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76 results found

no	title	author	magazine	year	volume	issue	page(s)	type
1	An eco-friendly catalytic system for multicomponent, one-pot synthesis of novel spiro-chromeno indoline-triones and their anti-prostate cancer potentials evaluated via alkaline phosphatase inhibition mechanism	Kumar, M. Rajesh		2018	81	C	p. 44-54	article
2	Aryl fluorosulfate analogues as potent antimicrobial agents: SAR, cytotoxicity and docking studies	Ravindar, Lekkala		2018	81	C	p. 107-118	article
3	A simple boronic acid-based fluorescent probe for selective detection of hydrogen peroxide in solutions and living cells	Han, Jialing		2018	81	C	p. 362-366	article
4	Benzylidine indane-1,3-diones: As novel urease inhibitors; synthesis, in vitro, and in silico studies	Bano, Bilquees		2018	81	C	p. 658-671	article
5	Bioactive compounds from sclerotia extract of Poria cocos that control adipocyte and osteoblast differentiation	Lee, Seulah		2018	81	C	p. 27-34	article
6	Bioactive seco-abietane rearranged diterpenoids from the aerial parts of Salvia prionitis	Li, Lingnan		2018	81	C	p. 454-460	article
7	Characterization of a α-l-rhamnosidase from Bacteroides thetaiotaomicron with high catalytic efficiency of epimedin C	Wu, Tao		2018	81	C	p. 461-467	article
8	Chemically induced degradation of CK2 by proteolysis targeting chimeras based on a ubiquitin–proteasome pathway	Chen, Hong		2018	81	C	p. 536-544	article
9	Conjugation of antifungal benzoic acid derivatives as a path for detoxification in Penicillium brasilianum, an endophyte from Melia azedarach	Fill, Taícia Pacheco		2018	81	C	p. 367-372	article
10	Coumarin-dithiocarbamate hybrids as novel multitarget AChE and MAO-B inhibitors against Alzheimer’s disease: Design, synthesis and biological evaluation	He, Qi		2018	81	C	p. 512-528	article
11	Cytotoxic ent-Abietane-type diterpenoids from the roots of Euphorbia ebracteolata	Han, Chunhui		2018	81	C	p. 93-97	article
12	Cytotoxic withanolides from the aerial parts of Tubocapsicum anomalum	Wang, Si-Bei		2018	81	C	p. 396-404	article
13	Design and synthesis of structurally defined heparan sulfate (HS)-FK506 conjugates as an exogenous approach to investigate biological functions of nucleus HS	Li, MaoLin		2018	81	C	p. 203-210	article
14	Design, synthesis and biological evaluation N 2-(2-alkyoxy-6-aliphatic aminopyridin-3-yl)-2,4-diaminepyrimidine derivatives bearing acylamino or DBTD ‘head’ as potential ALK inhibitors	Xing, Lingyun		2018	81	C	p. 689-699	article
15	Design, synthesis and evaluation of new classes of nonquaternary reactivators for acetylcholinesterase inhibited by organophosphates	Wei, Zhao		2018	81	C	p. 681-688	article
16	Design, synthesis, crystal structures and anticancer activity of 4-substituted quinolines to target PDK1	Vennila, K.N.		2018	81	C	p. 184-190	article
17	Development of new HO-1 inhibitors by a thorough scaffold-hopping analysis	Floresta, Giuseppe		2018	81	C	p. 334-339	article
18	4,5-Diazafluorene N-glycopyranosyl hydrazones as scaffolds for potential bioactive metallo-organic compounds: Synthesis, structural study and cytotoxic activity	Jäger, Sebastian		2018	81	C	p. 405-413	article
19	Dihydroactinidiolide, a natural product against Aβ25-35 induced toxicity in Neuro2a cells: Synthesis, in silico and in vitro studies	Das, Mamali		2018	81	C	p. 340-349	article
