nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A novel bi-functional chalcone inhibits multi-drug resistant Staphylococcus aureus and potentiates the activity of fluoroquinolones
|
Gupta, Vivek Kumar |
|
2019 |
83 |
C |
p. 214-225 |
artikel |
2 |
Antibacterial activity against drug-resistant microbial pathogens of cytochalasan alkaloids from the arthropod-associated fungus Chaetomium globosum TW1-1
|
Gao, Weixi |
|
2019 |
83 |
C |
p. 98-104 |
artikel |
3 |
Antileishmanial activity and ultrastructural changes of sesquiterpene lactones isolated from Calea pinnatifida (Asteraceae)
|
Caldas, Lhaís Araújo |
|
2019 |
83 |
C |
p. 348-353 |
artikel |
4 |
2-Aryl-quinazolin-4(3H)-ones as an inhibitor of leishmania folate pathway: In vitro biological evaluation, mechanism studies and molecular docking
|
Romero, Angel H. |
|
2019 |
83 |
C |
p. 145-153 |
artikel |
5 |
Assessment of novel azaanthraquinone derivatives as potent multi-target inhibitors of inflammation and amyloid-β aggregation in Alzheimer’s disease
|
Wang, Juan |
|
2019 |
83 |
C |
p. 477-486 |
artikel |
6 |
Bioactive monoterpene indole alkaloids from Nauclea officinalis
|
Liu, Yan-Ping |
|
2019 |
83 |
C |
p. 1-5 |
artikel |
7 |
Biology-oriented drug synthesis (BIODS), in vitro urease inhibitory activity, and in silico study of S-naproxen derivatives
|
Mohiuddin, Ghulam |
|
2019 |
83 |
C |
p. 29-46 |
artikel |
8 |
bioNMR-based identification of natural anti-Aβ compounds in Peucedanum ostruthium
|
Palmioli, Alessandro |
|
2019 |
83 |
C |
p. 76-86 |
artikel |
9 |
Carbazole and hydrazone derivatives as new competitive inhibitors of tyrosinase: Experimental clues to binuclear copper active site binding
|
Ghani, Usman |
|
2019 |
83 |
C |
p. 235-241 |
artikel |
10 |
Chemical fabrication of graphene oxide nanosheets attenuates biofilm formation of human clinical pathogens
|
Ramalingam, Vaikundamoorthy |
|
2019 |
83 |
C |
p. 326-335 |
artikel |
11 |
Design and synthesis of novel quinazolinone-1,2,3-triazole hybrids as new anti-diabetic agents: In vitro α-glucosidase inhibition, kinetic, and docking study
|
Saeedi, Mina |
|
2019 |
83 |
C |
p. 161-169 |
artikel |
12 |
Design, synthesis and anti-Alzheimer’s activity of novel 1,2,3-triazole-chromenone carboxamide derivatives
|
Rastegari, Arezoo |
|
2019 |
83 |
C |
p. 391-401 |
artikel |
13 |
Design, synthesis and bioevaluation of tricyclic fused ring system as dual binding site acetylcholinesterase inhibitors
|
Tanoli, Saba Tahir |
|
2019 |
83 |
C |
p. 336-347 |
artikel |
14 |
Design, synthesis, and biological activities of 1-aryl-(3-(2-styryl)phenyl)prop-2-en-1-ones
|
Shin, Soon Young |
|
2019 |
83 |
C |
p. 438-449 |
artikel |
15 |
Design, synthesis and in vitro apoptotic mechanism of novel pyrrolopyrimidine derivatives
|
Kilic-Kurt, Zühal |
|
2019 |
83 |
C |
p. 511-519 |
artikel |
16 |
Design, synthesis and molecular modeling study of certain VEGFR-2 inhibitors based on thienopyrimidne scaffold as cancer targeting agents
|
Ghith, Amna |
|
2019 |
83 |
C |
p. 111-128 |
artikel |
17 |
Design, synthesis and pharmacological evaluation of some substituted dihydropyrimidines with L-/T-type calcium channel blocking activities
|
Teleb, Mohamed |
|
2019 |
83 |
C |
p. 354-366 |
artikel |
18 |
Design, synthesis, structural characterization and in vitro evaluation of new 1,4-disubstituted-1,2,3-triazole derivatives against glioblastoma cells
|
da Silva, Veronica D. |
|
2019 |
83 |
C |
p. 87-97 |
artikel |
19 |
Discovery of novel quinazolines as potential anti-tubulin agents occupying three zones of colchicine domain
|
Li, Wenlong |
|
2019 |
83 |
C |
p. 380-390 |
artikel |
20 |
Dual effects of isoflavonoids from Pueraria lobata roots on estrogenic activity and anti-proliferation of MCF-7 human breast carcinoma cells
|
Ahn, Soo-Yeon |
|
2019 |
83 |
C |
p. 135-144 |
artikel |
