| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
5-Acetyl-6-methyl-4-aryl-3,4-dihydropyrimidin-2(1H)-ones: As potent urease inhibitors; synthesis, in vitro screening, and molecular modeling study
|
Shamim, Shahbaz
|
|
2018
|
76 |
C |
p. 37-52
|
artikel
|
| 2 |
Amino acids/peptides conjugated heterocycles: A tool for the recent development of novel therapeutic agents
|
Wang, Meng
|
|
2018
|
76 |
C |
p. 113-129
|
artikel
|
| 3 |
Aminoadamantanes containing monoterpene-derived fragments as potent tyrosyl-DNA phosphodiesterase 1 inhibitors
|
Ponomarev, Konstantin Yu.
|
|
2018
|
76 |
C |
p. 392-399
|
artikel
|
| 4 |
4-Aminopyridine based amide derivatives as dual inhibitors of tissue non-specific alkaline phosphatase and ecto-5′-nucleotidase with potential anticancer activity
|
Hassan, Sidra
|
|
2018
|
76 |
C |
p. 237-248
|
artikel
|
| 5 |
A simple and efficient synthesis of benzimidazoles containing piperazine or morpholine skeleton at C-6 position as glucosidase inhibitors with antioxidant activity
|
Özil, Musa
|
|
2018
|
76 |
C |
p. 468-477
|
artikel
|
| 6 |
Azole-hydrazone derivatives: Design, synthesis, in vitro biological evaluation, dual EGFR/HER2 inhibitory activity, cell cycle analysis and molecular docking study as anticancer agents
|
Labib, Madlen B.
|
|
2018
|
76 |
C |
p. 67-80
|
artikel
|
| 7 |
Bioactive polyoxygenated seco-cyclohexenes from Artabotrys hongkongensis
|
Liu, Yan-Ping
|
|
2018
|
76 |
C |
p. 386-391
|
artikel
|
| 8 |
Bioactivity evaluation of natural product α-mangostin as a novel xanthone-based lysine-specific demethylase 1 inhibitor to against tumor metastasis
|
Han, Chao
|
|
2018
|
76 |
C |
p. 415-419
|
artikel
|
| 9 |
Biocatalytic hydrolysis of chlorinated nicotinamides by a superior AS family amidase and its application in enzymatic production of 2-chloronicotinic acid
|
Zheng, Ren-Chao
|
|
2018
|
76 |
C |
p. 81-87
|
artikel
|
| 10 |
Biological evaluation of new imidazole derivatives tethered with indole moiety as potent α-glucosidase inhibitors
|
Naureen, Sadia
|
|
2018
|
76 |
C |
p. 365-369
|
artikel
|
| 11 |
Bovine Serum Albumin (BSA) coated iron oxide magnetic nanoparticles as biocompatible carriers for curcumin-anticancer drug
|
Nosrati, Hamed
|
|
2018
|
76 |
C |
p. 501-509
|
artikel
|
| 12 |
Carbazole alkaloids from Clausena hainanensis with their potential antiproliferative activities
|
Ma, Yan-Lei
|
|
2018
|
76 |
C |
p. 359-364
|
artikel
|
| 13 |
Chemical characterization of cytotoxic indole acetic acid derivative from mulberry fruit (Morus alba L.) against human cervical cancer
|
Yu, Jae Sik
|
|
2018
|
76 |
C |
p. 28-36
|
artikel
|
| 14 |
Design and synthesis of cell selective α/β-diastereomeric peptidomimetic with potent in vivo antibacterial activity against methicillin resistant S. Aureus
|
Dewangan, Rikeshwer Prasad
|
|
2018
|
76 |
C |
p. 538-547
|
artikel
|
| 15 |
Design and synthesis of tumor-targeting theranostic drug conjugates for SPECT and PET imaging studies
|
Wang, Tao
|
|
2018
|
76 |
C |
p. 458-467
|
artikel
|
| 16 |
Design, synthesis, and biological evaluation of deuterated phenylpropionic acid derivatives as potent and long-acting free fatty acid receptor 1 agonists
|
Li, Zheng
|
|
2018
|
76 |
C |
p. 303-313
|
artikel
|
| 17 |
Design, synthesis, and biological evaluation of novel substituted benzamide derivatives bearing a 1,2,3-triazole moiety as potent human dihydroorotate dehydrogenase inhibitors
|
Lu, Kuan
|
|
2018
|
76 |
C |
p. 528-537
|
artikel
|
| 18 |
Design, synthesis and evaluation of novel N-hydroxybenzamides/N-hydroxypropenamides incorporating quinazolin-4(3H)-ones as histone deacetylase inhibitors and antitumor agents
|
Hieu, Doan Thanh
|
|
2018
|
76 |
C |
p. 258-267
|
artikel
|
| 19 |
Design, synthesis and evaluation of resveratrol-indazole hybrids as novel monoamine oxidases inhibitors with amyloid-β aggregation inhibition
|
Lan, Jin-Shuai
|
|
2018
|
76 |
C |
p. 130-139
|
artikel
|
| 20 |
Design, synthesis, and initial evaluation of affinity-based small molecular probe for detection of WDR5
|
Chen, Wei-Lin
|
|
2018
|
76 |
C |
p. 380-385
|
artikel
|
| 21 |
Design, synthesis and molecular docking of thiazolidinedione based benzene sulphonamide derivatives containing pyrazole core as potential anti-diabetic agents
|
Naim, Mohd. Javed
|
|
2018
|
76 |
C |
p. 98-112
|
artikel
|
| 22 |
Design, synthesis and molecular modeling studies of new series of antitumor 1,2,4-triazines with potential c-Met kinase inhibitory activity
|
El-Wakil, Marwa H.
