| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
2-Aminopyrimidine derivatives as selective dual inhibitors of JAK2 and FLT3 for the treatment of acute myeloid leukemia
|
Xu, Sicong
|
|
|
134 |
C |
p.
|
artikel
|
| 2 |
An ultrasensitive GSH-specific fluorescent probe unveils celastrol-induced ccRCC ferroptosis
|
Li, Hongfang
|
|
|
134 |
C |
p.
|
artikel
|
| 3 |
A win-win scenario for antibacterial activity and skin mildness of cationic surfactants based on the modulation of host-guest supramolecular conformation
|
Wang, Xuejiao
|
|
|
134 |
C |
p.
|
artikel
|
| 4 |
Benzoxazole-appended piperidine derivatives as novel anticancer candidates against breast cancer
|
AboulWafa, Omaima M.
|
|
|
134 |
C |
p.
|
artikel
|
| 5 |
Chemical constituents isolated from Actinidia polygama and their α-glucosidase inhibitory activity and insulin secretion effect
|
Hwang, Hoseong
|
|
|
134 |
C |
p.
|
artikel
|
| 6 |
Chemoproteomics reveals arctigenin as a phagophore-closure blocker via targeting ESCRT-I subunit VPS28
|
Han, Jinyan
|
|
|
134 |
C |
p.
|
artikel
|
| 7 |
Design and synthesis of novel N-terminal peptides of integrin and aminopeptidase are new finding for anticancer activity
|
Krishnamoorthy, Rajavenkatesh
|
|
|
134 |
C |
p.
|
artikel
|
| 8 |
Design, synthesis and bioactivity evaluation of self-assembled PROTACs based on multi-target kinase inhibitors
|
Si, Ru
|
|
|
134 |
C |
p.
|
artikel
|
| 9 |
Design, synthesis and bioevaluation of 1,2,4-thiadiazolidine-3,5-dione derivatives as potential GSK-3β inhibitors for the treatment of Alzheimer's disease
|
Dong, Yongxi
|
|
|
134 |
C |
p.
|
artikel
|
| 10 |
Design, synthesis, and evaluation of N-methyl-propargylamine derivates as isoform-selective monoamine oxidases inhibitors for the treatment of nervous system diseases
|
Zhang, Kaicheng
|
|
|
134 |
C |
p.
|
artikel
|
| 11 |
Design, synthesis and pharmacological characterization of aminopyrimidine derivatives as BTK/FLT3 dual-target inhibitors against acute myeloid leukemia
|
Ran, Fansheng
|
|
|
134 |
C |
p.
|
artikel
|
| 12 |
Design, synthesis, antimicrobial screening and molecular modeling of novel 6,7 dimethylquinoxalin-2(1H)-one and thiazole derivatives targeting DNA gyrase enzyme
|
Alqurashi, Raghad M.
|
|
|
134 |
C |
p.
|
artikel
|
| 13 |
Design, synthesis, cytotoxic activities, and molecular docking of chalcone hybrids bearing 8-hydroxyquinoline moiety with dual tubulin/EGFR kinase inhibition
|
Amin, Mohammed M.
|
|
|
134 |
C |
p.
|
artikel
|
| 14 |
Design, synthesis, modeling studies and biological evaluation of pyrazole derivatives linked to oxime and nitrate moieties as nitric oxide donor selective COX-2 and aromatase inhibitors with dual anti-inflammatory and anti-neoplastic activities
|
A. A. Fadaly, Wael
|
|
|
134 |
C |
p.
|
artikel
|
| 15 |
Discovery of endosomalytic cell-penetrating peptides based on bacterial membrane-targeting sequences
|
An, Chuanjing
|
|
|
134 |
C |
p.
|
artikel
|
| 16 |
Discovery of new small molecule inhibitors of the BPTF bromodomain
|
Liang, Xiaochen
|
|
|
134 |
C |
p.
|
artikel
|
| 17 |
Editorial Board
|
|
|
|
134 |
C |
p.
|
artikel
|
| 18 |
Efficient synthesis and anticancer evaluation of spider toxin peptide LVTX-8-based analogues with enhanced stability
|
Chi, Qiao-Na
|
|
|
134 |
C |
p.
|
artikel
|
| 19 |
Engineered aldoxime dehydratase to enable the chemoenzymatic conversion of benzyl amines to aromatic nitriles
|
Xiao, Qinjie
|
|
|
134 |
C |
p.
|
artikel
|
| 20 |
Evaluation of honokiol, magnolol and of a library of new nitrogenated neolignans as pancreatic lipase inhibitors
|
Sciacca, Claudia
|
|
|
134 |
C |
p.
