nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A bifunctional agent for efficient imaging of PD-L1 and antimelanoma activity
|
Wang, Jin |
|
|
141 |
C |
p. |
artikel |
2 |
Advances in non-radioactive PSMA-targeted small molecule-drug conjugates in the treatment of prostate cancer
|
Chen, Min |
|
|
141 |
C |
p. |
artikel |
3 |
Ag/g-C3N4 nanocomposite: Green fabrication and its application as a catalyst in the synthesis of new series of depsipeptides as biologically active compounds and investigation on their anti-breast cancer activity
|
Shahi, Fatemeh |
|
|
141 |
C |
p. |
artikel |
4 |
A near-infrared fluorescent probe with remarkably large stokes shift for specifical imaging of peroxynitrite fluctuations in Hela cells
|
Lu, Zhengliang |
|
|
141 |
C |
p. |
artikel |
5 |
A novel class of pyrazole analogues as aurora kinase A inhibitor: design, synthesis, and anticancer evaluation
|
Yevale, Digambar B. |
|
|
141 |
C |
p. |
artikel |
6 |
Antimicrobial peptides fight against Pseudomonas aeruginosa at a sub-inhibitory concentration via anti-QS pathway
|
Li, Li |
|
|
141 |
C |
p. |
artikel |
7 |
Artificial intelligence in small molecule drug discovery from 2018 to 2023: Does it really work?
|
Lv, Qi |
|
|
141 |
C |
p. |
artikel |
8 |
Backbone N-methylation of peptides: Advances in synthesis and applications in pharmaceutical drug development
|
Li, Xuefei |
|
|
141 |
C |
p. |
artikel |
9 |
Battling colorectal cancer via s-triazine-based MMP-10/13 inhibitors armed with electrophilic warheads for concomitant ferroptosis induction; the first-in-class dual-acting agents
|
Morcos, Christine A. |
|
|
141 |
C |
p. |
artikel |
10 |
13C NMR-based dereplication using MixONat software to decipher potent anti-cholinesterase compounds in Mesua lepidota bark
|
Leong, Sow Tein |
|
|
141 |
C |
p. |
artikel |
11 |
Combination of quinoxaline with pentamethinium system: Mitochondrial staining and targeting
|
Kejík, Zdeněk |
|
|
141 |
C |
p. |
artikel |
12 |
Conjugates of nucleobases with triazole-hydroxamic acids for the reactivation of acetylcholinesterase and treatment of delayed neurodegeneration induced by organophosphate poisoning
|
Shulaeva, Marina M. |
|
|
141 |
C |
p. |
artikel |
13 |
Conjugation with glucagon like peptide-1 enables targeted protein degradation
|
Zhu, Liquan |
|
|
141 |
C |
p. |
artikel |
14 |
Corrigendum to “Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT” [Bioorg. Chem. 139 (2023) 106676]
|
Li, Peizhuo |
|
|
141 |
C |
p. |
artikel |
15 |
Corrigendum to “Synthesis and evaluation of antibacterial activity of transition metal-oleoyl amide complexes” [Bioorganic Chem. 140 (2023) 106786]
|
Farhan, Nesrain |
|
|
141 |
C |
p. |
artikel |
16 |
Derivative of cinnamic acid inhibits T3SS of Xanthomonas oryzae pv. oryzae through the HrpG-HrpX regulatory cascade
|
Shi, Yu |
|
|
141 |
C |
p. |
artikel |
17 |
Design and synthesis of 9-phenanthranilamide derivatives and the study of anti-inflammatory, antioxidant and neuroprotective activities
|
Du, Shuaishuai |
|
|
141 |
C |
p. |
artikel |
18 |
Design and synthesis of photoaffinity-based probes for labeling β-glucuronidase
|
Bi, Wen-Jing |
|
|
141 |
C |
p. |
artikel |
19 |
Design, synthesis and anti-osteosarcoma activity study of novel pyrido[2,3-d]pyrimidine derivatives by inhibiting DKK1-Wnt/β-catenin pathway
|
Shen, Yanni |
|
|
141 |
C |
p. |
artikel |
20 |
Design, synthesis and biological evaluation of novel 2,4-diaminopyrimidine cinnamyl derivatives as inhibitors of FAK with potent anti-gastric cancer activities
|
Liu, Yang |
|
|
141 |
C |
p. |
artikel |
21 |
Design, synthesis, biological evaluation, and docking study of new triazole-phenylacetamide derivatives as α-glucosidase inhibitors
|
Luo, Shuang |
|
|
141 |
C |
p. |
artikel |
22 |
Design, synthesis, in vitro and in silico evaluation of novel substituted 1,2,4-triazole analogues as dual human VEGFR-2 and TB-InhA inhibitors