21 |
Editorial Board
|
|
|
2019 |
83 |
C |
p. i |
artikel |
22 |
Introduction of Z-GP scaffold into procarbazine reduces spermatoxicity and myelosuppression
|
Wang, Rikang |
|
2019 |
83 |
C |
p. 461-467 |
artikel |
23 |
In vitro activities of a new fluoroquinolone derivative highly active against Chlamydia trachomatis
|
Vu, Thi Huyen |
|
2019 |
83 |
C |
p. 180-185 |
artikel |
24 |
Issue TOC
|
|
|
2019 |
83 |
C |
p. ii-xix |
artikel |
25 |
Molecular-docking-guided design and synthesis of new IAA-tacrine hybrids as multifunctional AChE/BChE inhibitors
|
Cheng, Zhi-Qiang |
|
2019 |
83 |
C |
p. 277-288 |
artikel |
26 |
Neuroprotective effects of triterpenoid saponins from Medicago sativa L. against H2O2-induced oxidative stress in SH-SY5Y cells
|
Liu, Xue-Gui |
|
2019 |
83 |
C |
p. 468-476 |
artikel |
27 |
New benzimidazothiazole derivatives as anti-inflammatory, antitumor active agents: Synthesis, in-vitro and in-vivo screening and molecular modeling studies
|
El-Kerdawy, Mohamed M. |
|
2019 |
83 |
C |
p. 250-261 |
artikel |
28 |
New iridal-type triterpenoid derivatives with cytotoxic activities from Belamcanda chinensis
|
Li, Jiayuan |
|
2019 |
83 |
C |
p. 20-28 |
artikel |
29 |
Novel dauricine derivatives suppress cancer via autophagy-dependent cell death
|
Zhou, Xiaobo |
|
2019 |
83 |
C |
p. 450-460 |
artikel |
30 |
Novel hybrids of benzothiazole-1,3,4-oxadiazole-4-thiazolidinone: Synthesis, in silico ADME study, molecular docking and in vivo anti-diabetic assessment
|
Bhutani, Rubina |
|
2019 |
83 |
C |
p. 6-19 |
artikel |
31 |
Novel nalidixic acid derivatives targeting topoisomerase II enzyme; Design, synthesis, anticancer activity and effect on cell cycle profile
|
Khalil, Omneya M. |
|
2019 |
83 |
C |
p. 262-276 |
artikel |
32 |
Novel 4-(3-phenylpropionamido), 4-(2-phenoxyacetamido) and 4-(cinnamamido) substituted benzamides bearing the pyrazole or indazole nucleus: synthesis, biological evaluation and mechanism of action
|
Raffa, Demetrio |
|
2019 |
83 |
C |
p. 367-379 |
artikel |
33 |
Novel tacrine-coumarin hybrids linked to 1,2,3-triazole as anti-Alzheimer’s compounds: In vitro and in vivo biological evaluation and docking study
|
Najafi, Zahra |
|
2019 |
83 |
C |
p. 303-316 |
artikel |
34 |
Potential bioisosteres of β-uracilalanines derived from 1H-1,2,3-triazole-C-carboxylic acids
|
Mironiuk-Puchalska, Ewa |
|
2019 |
83 |
C |
p. 500-510 |
artikel |
35 |
Preparation, characterization and in vitro activity of a docetaxel–albumin conjugate
|
Gao, Jing |
|
2019 |
83 |
C |
p. 154-160 |
artikel |
36 |
Proliferation inhibition of novel diphenylamine derivatives
|
Janovec, Ladislav |
|
2019 |
83 |
C |
p. 487-499 |
artikel |
37 |
α-Pyrones, secondary metabolites from fungus Cephalotrichum microsporum and their bioactivities
|
Zhu, He |
|
2019 |
83 |
C |
p. 129-134 |
artikel |
38 |
Rhamnocitrin isolated from Prunus padus var. seoulensis: A potent and selective reversible inhibitor of human monoamine oxidase A
|
Baek, Seung Cheol |
|
2019 |
83 |
C |
p. 317-325 |
artikel |
39 |
SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX
|
Eldehna, Wagdy M. |
|
2019 |
83 |
C |
p. 549-558 |
artikel |
40 |
4-Substituted benzenesulfonamides featuring cyclic imides moieties exhibit potent and isoform-selective carbonic anhydrase II/IX inhibition
|
Abdel-Aziz, Alaa A.-M. |
|
2019 |
83 |
C |
p. 198-204 |
artikel |
41 |
Syntheses, in vitro urease inhibitory activities of urea and thiourea derivatives of tryptamine, their molecular docking and cytotoxic studies
|
Kanwal, |
|
2019 |
83 |
C |
p. 595-610 |
artikel |
42 |
Synthesis and anti-proliferative activity of some new quinoline based 4,5-dihydropyrazoles and their thiazole hybrids as EGFR inhibitors
|
George, Riham F. |
|
2019 |
83 |
C |
p. 186-197 |
artikel |
43 |
