Digitale Bibliotheek
Sluiten Bladeren door artikelen uit een tijdschrift
     Tijdschrift beschrijving
       Alle jaargangen van het bijbehorende tijdschrift
         Alle afleveringen van het bijbehorende jaargang
                                       Alle artikelen van de bijbehorende aflevering
 
                             64 gevonden resultaten
nr titel auteur tijdschrift jaar jaarg. afl. pagina('s) type
1 Acylphloroglucinol trimers from Callistemon salignus seeds: Isolation, configurational assignment, hAChE inhibitory effects, and molecular docking studies Yu, Mu-Yuan

117 C p.
artikel
2 A designed cyclic peptide based on Trastuzumab used to construct peptide-drug conjugates for its HER2-targeting ability Zhou, Jiaqi

117 C p.
artikel
3 Amide-based xanthine oxidase inhibitors bearing an N-(1-alkyl-3-cyano-1H-indol-5-yl) moiety: Design, synthesis and structure-activity relationship investigation Zhang, Ting-jian

117 C p.
artikel
4 Anticancer profile and anti-inflammatory effect of new N-(2-((4-(1,3-diphenyl-1H-pyrazol-4-yl)pyridine sulfonamide derivatives Abdel-Maksoud, Mohammed S.

117 C p.
artikel
5 Artemicapillasins A–N, cytotoxic coumaric acid analogues against hepatic stellate cell LX2 from Artemisia capillaris (Yin-Chen) Gao, Zhen

117 C p.
artikel
6 Assessment of elementary derivatives of 1,5-benzodiazepine as anticancer agents with synergy potential Gawandi, Sinthiya J.

117 C p.
artikel
7 Biological effects of bis-hydrazone compounds bearing isovanillin moiety on the aldose reductase Yapar, Gönül

117 C p.
artikel
8 Caesalpinaxin, a cassane-type diterpenoid with a 21-carbon core skeleton from the seeds of Caesalpinia minax possessing pro-angiogenetic property Lou, Ruohan

117 C p.
artikel
9 β-Carboline tethered cinnamoyl 2-aminobenzamides as class I selective HDAC inhibitors: Design, synthesis, biological activities and modelling studies Namballa, Hari Krishna

117 C p.
artikel
10 Clavipyrrine A, a unique polycyclic nitrogenous meroterpenoid with promising anti-glioma effects isolated from the fungus Clitocybe clavipes Sun, Zhaocui

117 C p.
artikel
11 Clickable, selective, and cell-permeable activity-based probe of human cathepsin B – Minimalistic approach for enhanced selectivity Bhuiyan, Ashif I.

117 C p.
artikel
12 Continuous Sirtuin/HDAC (histone deacetylase) activity assay using thioamides as PET (Photoinduced Electron Transfer)–based fluorescence quencher Zessin, Matthes

117 C p.
artikel
13 Corrigendum to “Rational design-aided discovery of novel 1,2,4-oxadiazole derivatives as potential EGFR inhibitors” [Bioorg. Chem. 114 (2021) 105124] Unadkat, Vishal

117 C p.
artikel
14 Cytotoxic and apoptotic effects of 1,2-diborolanes with strong donor substitutes on human cancer cells Şahin, Yüksel

117 C p.
artikel
15 Design and synthesis of naphthylchalcones as novel anti-leukaemia agents Leitão, Emília P.T.

117 C p.
artikel
16 Design, parallel synthesis of Biginelli 1,4-dihydropyrimidines using PTSA as a catalyst, evaluation of anticancer activity and structure activity relationships via 3D QSAR studies Faizan, Syed

117 C p.
artikel
17 Design, synthesis and binding mode of interaction of novel small molecule o-hydroxy benzamides as HDAC3-selective inhibitors with promising antitumor effects in 4T1-Luc breast cancer xenograft model Routholla, Ganesh

117 C p.
artikel
18 Design, synthesis and biological evaluation of cinnamamide-quinazoline derivatives as potential EGFR inhibitors to reverse T790M mutation Zhang, Bin

