
Improving the catalytic efficiency of aldo-keto reductase KmAKR towards t-butyl 6-cyano-(3R,5R)-dihydroxyhexanoate via semi-rational design
|
Yu, Han |
|
2019 |
90 |
C |
p. |
artikel |
27 |
Investigation of potent inhibitors of cholinesterase based on thiourea and pyrazoline derivatives: Synthesis, inhibition assay and molecular modeling studies
|
Mumtaz, Amara |
|
2019 |
90 |
C |
p. |
artikel |
28 |
Isolation and characterization of three pairs of indolediketopiperazine enantiomers containing infrequent N-methoxy substitution from the marine algal-derived endophytic fungus Acrostalagmus luteoalbus TK-43
|
Cao, Jin |
|
2019 |
90 |
C |
p. |
artikel |
29 |
Issue TOC
|
|
|
2019 |
90 |
C |
p. |
artikel |
30 |
(±)-Meliviticines A and B: Rearranged prenylated acetophenone derivatives from Melicope viticina and their antimicrobial activity
|
Li, Wei |
|
2019 |
90 |
C |
p. |
artikel |
31 |
Muscle extract of Arothron immaculatus regulates the blood glucose level and the antioxidant system in high-fat diet and streptozotocin induced diabetic rats
|
Kaleshkumar, Karunanidhi |
|
2019 |
90 |
C |
p. |
artikel |
32 |
New phenolic Mannich bases with piperazines and their bioactivities
|
Gul, Halise Inci |
|
2019 |
90 |
C |
p. |
artikel |
33 |
New potent antifungal triazole alcohols containing N-benzylpiperazine carbodithioate moiety: Synthesis, in vitro evaluation and in silico study
|
Mahmoudi, Yaser |
|
2019 |
90 |
C |
p. |
artikel |
34 |
Novel cytisine derivatives exert anti-liver fibrosis effect via PI3K/Akt/Smad pathway
|
Tang, Sheng |
|
2019 |
90 |
C |
p. |
artikel |
35 |
Novel 12-hydroxydehydroabietylamine derivatives act as potent and selective butyrylcholinesterase inhibitors
|
Loesche, Anne |
|
2019 |
90 |
C |
p. |
artikel |
36 |
Novel Pyrazoloquinolin-2-ones: Design, synthesis, docking studies, and biological evaluation as antiproliferative EGFR-TK inhibitors
|
Elbastawesy, Mohammed A.I. |
|
2019 |
90 |
C |
p. |
artikel |
37 |
One-step synthesis of methylene-bridged bis-carbazole and evaluation of its antitumor activity and G-quadruplex DNA binding property
|
Li, Gang |
|
2019 |
90 |
C |
p. |
artikel |
38 |
Potential chemical transformation of phosphinic acid derivatives and their applications in the synthesis of drugs
|
Abdou, Moaz M. |
|
2019 |
90 |
C |
p. |
artikel |
39 |
Preface
|
Żymańczyk-Duda, Ewa |
|
2019 |
90 |
C |
p. |
artikel |
40 |
Probing the binding mechanism of capecitabine to human serum albumin using spectrometric methods, molecular modeling, and chemometrics approach
|
Mousavi, S. Fatemeh |
|
2019 |
90 |
C |
p. |
artikel |
41 |
Protective effect of hypoxylonol C and 4,5,4′,5′-tetrahydroxy-1,1′-binaphthyl isolated from Annulohypoxylon annulatum against streptozotocin-induced damage in INS-1 cells
|
Lee, Dahae |
|
2019 |
90 |
C |
p. |
artikel |
42 |
Repurposing the scorpion venom peptide VmCT1 into an active peptide against Gram-negative ESKAPE pathogens
|
Pedron, Cibele Nicolaski |
|
2019 |
90 |
C |
p. |
artikel |
43 |
Search for multifunctional agents against Alzheimer’s disease among non-imidazole histamine H3 receptor ligands. In vitro and in vivo pharmacological evaluation and computational studies of piperazine derivatives
|
Jończyk, Jakub |
|
2019 |
90 |
C |
p. |
artikel |
44 |
Substituted cinnamic anhydrides act as selective inhibitors of acetylcholinesterase
