| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Alkynyl and β-ketophosphonates: Selective and potent butyrylcholinesterase inhibitors
|
Cavallaro, Valeria
|
|
|
77 |
C |
p. 420-428
|
artikel
|
| 2 |
A new entry into the portfolio of α-glucosidase inhibitors as potent therapeutics for type 2 diabetes: Design, bioevaluation and one-pot multi-component synthesis of diamine-bridged coumarinyl oxadiazole conjugates
|
Kazmi, Madiha
|
|
|
77 |
C |
p. 190-202
|
artikel
|
| 3 |
A simple, cheap but reliable method for evaluation of zinc chelating properties
|
Catapano, Maria Carmen
|
|
|
77 |
C |
p. 287-292
|
artikel
|
| 4 |
Asymmetric synthesis, molecular modeling and biological evaluation of 5-methyl-3-aryloxazolidine-2,4-dione enantiomers as monoamine oxidase (MAO) inhibitors
|
Erol Gunal, Sule
|
|
|
77 |
C |
p. 608-618
|
artikel
|
| 5 |
Benzopyrone represents a privilege scaffold to identify novel adenosine A1/A2A receptor antagonists
|
van der Walt, Mietha M.
|
|
|
77 |
C |
p. 136-143
|
artikel
|
| 6 |
Bioactive triterpenoids from twigs of Betula schmidtii
|
Park, Kyoung Jin
|
|
|
77 |
C |
p. 527-533
|
artikel
|
| 7 |
4-Bromophenylhydrazinyl benzenesulfonylphenylureas as indoleamine 2,3-dioxygenase inhibitors with in vivo target inhibition and anti-tumor efficacy
|
Lin, Shu-Yu
|
|
|
77 |
C |
p. 600-607
|
artikel
|
| 8 |
Carbazole alkaloids with antiangiogenic activities from Clausena sanki
|
Wei, Rongrui
|
|
|
77 |
C |
p. 387-392
|
artikel
|
| 9 |
Characterization and structure-activity relationship studies of flavonoids as inhibitors against human carboxylesterase 2
|
Weng, Zi-Miao
|
|
|
77 |
C |
p. 320-329
|
artikel
|
| 10 |
Cholinesterase inhibitory alkaloids from the rhizomes of Coptis chinensis
|
Cao, Thao Quyen
|
|
|
77 |
C |
p. 625-632
|
artikel
|
| 11 |
8-Chrysoeriol, as a potential BCL-2 inhibitor triggers apoptosis of SW1990 pancreatic cancer cells
|
Zhang, Yiwen
|
|
|
77 |
C |
p. 478-484
|
artikel
|
| 12 |
Cunninghamella blakesleeana-mediated biotransformation of a contraceptive drug, desogestrel, and anti-MDR-Staphylococcus aureus activity of its metabolites
|
Atia-tul-Wahab,
|
|
|
77 |
C |
p. 152-158
|
artikel
|
| 13 |
Design and synthesis of novel coumarin-pyridinium hybrids: In vitro cholinesterase inhibitory activity
|
Vafadarnejad, Fahimeh
|
|
|
77 |
C |
p. 311-319
|
artikel
|
| 14 |
Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors
|
Lolak, Nabih
|
|
|
77 |
C |
p. 542-547
|
artikel
|
| 15 |
Design, synthesis and anticancer studies of novel aminobenzazolyl pyrimidines as tyrosine kinase inhibitors
|
Chikhale, Rupesh
|
|
|
77 |
C |
p. 84-100
|
artikel
|
| 16 |
Design, synthesis and biological evaluation of bitopic arylpiperazine-hexahydro-pyrazinoquinolines as preferential dopamine D3 receptor ligands
|
Zhou, Benhua
|
|
|
77 |
C |
p. 125-135
|
artikel
|
| 17 |
Design, synthesis and in vitro α-glucosidase inhibition of novel dihydropyrano[3,2-c]quinoline derivatives as potential anti-diabetic agents
|
Nikookar, Hamideh
|
|
|
77 |
C |
p. 280-286
|
artikel
|
| 18 |
Design, synthesis, characterization, antimicrobial evaluation and molecular modeling studies of some dehydroacetic acid-chalcone-1,2,3-triazole hybrids
|
Lal, Kashmiri
|
|
|
77 |
C |
p. 236-244
|
artikel
|
| 19 |
Development of novel synthesized phthalazinone-based PARP-1 inhibitors with apoptosis inducing mechanism in lung cancer
