| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A cathepsin B/GSH dual-responsive fluorinated peptide for effective siRNA delivery to cancer cells
|
Shi, Zhen
|
|
|
135 |
C |
p.
|
artikel
|
| 2 |
2-Aminobenzothiazoles in anticancer drug design and discovery
|
Huang, Guang
|
|
|
135 |
C |
p.
|
artikel
|
| 3 |
Antitumor activity and mechanisms of dual EGFR/DNA-targeting strategy for the treatment of lung cancer with EGFRL858R/T790M mutation
|
Dai, Lumei
|
|
|
135 |
C |
p.
|
artikel
|
| 4 |
Anti-tyrosinase flavone derivatives and their anti-melanogenic activities: Importance of the β-phenyl-α,β-unsaturated carbonyl scaffold
|
Lee, Jieun
|
|
|
135 |
C |
p.
|
artikel
|
| 5 |
Arylidine extensions of 3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-benzenesulfonamide derivatives: Synthesis, computational simulations and biological evaluation as tumor-associated carbonic anhydrase inhibitors
|
Metwally, Heba M.
|
|
|
135 |
C |
p.
|
artikel
|
| 6 |
A simple ratiometric fluorescent probe for two-photon imaging of carbon monoxide in living cells and zebrafish
|
Tang, Junshuai
|
|
|
135 |
C |
p.
|
artikel
|
| 7 |
B13, a well-tolerated inhibitor of hedgehog pathway, exhibited potent anti-tumor effects against colorectal carcinoma in vitro and in vivo
|
Wu, Huanxian
|
|
|
135 |
C |
p.
|
artikel
|
| 8 |
Cytotoxic C-20 non-oxygenated ent-kaurane diterpenoids from Isodon wardii
|
Tan, Qian
|
|
|
135 |
C |
p.
|
artikel
|
| 9 |
Design, synthesis, and biological evaluation of 6-(imidazo[1,2-a] pyridin-6-yl) quinazolin-4(3H)-one derivatives as potent anticancer agents by dual targeting Aurora kinase and ROR1
|
Fan, Yanhua
|
|
|
135 |
C |
p.
|
artikel
|
| 10 |
Design, synthesis, and biological evaluation of phenylurea indole derivatives as ABCG2 inhibitors
|
Ye, Gao-Jie
|
|
|
135 |
C |
p.
|
artikel
|
| 11 |
Design, synthesis, antiviral and fungicidal activities of novel polycarpine simplified analogues
|
Yan, Lili
|
|
|
135 |
C |
p.
|
artikel
|
| 12 |
Design, synthesis, characterization, crystal structure, in silico studies, and inhibitory properties of the PEPPSI type Pd(II)NHC complexes bearing chloro/fluorobenzyl group
|
Gök, Yetkin
|
|
|
135 |
C |
p.
|
artikel
|
| 13 |
Deuterated driven new chemical entities: An optimistic way to improve therapeutic efficacy
|
Chandra Mouli, H.M.
|
|
|
135 |
C |
p.
|
artikel
|
| 14 |
Development of certain aminoquinazoline scaffolds as potential multitarget anticancer agents with apoptotic and anti-proliferative effects: Design, synthesis and biological evaluation
|
Amin, Noha H.
|
|
|
135 |
C |
p.
|
artikel
|
| 15 |
Dianthrone derivatives from Polygonum multiflorum Thunb: Anti-diabetic activity, structure-activity relationships (SARs), and mode of action
|
Yang, Jian-Bo
|
|
|
135 |
C |
p.
|
artikel
|
| 16 |
Discovery of blood–brain barrier permeant amine-functionalized aurones as inhibitors of activated microglia
|
Chia, Shi Yi
|
|
|
135 |
C |
p.
|
artikel
|
| 17 |
Discovery of ergosterol derivative from Aspergillus sp. TJ507 that protects against hepatic ischemia/reperfusion injury
|
Hu, Hong
|
|
|
135 |
C |
p.
|
artikel
|
| 18 |
Discovery of novel (E)-1-methyl-9-(3-methylbenzylidene)-6,7,8,9-tetrahydropyrazolo[3,4-d]pyrido[1,2-a]pyrimidin-4(1H)-one as DDR2 kinase inhibitor: Synthesis, molecular docking, and anticancer properties
|
Ruzi, Zukela
|
|
|
135 |
C |
p.
|
artikel
|
| 19 |
Discovery of novel protein degraders based on bioorthogonal reaction-driven intracellular self-assembly strategy
|
Si, Ru
|
|
|
135 |
C |
p.
|
artikel
|
| 20 |
Editorial Board
|
|
|
|
135 |
C |
p.
|
artikel
|
| 21 |
Exploration of novel dihydroquinoxalinone derivatives as EGFRL858R/T790M tyrosine kinase inhibitors for the treatment of non-small-cell lung cancer
|
Cao, Yu
|
|
|
135 |
C |
p.
|
artikel
|
| 22 |
Ginsenoside Rh4 inhibits breast cancer growth through targeting histone deacetylase 2 to regulate immune microenvironment and apoptosis
|
Dong, Fangming
|
|
|
135 |
C |
p.