|
Zawal, Amira G. |
|
|
141 |
C |
p. |
artikel |
23 |
Dihydro-β-agarofuran-type sesquiterpenoids from the seeds of Tripterygium wilfordii (Thunder God Vine) and evaluation of their anti-osteoclastogenesis and immunosuppressive activities
|
Cao, Guangchao |
|
|
141 |
C |
p. |
artikel |
24 |
Discovery of a minimalistic DIE-based fluorescent probe for detection of parallel G-quadruplex forms
|
Dong, Yun |
|
|
141 |
C |
p. |
artikel |
25 |
Discovery of dolutegravir-1,2,3-triazole derivatives against prostate cancer via inducing DNA damage
|
Zhou, Shuyi |
|
|
141 |
C |
p. |
artikel |
26 |
Discovery of new DHA ethanolamine derivatives as potential anti-inflammatory agents targeting Nur77
|
Fang, Hua |
|
|
141 |
C |
p. |
artikel |
27 |
Discovery of novel cannabidiol derivatives with augmented antibacterial agents against methicillin-resistant Staphylococcus aureus
|
Zhang, Zhen |
|
|
141 |
C |
p. |
artikel |
28 |
Discovery of novel 4,5-diphenyl-imidazol-α-aminophosphonate hybrids as promising anti-diabetic agents: Design, synthesis, in vitro, and in silico enzymatic studies
|
Zareei, Samira |
|
|
141 |
C |
p. |
artikel |
29 |
Discovery of novel TLR4/MD-2 inhibitors: Receptor structure-based virtual screening studies and anti-inflammatory evaluation
|
Zhang, Tengyue |
|
|
141 |
C |
p. |
artikel |
30 |
Discovery of selective and potent USP22 inhibitors via structure-based virtual screening and bioassays exerting anti-tumor activity
|
Zhang, Yue |
|
|
141 |
C |
p. |
artikel |
31 |
Discovery of (S)-flurbiprofen-based novel azine derivatives as prostaglandin endoperoxide synthase-II inhibitors: Synthesis, in-vivo analgesic, anti-inflammatory activities, and their molecular docking
|
Alam, Aftab |
|
|
141 |
C |
p. |
artikel |
32 |
Editorial Board
|
|
|
|
141 |
C |
p. |
artikel |
33 |
Expanding the synthesis of a library of potent glucuronic acid glycodendrons for Dengue virus inhibition
|
Ramírez-López, Pedro |
|
|
141 |
C |
p. |
artikel |
34 |
Exploration of the novel phthalimide-hydroxypyridinone derivatives as multifunctional drug candidates against Alzheimer’s disease
|
Zhu, Xi |
|
|
141 |
C |
p. |
artikel |
35 |
Fluoroalkoxylated C-3 and C-9 (S)-12-bromostepholidine analogues with D1R antagonist activity
|
Namballa, Hari K. |
|
|
141 |
C |
p. |
artikel |
36 |
γ-Glutamyltranspeptidase-Activated Near-Infrared fluorescent probe for visualization of Drug-Induced liver injury
|
Liu, Feiyan |
|
|
141 |
C |
p. |
artikel |
37 |
Historical perspectives and recent advances in small molecule ligands of selective/biased/multi-targeted μ/δ/κ opioid receptor (2019–2022)
|
He, Ye |
|
|
141 |
C |
p. |
artikel |
38 |
Indoloquinazoline alkaloids suppress angiogenesis and inhibit metastasis of melanoma cells
|
Guo, Xingchen |
|
|
141 |
C |
p. |
artikel |
39 |
In vitro and in vivo anticancer activity of novel Rh(III) and Pd(II) complexes with pyrazolopyrimidine derivatives
|
Gu, Yun-Qiong |
|
|
141 |
C |
p. |
artikel |
40 |
Iridium(III) complex induces apoptosis in HeLa cells by regulating mitochondrial and PI3K/AKT signaling pathways: In vitro and in vivo experiments
|
He, Shu-fen |
|
|
141 |
C |
p. |
artikel |
41 |
Issue TOC
|
|
|
|
141 |
C |
p. |
artikel |
42 |
Molecular engineering and bioimaging applications of C2-alkenyl indole dyes with tunable emission wavelengths covering visible to NIR light
|
Liu, Yan |
|
|
141 |
C |
p. |
artikel |
43 |
mRNA incorporation of C(5)-halogenated pyrimidine ribonucleotides and induced high expression of corresponding protein for the development of mRNA vaccine
|
Dhurbachandra Singh, Chabungbam |
|
|
141 |
C |
p. |
artikel |
44 |
New 2-alkoxycyanopyridine derivatives as inhibitors of EGFR, HER2, and DHFR: Synthesis, anticancer evaluation, and molecular modeling studies
|
Hawas, Samia S. |
|
|
141 |
C |
p. |
artikel |
