nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Ac34FGlcNAz is an effective metabolic chemical reporter for O-GlcNAcylated proteins with decreased S-glyco-modification
|
Wang, Jiajia |
|
|
131 |
C |
p. |
artikel |
2 |
Advanced high-affinity glycoconjugate ligands of galectins
|
Hovorková, Michaela |
|
|
131 |
C |
p. |
artikel |
3 |
Allosteric quinoxaline-based inhibitors of the flavivirus NS2B/NS3 protease
|
Zephyr, Jacqueto |
|
|
131 |
C |
p. |
artikel |
4 |
A novel AIRE-based fluorescent ratiometric probe with endoplasmic reticulum-targeting ability for detection of hypochlorite and bioimaging
|
Yan, Jin-Long |
|
|
131 |
C |
p. |
artikel |
5 |
Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: Synthesis and biological evaluation
|
Carullo, Gabriele |
|
|
131 |
C |
p. |
artikel |
6 |
Chalcone derivatives as xanthine oxidase inhibitors: synthesis, binding mode investigation, biological evaluation, and ADMET prediction
|
Yang, Can |
|
|
131 |
C |
p. |
artikel |
7 |
Chemical constituents from the stems and leaves of Amomum villosum Lour. and their anti-inflammatory and antioxidant activities
|
Gao, Chengfeng |
|
|
131 |
C |
p. |
artikel |
8 |
Chromone-based benzohydrazide derivatives as potential α-glucosidase inhibitor: Synthesis, biological evaluation and molecular docking study
|
Fan, Meiyan |
|
|
131 |
C |
p. |
artikel |
9 |
Corrigendum to “[11]-chaetoglobosins with cytotoxic activities from Pseudeurotium bakeri” [Bioorg. Chem. 127 (2022) 106011]
|
Duan, Fangfang |
|
|
131 |
C |
p. |
artikel |
10 |
Corrigendum to “Design, synthesis and pharmacological evaluation of 2-arylurea-1,3,5-triazine derivative (XIN-9): A novel potent dual PI3K/mTOR inhibitor for cancer therapy” [Bioorg. Chem. 129 (2022) 106157]
|
Sun, Xin |
|
|
131 |
C |
p. |
artikel |
11 |
Cytotoxic steroidal saponins from the rhizomes of Paris fargesii var. Petiolata
|
Tian, Yun-Yuan |
|
|
131 |
C |
p. |
artikel |
12 |
Deciphering the biotransformation mechanism of dialkylresorcinols by CYP4F11
|
Shi, Yue |
|
|
131 |
C |
p. |
artikel |
13 |
Design and synthesis of 2-(2,2-diarylethyl)-cyclamine derivatives as M3 receptor antagonists and functional evaluation on COPD
|
Zhao, Yaopeng |
|
|
131 |
C |
p. |
artikel |
14 |
Design and synthesis of novel anti-multidrug-resistant staphylococcus aureus derivatives of glycyrrhetinic acid by blocking arginine biosynthesis, metabolic and H2S biogenesis
|
Cai, De-Sheng |
|
|
131 |
C |
p. |
artikel |
15 |
Design, synthesis and biological evaluation of alkynyl-containing maleimide derivatives for the treatment of drug-resistant tuberculosis
|
Li, Peng |
|
|
131 |
C |
p. |
artikel |
16 |
Design, synthesis, and biological evaluation of novel protopanoxadiol derivatives based PROTACs technology for the treatment of lung cancer
|
Wang, Peng |
|
|
131 |
C |
p. |
artikel |
17 |
Design, synthesis, and evaluation of JTE-013 derivatives as novel potent S1PR2 antagonists for recovering the sensitivity of colorectal cancer to 5-fluorouracil
|
Guo, Zhikun |
|
|
131 |
C |
p. |
artikel |
18 |
Design, synthesis, and metabolite identification of Tamoxifen esterase-activatable prodrugs
|
Elbagoury, Rahma M. |
|
|
131 |
C |
p. |
artikel |
19 |
Design, synthesis and molecular docking of novel substituted azepines as inhibitors of PI3K/Akt/TSC2/mTOR signaling pathway in colorectal carcinoma
|
Noser, Ahmed A. |
|
|
131 |
C |
p. |
artikel |
20 |
Design, synthesis and Molecular modeling study of certain EGFRinhibitors with a quinazolinone scaffold as anti-hepatocellular carcinoma and Radio-sensitizers
|
Ghorab, Walid M. |
|
|
131 |
C |
p. |
artikel |
21 |
