nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Albumin coated copper-cysteine nanozyme for reducing oxidative stress induced during sperm cryopreservation
|
Dashtestani, Fariba |
|
|
80 |
C |
p. 621-630 |
artikel |
2 |
11a-N-tosyl-5-carbapterocarpans: Synthesis, antineoplastic evaluation and in silico prediction of ADMETox properties
|
Mendes, Joseane A. |
|
|
80 |
C |
p. 585-590 |
artikel |
3 |
3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
|
Romagnoli, Romeo |
|
|
80 |
C |
p. 361-374 |
artikel |
4 |
Benzimidazole scaffold based hybrid molecules for various inflammatory targets: Synthesis and evaluation
|
Kaur, Gaganpreet |
|
|
80 |
C |
p. 24-35 |
artikel |
5 |
Bioactive secondary metabolites from the marine-associated fungus Aspergillus terreus
|
Liu, Mengting |
|
|
80 |
C |
p. 525-530 |
artikel |
6 |
Biological properties and structural study of new aminoalkyl derivatives of benzimidazole and benzotriazole, dual inhibitors of CK2 and PIM1 kinases
|
Chojnacki, K. |
|
|
80 |
C |
p. 266-275 |
artikel |
7 |
Characterization of inhibitory constituents of NO production from Catalpa ovata using LC-MS coupled with a cell-based assay
|
Park, Sangmin |
|
|
80 |
C |
p. 57-63 |
artikel |
8 |
Cytoprotective and antioxidant properties of organic selenides for the myelin-forming cells, oligodendrocytes
|
Shaaban, Saad |
|
|
80 |
C |
p. 43-56 |
artikel |
9 |
Cytotoxic macrocyclic diterpenoids from Jatropha multifida
|
Zhang, Jun-Sheng |
|
|
80 |
C |
p. 511-518 |
artikel |
10 |
Design and Amberlyst-15 mediated synthesis of novel thienyl-pyrazole carboxamides that potently inhibit Phospholipase A2 by binding to an allosteric site on the enzyme
|
Kumar, Achutha Dileep |
|
|
80 |
C |
p. 444-452 |
artikel |
11 |
Design and synthesis of donepezil analogues as dual AChE and BACE-1 inhibitors
|
Gabr, Moustafa T. |
|
|
80 |
C |
p. 245-252 |
artikel |
12 |
Design and synthesis of gallocyanine inhibitors of DKK1/LRP6 interactions for treatment of Alzheimer’s disease
|
Thysiadis, Savvas |
|
|
80 |
C |
p. 230-244 |
artikel |
13 |
Design and synthesis of novel imidazo[4,5-b]pyridine based compounds as potent anticancer agents with CDK9 inhibitory activity
|
Ghanem, Nada M. |
|
|
80 |
C |
p. 565-576 |
artikel |
14 |
Design, synthesis and activity of light deactivatable microRNA inhibitor
|
Yan, Hao |
|
|
80 |
C |
p. 492-497 |
artikel |
15 |
Design, synthesis and anticancer evaluation of 1H-pyrazolo[3,4-d]pyrimidine derivatives as potent EGFRWT and EGFRT790M inhibitors and apoptosis inducers
|
Gaber, Ahmed A. |
|
|
80 |
C |
p. 375-395 |
artikel |
16 |
Design, synthesis and anti leukemia cells proliferation activities of pyrimidylaminoquinoline derivatives as DOT1L inhibitors
|
Zhang, Li |
|
|
80 |
C |
p. 649-654 |
artikel |
17 |
Design, synthesis and antiplasmodial activity of novel imidazole derivatives based on 7-chloro-4-aminoquinoline
|
Kondaparla, Srinivasarao |
|
|
80 |
C |
p. 204-211 |
artikel |
18 |
Design, synthesis and biological evaluation of novel pyrrole derivatives as potential ClpP1P2 inhibitor against Mycobacterium tuberculosis
|
Liu, Pingxian |
|
|
80 |
C |
p. 422-432 |
artikel |
19 |
Design, synthesis and biological evaluation of novel 1,2,3-triazole linked coumarinopyrazole conjugates as potent anticholinesterase, anti-5-lipoxygenase, anti-tyrosinase and anti-cancer agents
|
Chekir, Samia |
|
|
80 |
C |
p. 189-194 |
artikel |
20 |
Design, synthesis and docking study of pyridine and thieno[2,3-b] pyridine derivatives as anticancer PIM-1 kinase inhibitors
|
Abdelaziz, Marwa E. |
|
|
80 |
C |