45 |
New 2,4-dihydro-1H-1,2,4-triazole-3-selones and 3,3′-di(4H-1,2,4-triazolyl)diselenides. Synthesis, biological evaluation, and in silico studies as antibacterial and fungicidal agents
|
oglu Askerov, Rizvan K. |
|
|
141 |
C |
p. |
artikel |
46 |
New imidazole-2-ones and their 2-thione analogues as anticancer agents and CAIX inhibitors: Synthesis, in silico ADME and molecular modeling studies
|
Ibrahim, Seham A. |
|
|
141 |
C |
p. |
artikel |
47 |
New phenothiazine conjugates as apoptosis inducing agents: Design, synthesis, In-vitro anti-cancer screening and 131I-radiolabeling for in-vivo evaluation
|
Sarhan, Mona O. |
|
|
141 |
C |
p. |
artikel |
48 |
Novel phenolate salts of bioactive agents: Cannabidiol phenolate salts
|
Guruprasad Reddy, Pulikanti |
|
|
141 |
C |
p. |
artikel |
49 |
Novel spirooxindole alkaloid derivatives from the medicinal insect Blaps japanensis and their biological evaluation
|
Yan, Yong-Ming |
|
|
141 |
C |
p. |
artikel |
50 |
Oligomeric phloroglucinols with hAChE inhibitory and antibacterial activities from tropic Rhodomyrtus tomentosa
|
Luo, E-E |
|
|
141 |
C |
p. |
artikel |
51 |
Oxidation of anti-thyroid drugs and their selenium analogs by ABTS radical cation
|
Frąckowiak-Wojtasek, Bożena |
|
|
141 |
C |
p. |
artikel |
52 |
Peptide Nucleic Acids: Recent Developments in the Synthesis and Backbone Modifications
|
Singh, Gurpreet |
|
|
141 |
C |
p. |
artikel |
53 |
Peptidomimetics based on ammonium decasubstituted pillar[5]arenes: Influence of the alpha-amino acid residue nature on cholinesterase inhibition
|
Nazarova, Anastasia |
|
|
141 |
C |
p. |
artikel |
54 |
Phenolic chalcones as agents against Trichomonas vaginalis
|
Oliveira, Lígia R. |
|
|
141 |
C |
p. |
artikel |
55 |
4-Phenylcoumarin derivatives as new HIV-1 NNRTIs: Design, synthesis, biological activities, and computational studies
|
Batran, Rasha Z. |
|
|
141 |
C |
p. |
artikel |
56 |
Potential natural product 3,4-seco-schitriterpenoids from Kadsura japonica L. as anti-neuroinflammatory agents
|
Liu, Shu-Hsiang |
|
|
141 |
C |
p. |
artikel |
57 |
Probing naphthalene diimide and 3-hydroxypropylphosphate as end-conjugating moieties for improved thrombin binding aptamers: Structural and biological effects
|
Riccardi, Claudia |
|
|
141 |
C |
p. |
artikel |
58 |
Protecting-group free synthesis of glycoconjugates displaying dual fungicidal and plant defense-eliciting activities
|
Noël, Nathan |
|
|
141 |
C |
p. |
artikel |
59 |
Prunolactones A-G, proangiogenic isocoumarin derivatives with an unusual 6/6/6/6/6 spiropentacyclic skeleton from the endophytic fungus Phomopsis prunorum
|
Zhang, Xue-Qing |
|
|
141 |
C |
p. |
artikel |
60 |
Pyrimidine-5-carbonitrile derivatives as sprout for CQDs proveniences: Antitumor and anti-inflammatory potentiality
|
Ahmed, Hanan B. |
|
|
141 |
C |
p. |
artikel |
61 |
Pyrimidine-morpholine hybrids as potent druggable therapeutics for Alzheimer’s disease: Synthesis, biochemical and in silico analyses
|
Zaib, Sumera |
|
|
141 |
C |
p. |
artikel |
62 |
Radiosynthesis, preclinical evaluation and pilot clinical PET imaging study of a 18F-labeled tracer targeting fibroblast activation protein
|
Fu, Lilan |
|
|
141 |
C |
p. |
artikel |
63 |
Rational design of β-carboline as an efficient type I/II photosensitizer to enable hypoxia-tolerant chemo-photodynamic therapy
|
Xu, Zhongyuan |
|
|
141 |
C |
p. |
artikel |
64 |
Recent advances in targeting leucine-rich repeat kinase 2 as a potential strategy for the treatment of Parkinson’s disease
|
Cao, Ruiwei |
|
|
141 |
C |
p. |
artikel |
65 |
Repurposing of conformationally-restricted cyclopentane-based AKT–inhibitors leads to discovery of potential and more selective antileishmanial agents than miltefosine
|
Hassan, Ahmed H.E. |
|
|
141 |
C |
p. |
artikel |
66 |
Silver(I) complexes with amino acid and dipeptide ligands – Chemical and antimicrobial relevant comparison (mini review)
