Digitale Bibliotheek
Sluiten Bladeren door artikelen uit een tijdschrift
 
Zoeken naar met titel:
ABCDEFGHIJKLMNOPQRSTUVWXYZ

     Tijdschrift beschrijving
       Alle jaargangen van het bijbehorende tijdschrift
         Alle afleveringen van het bijbehorende jaargang
                                       Alle artikelen van de bijbehorende aflevering
 
                             121 gevonden resultaten
nr titel auteur tijdschrift jaar jaarg. afl. pagina('s) type
1 Absolute configuration and protein tyrosine phosphatase 1B inhibitory activity of xanthoepocin, a dimeric naphtopyrone from Penicillium sp. IQ-429 Martínez-Aldino, Ingrid Y.
115 C p.
 artikel
2 Absolute configuration of polypropionate derivatives: Decempyrones A–J and their MptpA inhibition and anti-inflammatory activities Guo, Heng
115 C p.
 artikel
3 Alkaloid derivative ION-31a inhibits breast cancer metastasis and angiogenesis by targeting HSP90α Ni, Tian-Wen
115 C p.
 artikel
4 Analysis of Hsp90 allosteric modulators interactome reveals a potential dual action mode involving mitochondrial MDH2 Cassiano, Chiara
115 C p.
 artikel
5 A new ferroptosis inhibitor, isolated from Ajuga nipponensis, protects neuronal cells via activating NRF2-antioxidant response elements (AREs) pathway Tan, Qingyun
115 C p.
 artikel
6 An overall framework for the E. coli γ-glutamyltransferase-catalyzed transpeptidation reactions Somma, Valeria
115 C p.
 artikel
7 An overview of triazoloquinazolines: Pharmacological significance and recent developments Abuelizz, Hatem A.
115 C p.
 artikel
8 Anticancer effect evaluation in vitro and in vivo of iridium(III) polypyridyl complexes targeting DNA and mitochondria Zhang, Huiwen
115 C p.
 artikel
9 Antimicrobial properties of novel ionic liquids derived from imidazolium cation with phenolic functional groups Guzmán, Luis
115 C p.
 artikel
10 Benzimidazole analogues as efficient arsenals in war against methicillin-resistance staphylococcus aureus (MRSA) and its SAR studies Zha, Gao-Feng
115 C p.
 artikel
11 Beta-Carotene derivatives as novel therapy for the prevention and treatment of autistic symptoms Avraham, Yosefa
115 C p.
 artikel
12 Biphenylpiperazine Based MAO Inhibitors: Synthesis, Biological Evaluation, Reversibility and Molecular Modeling Studies El-Halaby, Lamiaa O.
115 C p.
 artikel
13 Biphenyl substituted lysine derivatives as recognition elements for the matrix metalloproteinases MMP-2 and MMP-9 Kirchhain, Arno
115 C p.
 artikel
14 Bisabolane, cadinane, and cyclonerane sesquiterpenes from an algicolous strain of Trichoderma asperelloides Zou, Ji-Xue
115 C p.
 artikel
15 Citral derivative activates cell cycle arrest and apoptosis signaling pathways in Candida albicans by generating oxidative stress Wani, Mohmmad Younus
115 C p.
 artikel
16 Computational design of binder as the LC3-p62 protein‐protein interaction Lyu, Weiping
115 C p.
 artikel
17 CuCl2-catalyzed inexpensive, faster and ligand/additive free synthesis of isoquinolin-1(2H)-one derivatives via the coupling–cyclization strategy: Evaluation of a new class of compounds as potential PDE4 inhibitors Thirupataiah, B.
115 C p.
 artikel
18 Current development of sigma-2 receptor radioligands as potential tumor imaging agents Shaghaghi, Zahra
115 C p.
 artikel
19 DD04107-Derived neuronal exocytosis inhibitor peptides: Evidences for synaptotagmin-1 as a putative target Butrón, Daniel
115 C p.
 artikel
20 Design and synthesis of novel conformationally constrained 7,12-dihydrodibenzo[b,h][1,6] naphthyridine and 7H-Chromeno[3,2-c] quinoline derivatives as topoisomerase I inhibitors: In vitro screening, molecular docking and ADME predictions Kardile, Ramakant A.