p. 674-692 |
artikel |
21 |
Design, synthesis and evaluation of some pyrazolo[3,4-d]pyrimidine derivatives bearing thiazolidinone moiety as anti-inflammatory agents
|
Tageldin, Gina N. |
|
|
80 |
C |
p. 164-173 |
artikel |
22 |
Design, synthesis and molecular modeling study of certain 4-Methylbenzenesulfonamides with CDK2 inhibitory activity as anticancer and radio-sensitizing agents
|
Ghorab, Mostafa M. |
|
|
80 |
C |
p. 276-287 |
artikel |
23 |
Design, synthesis, biological activities and DFT calculation of novel 1,2,4-triazole Schiff base derivatives
|
Jin, Ru-Yi |
|
|
80 |
C |
p. 253-260 |
artikel |
24 |
Design, synthesis, docking study, α-glucosidase inhibition, and cytotoxic activities of acridine linked to thioacetamides as novel agents in treatment of type 2 diabetes
|
Mohammadi-Khanaposhtani, Maryam |
|
|
80 |
C |
p. 288-295 |
artikel |
25 |
Design, synthesis, in-vitro thymidine phosphorylase inhibition, in-vivo antiangiogenic and in-silico studies of C-6 substituted dihydropyrimidines
|
Iftikhar, Fatima |
|
|
80 |
C |
p. 99-111 |
artikel |
26 |
Design, synthesis of novel azolyl flavonoids and their protein tyrosine Phosphatase-1B inhibitory activities
|
Zhang, Ling |
|
|
80 |
C |
p. 195-203 |
artikel |
27 |
Design, synthesis of novel isoindoline hybrids as COX-2 inhibitors: Anti-inflammatory, analgesic activities and docking study
|
Labib, Madlen B. |
|
|
80 |
C |
p. 70-80 |
artikel |
28 |
Development of dilipid polymyxins: Investigation on the effect of hydrophobicity through its fatty acyl component
|
Domalaon, Ronald |
|
|
80 |
C |
p. 639-648 |
artikel |
29 |
Dicoumarol derivatives: Green synthesis and molecular modelling studies of their anti-LOX activity
|
Simijonović, Dušica |
|
|
80 |
C |
p. 741-752 |
artikel |
30 |
Discovery of dihydrobenzofuran neolignans from Rubus ideaus L. with enantioselective anti-Aβ 1–42 aggregation activity
|
Zhou, Le |
|
|
80 |
C |
p. 64-69 |
artikel |
31 |
Discovery of polar spirocyclic orally bioavailable urea inhibitors of soluble epoxide hydrolase
|
Lukin, Alexey |
|
|
80 |
C |
p. 655-667 |
artikel |
32 |
Dual EGFR/HER2 inhibitors and apoptosis inducers: New benzo[g]quinazoline derivatives bearing benzenesulfonamide as anticancer and radiosensitizers
|
Ghorab, Mostafa M. |
|
|
80 |
C |
p. 611-620 |
artikel |
33 |
Editorial Board
|
|
|
|
80 |
C |
p. i |
artikel |
34 |
Efficient chemoenzymatic synthesis of (S)-α-amino-4-fluorobenzeneacetic acid using immobilized penicillin amidase
|
Lin, Chao-Ping |
|
|
80 |
C |
p. 174-179 |
artikel |
35 |
Efficient synthesis of the ketone body ester (R)-3-hydroxybutyryl-(R)-3-hydroxybutyrate and its (S,S) enantiomer
|
Budin, Noah |
|
|
80 |
C |
p. 560-564 |
artikel |
36 |
Enhancement in anti-tubercular activity of indole based thiosemicarbazones on complexation with copper(I) and silver(I) halides: Structure elucidation, evaluation and molecular modelling
|
Khan, Ashiq |
|
|
80 |
C |
p. 303-318 |
artikel |
37 |
Imidazopyridine linked triazoles as tubulin inhibitors, effectively triggering apoptosis in lung cancer cell line
|
Sayeed, Ibrahim Bin |
|
|
80 |
C |
p. 714-720 |
artikel |
38 |
Imidazo[2′,1′:2,3]thiazolo[4,5-d]pyridazinone as a new scaffold of DHFR inhibitors: Synthesis, biological evaluation and molecular modeling study
|
Ewida, Menna A. |
|
|
80 |
C |
p. 11-23 |
artikel |
39 |
Improvement of carbonyl reductase activity for the bioproduction of tert-butyl (3R,5S)-6-chloro-3,5-dihydroxyhexanoate
|
Liu, Zhi-Qiang |
|
|
80 |
C |
p. 733-740 |
artikel |
40 |
