nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Anticancer and DNA binding studies of potential amino acids based quinazolinone analogs: Synthesis, SAR and molecular docking
|
Rakesh, K.P. |
|
2019 |
87 |
C |
p. 252-264 |
artikel |
2 |
Anti-diabetic potential of Pueraria lobata root extract through promoting insulin signaling by PTP1B inhibition
|
Sun, Ran |
|
2019 |
87 |
C |
p. 12-15 |
artikel |
3 |
Antioxidant and angiotensin-converting enzyme (ACE) inhibitory activity of thymosin alpha-1 (Thα1) peptide
|
Kharazmi-Khorassani, Jasmin |
|
2019 |
87 |
C |
p. 743-752 |
artikel |
4 |
Antiproliferative effect, cell cycle arrest and apoptosis generation of novel synthesized anticancer heterocyclic derivatives based 4H-benzo[h]chromene
|
Alblewi, Fawzia F. |
|
2019 |
87 |
C |
p. 560-571 |
artikel |
5 |
Azacoccone E inhibits cancer cell growth by targeting 3-phosphoglycerate dehydrogenase
|
Guo, Jing |
|
2019 |
87 |
C |
p. 16-22 |
artikel |
6 |
Benzoxazinone-thiosemicarbazones as antidiabetic leads via aldose reductase inhibition: Synthesis, biological screening and molecular docking study
|
Shehzad, Muhammad Tariq |
|
2019 |
87 |
C |
p. 857-866 |
artikel |
7 |
Bioactive terpenoids from Euonymus verrucosus var. pauciflorus showing NO inhibitory activities
|
Yang, Yuling |
|
2019 |
87 |
C |
p. 447-456 |
artikel |
8 |
Bioassay-guided isolation of antioxidant and α-glucosidase inhibitory constituents from stem of Vigna angularis
|
Guo, Feng |
|
2019 |
87 |
C |
p. 312-320 |
artikel |
9 |
Characterization, quantitation, similarity evaluation and combination with Na+,K+-ATPase of cardiac glycosides from Streblus asper
|
Bai, Yidan |
|
2019 |
87 |
C |
p. 265-275 |
artikel |
10 |
Cucurbitane-type compounds from Momordica charantia: Isolation, in vitro antidiabetic, anti-inflammatory activities and in silico modeling approaches
|
Shivanagoudra, Siddanagouda R. |
|
2019 |
87 |
C |
p. 31-42 |
artikel |
11 |
Cytotoxic polyhydroxy serratene triterpenoids from Lycopodium complanatum
|
Dong, Qiuzhu |
|
2019 |
87 |
C |
p. 373-379 |
artikel |
12 |
Design and synthesis of mono-and di-pyrazolyl-s-triazine derivatives, their anticancer profile in human cancer cell lines, and in vivo toxicity in zebrafish embryos
|
Farooq, Muhammad |
|
2019 |
87 |
C |
p. 457-464 |
artikel |
13 |
Design and synthesis of novel PARP-1 inhibitors based on pyridopyridazinone scaffold
|
Elmasry, Ghada F. |
|
2019 |
87 |
C |
p. 655-666 |
artikel |
14 |
Design and synthesis of parthenolide-SAHA hybrids for intervention of drug-resistant acute myeloid leukemia
|
Ge, Weizhi |
|
2019 |
87 |
C |
p. 699-713 |
artikel |
15 |
Design, synthesis and biological evaluation of Helicobacter pylori inosine 5′-monophosphate dehydrogenase (HpIMPDH) inhibitors. Further optimization of selectivity towards HpIMPDH over human IMPDH2
|
Shah, Chetan P. |
|
2019 |
87 |
C |
p. 753-764 |
artikel |
16 |
Design, synthesis, and carbonic anhydrase inhibition activity of benzenesulfonamide-linked novel pyrazoline derivatives
|
Abdel-Aziz, Alaa A.-M. |
|
2019 |
87 |
C |
p. 425-431 |
artikel |
17 |
Design, synthesis and evaluation of a novel metal chelator as multifunctional agents for the treatment of Alzheimer’s disease
|
Wang, Yingying |
|
2019 |
87 |
C |
p. 720-727 |
artikel |
18 |
Design, synthesis and evaluation of chalcone Mannich base derivatives as multifunctional agents for the potential treatment of Alzheimer’s disease