115 C p.
 artikel
21 Design and synthesis of novel 4-fluorobenzamide-based derivatives as promising anti-inflammatory and analgesic agents with an enhanced gastric tolerability and COX-inhibitory activity Halim, Peter A.
115 C p.
 artikel
22 Design and synthesis of novel mitochondria-targeted CDDO derivatives as potential anti-cancer agents Ju, Wei
115 C p.
 artikel
23 Design, Hemiysnthesis, crystal structure and anticancer activity of 1, 2, 3-triazoles derivatives of totarol Laamari, Yassine
115 C p.
 artikel
24 Design, synthesis and antitumor activities of thiazole-containing mitochondrial targeting agents Zhang, Dongdong
115 C p.
 artikel
25 Design, synthesis and antitumor evaluation of novel chiral diaryl substituted azetidin-2-one derivatives as tubulin polymerization inhibitors Liang, Yuru
115 C p.
 artikel
26 Design, synthesis and bioevaluation of 2,7-diaryl-pyrazolo[1,5-a]pyrimidines as tubulin polymerization inhibitors Liu, Runlai
115 C p.
 artikel
27 Design, synthesis and biological evaluation of 2,3-dihydroimidazo[2,1-b]thiazoles as dual EGFR and IGF1R inhibitors Gadekar, Pradip K.
115 C p.
 artikel
28 Design, synthesis, and biological evaluation of novel FXR agonists based on auraptene Qiu, Qianqian
115 C p.
 artikel
29 Design, synthesis and biological evaluation of novel 5-(imidazolyl-methyl) thiazolidinediones as antidiabetic agents Shakour, Neda
115 C p.
 artikel
30 Design, synthesis and biological evaluation of novel pyrrolidone-based derivatives as potent p53-MDM2 inhibitors Si, Dongjuan
115 C p.
 artikel
31 Design, synthesis and evaluation of side-chain hydroxylated derivatives of lithocholic acid as potent agonists of the vitamin D receptor (VDR) González, Carmen M.
115 C p.
 artikel
32 Design, synthesis and evaluation of tetrahydrocarbazole derivatives as potential hypoglycemic agents Wang, Li-Li
115 C p.
 artikel
33 Design, synthesis, molecular docking and in silico ADMET profile of pyrano[2,3-d]pyrimidine derivatives as antimicrobial and anticancer agents Abd El-Sattar, Nour E.A.
115 C p.
 artikel
34 Development of coumarin-thiosemicarbazone hybrids as aldose reductase inhibitors: Biological assays, molecular docking, simulation studies and ADME evaluation Imran, Aqeel
115 C p.
 artikel
35 Dibenzocyclooctadiene lignans from Kadsura coccinea alleviate APAP-induced hepatotoxicity via oxidative stress inhibition and activating the Nrf2 pathway in vitro Yang, Yupei
115 C p.
 artikel
36 Discovery and evolution of 12N-substituted aloperine derivatives as anti-SARS-CoV-2 agents through targeting late entry stage Wang, Kun
115 C p.
 artikel
37 Discovery of a novel and selective cathepsin L inhibitor with anti-metastatic ability in vitro and in vivo against breast cancer cells Li, Yanchun
115 C p.
 artikel
38 Discovery of 4-benzyloxy and 4-(2-phenylethoxy) chalcone fibrate hybrids as novel PPARα agonists with anti-hyperlipidemic and antioxidant activities: Design, synthesis and in vitro/in vivo biological evaluation Hassan, Rasha M.
