| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A CuSO4/Bicinchoninic acid/Reducing sugar based stable and non-ROS catalyst system for the CuAAC reaction in bioanalysis
|
Wang, Yuchen
|
|
|
150 |
C |
p.
|
artikel
|
| 2 |
Amonafide-based H2O2-responsive theranostic prodrugs: Exploring the correlation between H2O2 level and anticancer efficacy
|
Yao, Xueyan
|
|
|
150 |
C |
p.
|
artikel
|
| 3 |
Amphiphilic coumarin-based probes for live-cell STED nanoscopy of plasma membrane
|
Kokot, Hana
|
|
|
150 |
C |
p.
|
artikel
|
| 4 |
A new strategy for the treatment of Parkinson’s disease: Discovery and bio-evaluation of the first central-targeting tyrosinase inhibitor
|
Qi, Shulei
|
|
|
150 |
C |
p.
|
artikel
|
| 5 |
A novel AIE fluorescent probe for the detection and imaging of hydrogen peroxide in living tumor cells and in vivo
|
Peng, Zihao
|
|
|
150 |
C |
p.
|
artikel
|
| 6 |
A quest for novel antimicrobial targets: Inhibition of Asp-tRNAAsn/Glu-tRNAGln amidotransferase (GatCAB) by synthetic analogs of aminoacyl-adenosine in vitro and live bacteria
|
Sangsuwan, Withsakorn
|
|
|
150 |
C |
p.
|
artikel
|
| 7 |
Axially chiral dihydrophenanthrene dimers from Pholidota yunnanensis with anti-neuroinflammatory activities
|
Qi, Jiaxin
|
|
|
150 |
C |
p.
|
artikel
|
| 8 |
Characterization of a small molecule inhibitor of the NLRP3 inflammasome and its potential use for acute lung injury
|
Xu, Yiming
|
|
|
150 |
C |
p.
|
artikel
|
| 9 |
Chemical sensors for the early diagnosis of bacterial resistance to β-lactam antibiotics
|
Canabal, Rafael
|
|
|
150 |
C |
p.
|
artikel
|
| 10 |
Chlorogenic acid can improve spermatogenic dysfunction in rats with varicocele by regulating mitochondrial homeostasis and inhibiting the activation of NLRP3 inflammasomes by oxidative mitochondrial DNA and cGAS/STING pathway
|
Jia, Zhi-chao
|
|
|
150 |
C |
p.
|
artikel
|
| 11 |
Comprehensive insights into fluorescent probes for the determination nitric oxide for diseases diagnosis
|
Ye, Chenqian
|
|
|
150 |
C |
p.
|
artikel
|
| 12 |
Computer-aided design of a fluorescent MAT2A inhibitor for visualized cancer synthetic lethality
|
Wang, Ziwei
|
|
|
150 |
C |
p.
|
artikel
|
| 13 |
Corrigendum to “Discovery of KRas G12C-IN-3 and Pomalidomide-based PROTACs as degraders of endogenous KRAS G12C with potent anticancer activity” [Bioorgan. Chem. 117 (2021) 105447]
|
Li, Ling
|
|
|
150 |
C |
p.
|
artikel
|
| 14 |
Corrigendum to “Sulfonamides as anticancer agents: A brief review on sulfonamide derivatives as inhibitors of various proteins overexpressed in cancer” [Bioorg. Chem. 147 (2024) 107409]
|
Elsayad, Khaled A.
|
|
|
150 |
C |
p.
|
artikel
|
| 15 |
Deciphering molecular mechanisms underlying the inhibition of β-glucuronidase by xanthones from Centaurium spicatum
|
Kamel, Emadeldin M.
|
|
|
150 |
C |
p.
|
artikel
|
| 16 |
Density functional theory and enzyme studies support interactions between angiotensin receptor blockers and angiotensin converting enzyme-2: Relevance to coronavirus 2019
|
Apostolopoulos, Vasso
|
|
|
150 |
C |
p.
|
artikel
|
| 17 |
Design and synthesis of hemicyanine-based NIRF probe for detecting Aβ aggregates in Alzheimer’s disease
|
Zhao, Xueqi
|
|
|
150 |
C |
p.
|
artikel
|
| 18 |
Designing NIR AIEgens for lysosomes targeting and efficient photodynamic therapy of tumors
|
Li, Yuanhang
|
|
|
150 |
C |
p.
