nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Acylphloroglucinol trimers from Callistemon salignus seeds: Isolation, configurational assignment, hAChE inhibitory effects, and molecular docking studies
|
Yu, Mu-Yuan |
|
|
117 |
C |
p. |
artikel |
2 |
A designed cyclic peptide based on Trastuzumab used to construct peptide-drug conjugates for its HER2-targeting ability
|
Zhou, Jiaqi |
|
|
117 |
C |
p. |
artikel |
3 |
Amide-based xanthine oxidase inhibitors bearing an N-(1-alkyl-3-cyano-1H-indol-5-yl) moiety: Design, synthesis and structure-activity relationship investigation
|
Zhang, Ting-jian |
|
|
117 |
C |
p. |
artikel |
4 |
Anticancer profile and anti-inflammatory effect of new N-(2-((4-(1,3-diphenyl-1H-pyrazol-4-yl)pyridine sulfonamide derivatives
|
Abdel-Maksoud, Mohammed S. |
|
|
117 |
C |
p. |
artikel |
5 |
Artemicapillasins A–N, cytotoxic coumaric acid analogues against hepatic stellate cell LX2 from Artemisia capillaris (Yin-Chen)
|
Gao, Zhen |
|
|
117 |
C |
p. |
artikel |
6 |
Assessment of elementary derivatives of 1,5-benzodiazepine as anticancer agents with synergy potential
|
Gawandi, Sinthiya J. |
|
|
117 |
C |
p. |
artikel |
7 |
Biological effects of bis-hydrazone compounds bearing isovanillin moiety on the aldose reductase
|
Yapar, Gönül |
|
|
117 |
C |
p. |
artikel |
8 |
Caesalpinaxin, a cassane-type diterpenoid with a 21-carbon core skeleton from the seeds of Caesalpinia minax possessing pro-angiogenetic property
|
Lou, Ruohan |
|
|
117 |
C |
p. |
artikel |
9 |
β-Carboline tethered cinnamoyl 2-aminobenzamides as class I selective HDAC inhibitors: Design, synthesis, biological activities and modelling studies
|
Namballa, Hari Krishna |
|
|
117 |
C |
p. |
artikel |
10 |
Clavipyrrine A, a unique polycyclic nitrogenous meroterpenoid with promising anti-glioma effects isolated from the fungus Clitocybe clavipes
|
Sun, Zhaocui |
|
|
117 |
C |
p. |
artikel |
11 |
Clickable, selective, and cell-permeable activity-based probe of human cathepsin B – Minimalistic approach for enhanced selectivity
|
Bhuiyan, Ashif I. |
|
|
117 |
C |
p. |
artikel |
12 |
Continuous Sirtuin/HDAC (histone deacetylase) activity assay using thioamides as PET (Photoinduced Electron Transfer)–based fluorescence quencher
|
Zessin, Matthes |
|
|
117 |
C |
p. |
artikel |
13 |
Corrigendum to “Rational design-aided discovery of novel 1,2,4-oxadiazole derivatives as potential EGFR inhibitors” [Bioorg. Chem. 114 (2021) 105124]
|
Unadkat, Vishal |
|
|
117 |
C |
p. |
artikel |
14 |
Cytotoxic and apoptotic effects of 1,2-diborolanes with strong donor substitutes on human cancer cells
|
Şahin, Yüksel |
|
|
117 |
C |
p. |
artikel |
15 |
Design and synthesis of naphthylchalcones as novel anti-leukaemia agents
|
Leitão, Emília P.T. |
|
|
117 |
C |
p. |
artikel |
16 |
Design, parallel synthesis of Biginelli 1,4-dihydropyrimidines using PTSA as a catalyst, evaluation of anticancer activity and structure activity relationships via 3D QSAR studies
|
Faizan, Syed |
|
|
117 |
C |
p. |
artikel |
17 |
Design, synthesis and binding mode of interaction of novel small molecule o-hydroxy benzamides as HDAC3-selective inhibitors with promising antitumor effects in 4T1-Luc breast cancer xenograft model
|
Routholla, Ganesh |
|
|
117 |
C |
p. |
artikel |
18 |
Design, synthesis and biological evaluation of cinnamamide-quinazoline derivatives as potential EGFR inhibitors to reverse T790M mutation
|
Zhang, Bin |
|
|
117 |
C |
p. |
artikel |
19 |
Design, synthesis, and evaluation of proliferation inhibitory activity of novel L-shaped ortho-quinone analogs as anticancer agents
|
Yu, Jia |
|
|
117 |
C |
p. |
artikel |
20 |
Design, synthesis and structure-activity evaluation of novel 2-pyridone-based inhibitors of α-synuclein aggregation with potentially improved BBB permeability
|