115 C p.
 artikel
39 Discovery of bioactive polycyclic polyprenylated acylphloroglucinols from Hypericum wilsonii Duan, Yulin
115 C p.
 artikel
40 Discovery of natural 15-LOX small molecule inhibitors from Chinese herbal medicine using virtual Screening, biological evaluation and molecular dynamics studies Li, Yatong
115 C p.
 artikel
41 Discovery of new anticancer thiourea-azetidine hybrids: design, synthesis, in vitro antiproliferative, SAR, in silico molecular docking against VEGFR-2, ADMET, toxicity, and DFT studies Parmar, Deepa R.
115 C p.
 artikel
42 Discovery of novel and potent safinamide-based derivatives as highly selective hMAO-B inhibitors for treatment of Parkinson's disease (PD): Design, synthesis, in vitro, in vivo and in silico biological studies Elkamhawy, Ahmed
115 C p.
 artikel
43 Discovery of novel inhibitors of human phosphoglycerate dehydrogenase by activity-directed combinatorial chemical synthesis strategy Zhou, Xia
115 C p.
 artikel
44 Discovery of potent and selective Cdc25 phosphatase inhibitors via rapid assembly and in situ screening of Quinonoid-focused libraries Tao, Yucen
115 C p.
 artikel
45 Discovery of 1,2,3-selenadiazole analogues as antifungal agents using a scaffold hopping approach Xu, Hang
115 C p.
 artikel
46 Discovery of small molecule acting as multitarget inhibitor of colorectal cancer by simultaneous blocking of the key COX-2, 5-LOX and PIM-1 kinase enzymes El-Miligy, Mostafa M.M.
115 C p.
 artikel
47 Divergent synthesis and elaboration of structure activity relationship for quinoline derivatives as highly selective NTPDase inhibitor Murtaza, Amna
115 C p.
 artikel
48 Editorial Board
115 C p.
 artikel
49 Eremophilane sesquiterpenoids from the whole plant of Parasenecio albus with immunosuppressive activity Zhou, Ming
115 C p.
 artikel
50 Essential moieties of myricetins, quercetins and catechins for binding and inhibitory activity against α-Glucosidase Fu, Minghai
115 C p.
 artikel
51 Evaluation of N-aryl-β-alanine derivatives as anticancer agents in triple-negative breast cancer and glioblastoma in vitro models Žukauskas, Mindaugas
115 C p.
 artikel
52 Exploring of tumor-associated carbonic anhydrase isoenzyme IX and XII inhibitory effects and cytotoxicities of the novel N-aryl-1-(4-sulfamoylphenyl)-5-(thiophen-2-yl)-1H-pyrazole-3-carboxamides Yamali, Cem
115 C p.
 artikel
53 Exploring phenylcarbamoylazinane-1,2,4-triazole thioethers as lipoxygenase inhibitors supported with in vitro, in silico and cytotoxic studies Shahid, Wardah
115 C p.
 artikel
54 Free energy perturbation guided Synthesis with Biological Evaluation of Substituted Quinoline derivatives as small molecule L858R/T790M/C797S mutant EGFR inhibitors targeting resistance in Non-Small Cell Lung Cancer (NSCLC) Karnik, Kshipra S.
115 C p.
 artikel
55 Identification, characterization and evaluation of novel antifungal cyclic peptides from Neobacillus drentensis Routhu, Sunitha Rani
115 C p.
 artikel
56 Identification of novel anti-cancer agents by the synthesis and cellular screening of a noscapine-based library Nemati, Faezeh
115 C p.
 artikel
57 Identification of phenylcarbamoylazinane-1,3,4-oxadiazole amides as lipoxygenase inhibitors with expression analysis and in silico studies Bashir, Bushra
115 C p.
 artikel
58 Inhibitory effect of triterpenoids from the mushroom Inonotus obliquus against α-glucosidase and their interaction: Inhibition kinetics and molecular stimulations Chen, Shao-Dan
115 C p.
 artikel
59 Integrating systematic pharmacology-based strategy and experimental validation to explore the synergistic pharmacological mechanisms of Guanxin V in treating ventricular remodeling Liang, Bo
115 C p.
 artikel
60 Issue TOC
115 C p.
 artikel
61 3-Methyl-imidazo[2,1-b]thiazole derivatives as a new class of antifolates: Synthesis, in vitro/in vivo bio-evaluation and molecular modeling simulations Ewida, Menna A.