|
artikel
|
| 23 |
Green and efficient one-pot three-component synthesis of novel drug-like furo[2,3-d]pyrimidines as potential active site inhibitors and putative allosteric hotspots modulators of both SARS-CoV-2 MPro and PLPro
|
Mousavi, Hossein
|
|
|
135 |
C |
p.
|
artikel
|
| 24 |
H2S-activated fluorescent probe enables dual-channel fluorescence tracking of drug release in tumor cells
|
Liu, Caiyun
|
|
|
135 |
C |
p.
|
artikel
|
| 25 |
Indoloquinazoline alkaloids with cardiomyocyte protective activity against cold ischemic injury from Aspergillus clavatonanicus
|
Jin, Xiaoqi
|
|
|
135 |
C |
p.
|
artikel
|
| 26 |
Interaction of ruthenium(Ⅱ) polypyridyl complexes [Ru(phen)2(L)]2+ (L = PIP, p-HPIP and m-HPIP) with RNA poly(A)•poly(U): Each complex unexpectedly exhibiting a destabilizing effect on RNA
|
Peng, Xing
|
|
|
135 |
C |
p.
|
artikel
|
| 27 |
Issue TOC
|
|
|
|
135 |
C |
p.
|
artikel
|
| 28 |
New ε-N-thioglutaryl-lysine derivatives as SIRT5 inhibitors: Chemical synthesis, kinetic and crystallographic studies
|
Deng, Ji
|
|
|
135 |
C |
p.
|
artikel
|
| 29 |
Novel 4-Amino-Quinazoline moieties ligated Platinum(IV) prodrugs overcome cisplatin resistance in EGFRWT human lung cancer
|
Li, Rui
|
|
|
135 |
C |
p.
|
artikel
|
| 30 |
Nucleus-targeted delivery of nitric oxide in human mesenchymal stem cells enhances osteogenic differentiation
|
Cho, Du-Hyong
|
|
|
135 |
C |
p.
|
artikel
|
| 31 |
Rational design, synthesis and biological evaluation of benzo[d]isoxazole derivatives as potent BET bivalent inhibitors for potential treatment of prostate cancer
|
Li, Junhua
|
|
|
135 |
C |
p.
|
artikel
|
| 32 |
Recent advances and future perspectives of noncompetitive proteasome inhibitors
|
Zeng, Gongruixue
|
|
|
135 |
C |
p.
|
artikel
|
| 33 |
SOS1-inspired hydrocarbon-stapled peptide as a pan-Ras inhibitor
|
Li, Anpeng
|
|
|
135 |
C |
p.
|
artikel
|
| 34 |
Structurally modified Cyclovirobuxine-D Buxus alkaloids as effective analgesic agents through Cav3.2 T-Type calcium channel inhibition
|
Munikishore, Rachakunta
|
|
|
135 |
C |
p.
|
artikel
|
| 35 |
Structure optimization of an F-indole-chalcone (FC116) on 4-methoxyphenyl group and therapeutic potential against colorectal cancers with low cytotoxicity
|
Du, Bolin
|
|
|
135 |
C |
p.
|
artikel
|
| 36 |
Synthesis and anti-SARS-CoV-2 evaluation of lipid prodrugs of β-D-N 4-hydroxycytidine (NHC) and a 3′-fluoro-substituted analogue of NHC
|
Wen, Zhao-Hui
|
|
|
135 |
C |
p.
|
artikel
|
| 37 |
Synthesis and biological evaluation of 1-phenyl-4,6-dihydrobenzo[b]pyrazolo[3,4-d]azepin-5(1H)-one/thiones as anticancer agents
|
Parupalli, Ramulu
|
|
|
135 |
C |
p.
|
artikel
|
| 38 |
Synthesis and evaluation of 99mTc-labeled 1-(2-Pyridyl)piperazine derivatives as radioligands for 5HT7 receptors
|
karimi, Maryam
|
|
|
135 |
C |
p.
|
artikel
|
| 39 |
Synthesis and structure–activity relationships of ticlopidine derivatives and analogs as inhibitors of ectonucleotidase CD39
|
Bi, Chunyang
|
|
|
135 |
C |
p.
|
artikel
|
| 40 |
Synthesis, DFT study, theoretical and experimental spectroscopy of fatty amides based on extra-virgin olive oil and their antibacterial activity
|
Farhan, Nesrain
|
|
|
135 |
C |
p.
|
artikel
|
| 41 |
Synthesis of novel oxazol-5-one derivatives containing chiral trifluoromethyl and isoxazole moieties as potent antitumor agents and the mechanism investigation
|
Wang, Mengqi
|
|
|
135 |
C |
p.
|
artikel
|
| 42 |
Synthesis of structurally diverse derivatives of aconitine-type diterpenoid alkaloids and their anti-proliferative effects on canine breast cancer cells
|
Zhang, Li
|
|
|
135 |
C |
p.
|
artikel
|
| 43 |
Targeting HER2-receptors with 177Lu-labeled triazole stapled cyclic peptidomimetic
|
Kumar Sharma, Amit
|
|
|
135 |
C |
p.
|
artikel
|
| 44 |
Towards the Development of Dual Hypouricemic and Anti-inflammatory Candidates: Design, Synthesis, Stability Studies and Biological Evaluation of Some Mutual Ester Prodrugs of Febuxostat-NSAIDs
|
Rashad, Aya Y.
|
|
|
135 |
C |
p.
|
artikel
|
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