|
Zhang, Xiaoyu |
|
2019 |
87 |
C |
p. 395-408 |
artikel |
19 |
Design, synthesis and evaluation of 2-(indolylmethylidene)-2,3-dihydro-1-benzofuran-3-one and 2-(indolyl)-4H-chromen-4-one derivatives as novel monoamine oxidases inhibitors
|
Takao, Koichi |
|
2019 |
87 |
C |
p. 594-600 |
artikel |
20 |
Development of a versatile DNMT and HDAC inhibitor C02S modulating multiple cancer hallmarks for breast cancer therapy
|
Yuan, Zigao |
|
2019 |
87 |
C |
p. 200-208 |
artikel |
21 |
Development of novel 2-substituted acylaminoethylsulfonamide derivatives as fungicides against Botrytis cinerea
|
Wang, Minlong |
|
2019 |
87 |
C |
p. 56-69 |
artikel |
22 |
Discovery of new inhibitors against both NF-κB and osteoclastogenesis from in-house library with α, β-unsaturated-enone fragment
|
Zhao, Chao |
|
2019 |
87 |
C |
p. 638-646 |
artikel |
23 |
Dual targeting of PTP1B and glucosidases with new bifunctional iminosugar inhibitors to address type 2 diabetes
|
Ferhati, Xhenti |
|
2019 |
87 |
C |
p. 534-549 |
artikel |
24 |
Editorial Board
|
|
|
2019 |
87 |
C |
p. i |
artikel |
25 |
Eight new glycosides with hepatoprotective activity isolated from the aerial parts of Morinda parvifolia
|
Su, Xianming |
|
2019 |
87 |
C |
p. 867-875 |
artikel |
26 |
Evaluation of angularly condensed diquinothiazines as potential anticancer agents
|
Jeleń, Małgorzata |
|
2019 |
87 |
C |
p. 810-820 |
artikel |
27 |
Evaluation of guanylhydrazone derivatives as inhibitors of Candida rugosa digestive lipase: Biological, biophysical, theoretical studies and biotechnological application
|
Santana, Camilla C. |
|
2019 |
87 |
C |
p. 169-180 |
artikel |
28 |
Fluorescent labeling of ursolic acid with FITC for investigation of its cytotoxic activity using confocal microscopy
|
Frolova, Tatiana S. |
|
2019 |
87 |
C |
p. 876-887 |
artikel |
29 |
Furofuran lignans as a new series of antidiabetic agents exerting α-glucosidase inhibition and radical scarvenging: Semisynthesis, kinetic study and molecular modeling
|
Worawalai, Wisuttaya |
|
2019 |
87 |
C |
p. 783-793 |
artikel |
30 |
Glycopentanolones A-D, four new geranylated quinolone alkaloids from Glycosmis pentaphylla
|
Choi, Yun-Hyeok |
|
2019 |
87 |
C |
p. 714-719 |
artikel |
31 |
Hyperpatulols A–I, spirocyclic acylphloroglucinol derivatives with anti-migration activities from the flowers of Hypericum patulum
|
Liu, Yang-Yang |
|
2019 |
87 |
C |
p. 409-416 |
artikel |
32 |
Inhibition of biofilm formation, quorum sensing activity and molecular docking study of isolated 3, 5, 7-Trihydroxyflavone from Alstonia scholaris leaf against P.aeruginosa
|
Abinaya, M. |
|
2019 |
87 |
C |
p. 291-301 |
artikel |
33 |
Interaction of C20-substituted derivative of pregnenolone acetate with copper (II) leads to ROS generation, DNA cleavage and apoptosis in cervical cancer cells: Therapeutic potential of copper chelation for cancer treatment
|
Zafar, Atif |
|
2019 |
87 |
C |
p. 276-290 |
artikel |
34 |
Introduction of amino moiety enhances the inhibitory potency of 1-tetralone chalcone derivatives against LPS-stimulated reactive oxygen species production in RAW 264.7 macrophages
|
Katila, Pramila |
|
2019 |
87 |
C |
p. 495-505 |
artikel |
35 |
Investigation of new quinoline derivatives as promising inhibitors of NTPDases: Synthesis, SAR analysis and molecular docking studies
|
Hayat, Komal |
|
2019 |
87 |
C |