|
Gießel, Josephine M. |
|
2019 |
90 |
C |
p. |
artikel |
45 |
Substituted phenyl[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetates/acetamides as alkaline phosphatase inhibitors: Synthesis, computational studies, enzyme inhibitory kinetics and DNA binding studies
|
Iqbal, Zafar |
|
2019 |
90 |
C |
p. |
artikel |
46 |
6-Substituted purines as ROCK inhibitors with anti-metastatic activity
|
Voller, Jiří |
|
2019 |
90 |
C |
p. |
artikel |
47 |
Synthesis and anticancer activity of bis-benzo[d][1,3]dioxol-5-yl thiourea derivatives with molecular docking study
|
Al-Harbi, Reem A.K. |
|
2019 |
90 |
C |
p. |
artikel |
48 |
Synthesis and antitumor activity of three novel ginsenoside M1 derivatives with 3′-ester modifications
|
Li, Ke-Ke |
|
2019 |
90 |
C |
p. |
artikel |
49 |
Synthesis and biological evaluation of indoloquinoline alkaloid cryptolepine and its bromo-derivative as dual cholinesterase inhibitors
|
Nuthakki, Vijay K. |
|
2019 |
90 |
C |
p. |
artikel |
50 |
Synthesis and biological evaluation of some new mono Mannich bases with piperazines as possible anticancer agents and carbonic anhydrase inhibitors
|
Tugrak, Mehtap |
|
2019 |
90 |
C |
p. |
artikel |
51 |
Synthesis and in vitro anti-tumor activity of carboranyl levodopa
|
Zhu, Yinghuai |
|
2019 |
90 |
C |
p. |
artikel |
52 |
Synthesis, anti-diabetic evaluation and molecular docking studies of 4-(1-aryl-1H-1, 2, 3-triazol-4-yl)-1,4-dihydropyridine derivatives as novel 11-β hydroxysteroid dehydrogenase-1 (11β-HSD1) inhibitors
|
Praveenkumar, E. |
|
2019 |
90 |
C |
p. |
artikel |
53 |
Synthesis, biological evaluation and in silico studies with 4-benzylidene-2-phenyl-5(4H)-imidazolone-based benzenesulfonamides as novel selective carbonic anhydrase IX inhibitors endowed with anticancer activity
|
Eldehna, Wagdy M. |
|
2019 |
90 |
C |
p. |
artikel |
54 |
Synthesis, modeling and biological evaluation of some pyrazolo[3,4-d]pyrimidinones and pyrazolo[4,3-e][1,2,4]triazolo[4,3-a]pyrimidinones as anti-inflammatory agents
|
Tageldin, Gina N. |
|
2019 |
90 |
C |
p. |
artikel |
55 |
Synthesis, molecular docking and kinetic studies of novel quinolinyl based acyl thioureas as mushroom tyrosinase inhibitors and free radical scavengers
|
Mustafa, Muhammad Naeem |
|
2019 |
90 |
C |
p. |
artikel |
56 |
5,6,7,8-Tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidine derivatives as inhibitors of full-length RORγt
|
Lao, Chuyu |
|
2019 |
90 |
C |
p. |
artikel |
57 |
The green synthesis and molecular docking of novel N-substituted rhodanines as effective inhibitors for carbonic anhydrase and acetylcholinesterase enzymes
|
Bayindir, Sinan |
|
2019 |
90 |
C |
p. |
artikel |
58 |
The stilbene derivatives, nucleosides, and nucleosides modified by stilbene derivatives
|
Krawczyk, Hanna |
|
2019 |
90 |
C |
p. |
artikel |
59 |
Triazole substituted metal-free, metallo-phthalocyanines and their water soluble derivatives as potential cholinesterases inhibitors: Design, synthesis and in vitro inhibition study
|
Arslan, Tayfun |
|
2019 |
90 |
C |
p. |
artikel |
60 |
Ultrasound-assisted synthesis of novel chalcone, heterochalcone and bis-chalcone derivatives and the evaluation of their antioxidant properties and as acetylcholinesterase inhibitors
|
Polo, Efraín |
|
2019 |
90 |
C |
p. |
artikel |