Mahía, Alejandro |
|
|
117 |
C |
p. |
artikel |
21 |
Design, synthesis, in vitro, and in silico studies of 1,2,4-triazole-piperazine hybrid derivatives as potential MAO inhibitors
|
Uslu, Harun |
|
|
117 |
C |
p. |
artikel |
22 |
Development of anti-breast cancer PI3K inhibitors based on 7-azaindole derivatives through scaffold hopping: Design, synthesis and in vitro biological evaluation
|
Yang, Chengbin |
|
|
117 |
C |
p. |
artikel |
23 |
Discovery of bletillain, an unusual benzyl polymer with significant autophagy-inducing effects in A549 lung cancer cells through the Akt/GSK-3β/β-catenin signaling pathway
|
Zhu, Huan |
|
|
117 |
C |
p. |
artikel |
24 |
Discovery of KRas G12C-IN-3 and Pomalidomide-based PROTACs as degraders of endogenous KRAS G12C with potent anticancer activity
|
Li, Ling |
|
|
117 |
C |
p. |
artikel |
25 |
Discovery of new 2-phenyl-1H-benzo[d]imidazole core-based potent α-glucosidase inhibitors: Synthesis, kinetic study, molecular docking, and in vivo anti-hyperglycemic evaluation
|
Li, Yue |
|
|
117 |
C |
p. |
artikel |
26 |
Discovery of novel ibrutinib analogues to treat malignant melanoma
|
Ren, Sumei |
|
|
117 |
C |
p. |
artikel |
27 |
Discovery of quinazolinyl-containing benzamides derivatives as novel HDAC1 inhibitors with in vitro and in vivo antitumor activities
|
Zhang, Zixue |
|
|
117 |
C |
p. |
artikel |
28 |
Diterpenoids from Euphorbia glomerulans with potential reversal activities against P-glycoprotein-mediated multidrug resistance
|
Hasan, Aobulikasimu |
|
|
117 |
C |
p. |
artikel |
29 |
Editorial Board
|
|
|
|
117 |
C |
p. |
artikel |
30 |
Growing the molecular architecture of imidazole-like ligands in HO-1 complexes
|
Floresta, Giuseppe |
|
|
117 |
C |
p. |
artikel |
31 |
Guided rational design with scaffold hopping leading to novel histamine H3 receptor ligands
|
Ghamari, Nakisa |
|
|
117 |
C |
p. |
artikel |
32 |
HDAC/MIF dual inhibitor inhibits NSCLC cell survival and proliferation by blocking the AKT pathway
|
Cao, Fangyuan |
|
|
117 |
C |
p. |
artikel |
33 |
Hepatoprotective, antioxidant and anti-inflammatory potentials of Vit-E/C@SeNPs in rats: Synthesis, characterization, biochemical, radio-biodistribution, molecular and histopathological studies
|
Aljuhr, Safa A. |
|
|
117 |
C |
p. |
artikel |
34 |
Indolin-2-one derivatives as selective Aurora B kinase inhibitors targeting breast cancer
|
Dokla, Eman M.E. |
|
|
117 |
C |
p. |
artikel |
35 |
Issue TOC
|
|
|
|
117 |
C |
p. |
artikel |
36 |
Meta-substituted piperlongumine derivatives attenuate inflammation in both RAW264.7 macrophages and a mouse model of colitis
|
Wang, Ziqing |
|
|
117 |
C |
p. |
artikel |
37 |
Molecular hybridization design and synthesis of novel spirooxindole-based MDM2 inhibitors endowed with BCL2 signaling attenuation; a step towards the next generation p53 activators
|
Lotfy, Gehad |
|
|
117 |
C |
p. |
artikel |
38 |
New α-pyrone derivatives with herbicidal activity from the endophytic fungus Alternaria brassicicola
|
Li, Fengli |
|
|
117 |
C |
p. |
artikel |
39 |
Novel 2,4-disubstituted quinazoline analogs as antibacterial agents with improved cytotoxicity profile: Optimization of the 2,4-substituents
|
Aboushady, Dina |
|
|
117 |
C |
p. |
artikel |
40 |
Novel natural scaffold as hURAT1 inhibitor identified by 3D-shape-based, docking-based virtual screening approach and biological evaluation
|
Chen, Xinhua |
|
|
117 |
C |
p. |
artikel |
41 |
Novel phenanthridine amide analogs as potential anti-leishmanial agents: In vitro and in silico insights
|
Nandikolla, Adinarayana |
|
|
117 |
C |
p. |
artikel |
42 |
Potential inhibitors and plant based technology: An alternative approach to treat corona virus
|
Sharma, Sachin |
|
|
117 |
C |
p. |
artikel |
43 |
Probing the Ca2+ mobilizing properties on primary cortical neurons of a new stable cADPR mimic