Design, synthesis, biological activity evaluation and structure-activity relationships of new steroidal aromatase inhibitors. The case of C-ring and 7β substituted steroids
|
Roleira, Fernanda M.F. |
|
|
131 |
C |
p. |
artikel |
22 |
Design, synthesis of 1,2,4-triazine derivatives as antidepressant and antioxidant agents: In vitro, in vivo and in silico studies
|
Pal, Rohit |
|
|
131 |
C |
p. |
artikel |
23 |
Development and challenges in the discovery of 5-HT1A and 5-HT7 receptor ligands
|
Singh, Deepika |
|
|
131 |
C |
p. |
artikel |
24 |
Development of new spiro[1,3]dithiine-4,11′-indeno[1,2-b]quinoxaline derivatives as S. aureus Sortase A inhibitors and radiosterilization with molecular modeling simulation
|
Ragab, Ahmed |
|
|
131 |
C |
p. |
artikel |
25 |
Discovery and structural optimization of 3-O-β-Chacotriosyl betulonic acid saponins as potent fusion inhibitors of Omicron virus infections
|
Liu, Mingjian |
|
|
131 |
C |
p. |
artikel |
26 |
Discovery of dioxo-benzo[b]thiophene derivatives as potent YAP-TEAD interaction inhibitors for treating breast cancer
|
Son, Youngchai |
|
|
131 |
C |
p. |
artikel |
27 |
Discovery of N-methylbenzo[d]oxazol-2-amine as new anthelmintic agent through scalable protocol for the synthesis of N-alkylbenzo[d]oxazol-2-amine and N-alkylbenzo[d]thiazol-2-amine derivatives
|
Laohapaisan, Pavitra |
|
|
131 |
C |
p. |
artikel |
28 |
Discovery of non-nucleoside oxindole derivatives as potent inhibitors against dengue RNA-dependent RNA polymerase
|
Maddipati, Venkatanarayana Chowdary |
|
|
131 |
C |
p. |
artikel |
29 |
Discovery of novel danshensu derivatives bearing pyrazolone moiety as potential anti-ischemic stroke agents with antioxidant activity
|
Li, Yi |
|
|
131 |
C |
p. |
artikel |
30 |
Discovery of two biotin-PEG4‑diarylidenyl piperidone prodrugs as potent antitumor agents with good efficacy, limited toxicity, and low resistance
|
Liu, Shuang-Qiang |
|
|
131 |
C |
p. |
artikel |
31 |
2,5-Disubstituted furan derivatives containing imidazole, triazole or tetrazole moiety as potent α-glucosidase inhibitors
|
He, Min |
|
|
131 |
C |
p. |
artikel |
32 |
Editorial Board
|
|
|
|
131 |
C |
p. |
artikel |
33 |
6-Heterocyclic carboxylic ester derivatives of gliotoxin lead to LSD1 inhibitors in gastric cancer cells
|
Shan, Lihong |
|
|
131 |
C |
p. |
artikel |
34 |
High-performance fluorescence probe for fast and specific visualization of norepinephrine in vivo and depression-like mice
|
Gu, Pengli |
|
|
131 |
C |
p. |
artikel |
35 |
Issue TOC
|
|
|
|
131 |
C |
p. |
artikel |
36 |
Length and rigidity of the spacer impact on aldose reductase inhibition of the 5F-like ARIs in a dual-occupied mode
|
Zeng, Yancong |
|
|
131 |
C |
p. |
artikel |
37 |
New tetrahydropyrimidine-1,2,3-triazole clubbed compounds: Antitubercular activity and Thymidine Monophosphate Kinase (TMPKmt) inhibition
|
El-Shoukrofy, Mai S. |
|
|
131 |
C |
p. |
artikel |
38 |
New thiourea and benzamide derivatives of 2-aminothiazole as multi-target agents against Alzheimer's disease: Design, synthesis, and biological evaluation
|
Kilic, Burcu |
|
|
131 |
C |
p. |
artikel |
39 |
Novel amino analogs of the trimethoxyphenyl ring in potent colchicine site ligands improve solubility by the masked polar group incorporation (MPGI) strategy
|
González, Myriam |
|
|
131 |
C |
p. |
artikel |
40 |
Novel dual-target μ‑opioid and TRPV1 ligands as potential pharmacotherapeutics for pain management
|
Gao, Mengkang |
|
|
131 |
C |
p. |
artikel |
41 |
Novel pyrazole-based COX-2 inhibitors as potential anticancer agents: Design, synthesis, cytotoxic effect against resistant cancer cells, cell cycle arrest, apoptosis induction and dual EGFR/Topo-1 inhibition
