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                             85 results found
no title author magazine year volume issue page(s) type
1 A bifunctional agent for efficient imaging of PD-L1 and antimelanoma activity Wang, Jin

141 C p.
article
2 Advances in non-radioactive PSMA-targeted small molecule-drug conjugates in the treatment of prostate cancer Chen, Min

141 C p.
article
3 Ag/g-C3N4 nanocomposite: Green fabrication and its application as a catalyst in the synthesis of new series of depsipeptides as biologically active compounds and investigation on their anti-breast cancer activity Shahi, Fatemeh

141 C p.
article
4 A near-infrared fluorescent probe with remarkably large stokes shift for specifical imaging of peroxynitrite fluctuations in Hela cells Lu, Zhengliang

141 C p.
article
5 A novel class of pyrazole analogues as aurora kinase A inhibitor: design, synthesis, and anticancer evaluation Yevale, Digambar B.

141 C p.
article
6 Antimicrobial peptides fight against Pseudomonas aeruginosa at a sub-inhibitory concentration via anti-QS pathway Li, Li

141 C p.
article
7 Artificial intelligence in small molecule drug discovery from 2018 to 2023: Does it really work? Lv, Qi

141 C p.
article
8 Backbone N-methylation of peptides: Advances in synthesis and applications in pharmaceutical drug development Li, Xuefei

141 C p.
article
9 Battling colorectal cancer via s-triazine-based MMP-10/13 inhibitors armed with electrophilic warheads for concomitant ferroptosis induction; the first-in-class dual-acting agents Morcos, Christine A.

141 C p.
article
10 13C NMR-based dereplication using MixONat software to decipher potent anti-cholinesterase compounds in Mesua lepidota bark Leong, Sow Tein

141 C p.
article
11 Combination of quinoxaline with pentamethinium system: Mitochondrial staining and targeting Kejík, Zdeněk

141 C p.
article
12 Conjugates of nucleobases with triazole-hydroxamic acids for the reactivation of acetylcholinesterase and treatment of delayed neurodegeneration induced by organophosphate poisoning Shulaeva, Marina M.

141 C p.
article
13 Conjugation with glucagon like peptide-1 enables targeted protein degradation Zhu, Liquan

141 C p.
article
14 Corrigendum to “Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT” [Bioorg. Chem. 139 (2023) 106676] Li, Peizhuo

141 C p.
article
15 Corrigendum to “Synthesis and evaluation of antibacterial activity of transition metal-oleoyl amide complexes” [Bioorganic Chem. 140 (2023) 106786] Farhan, Nesrain

141 C p.
article
16 Derivative of cinnamic acid inhibits T3SS of Xanthomonas oryzae pv. oryzae through the HrpG-HrpX regulatory cascade Shi, Yu

141 C p.
article
17 Design and synthesis of 9-phenanthranilamide derivatives and the study of anti-inflammatory, antioxidant and neuroprotective activities Du, Shuaishuai

141 C p.
article
18 Design and synthesis of photoaffinity-based probes for labeling β-glucuronidase Bi, Wen-Jing

141 C p.
article
19 Design, synthesis and anti-osteosarcoma activity study of novel pyrido[2,3-d]pyrimidine derivatives by inhibiting DKK1-Wnt/β-catenin pathway Shen, Yanni

141 C p.
article
20 Design, synthesis and biological evaluation of novel 2,4-diaminopyrimidine cinnamyl derivatives as inhibitors of FAK with potent anti-gastric cancer activities Liu, Yang

141 C p.
article
21 Design, synthesis, biological evaluation, and docking study of new triazole-phenylacetamide derivatives as α-glucosidase inhibitors Luo, Shuang

141 C p.
article
22 Design, synthesis, in vitro and in silico evaluation of novel substituted 1,2,4-triazole analogues as dual human VEGFR-2 and TB-InhA inhibitors Zawal, Amira G.

141 C p.
article
23 Dihydro-β-agarofuran-type sesquiterpenoids from the seeds of Tripterygium wilfordii (Thunder God Vine) and evaluation of their anti-osteoclastogenesis and immunosuppressive activities Cao, Guangchao

141 C p.
article
24 Discovery of a minimalistic DIE-based fluorescent probe for detection of parallel G-quadruplex forms Dong, Yun

141 C p.
article
25 Discovery of dolutegravir-1,2,3-triazole derivatives against prostate cancer via inducing DNA damage Zhou, Shuyi

141 C p.
article
26 Discovery of new DHA ethanolamine derivatives as potential anti-inflammatory agents targeting Nur77 Fang, Hua

141 C p.
article
27 Discovery of novel cannabidiol derivatives with augmented antibacterial agents against methicillin-resistant Staphylococcus aureus Zhang, Zhen

141 C p.
article
28 Discovery of novel 4,5-diphenyl-imidazol-α-aminophosphonate hybrids as promising anti-diabetic agents: Design, synthesis, in vitro, and in silico enzymatic studies Zareei, Samira

141 C p.
article
29 Discovery of novel TLR4/MD-2 inhibitors: Receptor structure-based virtual screening studies and anti-inflammatory evaluation Zhang, Tengyue