|
Vargová, Zuzana |
|
|
141 |
C |
p. |
artikel |
67 |
Small molecule tractable PARP inhibitors: Scaffold construction approaches, mechanistic insights and structure activity relationship
|
Thakur, Amandeep |
|
|
141 |
C |
p. |
artikel |
68 |
Structural diversity and biological activities of indole-diterpenoids from Penicillium janthinellum by co-culture with Paecilomyces formosus
|
Cao, Fei |
|
|
141 |
C |
p. |
artikel |
69 |
Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues
|
Shaikh, Ashif Y. |
|
|
141 |
C |
p. |
artikel |
70 |
Synthesis and biological evaluation of novel 3-(5-substituted-1H-indol-3-yl)pyrrolidine-2,5-dione derivatives with a dual affinity for serotonin 5-HT1A receptor and SERT
|
Wróbel, Martyna Z. |
|
|
141 |
C |
p. |
artikel |
71 |
Synthesis and chemical transformations of glycol nucleic acid (GNA) nucleosides
|
Kowalski, Konrad |
|
|
141 |
C |
p. |
artikel |
72 |
Synthesis and evaluation of highly potent HBV capsid assembly modulators (CAMs)
|
Amblard, Franck |
|
|
141 |
C |
p. |
artikel |
73 |
Synthesis and interaction with growth factors of sulfated oligosaccharides containing an anomeric fluorinated tail
|
de Paz, José L. |
|
|
141 |
C |
p. |
artikel |
74 |
Synthesis and structure-activity relationship studies of fusidic acid derivatives as anti-inflammatory agents for acute lung injury
|
Huang, Xing |
|
|
141 |
C |
p. |
artikel |
75 |
Synthesis by diastereomeric resolution, biochemical evaluation and molecular modelling of chiral 3-hydroxyl b-lactam microtubule-targeting agents for the treatment of triple negative breast and chemoresistant colorectal cancers
|
McLoughlin, Eavan C. |
|
|
141 |
C |
p. |
artikel |
76 |
Synthesis, characterization, biological activity, and in vitro digestion of selenium nanoparticles stabilized by Antarctic ice microalgae polypeptide
|
Zeng, Lixia |
|
|
141 |
C |
p. |
artikel |
77 |
Synthesis, characterization, in vitro antimycobacterial and cytotoxicity evaluation, DFT calculations, molecular docking and ADME studies of new isomeric benzimidazole-1,2,3-triazole-quinoline hybrid mixtures
|
Nyoni, Nombulelo T.P. |
|
|
141 |
C |
p. |
artikel |
78 |
Synthesis, docking studies and biological evaluation of 1H-1,2,3-triazole-7-chloroquinoline derivatives against SARS-CoV-2
|
Ng, Jerome P.L. |
|
|
141 |
C |
p. |
artikel |
79 |
Synthesis, evaluation and molecular dynamics study of human toll-like receptor 2/6 specific monoacyl lipopeptides as candidate immunostimulants
|
Zhu, Yueyue |
|
|
141 |
C |
p. |
artikel |
80 |
Synthesis, molecular modeling Insights, and anticancer assessment of novel polyfunctionalized Pyridine congeners
|
Abouelenein, Mohamed G. |
|
|
141 |
C |
p. |
artikel |
81 |
Synthesis of 3-sulfenylindole derivatives from 4-hydroxy-2H-chromene-2-thione and indole using oxidative cross-dehydrogenative coupling reaction and anti-proliferative activity study of some of their sulfone derivatives
|
Xalxo, Anjela |
|
|
141 |
C |
p. |
artikel |
82 |
The active phthalate metabolite, DHEP, induces proliferation and metastasis of prostate cancer cells via upregulation of β-catenin and downregulation of KLF7
|
Li, Hecheng |
|
|
141 |
C |
p. |
artikel |
83 |
Trypanocidal potential of synthetic p-aminochalcones: In silico and in vitro evaluation
|
Dutra Barroso Gomes, Naiara |
|
|
141 |
C |
p. |
artikel |
84 |
Two-dimensional chromatography for enantiomeric analysis of mitotane and its metabolite o,p′-DDA in patients with adrenocortical carcinoma indicates enantioselective metabolism
|
Stadler, Gabriela |
|
|
141 |
C |
p. |
artikel |
85 |
X-ray crystallography study and optimization of novel benzothiophene analogs as potent selective estrogen receptor covalent antagonists (SERCAs) with improved potency and safety profiles
|
Bai, Chengfeng |
|
|
141 |
C |
p. |
artikel |