|
artikel
|
| 19 |
Design, synthesis and anti-inflammatory assessment of certain substituted 1,2,4-triazoles bearing tetrahydroisoquinoline scaffold as COX 1/2-inhibitors
|
Abo-Elmagd, Mai I.
|
|
|
150 |
C |
p.
|
artikel
|
| 20 |
Design, synthesis and biological evaluation of novel naphthoquinothiazole derivatives as potent antitumor agents through inhibiting STAT3
|
Fan, Dongmei
|
|
|
150 |
C |
p.
|
artikel
|
| 21 |
Design, synthesis and cytotoxic evaluation of new thieno[2,3-d]pyrimidine analogues as VEGFR-2/AKT dual inhibitors, apoptosis and autophagy inducers
|
Abd El-Mawgoud, Heba K.
|
|
|
150 |
C |
p.
|
artikel
|
| 22 |
Design, synthesis, antineoplastic activity of new pyrazolo[3,4-d]pyrimidine derivatives as dual CDK2/GSK3β kinase inhibitors; molecular docking study, and ADME prediction
|
Nemr, Mohamed T.M.
|
|
|
150 |
C |
p.
|
artikel
|
| 23 |
Development and therapeutic potential of DNA-dependent protein kinase inhibitors
|
Hui, Zi
|
|
|
150 |
C |
p.
|
artikel
|
| 24 |
Discovery and characterization of novel FGFR1 inhibitors in triple-negative breast cancer via hybrid virtual screening and molecular dynamics simulations
|
Wang, Yuchen
|
|
|
150 |
C |
p.
|
artikel
|
| 25 |
Discovery of a first-in-class protein degrader for the c-ros oncogene 1 (ROS1)
|
Yang, Jiawen
|
|
|
150 |
C |
p.
|
artikel
|
| 26 |
Discovery of a highly selective fluorescent probe for hydrogen peroxide and its biocompatibility evaluation and bioimaging applications in cells and zebrafish
|
Li, Wenzhai
|
|
|
150 |
C |
p.
|
artikel
|
| 27 |
Discovery of cinnamamide/ester triazole hybrids as potential treatment for Alzheimer’s disease
|
Tan, Lin-Jie
|
|
|
150 |
C |
p.
|
artikel
|
| 28 |
Discovery of colchicine aryne cycloadduct as a potent molecule for the abrogation of epithelial to mesenchymal transition via modulating cell cycle regulatory CDK-2 and CDK-4 kinases in breast cancer cells
|
Iqbal Lone, Waseem
|
|
|
150 |
C |
p.
|
artikel
|
| 29 |
Discovery of 23,24-diols containing ergosterols with anti-neuroinflammatory activity from Penicillium citrinum TJ507
|
Zhang, Yeting
|
|
|
150 |
C |
p.
|
artikel
|
| 30 |
Discovery of (E)-3-(4-chlorophenyl)-N-(5-hydroxypentyl)acrylamide among N-substituted cinnamamide derivatives as a novel cosmetic ingredient for hyperpigmentation
|
Gunia-Krzyżak, Agnieszka
|
|
|
150 |
C |
p.
|
artikel
|
| 31 |
Discovery of natural AMPK activator from the fruits of Xanthium sibiricum Patr.: Xanthiumine A, protoberberine alkaloid with unique C28 skeleton
|
Yao, Tie
|
|
|
150 |
C |
p.
|
artikel
|
| 32 |
Discovery of novel CDK9 inhibitor with tridentate ligand: Design, synthesis and biological evaluation
|
Zhong, Ye
|
|
|
150 |
C |
p.
|
artikel
|
| 33 |
Discovery of novel chrysin derivatives as potential Anti-Psoriasis agents
|
Zhao, Xiujuan
|
|
|
150 |
C |
p.
|
artikel
|
| 34 |
Discovery of novel 1,8-naphthalimide piperazinamide based benzenesulfonamides derivatives as potent carbonic anhydrase IX inhibitors and ferroptosis inducers for the treatment of triple-negative breast cancer
|
Liang, Qiaoling
|
|
|
150 |
C |
p.
|
artikel
|
| 35 |
Discovery of piperine derivatives as inhibitors of human dihydroorotate dehydrogenase to induce ferroptosis in cancer cells
|
Zhang, Jian-Fei
|
|
|
150 |
C |
p.
|
artikel
|
| 36 |
Discovery of Protease-activated receptor 2 antagonists derived from phenylalanine for the treatment of breast cancer
|
Kim, Taegun
|
|
|
150 |
C |
p.