Investigation of salicylanilide and 4-chlorophenol-based N-monosubstituted carbamates as potential inhibitors of acetyl- and butyrylcholinesterase
|
Krátký, Martin |
|
|
80 |
C |
p. 668-673 |
artikel |
41 |
Issue TOC
|
|
|
|
80 |
C |
p. ii-xxiv |
artikel |
42 |
Lambertellin from Pycnoporus sanguineus MUCL 51321 and its anti-inflammatory effect via modulation of MAPK and NF-κB signaling pathways
|
Jouda, Jean-Bosco |
|
|
80 |
C |
p. 216-222 |
artikel |
43 |
Lipid reducing activity of novel cholic acid (CA) analogs: Design, synthesis and preliminary mechanism study
|
Luo, Guoshun |
|
|
80 |
C |
p. 396-407 |
artikel |
44 |
Multi-targetable chalcone analogs to treat deadly Alzheimer’s disease: Current view and upcoming advice
|
Zhang, Xu |
|
|
80 |
C |
p. 86-93 |
artikel |
45 |
Natural constituents from Cortex Mori Radicis as new pancreatic lipase inhibitors
|
Hou, Xu-Dong |
|
|
80 |
C |
p. 577-584 |
artikel |
46 |
New C-2 diastereomers of flavanone glycosides conjugated with 3-hydroxy-3-methylglutaric acid from the pericarp of Citrus grandis (L.) Osbeck
|
Ma, Shuang-Gang |
|
|
80 |
C |
p. 519-524 |
artikel |
47 |
New monoterpenoid by biotransformation of thymoquinone using Aspergillus niger
|
Mohammad, Mohammad Yasin |
|
|
80 |
C |
p. 212-215 |
artikel |
48 |
Nitric oxide inhibitory constituents from Siegesbeckia pubescens
|
Jang, Hari |
|
|
80 |
C |
p. 81-85 |
artikel |
49 |
Novel benzotriazole N-acylarylhydrazone hybrids: Design, synthesis, anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis and FAK inhibition
|
Kassab, Asmaa E. |
|
|
80 |
C |
p. 531-544 |
artikel |
50 |
Novel pyrrol-2(3H)-ones and pyridazin-3(2H)-ones carrying quinoline scaffold as anti-proliferative tubulin polymerization inhibitors
|
Abdelbaset, Mahmoud S. |
|
|
80 |
C |
p. 151-163 |
artikel |
51 |
Promiscuous enzyme-catalyzed cascade reaction: Synthesis of xanthone derivatives
|
Fu, Yajie |
|
|
80 |
C |
p. 555-559 |
artikel |
52 |
QM/MM study of the reaction mechanism of Cl-cis,cis-muconate with muconate lactonizing enzyme
|
Zhu, Ledong |
|
|
80 |
C |
p. 453-460 |
artikel |
53 |
Sam domain-based stapled peptides: Structural analysis and interaction studies with the Sam domains from the EphA2 receptor and the lipid phosphatase Ship2
|
Mercurio, Flavia Anna |
|
|
80 |
C |
p. 602-610 |
artikel |
54 |
2-S-cysteinylhydroquinone is an intermediate for the firefly luciferin biosynthesis that occurs in the pupal stage of the Japanese firefly, Luciola lateralis
|
Kanie, Shusei |
|
|
80 |
C |
p. 223-229 |
artikel |
55 |
Structural comparison of Mtb-DHFR and h-DHFR for design, synthesis and evaluation of selective non-pteridine analogues as antitubercular agents
|
Sharma, Kalicharan |
|
|
80 |
C |
p. 319-333 |
artikel |
56 |
Structure-based design of free fatty acid receptor 1 agonists bearing non-biphenyl scaffold
|
Li, Zheng |
|
|
80 |
C |
p. 296-302 |
artikel |
57 |
Structure-based design of some isonicotinic acid hydrazide analogues as potential antitubercular agents
|
Atta, Amal |
|
|
80 |
C |
p. 721-732 |
artikel |
58 |
Studies on the lipid-regulating mechanism of alisol-based compounds on lipoprotein lipase
|
Xu, Fei |
|
|
80 |
C |
p. 347-360 |
artikel |
59 |
Syntheses, antiviral activities and induced resistance mechanisms of novel quinazoline derivatives containing a dithioacetal moiety
|
Xie, Dandan |
|
|
80 |
C |
p. 433-443 |
artikel |
60 |
Synthesis, α-amylase inhibitory potential and molecular docking study of indole derivatives
|
Taha, Muhammad |
|
|
80 |
C |
p. 36-42 |
artikel |
61 |
Synthesis and biological evaluation of benzo[b]furo[3,4-e][1,4]diazepin-1-one derivatives as anti-cancer agents