|
D'Errico, Stefano |
|
|
117 |
C |
p. |
artikel |
44 |
Profiling sirtuin activity using Copper-free click chemistry
|
Curry, Alyson M. |
|
|
117 |
C |
p. |
artikel |
45 |
Property activity refinement of 2-anilino 4-amino substituted quinazolines as antimalarials with fast acting asexual parasite activity
|
Ashton, Trent D. |
|
|
117 |
C |
p. |
artikel |
46 |
Receptor mapping using methoxy phenyl piperazine derivative: Preclinical PET imaging
|
Mann, Garima |
|
|
117 |
C |
p. |
artikel |
47 |
Secoiridoid dimers and their biogenetic precursors from the fruits of Cornus officinalis with potential therapeutic effects on type 2 diabetes
|
Peng, Zhong-Can |
|
|
117 |
C |
p. |
artikel |
48 |
Site selective synthesis and anti-inflammatory evaluation of Spiro-isoxazoline stitched adducts of arteannuin B
|
Ur Rasool, Javeed |
|
|
117 |
C |
p. |
artikel |
49 |
Structurally diverse biflavonoids from the fruits of Citrus medica L. var. sarcodactylis Swingle and their hypolipidemic and immunosuppressive activities
|
Ma, Qin-Ge |
|
|
117 |
C |
p. |
artikel |
50 |
Structural simplification and bioisostere principle lead to Bis-benzodioxole-fibrate derivatives as potential hypolipidemic and hepatoprotective agents
|
Xie, Yundong |
|
|
117 |
C |
p. |
artikel |
51 |
Structure–activity relationship and biological evaluation of 12 N-substituted aloperine derivatives as PD-L1 down-regulatory agents through proteasome pathway
|
Zeng, Qing–Xuan |
|
|
117 |
C |
p. |
artikel |
52 |
Synthesis and biological evaluation of cationic TopFluor cholesterol analogues
|
Jurášek, Michal |
|
|
117 |
C |
p. |
artikel |
53 |
Synthesis and hyperglycemic, biochemical and histopathological evaluation of novel sulfonylbiguanide and sulfonylurea derivatives as potent anti-diabetic agents
|
Basyouni, Wahid M. |
|
|
117 |
C |
p. |
artikel |
54 |
Synthesis and in vitro evaluation of anti-inflammatory, antioxidant, and anti-fibrotic effects of new 8-aminopurine-2,6-dione-based phosphodiesterase inhibitors as promising anti-asthmatic agents
|
Wójcik-Pszczoła, Katarzyna |
|
|
117 |
C |
p. |
artikel |
55 |
Synthesis and in vitro evaluation of chlorogenic acid amides as potential hypoglycemic agents and their synergistic effect with acarbose
|
Cardullo, Nunzio |
|
|
117 |
C |
p. |
artikel |
56 |
Synthesis, biological evaluation and molecular docking of new sulfonamide-based indolinone derivatives as multitargeted kinase inhibitors against leukemia
|
El-Hussieny, Marwa |
|
|
117 |
C |
p. |
artikel |
57 |
Synthesis, biological evaluation, and molecular docking studies of deoxygenated C-glycosides as LpxC inhibitors
|
Dreger, Alexander |
|
|
117 |
C |
p. |
artikel |
58 |
Synthesis of a new series of pyrazolo[1,5-a]pyrimidines as CDK2 inhibitors and anti-leukemia
|
Almehmadi, Samar J. |
|
|
117 |
C |
p. |
artikel |
59 |
Synthesis of aspirin-curcumin mimic conjugates of potential antitumor and anti-SARS-CoV-2 properties
|
Srour, Aladdin M. |
|
|
117 |
C |
p. |
artikel |
60 |
The development of modulators for lysophosphatidic acid receptors: A comprehensive review
|
Liu, Wenjie |
|
|
117 |
C |
p. |
artikel |
61 |
The Mpro structure-based modifications of ebselen derivatives for improved antiviral activity against SARS-CoV-2 virus
|
Qiao, Zhen |
|
|
117 |
C |
p. |
artikel |
62 |
Triterpenoids and meroterpenoids with α-glucosidase inhibitory activities from the fruiting bodies of Ganoderma australe
|
Guo, Jiao-Cen |
|
|
117 |
C |
p. |
artikel |
63 |
Triterpenoid saponins from the leaves and stems of Pericampylus glaucus and their insulin mimetic activities
|
Lee, Hee-Ju |
|
|
117 |
C |
p. |
artikel |
64 |
Water-soluble pillar[5]arene sulfo-derivatives self-assemble into biocompatible nanosystems to stabilize therapeutic proteins
|
Shurpik, Dmitriy N. |
|
|
117 |
C |
p. |
artikel |