| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Annulated pyrazole derivatives as a novel class of urokinase (uPA) inhibitors: Green synthesis, anticancer activity, DNA-damage evaluation, and molecular modelling study
|
Farag, Paula S.
|
|
|
130 |
C |
p.
|
artikel
|
| 2 |
A simple protein histidine kinase activity assay for high-throughput inhibitor screening
|
Lee, Donghee
|
|
|
130 |
C |
p.
|
artikel
|
| 3 |
A toolbox of diverse arginine N-glycosylated peptides and specific antibodies
|
Jiang, Yanan
|
|
|
130 |
C |
p.
|
artikel
|
| 4 |
Based on 2-(difluoromethyl)-1-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]-1H-benzimidazole (ZSTK474), design, synthesis and biological evaluation of novel PI3Kα selective inhibitors
|
Wang, Yu
|
|
|
130 |
C |
p.
|
artikel
|
| 5 |
Chaetonigrisins A–L, a group of 3-Indole-1,2-Propanediol derived alkaloids from Chaetomium nigricolor YT-2
|
Qian, Xue-Qing
|
|
|
130 |
C |
p.
|
artikel
|
| 6 |
Characterization of a polysaccharide from Polygala tenuifolia willd. with immune activity via activation MAPKs pathway
|
Yu, Shasha
|
|
|
130 |
C |
p.
|
artikel
|
| 7 |
Chemical and biology of sulfur fluoride exchange (SuFEx) click chemistry for drug discovery
|
Wilson Lucas, Shadrack
|
|
|
130 |
C |
p.
|
artikel
|
| 8 |
Coumarin-4-yl‐1,2,3‐triazol‐4-yl-methyl-thiazolidine-2,4-diones: Synthesis, glucose uptake activity and cytotoxic evaluation
|
Metre, Tukaram V.
|
|
|
130 |
C |
p.
|
artikel
|
| 9 |
C-terminal modification of a de novo designed antimicrobial peptide via capping of macrolactam rings
|
Zeng, Ping
|
|
|
130 |
C |
p.
|
artikel
|
| 10 |
Design, synthesis, AML activity and molecular modeling of novel IDH2 inhibitors
|
Jin, Ruyi
|
|
|
130 |
C |
p.
|
artikel
|
| 11 |
Design, synthesis, and biological evaluation of novel HSP27 inhibitors to sensitize lung cancer cells to clinically available anticancer agents
|
Choi, Seul-Ki
|
|
|
130 |
C |
p.
|
artikel
|
| 12 |
Design, synthesis and biological evaluation of novel pyrazolo-pyrimidin-amines as potent and selective BTK inhibitors
|
Joshi, Darshan
|
|
|
130 |
C |
p.
|
artikel
|
| 13 |
Design, synthesis and evaluation of oxazolopyridinone derivatives as quorum sensing inhibitors
|
Chen, Weijin
|
|
|
130 |
C |
p.
|
artikel
|
| 14 |
Development of new 1, 3-dihydroxyacridone derivatives as Akt pathway inhibitors in skeletal muscle cells
|
Irazoqui, A. Paula
|
|
|
130 |
C |
p.
|
artikel
|
| 15 |
Discoidin domain receptor inhibitors as anticancer agents: A systematic review on recent development of DDRs inhibitors, their resistance and structure activity relationship
|
Shenoy, Ganesh Prasad
|
|
|
130 |
C |
p.
|
artikel
|
| 16 |
Discovery and mechanism of action of Thonzonium bromide from an FDA-approved drug library with potent and broad-spectrum inhibitory activity against main proteases of human coronaviruses
|
Wang, Ruyu
|
|
|
130 |
C |
p.
|
artikel
|
| 17 |
Editorial Board
|
|
|
|
130 |
C |
p.
|
artikel
|
| 18 |
Exploring the dual effect of novel 1,4-diarylpyranopyrazoles as antiviral and anti-inflammatory for the management of SARS-CoV-2 and associated inflammatory symptoms
|
Malebari, Azizah M.
|
|
|
130 |
C |
p.
|
artikel
|
| 19 |
Flavonoids dimers from the fruits of Psoralea corylifolia and their cytotoxicity against MCF-7 cells
|
Xu, Qing-Xia
|
|
|
130 |
C |
p.
|
artikel
|
| 20 |
Hybridization of amantadine with gardenamide A enhances NMDA antagonism and in vivo anti-PD effects
|
Zhu, Wenda
|
|
|
130 |
C |
p.
|
artikel
|
| 21 |
Identification of an N-phenylsulfonyl-2-(piperazin-1-yl)methyl-benzonitrile derivative as Zika virus entry inhibitor
|
Quan, Yanni
|
|
|
130 |
C |
p.
|
artikel
|
| 22 |
Identification of (N-aryl-N-arylsulfonyl)aminoacetohydroxamic acids as novel urease inhibitors and the mechanism exploration
|
Li, Su-Ya
|
|
|
130 |
C |
p.
|
artikel
|
| 23 |
In-situ construction of fluorescent probes for hydrogen peroxide detection in mitochondria and lysosomes with on-demand modular assembling and double turn-on features
|
Feng, Gang
|
|
|
130 |
C |
p.
|
artikel
|
| 24 |
Integrated transcriptomics and metabolomics analyses to investigate the anticancer mechanisms of cinobufagin against liver cancer through interfering with lipid, amino acid, carbohydrate, and nucleotide metabolism
|
Yang, Ailin
|
|
|
130 |
C |
p.
|
artikel
|
| 25 |
Investigation of the effects of isoeugenol-based phenolic compounds on migration and proliferation of HT29 colon cancer cells at cellular and molecular level
|
Bilgin, Sema
|
|
|
130 |
C |
p.