|
Malayeri, Sina Omid |
|
|
80 |
C |
p. 631-638 |
artikel |
62 |
Synthesis and biological evaluation of some N-(3-(1H-tetrazol-5-yl) phenyl)acetamide derivatives as novel non-carboxylic PTP1B inhibitors designed through bioisosteric modulation
|
Maheshwari, Neelesh |
|
|
80 |
C |
p. 145-150 |
artikel |
63 |
Synthesis and cholinesterase inhibitory activity of new 2-benzofuran carboxamide-benzylpyridinum salts
|
Abedinifar, Fahimeh |
|
|
80 |
C |
p. 180-188 |
artikel |
64 |
Synthesis and DNase I inhibitory properties of some 5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidines
|
Ts. Mavrova, Anelia |
|
|
80 |
C |
p. 693-705 |
artikel |
65 |
Synthesis and dopaminergic activity of a series of new 1-aryl tetrahydroisoquinolines and 2-substituted 1-aryl-3-tetrahydrobenzazepines
|
Lucena-Serrano, Cristina |
|
|
80 |
C |
p. 480-491 |
artikel |
66 |
Synthesis and molecular docking study of some novel 2,3-disubstituted quinazolin-4(3H)-one derivatives as potent inhibitors of urease
|
Akyüz, Gülay |
|
|
80 |
C |
p. 121-128 |
artikel |
67 |
Synthesis, biological activities, and molecular docking studies of 2-mercaptobenzimidazole based derivatives
|
Ali, Mumtaz |
|
|
80 |
C |
p. 472-479 |
artikel |
68 |
Synthesis, biological evaluation and docking study of 1,3,4-thiadiazole-thiazolidinone hybrids as anti-inflammatory agents with dual inhibition of COX-2 and 15-LOX
|
Omar, Yasser M. |
|
|
80 |
C |
p. 461-471 |
artikel |
69 |
Synthesis, characterization, monoamine oxidase inhibition, molecular docking and dynamic simulations of novel 2,1-benzothiazine-2,2-dioxide derivatives
|
Ahmad, Shakeel |
|
|
80 |
C |
p. 498-510 |
artikel |
70 |
Synthesis, in vitro and in silico evaluation of diaryl heptanones as potential 5LOX enzyme inhibitors
|
Meka, Bharani |
|
|
80 |
C |
p. 408-421 |
artikel |
71 |
Synthesis, in vitro urease inhibitory activity, and molecular docking studies of thiourea and urea derivatives
|
Bano, Bilquees |
|
|
80 |
C |
p. 129-144 |
artikel |
72 |
Synthesis of Bis-indolylmethane sulfonohydrazides derivatives as potent α-Glucosidase inhibitors
|
Gollapalli, Mohammed |
|
|
80 |
C |
p. 112-120 |
artikel |
73 |
Synthesis of C-2 and C-3 substituted quinolines and their evaluation as anti-HIV-1 agents
|
Shah, Purvi |
|
|
80 |
C |
p. 591-601 |
artikel |
74 |
Synthesis of novel isoindoline-1,3-dione-based oximes and benzenesulfonamide hydrazones as selective inhibitors of the tumor-associated carbonic anhydrase IX
|
Abdel-Aziz, Alaa A.-M. |
|
|
80 |
C |
p. 706-713 |
artikel |
75 |
Synthesis of spherical Fe2O3 nanoparticles from the thermal decomposition of iron (III) nano-structure complex: DFT studies and evaluation of the biological activity
|
Zare, Nahid |
|
|
80 |
C |
p. 334-346 |
artikel |
76 |
Targeting oncogenic transcriptional corepressor Nac1 POZ domain with conformationally constrained peptides by cyclization and stapling
|
Wu, Tao |
|
|
80 |
C |
p. 1-10 |
artikel |
77 |
Tetrahydroindolocarbazoles (THICZs) as new class of urokinase (uPA) inhibitors: Synthesis, anticancer evaluation, DNA-damage determination, and molecular modelling study
|
El-Sharief, Marwa A.M.Sh. |
|
|
80 |
C |
p. 545-554 |
artikel |
78 |
The first activation studies of the η-carbonic anhydrase from the malaria parasite Plasmodium falciparum with amines and amino acids
|
Angeli, Andrea |
|
|
80 |
C |
p. 94-98 |
artikel |
79 |
The zinc – but not cadmium – containing ζ-carbonic from the diatom Thalassiosira weissflogii is potently activated by amines and amino acids
|
Angeli, Andrea |
|
|
80 |
C |
p. 261-265 |
artikel |