|
|
2018
|
76 |
C |
p. 154-165
|
artikel
|
| 23 |
Design, synthesis, antibacterial evaluation and molecular docking studies of some new quinoxaline derivatives targeting dihyropteroate synthase enzyme
|
El-Attar, Maryam A.Z.
|
|
2018
|
76 |
C |
p. 437-448
|
artikel
|
| 24 |
Design, synthesis, anti-inflammatory antitumor activities, molecular modeling and molecular dynamics simulations of potential naprosyn® analogs as COX-1 and/or COX-2 inhibitors
|
El Sayed, Mardia T.
|
|
2018
|
76 |
C |
p. 188-201
|
artikel
|
| 25 |
Design, synthesis, molecular docking of new lipophilic acetamide derivatives affording potential anticancer and antimicrobial agents
|
Ahmed, Hany E.A.
|
|
2018
|
76 |
C |
p. 332-342
|
artikel
|
| 26 |
Design, synthesis, monoamine oxidase inhibition and docking studies of new dithiocarbamate derivatives bearing benzylamine moiety
|
Kaya Çavuşoğlu, Betül
|
|
2018
|
76 |
C |
p. 177-187
|
artikel
|
| 27 |
Design, synthesis of novel Triazolones and bis-Triazolones derivatives under ultrasound irradiation and evaluation as potent angiotensin converting enzyme (ACE) inhibitors
|
Ben Salah, Bochra
|
|
2018
|
76 |
C |
p. 147-153
|
artikel
|
| 28 |
Development of optimized conditions for Glaser-Hay bioconjugations
|
Nimmo, Zachary M.
|
|
2018
|
76 |
C |
p. 326-331
|
artikel
|
| 29 |
Development of pyrrolo[2,1-c][1,4]benzodiazepine β-glucoside prodrugs for selective therapy of cancer
|
Adiyala, Praveen Reddy
|
|
2018
|
76 |
C |
p. 288-293
|
artikel
|
| 30 |
Editorial Board
|
|
|
2018
|
76 |
C |
p. i
|
artikel
|
| 31 |
Effects of adamantane alterations on soluble epoxide hydrolase inhibition potency, physical properties and metabolic stability
|
Burmistrov, Vladimir
|
|
2018
|
76 |
C |
p. 510-527
|
artikel
|
| 32 |
Efficient one-pot enzymatic synthesis of dephospho coenzyme A
|
Sapkota, Krishna
|
|
2018
|
76 |
C |
p. 23-27
|
artikel
|
| 33 |
First evaluation of organotellurium derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors
|
Angeli, Andrea
|
|
2018
|
76 |
C |
p. 268-272
|
artikel
|
| 34 |
Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and membrane-bound hCA IX isoforms
|
Krasavin, Mikhail
|
|
2018
|
76 |
C |
p. 88-97
|
artikel
|
| 35 |
Improving the carbonic anhydrase inhibition profile of the sulfamoylphenyl pharmacophore by attachment of carbohydrate moieties
|
Riafrecha, Leonardo E.
|
|
2018
|
76 |
C |
p. 61-66
|
artikel
|
| 36 |
Issue TOC
|
|
|
2018
|
76 |
C |
p. ii-xv
|
artikel
|
| 37 |
Modification of Bischler-Möhlau indole derivatives through palladium catalyzed Suzuki reaction as effective cholinesterase inhibitors, their kinetic and molecular docking studies
|
Parveen, Shaista
|
|
2018
|
76 |
C |
p. 166-176
|
artikel
|
| 38 |
Nitric oxide inhibitors with a spiro diterpenoid skeleton from Scutellaria formosana: Structures, NO inhibitory effects, and interactions with iNOS
|
Wang, Peixia
|
|
2018
|
76 |
C |
p. 53-60
|
artikel
|
| 39 |
NO inhibitory constituents as potential anti-neuroinflammatory agents for AD from Blumea balsamifera
|
Ma, Jun
|
|
2018
|
76 |
C |
p. 449-457
|
artikel
|
| 40 |
Novel 1,2,4-triazole derivatives as potential anticancer agents: Design, synthesis, molecular docking and mechanistic studies
|
El-Sherief, Hany A.M.