p. 218-226 |
artikel |
36 |
In vitro and in silico studies of novel synthetic ACE-inhibitory peptides derived from Saccharomyces cerevisiae protein hydrolysate
|
Mirzaei, Mahta |
|
2019 |
87 |
C |
p. 647-654 |
artikel |
37 |
Iridoids from Valeriana jatamansi induce autophagy-associated cell death via the PDK1/Akt/mTOR pathway in HCT116 human colorectal carcinoma cells
|
Tan, Yu-Zhu |
|
2019 |
87 |
C |
p. 136-141 |
artikel |
38 |
Isoindolin-1-one derivatives as urease inhibitors: Design, synthesis, biological evaluation, molecular docking and in-silico ADME evaluation
|
Peytam, Fariba |
|
2019 |
87 |
C |
p. 1-11 |
artikel |
39 |
Issue TOC
|
|
|
2019 |
87 |
C |
p. ii-xxvii |
artikel |
40 |
Lithocarols A-F, six tenellone derivatives from the deep-sea derived fungus Phomopsis lithocarpus FS508
|
Xu, Jianlin |
|
2019 |
87 |
C |
p. 728-735 |
artikel |
41 |
Mechanistic investigation of anthocyanidin derivatives as α-glucosidase inhibitors
|
Kim, Jang Hoon |
|
2019 |
87 |
C |
p. 803-809 |
artikel |
42 |
Meglumine as a green, efficient and reusable catalyst for synthesis and molecular docking studies of bis(indolyl)methanes as antioxidant agents
|
Nemallapudi, Bakthavatchala Reddy |
|
2019 |
87 |
C |
p. 465-473 |
artikel |
43 |
Multi-target-directed triazole derivatives as promising agents for the treatment of Alzheimer’s disease
|
Kaur, Anupamjeet |
|
2019 |
87 |
C |
p. 572-584 |
artikel |
44 |
Natural and semisynthetic oxyprenylated aromatic compounds as stimulators or inhibitors of melanogenesis
|
Genovese, Salvatore |
|
2019 |
87 |
C |
p. 181-190 |
artikel |
45 |
Natural flavonoid α-glucosidase inhibitors from Retama raetam: Enzyme inhibition and molecular docking reveal important interactions with the enzyme active site
|
Ghani, Usman |
|
2019 |
87 |
C |
p. 736-742 |
artikel |
46 |
Natural product-based design, synthesis and biological evaluation of 2′,3,4,4′-tetrahydrochalcone analogues as antivitiligo agents
|
Zhong, Hui |
|
2019 |
87 |
C |
p. 523-533 |
artikel |
47 |
New benzyl pyridinium derivatives bearing 2,4-dioxochroman moiety as potent agents for treatment of Alzheimer’s disease: Design, synthesis, biological evaluation, and docking study
|
Mollazadeh, Marjan |
|
2019 |
87 |
C |
p. 506-515 |
artikel |
48 |
New phosphate derivatives of betulin as anticancer agents: Synthesis, crystal structure, and molecular docking study
|
Chrobak, Elwira |
|
2019 |
87 |
C |
p. 613-628 |
artikel |
49 |
Nitrogen-containing derivatives of O-tetramethylquercetin: Synthesis and biological profiles in prostate cancer cell models
|
Rajaram, Pravien |
|
2019 |
87 |
C |
p. 227-239 |
artikel |
50 |
NO inhibitory phytochemicals as potential anti-inflammatory agents from the twigs of Trigonostemon heterophyllus
|
Xi, Yaru |
|
2019 |
87 |
C |
p. 417-424 |
artikel |
51 |
Novel 8-amino-1,2,4-triazolo[4,3-a]pyrazin-3-one derivatives as potent human adenosine A1 and A2A receptor antagonists. Evaluation of their protective effect against β-amyloid-induced neurotoxicity in SH-SY5Y cells
|
Falsini, Matteo |
|
2019 |
87 |
C |
p. 380-394 |
artikel |
52 |
Novel synthesized SLC-0111 thiazole and thiadiazole analogues: Determination of their carbonic anhydrase inhibitory activity and molecular modeling studies
|
Abo-Ashour, Mahmoud F. |
|
2019 |
87 |
C |
p. 794-802 |
artikel |
53 |
Organometallic ruthenium(II)-arene complexes with triphenylphosphine amino acid bioconjugates: Synthesis, characterization and biological properties