20	Discovery of novel cathepsin inhibitors with potent anti-metastatic effects in breast cancer cells	Yuan, Lei		2018	81	C	p. 672-680	article
21	Discovery of Wogonin-based PROTACs against CDK9 and capable of achieving antitumor activity	Bian, Jinlei		2018	81	C	p. 373-381	article
22	DNA-binding, enzyme inhibition, and photochemical properties of chalcone-containing metallophthalocyanine compounds	Özen, Furkan		2018	81	C	p. 71-78	article
23	Editorial Board			2018	81	C	p. i	article
24	Flurbiprofen derivatives as novel α-amylase inhibitors: Biology-oriented drug synthesis (BIODS), in vitro, and in silico evaluation	Khan, Momin		2018	81	C	p. 157-167	article
25	Ginkgolic acid as a dual-targeting inhibitor for protein tyrosine phosphatases relevant to insulin resistance	Yoon, Sun-Young		2018	81	C	p. 264-269	article
26	α-Glucosidase inhibitory effects of polyphenols from Geranium asphodeloides: Inhibition kinetics and mechanistic insights through in vitro and in silico studies	Renda, Gülin		2018	81	C	p. 545-552	article
27	Helix-loop-helix peptide foldamers and their use in the construction of hydrolase mimetics	Drewniak, Magda		2018	81	C	p. 356-361	article
28	Highly functionalized 2-amino-4H-pyrans as potent cholinesterase inhibitors	Kumar, Raju Suresh		2018	81	C	p. 134-143	article
29	Identification and characterization of a highly S-enantioselective halohydrin dehalogenase from Tsukamurella sp. 1534 for kinetic resolution of halohydrins	Wan, Nanwei		2018	81	C	p. 529-535	article
30	Identification of 5-benzylidene-2-phenylthiazolones as potent PRMT5 inhibitors by virtual screening, structural optimization and biological evaluations	Zhu, Kongkai		2018	81	C	p. 289-298	article
31	Identification of human, rat and mouse hydrolyzing enzymes bioconverting amino acid ester prodrug of ketoprofen	Huttunen, K.M.		2018	81	C	p. 494-503	article
32	Identification of new pyrrolo[2,3-d]pyrimidines as potent VEGFR-2 tyrosine kinase inhibitors: Design, synthesis, biological evaluation and molecular modeling	Adel, Mai		2018	81	C	p. 612-629	article
33	Identification of novel and selective non-peptide inhibitors targeting the polo-box domain of polo-like kinase 1	Chen, Yanhong		2018	81	C	p. 278-288	article
34	Inhibitory properties of aromatic thiosemicarbazones on mushroom tyrosinase: Synthesis, kinetic studies, molecular docking and effectiveness in melanogenesis inhibition	Hałdys, K.		2018	81	C	p. 577-586	article
35	Issue TOC			2018	81	C	p. ii-xxii	article
36	Modulation of the mobility of a key region in human galactokinase: Impacts on catalysis and stability	McAuley, Margaret		2018	81	C	p. 649-657	article
37	Multi-targeted dihydrazones as potent biotherapeutics	Li, Chen		2018	81	C	p. 389-395	article
38	New azafluorenones with cytotoxic and carbonic anhydrase inhibitory properties: 2-Aryl-4-(4-hydroxyphenyl)-5H-indeno[1,2-b]pyridin-5-ones	Tugrak, Mehtap		2018	81	C	p. 433-439	article
39	New bio-sensitive and biologically active single crystal of pyrimidine scaffold ligand and its gold and platinum complexes: DFT, antimicrobial, antioxidant, DNA interaction, molecular docking with DNA/BSA and anticancer studies	Sankarganesh, Murugesan		2018	81	C	p. 144-156	article
40	New indole based hybrid oxadiazole scaffolds with N-substituted acetamides: As potent anti-diabetic agents	Nazir, Majid		2018	81	C	p. 253-263	article