115 C p.
 artikel
62 Microwave prompted solvent-free synthesis of new series of heterocyclic tagged 7-arylidene indanone hybrids and their computational, antifungal, antioxidant, and cytotoxicity study Adole, Vishnu A.
115 C p.
 artikel
63 Molecular modelling, synthesis and antimicrobial evaluation of benzimidazole nucleoside mimetics Chaurasia, Himani
115 C p.
 artikel
64 Multicomponent reaction for the synthesis of new 1,3,4-thiadiazole-thiazolidine-4-one molecular hybrids as promising antidiabetic agents through α-glucosidase and α-amylase inhibition Gummidi, Lalitha
115 C p.
 artikel
65 Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery Prasad, Mayuri S.
115 C p.
 artikel
66 Natural STAT3 inhibitors: A mini perspective Wang, Zhuo
115 C p.
 artikel
67 N-(3-cyano-1H-indol-5-yl)isonicotinamide and N-(3-cyano-1H-indol-5-yl)-1H-benzo[d]imidazole-5-carboxamide derivatives: Novel amide-based xanthine oxidase inhibitors Tu, Shun
115 C p.
 artikel
68 Neuropathic pain-alleviating activity of novel 5-HT6 receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamide Drop, Marcin
115 C p.
 artikel
69 New alkali tolerant β-galactosidase from Paracoccus marcusii KGP – A promising biocatalyst for the synthesis of oligosaccharides derived from lactulose (OsLu), the new generation prebiotics Kalathinathan, Pooja
115 C p.
 artikel
70 New diphenyl ethers from a fungus Epicoccum sorghinum L28 and their antifungal activity against phytopathogens Zhu, Junjie
115 C p.
 artikel
71 New lignans from the fruits of Leonurus japonicus and their hepatoprotective activities Tian, Zhi-Hao
115 C p.
 artikel
72 New N-(1,3,4-thiadiazol-2-yl)furan-2-carboxamide derivatives as potential inhibitors of the VEGFR-2 Hekal, Mohamed H.
115 C p.
 artikel
73 New thieno[3,2-d]pyrimidine-based derivatives: Design, synthesis and biological evaluation as antiproliferative agents, EGFR and ARO inhibitors inducing apoptosis in breast cancer cells Farghaly, Ahmed M.
115 C p.
 artikel
74 Novel Dy2O3/ZnO-Au ternary nanocomposites: Green synthesis using pomegranate fruit extract, characterization and their photocatalytic and antibacterial properties Khormali, Keyvan
115 C p.
 artikel
75 Novel insights on the molecular mechanism of action of the anti-angiogenic pyrazolyl-urea GeGe-3 by functional proteomics Morretta, Elva
115 C p.
 artikel
76 Novel manganese carbon quantum dots as a nano-probe: Facile synthesis, characterization and their application in naproxen delivery (Mn/CQD/SiO2@naproxen) Ardestani, Mehdi Shafiee
115 C p.
 artikel
77 Novel piperazine urea derivatives as highly potent transient receptor potential vanilloid 1 (TRPV1) antagonists Hu, Jing
115 C p.
 artikel
78 Novel, selective acrylamide linked quinazolines for the treatment of double mutant EGFR-L858R/T790M Non-Small-Cell lung cancer (NSCLC) Pawara, Rahul
115 C p.
 artikel
79 Novel tetrahydrobenzo[b]thiophen-2-yl)urea derivatives as novel α-glucosidase inhibitors: Synthesis, kinetics study, molecular docking, and in vivo anti-hyperglycemic evaluation Xie, Hong-Xu