|
artikel
|
| 26 |
Isolation and identification of hemostatic steroidal glycosides from Ypsilandra thibetica
|
Ma, Wen-Yi
|
|
|
130 |
C |
p.
|
artikel
|
| 27 |
Issue TOC
|
|
|
|
130 |
C |
p.
|
artikel
|
| 28 |
Light and hydrogen peroxide dual-responsive DNA interstrand crosslink precursors with potent cytotoxicity
|
Jia, Yuanyuan
|
|
|
130 |
C |
p.
|
artikel
|
| 29 |
Mitochondria-targeted pentacyclic triterpenoid carbon dots for selective cancer cell destruction via inducing autophagy, apoptosis, as well as ferroptosis
|
Tian, Luyao
|
|
|
130 |
C |
p.
|
artikel
|
| 30 |
Modulating the affinity and signaling bias of cannabinoid receptor 1 antagonists
|
Hsiao, Wen-Chi
|
|
|
130 |
C |
p.
|
artikel
|
| 31 |
Multifunctional organic nanomaterials with ultra-high photothermal conversion efficiency for photothermal therapy and inhibition of cancer metastasis
|
Yang, Xiao-Zhen
|
|
|
130 |
C |
p.
|
artikel
|
| 32 |
Nematocidal alkaloids from the roots of Stemona mairei (H.Lév.)K.Krause and identification of their pharmacophoric moiety
|
Shi, Bao-Bao
|
|
|
130 |
C |
p.
|
artikel
|
| 33 |
New amides derived from sclareolide as anticholinesterase agents
|
Silva, Júnio G.
|
|
|
130 |
C |
p.
|
artikel
|
| 34 |
Novel 6-amino-1,3,5-triazine derivatives as potent BTK inhibitors: structure-activity relationship (SAR) analysis and preliminary mechanism investigation
|
Xiao, Maoxu
|
|
|
130 |
C |
p.
|
artikel
|
| 35 |
Novel AP2238-clorgiline hybrids as multi-target agents for the treatment of Alzheimer's disease: Design, synthesis, and biological evaluation
|
Zhong, Guohui
|
|
|
130 |
C |
p.
|
artikel
|
| 36 |
Novel quinazolinone disulfide analogues as pqs quorum sensing inhibitors against Pseudomonas aeruginosa
|
Sabir, Shekh
|
|
|
130 |
C |
p.
|
artikel
|
| 37 |
OSMAC strategy integrated with molecular networking discovery peniciacetals A−I, nine new meroterpenoids from the mangrove-derived fungus Penicillium sp. HLLG-122
|
Qin, Yuyue
|
|
|
130 |
C |
p.
|
artikel
|
| 38 |
Schisandrin B ameliorates acute liver injury by regulating EGFR-mediated activation of autophagy
|
Li, Xiankuan
|
|
|
130 |
C |
p.
|
artikel
|
| 39 |
Structural optimization of novel Ras modulator for treatment of Colorectal cancer by promoting β-catenin and Ras degradation
|
Choi, Seonghwi
|
|
|
130 |
C |
p.
|
artikel
|
| 40 |
Structure-activity relationship study of a series of nucleoside derivatives bearing sulfonamide scaffold as potent and selective PRMT5 inhibitors
|
Chen, Yuting
|
|
|
130 |
C |
p.
|
artikel
|
| 41 |
Studies on crystal structures, optical, dyeing and biological properties of protoberberine alkaloids and their supramolecular salts
|
Du, Haijuan
|
|
|
130 |
C |
p.
|
artikel
|
| 42 |
Synthesis, characterization, in-silico, and pharmacological evaluation of new 2-amino-6‑trifluoromethoxy benzothiazole derivatives
|
Malik, Sumra
|
|
|
130 |
C |
p.
|
artikel
|
| 43 |
Synthesis, larvicidal efficiency and molecular docking studies of novel annulated pyrano[2,3-c]pyrazoles against Culex pipiens L. and Musca domestica L. larvae
|
El-Sayed, Mahmoud K.F.
|
|
|
130 |
C |
p.
|
artikel
|
| 44 |
Synthesis, radiolabeling and evaluation of [99mTc][Tc-HYNIC/EDDA]-Met(O) as a early agent for amino acid metabolic imaging in C6 glioblastoma tumor
|
Dinmohammadi, Fahimeh
|
|
|
130 |
C |
p.
|
artikel
|
| 45 |
Synthetic amino acids-derived peptides target Cryptococcus neoformans by inducing cell membrane disruption
|
Sharma, Komal
|
|
|
130 |
C |
p.
|
artikel
|
| 46 |
Targeting phosphodiesterase 4 as a therapeutic strategy for cognitive improvement
|
Wei, Xuemei
|
|
|
130 |
C |
p.
|
artikel
|
| 47 |
tLyp–1: A peptide suitable to target NRP–1 receptor
|
Larue, Ludivine
|
|
|
130 |
C |
p.
|
artikel
|
| 48 |
Towards Alzheimer’s disease-related targets: One-pot Cu(I)- mediated synthesis of new nitroindazolyltriazoles
|
Eddahmi, Mohammed
|
|
|
130 |
C |
p.
|
artikel
|
| 49 |
Uncariphyllin A-J, indole alkaloids from Uncaria rhynchophylla as antagonists of dopamine D2 and Mu opioid receptors
|
Xu, Yang
|
|
|
130 |
C |
p.
|
artikel
|
| 50 |
Unraveling the therapeutic potential of carbamoyl phosphate synthetase 1 (CPS1) in human diseases
|
Zhang, Lan
|
|
|
130 |
C |
p.
|
artikel
|
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