Synthesis, and anti-proliferative, Pim-1 kinase inhibitors and molecular docking of thiophenes derived from estrone
|
Mohareb, Rafat M. |
|
2019 |
83 |
C |
p. 402-413 |
artikel |
44 |
Synthesis and biological evaluation of 1-benzyl-N-(2-(phenylamino)pyridin-3-yl)-1H-1,2,3-triazole-4-carboxamides as antimitotic agents
|
Prasad, Budaganaboyina |
|
2019 |
83 |
C |
p. 535-548 |
artikel |
45 |
Synthesis and biological evaluation of new N-benzylpyridinium-based benzoheterocycles as potential anti-Alzheimer’s agents
|
Salehi, Naeimeh |
|
2019 |
83 |
C |
p. 559-568 |
artikel |
46 |
Synthesis and biological evaluation of new quinoline derivatives as antileishmanial and antitrypanosomal agents
|
Chanquia, Santiago N. |
|
2019 |
83 |
C |
p. 526-534 |
artikel |
47 |
Synthesis and biological evaluation of new 2,4,6-trisubstituted pyrimidines and their N-alkyl derivatives
|
Kahriman, Nuran |
|
2019 |
83 |
C |
p. 580-594 |
artikel |
48 |
Synthesis and biological evaluation of N-glucosyl indole derivatives as sodium-dependent glucose co-transporter 2 inhibitors
|
Chu, Kuang-Feng |
|
2019 |
83 |
C |
p. 520-525 |
artikel |
49 |
Synthesis and biological evaluation of pyrano[4,3-b][1]benzopyranone derivatives as monoamine oxidase and cholinesterase inhibitors
|
Takao, Koichi |
|
2019 |
83 |
C |
p. 432-437 |
artikel |
50 |
Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates
|
Küçükbay, Hasan |
|
2019 |
83 |
C |
p. 414-423 |
artikel |
51 |
Synthesis and DNA binding profile of monomeric, dimeric, and trimeric derivatives of crystal violet
|
Nuñez, Omar |
|
2019 |
83 |
C |
p. 297-302 |
artikel |
52 |
Synthesis and 2D-QSAR study of dispiropyrrolodinyl-oxindole based alkaloids as cholinesterase inhibitors
|
Srour, Aladdin M. |
|
2019 |
83 |
C |
p. 226-234 |
artikel |
53 |
Synthesis and evaluation of an AZD2461 [18F]PET probe in non-human primates reveals the PARP-1 inhibitor to be non-blood-brain barrier penetrant
|
Reilly, Sean W. |
|
2019 |
83 |
C |
p. 242-249 |
artikel |
54 |
Synthesis and evaluation of new 4-oxoquinazolin-3(4H)-yl)benzoic acid and benzamide derivatives as potent antibacterial agents effective against multidrug resistant Staphylococcus aureus
|
Gatadi, Srikanth |
|
2019 |
83 |
C |
p. 569-579 |
artikel |
55 |
Synthesis, characterization, crystal structure of the coordination polymer Zn(II) with thiosemicarbazone of glyoxalic acid and their inhibitory properties against some metabolic enzymes
|
Huseynova, Mansura |
|
2019 |
83 |
C |
p. 55-62 |
artikel |
56 |
Synthesis, in vitro urease inhibition and molecular docking studies of some novel quinazolin-4(3H)-one derivatives containing triazole, thiadiazole and thiosemicarbazide functionalities
|
Menteşe, Emre |
|
2019 |
83 |
C |
p. 289-296 |
artikel |
57 |
Synthesis of N-benzyl substituted 1,4-imino-l-lyxitols with a basic functional group as selective inhibitors of Golgi α-mannosidase IIb
|
Klunda, Tomáš |
|
2019 |
83 |
C |
p. 424-431 |
artikel |
58 |
Synthesis of new pyrazoles and pyrozolo [3,4-b] pyridines as anti-inflammatory agents by inhibition of COX-2 enzyme
|
Mohamed, Lamia W. |
|
2019 |
83 |
C |
p. 47-54 |
artikel |
59 |
Synthesis of novel N-(1,3-thiazol-2-yl)benzamide clubbed oxadiazole scaffolds: Urease inhibition, Lipinski rule and molecular docking analyses
|
Athar Abbasi, Muhammad |
|
2019 |
83 |
C |
p. 63-75 |
artikel |
60 |
Synthesis of 1,2,4-triazole-5-on derivatives and determination of carbonic anhydrase II isoenzyme inhibition effects
|
Akin, Safak |
|
2019 |
83 |
C |
p. 170-179 |
artikel |
61 |
Trichosanhemiketal A and B: Two 13,14-seco-13,14-epoxyporiferastanes from the root of Trichosanthes kirilowii Maxim.
|
Ha, Manh Tuan |
|
2019 |
83 |
C |
p. 105-110 |
artikel |
62 |
Understanding the cytotoxic effects of new isovanillin derivatives through phospholipid Langmuir monolayers
|
de Carvalho, Ana C. |
|
2019 |
83 |
C |
p. 205-213 |
artikel |