|
|
2018
|
76 |
C |
p. 314-325
|
artikel
|
| 41 |
Oxindole based oxadiazole hybrid analogs: Novel α-glucosidase inhibitors
|
Taha, Muhammad
|
|
2018
|
76 |
C |
p. 273-280
|
artikel
|
| 42 |
Pharmacokinetic studies of naproxen amides of some amino acid esters with promising colorectal cancer chemopreventive activity
|
Aboul-Fadl, Tarek
|
|
2018
|
76 |
C |
p. 370-379
|
artikel
|
| 43 |
Pharmacophore-based drug design for potential AChE inhibitors from Traditional Chinese Medicine Database
|
Jiang, Yingying
|
|
2018
|
76 |
C |
p. 400-414
|
artikel
|
| 44 |
Preventing the N-terminal processing of human interferon α-2b and its chimeric derivatives expressed in Escherichia coli
|
Ahsan, Fatima
|
|
2018
|
76 |
C |
p. 294-302
|
artikel
|
| 45 |
Protonography and anion inhibition profile of the α-carbonic anhydrase (CruCA4) identified in the Mediterranean red coral Corallium rubrum
|
Del Prete, Sonia
|
|
2018
|
76 |
C |
p. 281-287
|
artikel
|
| 46 |
Structural modeling of osteoarthritis ADAMTS4 complex with its cognate inhibitory protein TIMP3 and rational derivation of cyclic peptide inhibitors from the complex interface to target ADAMTS4
|
Zhang, Wei
|
|
2018
|
76 |
C |
p. 13-22
|
artikel
|
| 47 |
Sulfonamides containing curcumin scaffold: Synthesis, characterization, carbonic anhydrase inhibition and molecular docking studies
|
Ahmed, Mahmood
|
|
2018
|
76 |
C |
p. 218-227
|
artikel
|
| 48 |
Synthesis and biological evaluation of new oxopyrrolidine derivatives as inhibitors of acetyl cholinesterase and β amyloid protein as anti – Alzheimer’s agents
|
Mohamed, Lamia W.
|
|
2018
|
76 |
C |
p. 210-217
|
artikel
|
| 49 |
Synthesis and molecular docking study of new benzofuran and furo[3,2-g]chromone-based cytotoxic agents against breast cancer and p38α MAP kinase inhibitors
|
Amin, Kamelia M.
|
|
2018
|
76 |
C |
p. 487-500
|
artikel
|
| 50 |
Synthesis, anti-inflammatory, p38α MAP kinase inhibitory activities and molecular docking studies of quinoxaline derivatives containing triazole moiety
|
Tariq, Sana
|
|
2018
|
76 |
C |
p. 343-358
|
artikel
|
| 51 |
Synthesis, biological evaluation and molecular docking studies of a new series of chalcones containing naphthalene moiety as anticancer agents
|
Wang, Guangcheng
|
|
2018
|
76 |
C |
p. 249-257
|
artikel
|
| 52 |
Synthesis, molecular docking and biological evaluation of some benzimidazole derivatives as potent pancreatic lipase inhibitors
|
Menteşe, Emre
|
|
2018
|
76 |
C |
p. 478-486
|
artikel
|
| 53 |
Synthesis of benzo[d]imidazo[2,1-b]thiazole-chalcone conjugates as microtubule targeting and apoptosis inducing agents
|
Sultana, Faria
|
|
2018
|
76 |
C |
p. 1-12
|
artikel
|
| 54 |
Synthesis of derivatives of cleistopholine and their anti-acetylcholinesterase and anti-β-amyloid aggregation activity
|
Wu, Zhenhua
|
|
2018
|
76 |
C |
p. 228-236
|
artikel
|
| 55 |
Synthesis of imidazo-thiadiazole linked indolinone conjugates and evaluated their microtubule network disrupting and apoptosis inducing ability
|
Narasimha Rao, M.P.
|
|
2018
|
76 |
C |
p. 420-436
|
artikel
|
| 56 |
The “Janus face” of the thrombin binding aptamer: Investigating the anticoagulant and antiproliferative properties through straightforward chemical modifications
|
Esposito, Veronica
|
|
2018
|
76 |
C |
p. 202-209
|
artikel
|
| 57 |
Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors
|
Sapegin, Alexander
|
|
2018
|
76 |
C |
p. 140-146
|
artikel
|
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