|
Halim, Peter A. |
|
|
131 |
C |
p. |
artikel |
42 |
Optimisation of pyrazolo[1,5-a]pyrimidin-7(4H)-one derivatives as novel Hsp90 C-terminal domain inhibitors against Ewing sarcoma
|
Zajec, Živa |
|
|
131 |
C |
p. |
artikel |
43 |
Phytochemical composition, bioactive properties, and toxicological profile of Tetrapleura tetraptera
|
Anyamele, ThankGod |
|
|
131 |
C |
p. |
artikel |
44 |
Profiling of the chemical space on the phenyl group of substituted benzothiazole RIPK3 inhibitors
|
Xu, Yue |
|
|
131 |
C |
p. |
artikel |
45 |
P-Y/G@NHs sensitizes non-small cell lung cancer cells to radiotherapy via blockage of the PI3K/AKT signaling pathway
|
Zhang, Lu |
|
|
131 |
C |
p. |
artikel |
46 |
Rice peroxygenase catalyzes lipoxygenase-dependent regiospecific epoxidation of lipid peroxides in the response to abiotic stressors
|
Tran, Anh Duc |
|
|
131 |
C |
p. |
artikel |
47 |
Schiff bases as linker in the development of quinoline-sulfonamide hybrids as selective cancer-associated carbonic anhydrase isoforms IX/XII inhibitors: A new regioisomerism tactic
|
El-Malah, Afaf |
|
|
131 |
C |
p. |
artikel |
48 |
seco-Sesquiterpenes and acorane-type sesquiterpenes with antiviral activity from the twigs and leaves of Illicium henryi Diels
|
Yong, Jin-Yao |
|
|
131 |
C |
p. |
artikel |
49 |
Sequence and structure-guided discovery of a novel NADH-dependent 7β-hydroxysteroid dehydrogenase for efficient biosynthesis of ursodeoxycholic acid
|
Huang, Bin |
|
|
131 |
C |
p. |
artikel |
50 |
Solid lipid nanoparticles (SLNs), the potential novel vehicle for enhanced in vivo efficacy of hesperidin as an anti-inflammatory agent
|
Shahraki, Omolbanin |
|
|
131 |
C |
p. |
artikel |
51 |
State of art in the chemistry of nucleoside-based Pt(II) complexes
|
D'Errico, Stefano |
|
|
131 |
C |
p. |
artikel |
52 |
Structural characteristics of a low molecular weight velvet antler protein and the anti-tumor activity on S180 tumor-bearing mice
|
Cao, Tian-qi |
|
|
131 |
C |
p. |
artikel |
53 |
Synthesis and cytotoxicity evaluation of DNA-interactive β-carboline indolyl-3-glyoxamide derivatives: Topo-II inhibition and in silico modelling studies
|
Soni, Jay Prakash |
|
|
131 |
C |
p. |
artikel |
54 |
Synthesis, antiproliferative and anti-MDR activities of lathyrane diterpene derivatives based on configuration inversion strategy
|
Xiao, Yao |
|
|
131 |
C |
p. |
artikel |
55 |
Synthesis, biological evaluation, and molecular docking studies of aldotetronic acid-based LpxC inhibitors
|
Wimmer, Stefan |
|
|
131 |
C |
p. |
artikel |
56 |
Synthesis of Cy5-Labelled C5-Alkynyl-modified cytidine triphosphates via Sonogashira coupling for DNA labelling
|
Kuznetsova, Viktoriya E. |
|
|
131 |
C |
p. |
artikel |
57 |
Synthesis of new phenoxymethylcoumarin clubbed 4-arylthiazolylhydrazines as α-glucosidase inhibitors and their kinetics and molecular docking studies
|
ul Ain, Qurat |
|
|
131 |
C |
p. |
artikel |
58 |
Synthesis, pharmacological evaluation, DFT calculation, and theoretical investigation of spirocyclohexane derivatives
|
Abdel Hamid, Atef M. |
|
|
131 |
C |
p. |
artikel |
59 |
The dual FAK-HDAC inhibitor MY-1259 displays potent activities in gastric cancers in vitro and in vivo
|
Song, Jian |
|
|
131 |
C |
p. |
artikel |
60 |
The metal ion hypothesis of Alzheimer’s disease and the anti-neuroinflammatory effect of metal chelators
|
Chen, Li-Lin |
|
|
131 |
C |
p. |
artikel |
61 |
Triazole-based estradiol dimers prepared via CuAAC from 17α-ethinyl estradiol with five-atom linkers causing G2/M arrest and tubulin inhibition
|
Jurášek, Michal |
|
|
131 |
C |
p. |
artikel |