|
Almahli, Hadia
|
|
|
77 |
C |
p. 443-456
|
artikel
|
| 20 |
Development of thermostable amylase enzyme from Bacillus cereus for potential antibiofilm activity
|
Vaikundamoorthy, Ramalingam
|
|
|
77 |
C |
p. 494-506
|
artikel
|
| 21 |
5,6-Dihydropyrimidine-1(2H)-carbothioamides: Synthesis, in vitro GABA-AT screening, anticonvulsant activity and molecular modelling study
|
Sahu, Meeta
|
|
|
77 |
C |
p. 56-67
|
artikel
|
| 22 |
1,3-Diphenylpropanes from Daphne giraldii induced apoptosis in hepatocellular carcinoma cells through nuclear factor kappa-B inhibition
|
Yao, Guo-Dong
|
|
|
77 |
C |
p. 619-624
|
artikel
|
| 23 |
Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors
|
Nocentini, Alessio
|
|
|
77 |
C |
p. 293-299
|
artikel
|
| 24 |
Discovery of thinopyrimidine-triazole conjugates as c-Met targeting and apoptosis inducing agents
|
Wang, Linxiao
|
|
|
77 |
C |
p. 370-380
|
artikel
|
| 25 |
Diterpenoids from the roots of Euphorbia ebracteolata and their anti-tuberculosis effects
|
Yu, Zhenlong
|
|
|
77 |
C |
p. 471-477
|
artikel
|
| 26 |
Editorial Board
|
|
|
|
77 |
C |
p. i
|
artikel
|
| 27 |
Enantiomeric lignans with anti-β-amyloid aggregation activity from the twigs and leaves of Pithecellobium clypearia Benth
|
Wang, Yu-Xi
|
|
|
77 |
C |
p. 579-585
|
artikel
|
| 28 |
Engineering of Talaromyces thermophilus lipase by altering its crevice-like binding site for highly efficient biocatalytic synthesis of chiral intermediate of Pregablin
|
Ding, Xu
|
|
|
77 |
C |
p. 330-338
|
artikel
|
| 29 |
3-(E)-Styryl-2H-chromene derivatives as potent and selective monoamine oxidase B inhibitors
|
Takao, Koichi
|
|
|
77 |
C |
p. 436-442
|
artikel
|
| 30 |
Evaluating hydrophobic galactonoamidines as transition state analogs for enzymatic β-galactoside hydrolysis
|
Pickens, Jessica B.
|
|
|
77 |
C |
p. 144-151
|
artikel
|
| 31 |
Evaluation of α-glucosidase inhibiting potentials with docking calculations of synthesized arylidene-pyrazolones
|
Chaudhry, Faryal
|
|
|
77 |
C |
p. 507-514
|
artikel
|
| 32 |
Exploiting the biological efficacy of benzimidazole based Schiff base complexes with l-Histidine as a co-ligand: Combined molecular docking, DNA interaction, antimicrobial and cytotoxic studies
|
Kumaravel, Ganesan
|
|
|
77 |
C |
p. 269-279
|
artikel
|
| 33 |
Fungal synthesis of chiral phosphonic synthetic platform – Scope and limitations of the method
|
Serafin-Lewańczuk, Monika
|
|
|
77 |
C |
p. 402-410
|
artikel
|
| 34 |
Influence of the d/l configuration of N-acyl-homoserine lactones (AHLs) and analogues on their Lux-R dependent quorum sensing activity
|
Li, Si-Zhe
|
|
|
77 |
C |
p. 215-222
|
artikel
|
| 35 |
In-vitro evaluation of antioxidant, anti-elastase, anti-collagenase, anti-hyaluronidase activities of safranal and determination of its sun protection factor in skin photoaging
|
Madan, Kumud
|
|
|
77 |
C |
p. 159-167
|
artikel
|
| 36 |
Ionic liquid-enabled synthesis, cholinesterase inhibitory activity, and molecular docking study of highly functionalized tetrasubstituted pyrrolidines
|
Kumar, Raju Suresh
|
|
|
77 |
C |
p. 263-268
|
artikel
|
| 37 |
Issue TOC
|
|
|
|
77 |
C |
p. ii-xix
|
artikel
|
| 38 |
Molecular docking simulation, synthesis and 3D pharmacophore studies of novel 2-substituted-5-nitro-benzimidazole derivatives as anticancer agents targeting VEGFR-2 and c-Met
|
Ibrahim, Heba A.