115 C p.
 artikel
80 Novel 1,3,4-thiadiazole/oxadiazole-linked honokiol derivatives suppress cancer via inducing PI3K/Akt/mTOR-dependent autophagy Xu, Ting
115 C p.
 artikel
81 Novel thiomorpholine tethered isatin hydrazones as potential inhibitors of resistant Mycobacterium tuberculosis Karunanidhi, Sivanandhan
115 C p.
 artikel
82 N-salicyloyl tryptamine derivatives as potential therapeutic agents for Alzheimer's disease with neuroprotective effects Bai, Yinliang
115 C p.
 artikel
83 Nucleus-targeting imaging and enhanced cytotoxicity based on naphthalimide derivatives Wang, Shan-Shan
115 C p.
 artikel
84 Optimisation of 2-(N-phenyl carboxamide) triazolopyrimidine antimalarials with moderate to slow acting erythrocytic stage activity Bailey, Brodie L.
115 C p.
 artikel
85 Pentacyclic triterpene carboxylic acids derivatives integrated piperazine-amino acid complexes for α-glucosidase inhibition in vitro Huang, Jinxiang
115 C p.
 artikel
86 Phomaligols F–I, polyoxygenated cyclohexenone derivatives from marine-derived fungus Aspergillus flavus BB1 Liu, Xiao-Jing
115 C p.
 artikel
87 Photochemical synthesis, intercalation with DNA and antitumor evaluation in vitro of benzo[d]thiazolo[3,2-a]quinolin-10-ium derivatives Saifutiarova, Alina E.
115 C p.
 artikel
88 Potent antiplasmodial alkaloids from the rhizobacterium Pantoea agglomerans as hemozoin modulators Thissera, Bathini
115 C p.
 artikel
89 Preparation, spectroscopic, characterizations and biological studies of new charge transfer complexes formed between fluconazole drug with various acceptors Ali, Mahmoud M.
115 C p.
 artikel
90 Promising potential of a 18F-labelled small-molecular radiotracer to evaluate PD-L1 expression in tumors by PET imaging Lv, Gaochao
115 C p.
 artikel
91 Pseudopeptides with aldehyde or vinylsulfone warheads: Synthesis and antiproteasomal activity Jorda, Radek
115 C p.
 artikel
92 Purified recombinant human Chromogranin A N46 peptide with remarkable anticancer effect on human colon cancer cells Okasha, Hend
115 C p.
 artikel
93 Pyridazinones containing dithiocarbamoyl moieties as a new class of selective MAO-B inhibitors Besada, Pedro
115 C p.
 artikel
94 Quinazolinone dimers as a potential new class of safer Kv1 inhibitors: Overcoming hERG, sodium and calcium channel affinities Emam, Aya M.
115 C p.
 artikel
95 Ronald C.D. Breslow (1931–2017): A career in review Joseph, Vincent
115 C p.
 artikel
96 Selective inhibition of Helicobacter pylori methionine aminopeptidase by azaindole hydroxamic acid derivatives: Design, synthesis, in vitro biochemical and structural studies Bala, Sandeepchowdary
115 C p.
 artikel
97 Selective MOR activity of DAPEA and Endomorphin-2 analogues containing a (R)-γ-Freidinger lactam in position two Della Valle, Alice
115 C p.
 artikel
98 Selective targeting of cancer cells using a hydrogen peroxide-activated Hsp90 inhibitor Oh, Yong Jin
115 C p.
 artikel
99 Semicarbazones, thiosemicarbazone, thiazole and oxazole analogues as monoamine oxidase inhibitors: Synthesis, characterization, biological evaluation, molecular docking, and kinetic studies Qazi, Syeda Uroos
115 C p.
 artikel
100 Squaraine dyes as serum albumins probes: Synthesis, photophysical experiments and molecular docking studies S.D. Gomes, Vanessa
115 C p.
 artikel
101 Stelleranoids A–M, guaiane-type sesquiterpenoids based on [5,7] bicyclic system from Stellera chamaejasme and their cytotoxic activity Pan, Jun