|
artikel
|
| 37 |
Discovery of TCP-(MP)-caffeic acid analogs as a new class of agents for treatment of osteoclastic bone loss
|
Chen, Zhihao
|
|
|
150 |
C |
p.
|
artikel
|
| 38 |
DMF-DMA catalyzed Synthesis, molecular docking, in-vitro, in-silico design, and binding free energy studies of novel thiohydantoin derivatives as antioxidant and antiproliferative agents targeting EGFR tyrosine kinase and aromatase cytochrome P450 enzyme
|
Seliem, Israa A.
|
|
|
150 |
C |
p.
|
artikel
|
| 39 |
Editorial Board
|
|
|
|
150 |
C |
p.
|
artikel
|
| 40 |
Endophytic Fungi: Cellular factories of novel medicinal chemistries
|
Pokhriyal, Ankita
|
|
|
150 |
C |
p.
|
artikel
|
| 41 |
Enhanced binding interaction and antibacterial inhibition for nanometal oxide particles activated with Aloe Vulgarize through one-pot ultrasonication techniques
|
Dzulkharnien, Nur Syafiqah Farhanah
|
|
|
150 |
C |
p.
|
artikel
|
| 42 |
Evaluation of antifungal potentials of Albizia kalkora extract as a natural fungicide: In vitro and computational studies
|
Hassan, Ahmad
|
|
|
150 |
C |
p.
|
artikel
|
| 43 |
α-Glucosidase inhibition assay of galbanic acid and it amide derivatives: New excellent semi-synthetic α-glucosidase inhibitors
|
Mohammadi-Khanaposhtani, Maryam
|
|
|
150 |
C |
p.
|
artikel
|
| 44 |
Gypenoside L inhibits hepatocellular carcinoma by targeting the SREBP2-HMGCS1 axis and enhancing immune response
|
Xiao, Man-Yu
|
|
|
150 |
C |
p.
|
artikel
|
| 45 |
Highly potent anti-melanogenic effect of 2-thiobenzothiazole derivatives through nanomolar tyrosinase activity inhibition
|
Jin Jung, Hee
|
|
|
150 |
C |
p.
|
artikel
|
| 46 |
Homo and Hetero-Branched Lipopeptide Dendrimers: Synthesis and Antimicrobial Activity
|
Lamba, Saurabh
|
|
|
150 |
C |
p.
|
artikel
|
| 47 |
(±)-Hypernumqulins A–H: Eight pairs of unexpected [2+2] cycloaddition sesquiterpenoid alkaloid with 6/6/6/4/10 ring system from Hypericum monogynum L.
|
Dong, Zhaoyue
|
|
|
150 |
C |
p.
|
artikel
|
| 48 |
Identification of novel 4-substituted 7H-pyrrolo[2,3-d]pyrimidine derivatives as new FtsZ inhibitors: Bioactivity evaluation and computational simulation
|
Li, Ting
|
|
|
150 |
C |
p.
|
artikel
|
| 49 |
Impact of sulfur substitution on biotin binding affinity to streptavidin
|
Groaz, Elisabetta
|
|
|
150 |
C |
p.
|
artikel
|
| 50 |
Inhibition of the STAT3-EPHX2 axis promotes regression of ulcerative colitis by treatment with novel porphyrin derivative
|
Xu, Bin
|
|
|
150 |
C |
p.
|
artikel
|
| 51 |
Issue TOC
|
|
|
|
150 |
C |
p.
|
artikel
|
| 52 |
Molecular mechanisms of EGCG-CSH/n-HA/CMC in promoting osteogenic differentiation and macrophage polarization
|
Jia, Bei
|
|
|
150 |
C |
p.
|
artikel
|
| 53 |
New coumarin linked thiazole derivatives as antimycobacterial agents: Design, synthesis, enoyl acyl carrier protein reductase (InhA) inhibition and molecular modeling
|
Kassem, Asmaa F.
|
|
|
150 |
C |
p.
|
artikel
|
| 54 |
Novel acyl hydrazide derivatives of polyhydroquinoline as potent anti-diabetic and anti-glycating agents: Synthesis, in vitro α-amylase, α-glucosidase inhibition and anti-glycating activity with molecular docking insights
|
Ur Rahman, Sajjad
|
|
|
150 |
C |
p.