|
|
|
77 |
C |
p. 457-470
|
artikel
|
| 39 |
Neuroprotection by new ligustrazine-cinnamon acid derivatives on CoCl2-induced apoptosis in differentiated PC12 cells
|
Wang, Penglong
|
|
|
77 |
C |
p. 360-369
|
artikel
|
| 40 |
New acrylamide-substituted quinazoline derivatives with enhanced potency for the treatment of EGFR T790M-mutant non-small-cell lung cancers
|
Liu, Zhuo
|
|
|
77 |
C |
p. 593-599
|
artikel
|
| 41 |
New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors
|
Gul, Halise Inci
|
|
|
77 |
C |
p. 411-419
|
artikel
|
| 42 |
NO inhibitors function as potential anti-neuroinflammatory agents for AD from the flowers of Inula japonica
|
Liu, Feng
|
|
|
77 |
C |
p. 168-175
|
artikel
|
| 43 |
Non-acidic 1,3,4-trisubstituted-pyrazole derivatives as lonazolac analogs with promising COX-2 selectivity, anti-inflammatory activity and gastric safety profile
|
Abdellatif, Khaled R.A.
|
|
|
77 |
C |
p. 568-578
|
artikel
|
| 44 |
Novel pyrimidine-pyridine hybrids: Synthesis, cyclooxygenase inhibition, anti-inflammatory activity and ulcerogenic liability
|
Abdelgawad, Mohamed A.
|
|
|
77 |
C |
p. 339-348
|
artikel
|
| 45 |
Novel sulfonamide incorporating piperazine, aminoalcohol and 1,3,5-triazine structural motifs with carbonic anhydrase I, II and IX inhibitory action
|
Havránková, Eva
|
|
|
77 |
C |
p. 25-37
|
artikel
|
| 46 |
Potent ACE inhibitors from 5-hydroxy indanone derivatives
|
Vulupala, Hanmanth Reddy
|
|
|
77 |
C |
p. 660-665
|
artikel
|
| 47 |
Potent dialkyl substrate-product analogue inhibitors and inactivators of α-methylacyl-coenzyme A racemase from Mycobacterium tuberculosis by rational design
|
Pal, Mohan
|
|
|
77 |
C |
p. 640-650
|
artikel
|
| 48 |
Probing the β-pocket of the active site of human liver glycogen phosphorylase with 3-(C-β-d-glucopyranosyl)-5-(4-substituted-phenyl)-1, 2, 4-triazole inhibitors
|
Kyriakis, Efthimios
|
|
|
77 |
C |
p. 485-493
|
artikel
|
| 49 |
Purification and characterization of β-galactosidase from probiotic Pediococcus acidilactici and its use in milk lactose hydrolysis and galactooligosaccharide synthesis
|
Chanalia, Preeti
|
|
|
77 |
C |
p. 176-189
|
artikel
|
| 50 |
Pyridazinone hybrids: Design, synthesis and evaluation as potential anticonvulsant agents
|
Partap, Sangh
|
|
|
77 |
C |
p. 74-83
|
artikel
|
| 51 |
Rupestrines A-D, alkaloids from the aerial parts of Corydalis rupestris
|
Naseri, Maryam
|
|
|
77 |
C |
p. 651-659
|
artikel
|
| 52 |
Silibinin phosphodiester glyco-conjugates: Synthesis, redox behaviour and biological investigations
|
Romanucci, Valeria
|
|
|
77 |
C |
p. 349-359
|
artikel
|
| 53 |
Structure-based optimization of free fatty acid receptor 1 agonists bearing thiazole scaffold
|
Li, Zheng
|
|
|
77 |
C |
p. 429-435
|
artikel
|
| 54 |
Synthesis and biological evaluation of imidazo[2,1-b]thiazole-benzimidazole conjugates as microtubule-targeting agents
|
Baig, Mirza Feroz
|
|
|
77 |
C |
p. 515-526
|
artikel
|
| 55 |
Synthesis and biological evaluation of naphthalimide-polyamine conjugates modified by alkylation as anticancer agents through p53 pathway
|
Dai, Fujun
|
|
|
77 |
C |
p. 16-24
|
artikel
|
| 56 |
Synthesis and biological evaluation of novel N,N′-diaryl cyanoguanidines acting as potent and selective carbonic anhydrase II inhibitors
|
Akocak, Suleyman
|
|
|
77 |
C |
p. 245-251
|
artikel
|
| 57 |
Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy
|
Nocentini, Alessio
|
|
|
77 |
C |
p. 633-639
|
artikel
|
| 58 |
Synthesis and properties of the para-trimethylammonium analogues of green fluorescence protein (GFP) chromophore: The mimic of protonated GFP chromophore
|
Fanjiang, Ming-Wei
|
|
|
77 |
C |
p. 300-310
|
artikel
|
| 59 |
Synthesis and structure-activity relationship study of multi-target triazine derivatives as innovative candidates for treatment of Alzheimer's disease
|
Iraji, Aida
|
|
|
77 |
C |
p. 223-235
|
artikel
|
| 60 |
Synthesis, anticancer assessment on human breast, liver and colon carcinoma cell lines and molecular modeling study using novel pyrazolo[4,3-c]pyridine derivatives
|
Metwally, Nadia Hanafy
|
|
|
77 |
C |
p. 203-214
|
artikel
|
| 61 |
Synthesis, biological evaluation and computational studies of novel iminothiazolidinone benzenesulfonamides as potent carbonic anhydrase II and IX inhibitors
|
Mahmood, Shams-ul
|
|
|
77 |
C |
p. 381-386
|
artikel
|
| 62 |
Synthesis, biological evaluation and molecular modeling of novel thienopyrimidinone and triazolothienopyrimidinone derivatives as dual anti-inflammatory antimicrobial agents
|
Bekhit, Adnan A.
|
|
|
77 |
C |
p. 38-46
|
artikel
|
| 63 |
Synthesis, biological evaluation and molecular modeling studies of phenyl-/benzhydrylpiperazine derivatives as potential MAO inhibitors
|
Kumar, Bhupinder
|
|
|
77 |
C |
p. 252-262
|
artikel
|
| 64 |
Synthesis, α-glucosidase inhibition and molecular docking study of coumarin based derivatives
|
Taha, Muhammad
|
|
|
77 |
C |
p. 586-592
|
artikel
|
| 65 |
Synthesis, molecular modelling studies and ADME prediction of benzothiazole clubbed oxadiazole-Mannich bases, and evaluation of their anti-diabetic activity through in vivo model
|
Bhutani, Rubina
|
|
|
77 |
C |
p. 6-15
|
artikel
|
| 66 |
Synthesis of benzimidazole-linked-1,3,4-oxadiazole carboxamides as GSK-3β inhibitors with in vivo antidepressant activity
|
Tantray, Mushtaq A.
|
|
|
77 |
C |
p. 393-401
|
artikel
|
| 67 |
Synthesis of novel 5-amino-1,3,4-thiadiazole-2-sulfonamide containing acridine sulfonamide/carboxamide compounds and investigation of their inhibition effects on human carbonic anhydrase I, II, IV and VII
|
Aday, Burak
|
|
|
77 |
C |
p. 101-105
|
artikel
|
| 68 |
Synthesis of pyrazole acrylic acid based oxadiazole and amide derivatives as antimalarial and anticancer agents
|
Verma, Garima
|
|
|
77 |
C |
p. 106-124
|
artikel
|
| 69 |
Synthesis: Small library of hybrid scaffolds of benzothiazole having hydrazone and evaluation of their β-glucuronidase activity
|
Taha, Muhammad
|
|
|
77 |
C |
p. 47-55
|
artikel
|
| 70 |
Taurine as a green bio-organic catalyst for the preparation of bio-active barbituric and thiobarbituric acid derivatives in water media
|
Daneshvar, Nader
|
|
|
77 |
C |
p. 68-73
|
artikel
|
| 71 |
The γ-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae is potently activated by amines and amino acids
|
Angeli, Andrea
|
|
|
77 |
C |
p. 1-5
|
artikel
|
| 72 |
Thiazole-substituted benzenesulfonamides as inhibitors of 12 human carbonic anhydrases
|
Čapkauskaitė, Edita
|
|
|
77 |
C |
p. 534-541
|
artikel
|
| 73 |
Thiazolidinediones as antidiabetic agents: A critical review
|
Nanjan, M.J.
|
|
|
77 |
C |
p. 548-567
|
artikel
|
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