|
Pernar, Margareta |
|
2019 |
87 |
C |
p. 432-446 |
artikel |
54 |
Phenylsulfonyl piperazine bridged [1,3]dioxolo[4,5-g]chromenones as promising antiproliferative and antioxidant agents
|
Patel, Rahul V. |
|
2019 |
87 |
C |
p. 23-30 |
artikel |
55 |
Pomalidomide hybrids act as proteolysis targeting chimeras: Synthesis, anticancer activity and B-Raf degradation
|
Chen, Hong |
|
2019 |
87 |
C |
p. 191-199 |
artikel |
56 |
Probing the antibacterial and anticancer potential of tryptamine based mixed ligand Schiff base Ruthenium(III) complexes
|
Malik, Manzoor Ahmad |
|
2019 |
87 |
C |
p. 773-782 |
artikel |
57 |
Promising anti-inflammatory effects of chalcones via inhibition of cyclooxygenase, prostaglandin E2, inducible NO synthase and nuclear factor κb activities
|
ur Rashid, Haroon |
|
2019 |
87 |
C |
p. 335-365 |
artikel |
58 |
Rhamnolipid inspired lipopeptides effective in preventing adhesion and biofilm formation of Candida albicans
|
Jovanovic, Milos |
|
2019 |
87 |
C |
p. 209-217 |
artikel |
59 |
Sanggenon O induced apoptosis of A549 cells is counterbalanced by protective autophagy
|
Li, Zhong-Rui |
|
2019 |
87 |
C |
p. 688-698 |
artikel |
60 |
Semi-synthetic isoflavones as BACE-1 inhibitors against Alzheimer’s disease
|
Ribaudo, Giovanni |
|
2019 |
87 |
C |
p. 474-483 |
artikel |
61 |
Sesquiterpenes from Curcuma zedoaria rhizomes and their cytotoxicity against human gastric cancer AGS cells
|
Lee, Tae Kyoung |
|
2019 |
87 |
C |
p. 117-122 |
artikel |
62 |
Structure-based design, synthesis and biological evaluation of a newer series of pyrazolo[1,5-a]pyrimidine analogues as potential anti-tubercular agents
|
Modi, Palmi |
|
2019 |
87 |
C |
p. 240-251 |
artikel |
63 |
Sulfenamide derivatives can improve transporter-mediated cellular uptake of metformin and induce cytotoxicity in human breast adenocarcinoma cell lines
|
Markowicz-Piasecka, Magdalena |
|
2019 |
87 |
C |
p. 321-334 |
artikel |
64 |
Sulfur, selenium and tellurium containing amines act as effective carbonic anhydrase activators
|
Tanini, Damiano |
|
2019 |
87 |
C |
p. 516-522 |
artikel |
65 |
Synthesis and antiproliferative activity of new 2-glyco-3-nitro-2H-chromenes
|
Luque-Agudo, Verónica |
|
2019 |
87 |
C |
p. 112-116 |
artikel |
66 |
Synthesis and biological evaluation of coumarin-1,3,4-oxadiazole hybrids as selective carbonic anhydrase IX and XII inhibitors
|
Narella, Sridhar Goud |
|
2019 |
87 |
C |
p. 765-772 |
artikel |
67 |
Synthesis and biological evaluation of new bisindole-imidazopyridine hybrids as apoptosis inducers
|
Sunkari, Satish |
|
2019 |
87 |
C |
p. 484-494 |
artikel |
68 |
Synthesis and biological evaluation of purine-pyrazole hybrids incorporating thiazole, thiazolidinone or rhodanine moiety as 15-LOX inhibitors endowed with anticancer and antioxidant potential
|
Afifi, Ola S. |
|
2019 |
87 |
C |
p. 821-837 |
artikel |
69 |
Synthesis and characterization of new thiosemicarbazones, as potent urease inhibitors: In vitro and in silico studies
|
Islam, Muhammad |
|
2019 |
87 |
C |
p. 155-162 |
artikel |
70 |
Synthesis and characterization of novel bromophenols: Determination of their anticholinergic, antidiabetic and antioxidant activities
|
Öztaşkın, Necla |
|
2019 |
87 |
C |
p. 91-102 |
artikel |
71 |
Synthesis and evaluation of novel benzotropolones as Atg4B inhibiting autophagy blockers