|
artikel
|
| 55 |
Novel antibody-antibiotic conjugate using KRM-1657 as payload eliminates intracellular MRSA in vitro and in vivo
|
Fan, Shiyong
|
|
|
150 |
C |
p.
|
artikel
|
| 56 |
Novel insight into mitochondrial dynamin-related protein-1 as a new chemo-sensitizing target in resistant cancer cells
|
Sami Alkafaas, Samar
|
|
|
150 |
C |
p.
|
artikel
|
| 57 |
Novel 131-iodine labeled and ultrasound-responsive nitric oxide and reactive oxygen species controlled released nanoplatform for synergistic sonodynamic/nitric oxide/chemodynamic/radionuclide therapy
|
Ma, Sufang
|
|
|
150 |
C |
p.
|
artikel
|
| 58 |
Novel isoniazid-hydrazone derivatives induce cell growth inhibition, cell cycle arrest and apoptosis via mitochondria-dependent caspase activation and PI3K/AKT inhibition
|
Rouzi, Khouloud
|
|
|
150 |
C |
p.
|
artikel
|
| 59 |
Novel quinazoline sulfonamide-based scaffolds modulate methicillin-resistant Staphylococcus aureus (MRSA) pneumonia in immunodeficient irradiated model: Regulatory role of TGF-β
|
Soliman, Aiten M.
|
|
|
150 |
C |
p.
|
artikel
|
| 60 |
Novel tropane analogues as Hsp90 inhibitors targeting colon cancer: Synthesis, biological estimation, and molecular docking study
|
Almehmadi, Samar J.
|
|
|
150 |
C |
p.
|
artikel
|
| 61 |
Protective effects of baicalin against phenylarsine oxide-induced cytotoxicity in human skin keratinocytes
|
Li, Mengling
|
|
|
150 |
C |
p.
|
artikel
|
| 62 |
Pseudo-Natural Products: Expanding chemical and biological space by surpassing natural constraints
|
Ahamad, Shakir
|
|
|
150 |
C |
p.
|
artikel
|
| 63 |
Pyrazolone compounds could inhibit CES1 and ameliorates fat accumulation during adipocyte differentiation
|
Wang, Dan-Dan
|
|
|
150 |
C |
p.
|
artikel
|
| 64 |
Reactivators of butyrylcholinesterase inhibited by organophosphorus compounds
|
Kohoutova, Zuzana
|
|
|
150 |
C |
p.
|
artikel
|
| 65 |
Recent advances in small molecule Nav 1.7 inhibitors for cancer pain management
|
Yu, Xiaoquan
|
|
|
150 |
C |
p.
|
artikel
|
| 66 |
Recent advances in the development of bacterial response regulators inhibitors as antibacterial and/or antibiotic adjuvant agent: A new approach to combat bacterial resistance
|
Majdi, Chaimae
|
|
|
150 |
C |
p.
|
artikel
|
| 67 |
Recent efforts in the development of glycoconjugate vaccine and available treatment for tuberculosis
|
Banoo, Sajida
|
|
|
150 |
C |
p.
|
artikel
|
| 68 |
RNase H-sensitive multifunctional ASO-based constructs as promising tools for the treatment of multifactorial complex pathologies
|
Mata-Ventosa, Aida
|
|
|
150 |
C |
p.
|
artikel
|
| 69 |
(5S)-5-Benzylswainsonines as potent and selective inhibitors of Golgi α-mannosidase II: synthesis, enzyme evaluation and molecular modelling
|
Kalník, Martin
|
|
|
150 |
C |
p.
|
artikel
|
| 70 |
sp2-Iminosugar azobenzene O-glycosides: Light-sensitive glycosidase inhibitors with unprecedented tunability and switching factors
|
Rivero-Barbarroja, Gonzalo
|
|
|
150 |
C |
p.
|
artikel
|
| 71 |
Stable ubiquitin conjugation for biological interrogation of ubiquitinated tau repeat domain
|
Viola, Giovanna
|
|
|
150 |
C |
p.
|
artikel
|
| 72 |
Stilbene-pyridazinone hybrids: design, synthesis and in vitro antiplatelet activity screening
|
Costas-Lago, Maria Carmen
|
|
|
150 |
C |
p.
|
artikel
|
| 73 |
Structure-activity relationships of natural and synthetic lathyrane-based diterpenoids for suppression of NLRP3-driven inflammation and gouty arthritis
|
Zhuang, Yuqing
|
|
|
150 |
C |
p.
