nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A comparative study of diaryl urea molecules with and without sulfonamide group on Carbonic anhydrase IX and XII inhibition and its consequence on breast cancer cells
|
Debnath, Joy |
|
|
145 |
C |
p. |
artikel |
2 |
3-Amide-β-carbolines block the cell cycle by targeting CDK2 and DNA in tumor cells potentially as anti-mitotic agents
|
Zhi, Dongming |
|
|
145 |
C |
p. |
artikel |
3 |
A novel NIR fluorescent probe inhibits melanoma progression through apoptosis and ERK/DRP1-mediated mitochondrial fission
|
He, Qingqing |
|
|
145 |
C |
p. |
artikel |
4 |
Anti-diabetic and anti-inflammatory indole diterpenes from the marine-derived fungus Penicillium sp. ZYX-Z-143
|
Dai, Lu-Ting |
|
|
145 |
C |
p. |
artikel |
5 |
Astraoleanosides E–P, oleanane-type triterpenoid saponins from the aerial parts of Astragalus membranaceus Bunge and their β-glucuronidase inhibitory activity
|
Nguyen, Manh Khoa |
|
|
145 |
C |
p. |
artikel |
6 |
Bibenzyl and naphthalene derivatives from Dendrobium chrysanthum and their anti-hepatic-steatosis activities
|
Zhang, Zi-Mo |
|
|
145 |
C |
p. |
artikel |
7 |
Biologically active isoquinoline alkaloids covering 2019–2022
|
Wang, Dengtuo |
|
|
145 |
C |
p. |
artikel |
8 |
Buffalo colostrum peptide mitigates Parkinson's disease pathophysiology through Cullin-3 inhibition
|
Ashok, Arpitha |
|
|
145 |
C |
p. |
artikel |
9 |
Chemical proteomics unveils that seventy flavors pearl pill ameliorates ischemic stroke by regulating oxidative phosphorylation
|
Ma, Ruyun |
|
|
145 |
C |
p. |
artikel |
10 |
Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases
|
Fuentes-Aguilar, Alma |
|
|
145 |
C |
p. |
artikel |
11 |
Counterion influence on near-infrared-II heptamethine cyanine salts for photothermal therapy
|
Zheng, Yilin |
|
|
145 |
C |
p. |
artikel |
12 |
Cyclic peptide conjugated photosensitizer for targeted phototheranostics of gram-negative bacterial infection
|
Wu, Minghao |
|
|
145 |
C |
p. |
artikel |
13 |
Design, synthesis, and anticancer evaluation of N-sulfonylpiperidines as potential VEGFR-2 inhibitors, apoptotic inducers
|
Elgammal, Walid E. |
|
|
145 |
C |
p. |
artikel |
14 |
Design, synthesis, and biological evaluation of gambogenic acid derivatives: Unraveling their anti-cancer effects by inducing pyroptosis
|
Huang, Qing |
|
|
145 |
C |
p. |
artikel |
15 |
Design, synthesis, and biological evaluation of some new 2-phenyl-3,6-pyridazinedione derivatives as PDE-5 inhibitors
|
Abd-Rabo, Zeinab S. |
|
|
145 |
C |
p. |
artikel |
16 |
Design, synthesis, biological evaluation and docking study of some new aryl and heteroaryl thiomannosides as FimH antagonists
|
Mohammed, Anber F. |
|
|
145 |
C |
p. |
artikel |
17 |
Discovery of a doublecortin-like kinase 1 inhibitor to prevent inflammatory responses in acute lung injury
|
Cai, Binhao |
|
|
145 |
C |
p. |
artikel |
18 |
Discovery of a stilbenoid-flavanone hybrid as an antitumor Wnt/β-catenin signaling pathway inhibitor
|
Hassan, Ahmed H.E. |
|
|
145 |
C |
p. |
artikel |
19 |