117 C p.
artikel
19 Design, synthesis, and evaluation of proliferation inhibitory activity of novel L-shaped ortho-quinone analogs as anticancer agents Yu, Jia

117 C p.
artikel
20 Design, synthesis and structure-activity evaluation of novel 2-pyridone-based inhibitors of α-synuclein aggregation with potentially improved BBB permeability Mahía, Alejandro

117 C p.
artikel
21 Design, synthesis, in vitro, and in silico studies of 1,2,4-triazole-piperazine hybrid derivatives as potential MAO inhibitors Uslu, Harun

117 C p.
artikel
22 Development of anti-breast cancer PI3K inhibitors based on 7-azaindole derivatives through scaffold hopping: Design, synthesis and in vitro biological evaluation Yang, Chengbin

117 C p.
artikel
23 Discovery of bletillain, an unusual benzyl polymer with significant autophagy-inducing effects in A549 lung cancer cells through the Akt/GSK-3β/β-catenin signaling pathway Zhu, Huan

117 C p.
artikel
24 Discovery of KRas G12C-IN-3 and Pomalidomide-based PROTACs as degraders of endogenous KRAS G12C with potent anticancer activity Li, Ling

117 C p.
artikel
25 Discovery of new 2-phenyl-1H-benzo[d]imidazole core-based potent α-glucosidase inhibitors: Synthesis, kinetic study, molecular docking, and in vivo anti-hyperglycemic evaluation Li, Yue

117 C p.
artikel
26 Discovery of novel ibrutinib analogues to treat malignant melanoma Ren, Sumei

117 C p.
artikel
27 Discovery of quinazolinyl-containing benzamides derivatives as novel HDAC1 inhibitors with in vitro and in vivo antitumor activities Zhang, Zixue

117 C p.
artikel
28 Diterpenoids from Euphorbia glomerulans with potential reversal activities against P-glycoprotein-mediated multidrug resistance Hasan, Aobulikasimu

117 C p.
artikel
29 Editorial Board
117 C p.
artikel
30 Growing the molecular architecture of imidazole-like ligands in HO-1 complexes Floresta, Giuseppe

117 C p.
artikel
31 Guided rational design with scaffold hopping leading to novel histamine H3 receptor ligands Ghamari, Nakisa

117 C p.
artikel
32 HDAC/MIF dual inhibitor inhibits NSCLC cell survival and proliferation by blocking the AKT pathway Cao, Fangyuan

117 C p.
artikel
33 Hepatoprotective, antioxidant and anti-inflammatory potentials of Vit-E/C@SeNPs in rats: Synthesis, characterization, biochemical, radio-biodistribution, molecular and histopathological studies Aljuhr, Safa A.

117 C p.
artikel
34 Indolin-2-one derivatives as selective Aurora B kinase inhibitors targeting breast cancer Dokla, Eman M.E.

117 C p.
artikel
35 Issue TOC
117 C p.
artikel
36 Meta-substituted piperlongumine derivatives attenuate inflammation in both RAW264.7 macrophages and a mouse model of colitis Wang, Ziqing

117 C p.
artikel
37 Molecular hybridization design and synthesis of novel spirooxindole-based MDM2 inhibitors endowed with BCL2 signaling attenuation; a step towards the next generation p53 activators Lotfy, Gehad

117 C p.
artikel
38 New α-pyrone derivatives with herbicidal activity from the endophytic fungus Alternaria brassicicola Li, Fengli

117 C p.
artikel
39 Novel 2,4-disubstituted quinazoline analogs as antibacterial agents with improved cytotoxicity profile: Optimization of the 2,4-substituents Aboushady, Dina

117 C p.
artikel
40 Novel natural scaffold as hURAT1 inhibitor identified by 3D-shape-based, docking-based virtual screening approach and biological evaluation Chen, Xinhua

117 C p.
artikel
41 Novel phenanthridine amide analogs as potential anti-leishmanial agents: In vitro and in silico insights Nandikolla, Adinarayana

117 C p.
artikel
42 Potential inhibitors and plant based technology: An alternative approach to treat corona virus Sharma, Sachin

117 C p.
artikel
43 Probing the Ca2+ mobilizing properties on primary cortical neurons of a new stable cADPR mimic D'Errico, Stefano

117 C p.
artikel
44 Profiling sirtuin activity using Copper-free click chemistry Curry, Alyson M.

117 C p.
artikel
45 Property activity refinement of 2-anilino 4-amino substituted quinazolines as antimalarials with fast acting asexual parasite activity Ashton, Trent D.