|
Tanc, Muhammet |
|
2019 |
87 |
C |
p. 163-168 |
artikel |
72 |
Synthesis and evaluation of novel α-substituted chalcones with potent anti-cancer activities and ability to overcome multidrug resistance
|
Riaz, Sharon |
|
2019 |
87 |
C |
p. 123-135 |
artikel |
73 |
Synthesis, bioactivity and molecular modeling studies on potential anti-Alzheimer piperidinehydrazide-hydrazones
|
Parlar, Sulunay |
|
2019 |
87 |
C |
p. 888-900 |
artikel |
74 |
Synthesis, biological activity and multiscale molecular modeling studies of bis-coumarins as selective carbonic anhydrase IX and XII inhibitors with effective cytotoxicity against hepatocellular carcinoma
|
Kurt, Belma Zengin |
|
2019 |
87 |
C |
p. 838-850 |
artikel |
75 |
Synthesis, biological evaluation and molecular modelling studies of 1,3,7,8-tetrasubstituted xanthines as potent and selective A2A AR ligands with in vivo efficacy against animal model of Parkinson’s disease
|
Rohilla, Suman |
|
2019 |
87 |
C |
p. 601-612 |
artikel |
76 |
Synthesis, evaluation and docking of novel pyrazolo pyrimidines as potent p38α MAP kinase inhibitors with improved anti-inflammatory, ulcerogenic and TNF-α inhibitory properties
|
Somakala, Kanagasabai |
|
2019 |
87 |
C |
p. 550-559 |
artikel |
77 |
Synthesis, molecular docking studies, and antimicrobial evaluation of new structurally diverse ureas
|
Patil, Mahadev |
|
2019 |
87 |
C |
p. 302-311 |
artikel |
78 |
Synthesis of benzensulfonamides linked to quinazoline scaffolds as novel carbonic anhydrase inhibitors
|
El-Azab, Adel S. |
|
2019 |
87 |
C |
p. 78-90 |
artikel |
79 |
Synthesis of CC, CN coupled novel substituted dibutyl benzothiazepinone derivatives and evaluation of their thrombin inhibitory activity
|
Baburajeev, C.P. |
|
2019 |
87 |
C |
p. 142-154 |
artikel |
80 |
Synthesis of compounds having antimicrobial activity from alginate
|
Salem, Dalia M.S.A. |
|
2019 |
87 |
C |
p. 103-111 |
artikel |
81 |
Synthesis of TPEN variants to improve cancer cells selective killing capacity
|
Schaefer-Ramadan, Stephanie |
|
2019 |
87 |
C |
p. 366-372 |
artikel |
82 |
The comparative study of the DNA binding and biological activities of the quaternized dicnq as a dicationic form and its platinum(II) heteroleptic cationic complex
|
Yıldız, Ufuk |
|
2019 |
87 |
C |
p. 70-77 |
artikel |
83 |
5-Thioxoimidazolidine-2-one derivatives: Synthesis, anti-inflammatory activity, analgesic activity, COX inhibition assay and molecular modelling study
|
El-Sharief, Marwa A.M.Sh. |
|
2019 |
87 |
C |
p. 679-687 |
artikel |
84 |
Tick-borne flavivirus reproduction inhibitors based on isoxazole core linked with adamantane
|
Vasilenko, Dmitry A. |
|
2019 |
87 |
C |
p. 629-637 |
artikel |
85 |
Tyrosinase inhibition and anti-melanin generation effect of cinnamamide analogues
|
Ullah, Sultan |
|
2019 |
87 |
C |
p. 43-55 |
artikel |
86 |
Unveiling novel diphenyl-1H-pyrazole based acrylates tethered to 1,2,3-triazole as promising apoptosis inducing cytotoxic and anti-inflammatory agents
|
Khan, Mohemmed Faraz |
|
2019 |
87 |
C |
p. 667-678 |
artikel |
87 |
Withanolides from Physalis peruviana showing nitric oxide inhibitory effects and affinities with iNOS
|
Dong, Bangjian |
|
2019 |
87 |
C |
p. 585-593 |
artikel |
88 |
Xanthine oxidase inhibitors from an endophytic fungus Lasiodiplodia pseudotheobromae
|
Kumar, Sanjay |
|
2019 |
87 |
C |
p. 851-856 |
artikel |