41	Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX	Mikuš, Peter		2018	81	C	p. 241-252	article
42	Novel thymol bearing oxypropanolamine derivatives as potent some metabolic enzyme inhibitors – Their antidiabetic, anticholinergic and antibacterial potentials	Zengin, Mustafa		2018	81	C	p. 119-126	article
43	Oxadiazolone derivatives, new promising multi-target inhibitors against M. tuberculosis	Nguyen, Phuong Chi		2018	81	C	p. 414-424	article
44	Pharmacophore mapping, molecular docking, chemical synthesis of some novel pyrrolyl benzamide derivatives and evaluation of their inhibitory activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis	Joshi, Shrinivas D.		2018	81	C	p. 440-453	article
45	Piperazine: An excellent catalyst for the synthesis of 2-amino-3-cyano-4H-pyrans derivatives in aqueous medium	Yousefi, Maryam Rastgoo		2018	81	C	p. 326-333	article
46	Polyamine derivatives from the bee pollen of Quercus mongolica with tyrosinase inhibitory activity	Kim, Seon Beom		2018	81	C	p. 127-133	article
47	Rational design and synthesis of new tetralin-sulfonamide derivatives as potent anti-diabetics and DPP-4 inhibitors: 2D & 3D QSAR, in vivo radiolabeling and bio distribution studies	Abd El-Karim, Somaia S.		2018	81	C	p. 481-493	article
48	Searching for improved mimetic peptides inhibitors preventing conformational transition of amyloid-β42 monomer	Gera, János		2018	81	C	p. 211-221	article
49	Six kanshone C-derived sesquiterpenoid hybrids nardochalaristolones A–D, nardoflavaristolone A and dinardokanshone F from Nardostachys jatamansi DC.	Deng, Xu		2018	81	C	p. 35-43	article
50	Stereoisomeric guaiacylglycerol-β-coniferyl aldehyde ether induces distinctive apoptosis by downregulation of MEK/ERK pathway in hepatocellular carcinoma cells	Yao, Guo-Dong		2018	81	C	p. 382-388	article
51	Synthesis and biological evaluation of (3′-amino-[1,1′-biphenyl]-4-yl) sulfamic acid derivatives as novel HPTPβ inhibitors	Zhang, Wenjuan		2018	81	C	p. 270-277	article
52	Synthesis and biological evaluation of N-aryl-2-phenyl-hydrazinecarbothioamides: Experimental and theoretical analysis on tyrosinase inhibition and interaction with HSA	Sousa-Pereira, Danilo		2018	81	C	p. 79-87	article
53	Synthesis and biological screening of new thiazolo[4,5-d]pyrimidine and dithiazolo[3,2-a:5′,4′-e]pyrimidinone derivatives as antimicrobial, antiquorum-sensing and antitumor agents	Abd Elhameed, Alaa A.		2018	81	C	p. 299-310	article
54	Synthesis and in vitro antitumor evaluation of some new thiophenes and thieno[2,3-d]pyrimidine derivatives	Fouad, Mahasen M.		2018	81	C	p. 587-598	article
55	Synthesis, antimicrobial activity and molecular modeling study of 3-(5-amino-(2H)-1,2,4-triazol-3-yl]-naphthyridinones as potential DNA-gyrase inhibitors	Mohamed, Noha G.		2018	81	C	p. 599-611	article
56	Synthesis, antiproliferative activity and molecular docking of thiocolchicine urethanes	Majcher, Urszula		2018	81	C	p. 553-566	article
57	Synthesis, biological activity and structure activity relationship studies of novel conazole analogues via conventional, microwave and ultrasound mediated techniques	Mermer, Arif		2018	81	C	p. 55-70	article
58	Synthesis, biological evaluation and docking study of N-(2-(3,4,5-trimethoxybenzyl)benzoxazole-5-yl) benzamide derivatives as selective COX-2 inhibitor and anti-inflammatory agents	Kaur, Avneet		2018	81	C	p. 191-202	article