Discovery of the 2,4-disubstituted quinazoline derivative as a novel neddylation inhibitor for tumor therapy
|
Su, Jingtian |
|
|
145 |
C |
p. |
artikel |
20 |
Diterpenoids from Euphorbia peplus possessing cytotoxic and anti-inflammatory activities
|
Li, Ying |
|
|
145 |
C |
p. |
artikel |
21 |
Editorial Board
|
|
|
|
145 |
C |
p. |
artikel |
22 |
Effect of N-o-nitrobenzylation on conformation and membrane permeability of linear peptides
|
Huang, Zhihan |
|
|
145 |
C |
p. |
artikel |
23 |
Effects of selenium nanoparticles produced by Lactobacillus acidophilus HN23 on lipid deposition in WRL68 cells
|
Lei, Xianglan |
|
|
145 |
C |
p. |
artikel |
24 |
Enzymatic properties and immobilization of a thermostable prenyltransferase from Aspergillus fumigatiaffinis for the production of prenylated naringenin
|
Li, Wenbo |
|
|
145 |
C |
p. |
artikel |
25 |
Expansion of targeted degradation by Gilteritinib-Warheaded PROTACs to ALK fusion proteins
|
Yokoo, Hidetomo |
|
|
145 |
C |
p. |
artikel |
26 |
Exploiting the biocatalytic potential of co-expressed l-fucose isomerase and d-tagatose 3-epimerase for the biosynthesis of 6-deoxy-l-sorbose
|
Waheed Iqbal, Muhammad |
|
|
145 |
C |
p. |
artikel |
27 |
Genetic loss of Nrf1 and Nrf2 leads to distinct metabolism reprogramming of HepG2 cells by opposing regulation of the PI3K-AKT-mTOR signalling pathway
|
Deng, Rongzhen |
|
|
145 |
C |
p. |
artikel |
28 |
Glycomimetic inhibitors of tandem-repeat galectins: Simple and efficient
|
Vrbata, David |
|
|
145 |
C |
p. |
artikel |
29 |
Green synthesis of zinc oxide nanoparticles using ethanolic extract of Gliricidia sepium (Jacq.) Kunth. ex. Walp., stem: Characterizations and their gastroprotective effect on ethanol-induced gastritis in rats
|
Wafaey, Aya A. |
|
|
145 |
C |
p. |
artikel |
30 |
Hybrid pharmacophore design and synthesis of donepezil-inspired aurone derivative salts as multifunctional acetylcholinesterase inhibitors
|
Funahashi, Rei |
|
|
145 |
C |
p. |
artikel |
31 |
Hydrocarbon stapled temporin-L analogue as potential antibacterial and antiendotoxin agents with enhanced protease stability
|
Mahto, Aman Kumar |
|
|
145 |
C |
p. |
artikel |
32 |
Identification and anti-oxidative potential of milk fat globule membrane (MFGM)-derived bioactive peptides released through in vitro gastrointestinal digestion
|
Li, He |
|
|
145 |
C |
p. |
artikel |
33 |
Identification and structural modification of ent-rosane diterpenoids from Euphorbia milii inhibiting RANKL-induced osteoclastogenesis
|
Peng, Xing |
|
|
145 |
C |
p. |
artikel |
34 |
Identification of new 5-(2,6-dichlorophenyl)-3-oxo-2,3-dihydro-5H-thiazolo[3,2-a]pyrimidine-7-carboxylic acids as p38α MAPK inhibitors: Design, synthesis, antitumor evaluation, molecular docking and in silico studies
|
El-Wakil, Marwa H. |
|
|
145 |
C |
p. |
artikel |
35 |
Identification of novel human CC chemokine receptor 8 (CCR8) antagonists via the synthesis of naphthalene amide and sulfonamide isosteres
|
Verhaegen, Yenthel |
|
|
145 |
C |
p. |
artikel |
36 |
Identification of Phytochemicals with Inhibitory Potential Against Beta-lactamase Enzymes via Computer-aided Approach