141 C p.
article
30 Discovery of selective and potent USP22 inhibitors via structure-based virtual screening and bioassays exerting anti-tumor activity Zhang, Yue

141 C p.
article
31 Discovery of (S)-flurbiprofen-based novel azine derivatives as prostaglandin endoperoxide synthase-II inhibitors: Synthesis, in-vivo analgesic, anti-inflammatory activities, and their molecular docking Alam, Aftab

141 C p.
article
32 Editorial Board
141 C p.
article
33 Expanding the synthesis of a library of potent glucuronic acid glycodendrons for Dengue virus inhibition Ramírez-López, Pedro

141 C p.
article
34 Exploration of the novel phthalimide-hydroxypyridinone derivatives as multifunctional drug candidates against Alzheimer’s disease Zhu, Xi

141 C p.
article
35 Fluoroalkoxylated C-3 and C-9 (S)-12-bromostepholidine analogues with D1R antagonist activity Namballa, Hari K.

141 C p.
article
36 γ-Glutamyltranspeptidase-Activated Near-Infrared fluorescent probe for visualization of Drug-Induced liver injury Liu, Feiyan

141 C p.
article
37 Historical perspectives and recent advances in small molecule ligands of selective/biased/multi-targeted μ/δ/κ opioid receptor (2019–2022) He, Ye

141 C p.
article
38 Indoloquinazoline alkaloids suppress angiogenesis and inhibit metastasis of melanoma cells Guo, Xingchen

141 C p.
article
39 In vitro and in vivo anticancer activity of novel Rh(III) and Pd(II) complexes with pyrazolopyrimidine derivatives Gu, Yun-Qiong

141 C p.
article
40 Iridium(III) complex induces apoptosis in HeLa cells by regulating mitochondrial and PI3K/AKT signaling pathways: In vitro and in vivo experiments He, Shu-fen

141 C p.
article
41 Issue TOC
141 C p.
article
42 Molecular engineering and bioimaging applications of C2-alkenyl indole dyes with tunable emission wavelengths covering visible to NIR light Liu, Yan

141 C p.
article
43 mRNA incorporation of C(5)-halogenated pyrimidine ribonucleotides and induced high expression of corresponding protein for the development of mRNA vaccine Dhurbachandra Singh, Chabungbam

141 C p.
article
44 New 2-alkoxycyanopyridine derivatives as inhibitors of EGFR, HER2, and DHFR: Synthesis, anticancer evaluation, and molecular modeling studies Hawas, Samia S.

141 C p.
article
45 New 2,4-dihydro-1H-1,2,4-triazole-3-selones and 3,3′-di(4H-1,2,4-triazolyl)diselenides. Synthesis, biological evaluation, and in silico studies as antibacterial and fungicidal agents oglu Askerov, Rizvan K.

141 C p.
article
46 New imidazole-2-ones and their 2-thione analogues as anticancer agents and CAIX inhibitors: Synthesis, in silico ADME and molecular modeling studies Ibrahim, Seham A.

141 C p.
article
47 New phenothiazine conjugates as apoptosis inducing agents: Design, synthesis, In-vitro anti-cancer screening and 131I-radiolabeling for in-vivo evaluation Sarhan, Mona O.

141 C p.
article
48 Novel phenolate salts of bioactive agents: Cannabidiol phenolate salts Guruprasad Reddy, Pulikanti

141 C p.
article
49 Novel spirooxindole alkaloid derivatives from the medicinal insect Blaps japanensis and their biological evaluation Yan, Yong-Ming

141 C p.
article
50 Oligomeric phloroglucinols with hAChE inhibitory and antibacterial activities from tropic Rhodomyrtus tomentosa Luo, E-E

141 C p.
article
51 Oxidation of anti-thyroid drugs and their selenium analogs by ABTS radical cation Frąckowiak-Wojtasek, Bożena

141 C p.
article
52 Peptide Nucleic Acids: Recent Developments in the Synthesis and Backbone Modifications Singh, Gurpreet

141 C p.
article
53 Peptidomimetics based on ammonium decasubstituted pillar[5]arenes: Influence of the alpha-amino acid residue nature on cholinesterase inhibition Nazarova, Anastasia

141 C p.
article
54 Phenolic chalcones as agents against Trichomonas vaginalis Oliveira, Lígia R.

141 C p.
article
55 4-Phenylcoumarin derivatives as new HIV-1 NNRTIs: Design, synthesis, biological activities, and computational studies Batran, Rasha Z.

141 C p.
article
56 Potential natural product 3,4-seco-schitriterpenoids from Kadsura japonica L. as anti-neuroinflammatory agents Liu, Shu-Hsiang

141 C p.
article
57 Probing naphthalene diimide and 3-hydroxypropylphosphate as end-conjugating moieties for improved thrombin binding aptamers: Structural and biological effects Riccardi, Claudia

141 C p.
article
58 Protecting-group free synthesis of glycoconjugates displaying dual fungicidal and plant defense-eliciting activities Noël, Nathan

141 C p.
article
59 Prunolactones A-G, proangiogenic isocoumarin derivatives with an unusual 6/6/6/6/6 spiropentacyclic skeleton from the endophytic fungus Phomopsis prunorum Zhang, Xue-Qing

141 C p.
article
60 Pyrimidine-5-carbonitrile derivatives as sprout for CQDs proveniences: Antitumor and anti-inflammatory potentiality Ahmed, Hanan B.