59	Synthesis of different thio-scaffolds bearing sulfonamide with subnanomolar carbonic anhydrase II and IX inhibitory properties and X-ray investigations for their inhibitory mechanism	Angeli, Andrea		2018	81	C	p. 642-648	article
60	Synthesis of 1H-1,2,3-triazole derivatives as new α-glucosidase inhibitors and their molecular docking studies	Avula, Satya Kumar		2018	81	C	p. 98-106	article
61	Synthesis of matrinic amide derivatives containing 1,3,4-thiadiazole scaffold as insecticidal/acaricidal agents	Lv, Min		2018	81	C	p. 88-92	article
62	Synthesis of new 3-phenylquinazolin-4(3H)-one derivatives as potent antibacterial agents effective against methicillin- and vancomycin-resistant Staphylococcus aureus (MRSA and VRSA)	Gatadi, Srikanth		2018	81	C	p. 175-183	article
63	Synthesis of novel 1,2-bis-quinolinyl-1,4-naphthoquinones: ERK2 inhibition, cytotoxicity and molecular docking studies	Aly, Ashraf A.		2018	81	C	p. 700-712	article
64	Synthesis of novel dipeptide sulfonamide conjugates with effective carbonic anhydrase I, II, IX, and XII inhibitory properties	Buğday, Nesrin		2018	81	C	p. 311-318	article
65	The azatryptophan-based fluorescent platform for in vitro rapid screening of inhibitors disrupting IKKβ-NEMO interaction	Chao, Wei-Chih		2018	81	C	p. 504-511	article
66	Thiazolo[3,2-a]pyrimidin-5-one derivatives as a novel class of 11β-hydroxysteroid dehydrogenase inhibitors	Studzińska, Renata		2018	81	C	p. 21-26	article
67	1,2,4-Triazole-based benzothiazole/benzoxazole derivatives: Design, synthesis, p38α MAP kinase inhibition, anti-inflammatory activity and molecular docking studies	Tariq, Sana		2018	81	C	p. 630-641	article
68	1,2,3-triazole tethered Indole-3-glyoxamide derivatives as multiple inhibitors of 5-LOX, COX-2 & tubulin: Their anti-proliferative & anti-inflammatory activity	Naaz, Fatima		2018	81	C	p. 1-20	article
69	Trichocarotins A–H and trichocadinin A, nine sesquiterpenes from the marine-alga-epiphytic fungus Trichoderma virens	Shi, Zhen-Zhen		2018	81	C	p. 319-325	article
70	Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer	Eldehna, Wagdy M.		2018	81	C	p. 425-432	article
71	Tyrosinase inhibition by some flavonoids: Inhibitory activity, mechanism by in vitro and in silico studies	Şöhretoğlu, Didem		2018	81	C	p. 168-174	article
72	Ugi multicomponent-reaction: Syntheses of cytotoxic dehydroabietylamine derivatives	Wiemann, Jana		2018	81	C	p. 567-576	article
73	Unexpected effect of cyclodepsipeptides bearing a sulfonylhydrazide moiety towards histone deacetylase activity	Létévé, Mathieu		2018	81	C	p. 222-233	article
74	Unusual ent-atisane type diterpenoids with 2-oxopropyl skeleton from the roots of Euphorbia ebracteolata and their antiviral activity against human rhinovirus 3 and enterovirus 71	Wang, Bo		2018	81	C	p. 234-240	article
75	Unveiling novel 2-cyclopropyl-3-ethynyl-4-(4-fluorophenyl)quinolines as GPCR ligands via PI3-kinase/PAR-1 antagonism and platelet aggregation valuations; development of a new class of anticancer drugs with thrombolytic effects	Thangarasu, P.		2018	81	C	p. 468-480	article
76	Xylarianins A-D from the endophytic fungus Xylaria sp. SYPF 8246 as natural inhibitors of human carboxylesterase 2	Zhang, Juan		2018	81	C	p. 350-355	article

76 results found

Koninklijke Bibliotheek - National Library of the Netherlands