|
Nwokebu, Goodness Chizorom |
|
|
145 |
C |
p. |
artikel |
37 |
Issue TOC
|
|
|
|
145 |
C |
p. |
artikel |
38 |
Macrolide sesquiterpene pyridine alkaloids from Celastrus monospermus and evaluation of their immunosuppressive and anti-osteoclastogenesis activities
|
Ning, Ruonan |
|
|
145 |
C |
p. |
artikel |
39 |
Monoamine oxidase B activatable red fluorescence probe for bioimaging in cells and zebrafish
|
Yang, Zhengmin |
|
|
145 |
C |
p. |
artikel |
40 |
Multi-target rational design and synthesis of novel diphenyl-tethered pyrazolopyrimidines targeting EGFR and topoisomerase II with potential DNA intercalation and apoptosis induction
|
Gaber, Ahmed A |
|
|
145 |
C |
p. |
artikel |
41 |
N- and s-substituted Pyrazolopyrimidines: A promising new class of potent c-Src kinase inhibitors with prominent antitumor activity
|
Awaji, Aeshah A. |
|
|
145 |
C |
p. |
artikel |
42 |
New daphnane diterpenoidal 1,3,4-oxdiazole derivatives as potential anti-hepatoma agents: Synthesis, biological evaluation and molecular modeling studies
|
Wang, Xinyi |
|
|
145 |
C |
p. |
artikel |
43 |
New 2-oxoindole derivatives as multiple PDGFRα/ß and VEGFR-2 tyrosine kinase inhibitors
|
Ezelarab, Hend A.A. |
|
|
145 |
C |
p. |
artikel |
44 |
Novel drimane-type sesquiterpenoids and nucleosides from the Helicoma septoconstrictum suppress the growth of ovarian cancer cells
|
Zheng, Wen |
|
|
145 |
C |
p. |
artikel |
45 |
Novel multi-target angiogenesis inhibitors as potential anticancer agents: Design, synthesis and preliminary activity evaluation
|
Zhang, Qingqing |
|
|
145 |
C |
p. |
artikel |
46 |
Novel Pyrimidine-5-Carbonitriles as potential apoptotic and antiproliferative agents by dual inhibition of EGFRWT/T790M and PI3k enzymes; Design, Synthesis, biological Evaluation, and docking studies
|
Reda, Nada |
|
|
145 |
C |
p. |
artikel |
47 |
Novel spiroindoline derivatives targeting aldose reductase against diabetic complications: Bioactivity, cytotoxicity, and molecular modeling studies
|
Güleç, Özcan |
|
|
145 |
C |
p. |
artikel |
48 |
Phenolics and terpenoids with good anti-inflammatory activity from the fruits of Amomum villosum and the anti-inflammatory mechanism of active diterpene
|
Xu, Yang |
|
|
145 |
C |
p. |
artikel |
49 |
Proteasome activation: A novel strategy for targeting undruggable intrinsically disordered proteins
|
Yu, Qian |
|
|
145 |
C |
p. |
artikel |
50 |
Pyrano[2,3-b]chromone derivatives as novel dual inhibitors of α-glucosidase and α-amylase: Design, synthesis, biological evaluation, and in silico studies
|
Farzaneh, Elnaz |
|
|
145 |
C |
p. |
artikel |
51 |
Recent advances in antimicrobial peptide-based therapy
|
Mulukutla, Aditya |
|
|
145 |
C |
p. |
artikel |
52 |
Recent developments on the synthesis of biologically active glycohybrids
|
Mishra, Vinay Kumar |
|
|
145 |
C |
p. |
artikel |
53 |
Sequential release of interacting proteins and Ub-modifying enzymes by disulfide heterotypic ubiquitin reagents
|
Cai, Hongyi |
|
|
145 |
C |
p. |
artikel |
54 |
SETDB1: Progress and prospects in cancer treatment potential and inhibitor research