|
artikel
|
| 21 |
Exploring chromone sulfonamides and sulfonylhydrazones as highly selective ectonucleotidase inhibitors: Synthesis, biological evaluation and in silico study
|
Younus, Hafiza Amna
|
|
|
134 |
C |
p.
|
artikel
|
| 22 |
Fusion of Michael-acceptors enhances the anti-inflammatory activity of ginsenosides as potential modulators of the NLRP3 signaling pathway
|
Yang, Gangqiang
|
|
|
134 |
C |
p.
|
artikel
|
| 23 |
Hypoglycemic oligostilbenes from the stems of Caragana sinica
|
Sun, Xing-Yan
|
|
|
134 |
C |
p.
|
artikel
|
| 24 |
Immunosuppressive diarylpropane dimer and spirocyclic-monomers from Horsfieldia kingii
|
Wang, Chao-Fan
|
|
|
134 |
C |
p.
|
artikel
|
| 25 |
Introduction of a β-leucine residue instead of leucine9 and glycine10 residues in Temporin L for improved cell selectivity, stability and activity against planktonic and biofilm of methicillin resistant S. aureus
|
Verma, Neeraj Kumar
|
|
|
134 |
C |
p.
|
artikel
|
| 26 |
Issue TOC
|
|
|
|
134 |
C |
p.
|
artikel
|
| 27 |
New chromones from the roots of Saposhnikovia divaricata (Turcz.) Schischk with anti-inflammatory activity
|
Sun, Yan
|
|
|
134 |
C |
p.
|
artikel
|
| 28 |
Novel lignans from Zanthoxylum nitidum and antiproliferation activity of sesaminone in osimertinib-resistant non-small cell lung cancer cells
|
Wang, Cai Yi
|
|
|
134 |
C |
p.
|
artikel
|
| 29 |
Novel NQO1 substrates bearing two nitrogen redox centers: Design, synthesis, molecular dynamics simulations, and antitumor evaluation
|
Gong, Qijie
|
|
|
134 |
C |
p.
|
artikel
|
| 30 |
Oxazolo[5,4-f]quinoxaline-type selective inhibitors of glycogen synthase kinase-3α (GSK-3α): Development and impact on temozolomide treatment of glioblastoma cells
|
Hasyeoui, Mohamed
|
|
|
134 |
C |
p.
|
artikel
|
| 31 |
Phenyldivinylsulfonamides for the construction of antibody–drug conjugates with controlled four payloads
|
Wei, Ding
|
|
|
134 |
C |
p.
|
artikel
|
| 32 |
Rapid discovery and crystallography study of highly potent and selective butylcholinesterase inhibitors based on oxime-containing libraries and conformational restriction strategies
|
Jing, Lanlan
|
|
|
134 |
C |
p.
|
artikel
|
| 33 |
Recent advances of LSD1/KDM1A inhibitors for disease therapy
|
Zhang, Chaofeng
|
|
|
134 |
C |
p.
|
artikel
|
| 34 |
SAR-guided development of indole-matrine hybrids as potential anticancer agents via mitochondrial stress/cytochrome c/caspase 3 signaling pathway
|
Li, Lingyu
|
|
|
134 |
C |
p.
|
artikel
|
| 35 |
Spectroscopic analysis, kinetic mechanism, computational docking, and molecular dynamics of active metabolites from the aerial parts of Astragalus membranaceus Bunge as tyrosinase inhibitors
|
Manh Khoa, Nguyen
|
|
|
134 |
C |
p.
|
artikel
|
| 36 |
Structurally diverse new eudesmane sesquiterpenoids with anti-inflammatory activity from the fruits of Alpinia oxyphylla
|
Dong, Jie
|
|
|
134 |
C |
p.
|
artikel
|
| 37 |
Structural optimization of tetrahydroisoquinoline-hydroxamate hybrids as potent dual ERα degraders and HDAC inhibitors
|
Xiong, Shuangshuang
|
|
|
134 |
C |
p.
|
artikel
|
| 38 |
Synthesis, in-Silico studies and biological evaluation of pyrimidine based thiazolidinedione derivatives as potential anti-diabetic agent
|
Amin, Shaista
|
|
|
134 |
C |
p.
|
artikel
|
| 39 |
Ugi reaction-assisted assembly of covalent PROTACs against glutathione peroxidase 4
|
Zhu, Liquan
|
|
|
134 |
C |
p.
|
artikel
|
| 40 |
Wang resin catalysed sonochemical synthesis of pyrazolo[4,3-d]pyrimidinones and 2,3-dihydroquinazolin-4(1H)-ones: Identification of chorismate mutase inhibitors having effects on Mycobacterium tuberculosis cell viability
|
Shukla, Sharda
|
|
|
134 |
C |
p.
|
artikel
|
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