|
artikel
|
| 74 |
Structures, biosynthesis and biological activities of benastatins, anthrabenzoxocinones and fredericamycins
|
Tsakem, Bienvenu
|
|
|
150 |
C |
p.
|
artikel
|
| 75 |
Structure, unique biological properties, and mechanisms of action of transforming growth factor β
|
Zelisko, Nataliya
|
|
|
150 |
C |
p.
|
artikel
|
| 76 |
Synthesis and anti-proliferative effect of novel 4-Aryl-1, 3-Thiazole-TPP conjugates via mitochondrial uncoupling process
|
Hu, Yixin
|
|
|
150 |
C |
p.
|
artikel
|
| 77 |
Synthesis and characterization of organoselenium based BODIPY and its application in living cells
|
Shelar, Divyesh S.
|
|
|
150 |
C |
p.
|
artikel
|
| 78 |
Synthesis and pharmacological evaluation of novel N-aryl-cinnamoyl-hydrazone hybrids designed as neuroprotective agents for the treatment of Parkinson’s disease
|
de Freitas Silva, Matheus
|
|
|
150 |
C |
p.
|
artikel
|
| 79 |
Synthesis, biological evaluation, theoretical calculations, QSAR and molecular docking studies of novel arylaminonaphthols as potent antioxidants and BChE inhibitors
|
Benoune, Racha Amira
|
|
|
150 |
C |
p.
|
artikel
|
| 80 |
Synthesis, COX-2 inhibition, anti-inflammatory activity, molecular docking, and histopathological studies of new pyridazine derivatives
|
Ewieda, Sara Y.
|
|
|
150 |
C |
p.
|
artikel
|
| 81 |
Synthesis, insecticidal Activity, and molecular docking analysis of some benzo[h]quinoline derivatives against Culex pipiens L. Larvae
|
El-Helw, Eman A.E.
|
|
|
150 |
C |
p.
|
artikel
|
| 82 |
Synthesis, molecular modeling simulations and anticancer activity of some new Imidazo[2,1-b]thiazole analogues as EGFR/HER2 and DHFR inhibitors
|
Moharram, Esraa A.
|
|
|
150 |
C |
p.
|
artikel
|
| 83 |
Synthesis of amino juglone derivatives with adjuvant activity against clinical isolated methicillin-resistant staphylococcus aureus strains
|
Majdi, Chaimae
|
|
|
150 |
C |
p.
|
artikel
|
| 84 |
Targeting MDM2-p53 interaction in Glioblastoma: Transcriptomic analysis and Peptide-Based inhibition strategy
|
Han, Manman
|
|
|
150 |
C |
p.
|
artikel
|
| 85 |
Tetrazine–trans-cyclooctene ligation: Unveiling the chemistry and applications within the human body
|
Tomarchio, Elisabetta Grazia
|
|
|
150 |
C |
p.
|
artikel
|
| 86 |
The cytotoxic natural compound erianin binds to colchicine site of β-tubulin and overcomes taxane resistance
|
Yan, Wei
|
|
|
150 |
C |
p.
|
artikel
|
| 87 |
The flavonoids from the fruits of Psoralea corylifolia and their potential in inhibiting metastasis of human non-small cell lung cancers
|
Shi, Peixin
|
|
|
150 |
C |
p.
|
artikel
|
| 88 |
The proof of concept of 2-{3-[N-(1-benzylpiperidin-4-yl)propyl]amino}-6-[N-methyl-N-(prop-2-yn-1-yl)amino]-4-phenylpyridine-3,5-dicarbonitrile for the therapy of neuropathic pain
|
Entrena, José M.
|
|
|
150 |
C |
p.
|
artikel
|
| 89 |
Triazole derivatives inhibit the VOR complex-mediated nuclear transport of extracellular particles: Potential application in cancer and HIV-1 infection
|
Carbone, Daniela
|
|
|
150 |
C |
p.
|
artikel
|
| 90 |
Tripeptide linked dispiro cyclotriphosphazene conjugates: Synthesis, molecular docking analysis of compounds binding within cancer cell line receptors and in vitro cytotoxic and genotoxic activities
|
Çalışkan, Eray
|
|
|
150 |
C |
p.
|
artikel
|
| 91 |
Unveiling a new strategy for PDIA1 inhibition: Integration of activity-based probes profiling and targeted degradation
|
Zhang, Bei
|
|
|
150 |
C |
p.
|
artikel
|
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