115 C p.
 artikel
102 Stereoselective synthesis of (26R)-26-hydroxydiosgenin and its effect on the regulation of rat ovarian function Hilario-Martínez, J. Ciciolil
115 C p.
 artikel
103 Steroidal saponins with cytotoxic effects from the rhizomes of Asparagus cochinchinensis Liu, Bo
115 C p.
 artikel
104 Structurally diversified ent-kaurane and abietane diterpenoids from the stems of Tripterygium wilfordii and their anti-inflammatory activity Zhou, Xiao-Qiong
115 C p.
 artikel
105 Structural optimization, synthesis and in vitro synergistic anticancer activities of combinations of new N3-substituted dihydropyrimidine calcium channel blockers with cisplatin and etoposide El-Wakil, Marwa H.
115 C p.
 artikel
106 Structure-guided discovery of novel potent and efficacious proteolysis targeting chimera (PROTAC) degrader of BRD4 Xiang, Wang
115 C p.
 artikel
107 Synergistic effect of curcumin-Cu and curcumin-Ag nanoparticle loaded niosome: Enhanced antibacterial and anti-biofilm activities Targhi, Arefeh Abolhassani
115 C p.
 artikel
108 Synthesis and evaluation of a novel class of ethacrynic acid derivatives containing triazoles as potent anticancer agents El Abbouchi, Abdelmoula
115 C p.
 artikel
109 Synthesis and evaluation of curcumin-based near-infrared fluorescent probes for the in vivo optical imaging of amyloid-β plaques Park, Yong Dae
115 C p.
 artikel
110 Synthesis and kinetic characterization of hyperbolic inhibitors of human cathepsins K and S based on a succinimide scaffold Goričan, Tjaša
115 C p.
 artikel
111 Synthesis, antiepileptic effects, and structure-activity relationships of α-asarone derivatives: In vitro and in vivo neuroprotective effect of selected derivatives Zhang, Jian
115 C p.
 artikel
112 Synthesis, antitubercular, antimicrobial activities and molecular docking study of quinoline bearing dihydropyrimidines Desai, Nisheeth C.
115 C p.
 artikel
113 Synthesis, biological evaluation (antioxidant, antimicrobial, enzyme inhibition, and cytotoxic) and molecular docking study of hydroxy methoxy benzoin/benzil analogous Yaylı, Nurettin
115 C p.
 artikel
114 Synthesis, characterization, cytotoxicity studies, theoretical approach of adsorptive removal and molecular calculations of four new phosphoramide derivatives and related graphene oxide Gholivand, Khodayar
115 C p.
 artikel
115 Synthesis, in vitro antiurease, in vivo antinematodal activity of quinoline analogs and their in-silico study Zaman, Khalid
115 C p.
 artikel
116 Synthesis, molecular docking, and evaluation of antibacterial activity of 1,2,4-triazole-norfloxacin hybrids Yang, Ping
115 C p.
 artikel
117 Synthesis, molecular docking and molecular dynamics studies of novel tacrine-carbamate derivatives as potent cholinesterase inhibitors Ozten, Ozge
115 C p.
 artikel
118 Synthesis of new 2-(thiazol-4-yl)thiazolidin-4-one derivatives as potential anti-mycobacterial agents Abhale, Yogita K.
115 C p.
 artikel
119 Synthesis of trans- methyl ferulate bearing an oxadiazole ether as potential activators for controlling plant virus He, Feng
115 C p.
 artikel
120 Thiazolidinone-linked1,2,3-triazoles with monoterpenic skeleton as new potential anticancer agents: Design, synthesis and molecular docking studies Oubella, Ali
115 C p.
 artikel
121 Voltage gated sodium channel inhibitors as anticonvulsant drugs: A systematic review on recent developments and structure activity relationship studies Pal, Rohit
115 C p.
 artikel
                             121 gevonden resultaten
 
 Koninklijke Bibliotheek - Nationale Bibliotheek van Nederland