|
Ma, Tingnan |
|
|
145 |
C |
p. |
artikel |
55 |
Small-molecule modulators of tumor immune microenvironment
|
Zhang, Jing |
|
|
145 |
C |
p. |
artikel |
56 |
Structural modification of natural axinelline A: Achieving reduced colitis side effects through balanced COX inhibition
|
Ju, Zhiran |
|
|
145 |
C |
p. |
artikel |
57 |
Structural optimization and biological evaluation of ML364 based derivatives as USP2a inhibitors
|
Son, Youngchai |
|
|
145 |
C |
p. |
artikel |
58 |
Structure-Affinity relationships of novel σ2R/TMEM97 ligands
|
Walby, Grant D. |
|
|
145 |
C |
p. |
artikel |
59 |
Sulfur (SⅥ)-containing heterocyclic hybrids as antibacterial agents against methicillin-resistant Staphylococcus aureus (MRSA) and its SAR
|
Verma, Santosh Kumar |
|
|
145 |
C |
p. |
artikel |
60 |
Synthesis and bio-evaluation of newer dihydropyridines and tetrahydropyridines based glycomimetic azasugars
|
Deswal, Nidhi |
|
|
145 |
C |
p. |
artikel |
61 |
Synthesis and evaluation of novel N1-acylated 5-(4-pyridinyl)indazole derivatives as potent and selective haspin inhibitors
|
Shawky, Mona M. |
|
|
145 |
C |
p. |
artikel |
62 |
Synthesis and preclinical evaluation of a novel molecular probe [18F]AlF-NOTA-PEG2-Asp2-PDL1P for PET imaging of PD-L1 positive tumor
|
Sun, Penghui |
|
|
145 |
C |
p. |
artikel |
63 |
Tailored quinoline hybrids as promising COX-2/15-LOX dual inhibitors endowed with diverse safety profile: Design, synthesis, SAR, and histopathological study
|
Hegazy, Mohamed E. |
|
|
145 |
C |
p. |
artikel |
64 |
Targeting dihydroceramide desaturase 1 (Des1): Syntheses of ceramide analogues with a rigid scaffold, inhibitory assays, and AlphaFold2-assisted structural insights reveal cyclopropenone PR280 as a potent inhibitor
|
Rivero, Pablo |
|
|
145 |
C |
p. |
artikel |
65 |
The antimicrobial potential of adarotene derivatives against Staphylococcus aureus strains
|
Princiotto, Salvatore |
|
|
145 |
C |
p. |
artikel |
66 |
The binding selectivity of quercetin and its structure-related polyphenols to human serum albumin using a fluorescent dye cocktail for multiplex drug-site mapping
|
Mukai, Rie |
|
|
145 |
C |
p. |
artikel |
67 |
The first-in-class pyrazole-based dual InhA-VEGFR inhibitors towards integrated antitubercular host-directed therapy
|
Shaaban, Marwa M. |
|
|
145 |
C |
p. |
artikel |
68 |
Transmembrane modification of tumor vascular targeting peptide A7R as molecular cargo delivery tool
|
Zhang, Qingqing |
|
|
145 |
C |
p. |
artikel |
69 |
Triphenylphosphonium-linked derivative of hecogenin with enhanced antiproliferative activity: Design, synthesis, and biological evaluation
|
Zhang, Jinling |
|
|
145 |
C |
p. |
artikel |
70 |
Unleashing the potential of vanillic acid: A new twist on nature's recipe to fight inflammation and circumvent azole-resistant fungal infections
|
Khan, Farooq-Ahmad |
|
|
145 |
C |
p. |
artikel |
71 |
Utilizing microbial metabolite in catalytic cascade synthesis of conjugated oligomers for In-Situ regulation of biological activity
|
Li, Yuke |
|
|
145 |
C |
p. |
artikel |