141 C p.
article
61 Pyrimidine-morpholine hybrids as potent druggable therapeutics for Alzheimer’s disease: Synthesis, biochemical and in silico analyses Zaib, Sumera

141 C p.
article
62 Radiosynthesis, preclinical evaluation and pilot clinical PET imaging study of a 18F-labeled tracer targeting fibroblast activation protein Fu, Lilan

141 C p.
article
63 Rational design of β-carboline as an efficient type I/II photosensitizer to enable hypoxia-tolerant chemo-photodynamic therapy Xu, Zhongyuan

141 C p.
article
64 Recent advances in targeting leucine-rich repeat kinase 2 as a potential strategy for the treatment of Parkinson’s disease Cao, Ruiwei

141 C p.
article
65 Repurposing of conformationally-restricted cyclopentane-based AKT–inhibitors leads to discovery of potential and more selective antileishmanial agents than miltefosine Hassan, Ahmed H.E.

141 C p.
article
66 Silver(I) complexes with amino acid and dipeptide ligands – Chemical and antimicrobial relevant comparison (mini review) Vargová, Zuzana

141 C p.
article
67 Small molecule tractable PARP inhibitors: Scaffold construction approaches, mechanistic insights and structure activity relationship Thakur, Amandeep

141 C p.
article
68 Structural diversity and biological activities of indole-diterpenoids from Penicillium janthinellum by co-culture with Paecilomyces formosus Cao, Fei

141 C p.
article
69 Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues Shaikh, Ashif Y.

141 C p.
article
70 Synthesis and biological evaluation of novel 3-(5-substituted-1H-indol-3-yl)pyrrolidine-2,5-dione derivatives with a dual affinity for serotonin 5-HT1A receptor and SERT Wróbel, Martyna Z.

141 C p.
article
71 Synthesis and chemical transformations of glycol nucleic acid (GNA) nucleosides Kowalski, Konrad

141 C p.
article
72 Synthesis and evaluation of highly potent HBV capsid assembly modulators (CAMs) Amblard, Franck

141 C p.
article
73 Synthesis and interaction with growth factors of sulfated oligosaccharides containing an anomeric fluorinated tail de Paz, José L.

141 C p.
article
74 Synthesis and structure-activity relationship studies of fusidic acid derivatives as anti-inflammatory agents for acute lung injury Huang, Xing

141 C p.
article
75 Synthesis by diastereomeric resolution, biochemical evaluation and molecular modelling of chiral 3-hydroxyl b-lactam microtubule-targeting agents for the treatment of triple negative breast and chemoresistant colorectal cancers McLoughlin, Eavan C.

141 C p.
article
76 Synthesis, characterization, biological activity, and in vitro digestion of selenium nanoparticles stabilized by Antarctic ice microalgae polypeptide Zeng, Lixia

141 C p.
article
77 Synthesis, characterization, in vitro antimycobacterial and cytotoxicity evaluation, DFT calculations, molecular docking and ADME studies of new isomeric benzimidazole-1,2,3-triazole-quinoline hybrid mixtures Nyoni, Nombulelo T.P.

141 C p.
article
78 Synthesis, docking studies and biological evaluation of 1H-1,2,3-triazole-7-chloroquinoline derivatives against SARS-CoV-2 Ng, Jerome P.L.

141 C p.
article
79 Synthesis, evaluation and molecular dynamics study of human toll-like receptor 2/6 specific monoacyl lipopeptides as candidate immunostimulants Zhu, Yueyue

141 C p.
article
80 Synthesis, molecular modeling Insights, and anticancer assessment of novel polyfunctionalized Pyridine congeners Abouelenein, Mohamed G.

141 C p.
article
81 Synthesis of 3-sulfenylindole derivatives from 4-hydroxy-2H-chromene-2-thione and indole using oxidative cross-dehydrogenative coupling reaction and anti-proliferative activity study of some of their sulfone derivatives Xalxo, Anjela

141 C p.
article
82 The active phthalate metabolite, DHEP, induces proliferation and metastasis of prostate cancer cells via upregulation of β-catenin and downregulation of KLF7 Li, Hecheng

141 C p.
article
83 Trypanocidal potential of synthetic p-aminochalcones: In silico and in vitro evaluation Dutra Barroso Gomes, Naiara

141 C p.
article
84 Two-dimensional chromatography for enantiomeric analysis of mitotane and its metabolite o,p′-DDA in patients with adrenocortical carcinoma indicates enantioselective metabolism Stadler, Gabriela

141 C p.
article
85 X-ray crystallography study and optimization of novel benzothiophene analogs as potent selective estrogen receptor covalent antagonists (SERCAs) with improved potency and safety profiles Bai, Chengfeng

141 C p.
article
                             85 results found
 
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