117 C p.
artikel
46 Receptor mapping using methoxy phenyl piperazine derivative: Preclinical PET imaging Mann, Garima

117 C p.
artikel
47 Secoiridoid dimers and their biogenetic precursors from the fruits of Cornus officinalis with potential therapeutic effects on type 2 diabetes Peng, Zhong-Can

117 C p.
artikel
48 Site selective synthesis and anti-inflammatory evaluation of Spiro-isoxazoline stitched adducts of arteannuin B Ur Rasool, Javeed

117 C p.
artikel
49 Structurally diverse biflavonoids from the fruits of Citrus medica L. var. sarcodactylis Swingle and their hypolipidemic and immunosuppressive activities Ma, Qin-Ge

117 C p.
artikel
50 Structural simplification and bioisostere principle lead to Bis-benzodioxole-fibrate derivatives as potential hypolipidemic and hepatoprotective agents Xie, Yundong

117 C p.
artikel
51 Structure–activity relationship and biological evaluation of 12 N-substituted aloperine derivatives as PD-L1 down-regulatory agents through proteasome pathway Zeng, Qing–Xuan

117 C p.
artikel
52 Synthesis and biological evaluation of cationic TopFluor cholesterol analogues Jurášek, Michal

117 C p.
artikel
53 Synthesis and hyperglycemic, biochemical and histopathological evaluation of novel sulfonylbiguanide and sulfonylurea derivatives as potent anti-diabetic agents Basyouni, Wahid M.

117 C p.
artikel
54 Synthesis and in vitro evaluation of anti-inflammatory, antioxidant, and anti-fibrotic effects of new 8-aminopurine-2,6-dione-based phosphodiesterase inhibitors as promising anti-asthmatic agents Wójcik-Pszczoła, Katarzyna

117 C p.
artikel
55 Synthesis and in vitro evaluation of chlorogenic acid amides as potential hypoglycemic agents and their synergistic effect with acarbose Cardullo, Nunzio

117 C p.
artikel
56 Synthesis, biological evaluation and molecular docking of new sulfonamide-based indolinone derivatives as multitargeted kinase inhibitors against leukemia El-Hussieny, Marwa

117 C p.
artikel
57 Synthesis, biological evaluation, and molecular docking studies of deoxygenated C-glycosides as LpxC inhibitors Dreger, Alexander

117 C p.
artikel
58 Synthesis of a new series of pyrazolo[1,5-a]pyrimidines as CDK2 inhibitors and anti-leukemia Almehmadi, Samar J.

117 C p.
artikel
59 Synthesis of aspirin-curcumin mimic conjugates of potential antitumor and anti-SARS-CoV-2 properties Srour, Aladdin M.

117 C p.
artikel
60 The development of modulators for lysophosphatidic acid receptors: A comprehensive review Liu, Wenjie

117 C p.
artikel
61 The Mpro structure-based modifications of ebselen derivatives for improved antiviral activity against SARS-CoV-2 virus Qiao, Zhen

117 C p.
artikel
62 Triterpenoids and meroterpenoids with α-glucosidase inhibitory activities from the fruiting bodies of Ganoderma australe Guo, Jiao-Cen

117 C p.
artikel
63 Triterpenoid saponins from the leaves and stems of Pericampylus glaucus and their insulin mimetic activities Lee, Hee-Ju

117 C p.
artikel
64 Water-soluble pillar[5]arene sulfo-derivatives self-assemble into biocompatible nanosystems to stabilize therapeutic proteins Shurpik, Dmitriy N.

117 C p.
artikel
                             64 gevonden resultaten
 
 Koninklijke Bibliotheek - Nationale Bibliotheek van Nederland