nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Advancements in folate receptor targeting for anti-cancer therapy: A small molecule-drug conjugate approach
|
Rana, Abhilash |
|
|
112 |
C |
p. |
artikel |
2 |
Amiridine-piperazine hybrids as cholinesterase inhibitors and potential multitarget agents for Alzheimer's disease treatment
|
Makhaeva, Galina F. |
|
|
112 |
C |
p. |
artikel |
3 |
A novel β-hairpin peptide derived from the ARC repressor selectively interacts with the major groove of B-DNA
|
Stefanucci, Azzurra |
|
|
112 |
C |
p. |
artikel |
4 |
Anti-inflammatory effect of luteolin is related to the changes in the gut microbiota and contributes to preventing the progression from simple steatosis to nonalcoholic steatohepatitis
|
Sun, Wen-Long |
|
|
112 |
C |
p. |
artikel |
5 |
A study on MAPK/ERK and CDK2-Cyclin-E signal switch “on and off” in cell proliferation by bis urea derivatives of 1, 4-Diisocyanatobenzene
|
Nagalakshmamma, Vadabingi |
|
|
112 |
C |
p. |
artikel |
6 |
Benzosuberene-sulfone analogues synthesis from Cedrus deodara oil and their therapeutic evaluation by computational analysis to treat type 2 diabetes
|
Bharti, Richa |
|
|
112 |
C |
p. |
artikel |
7 |
Bioactive monoterpene phenol dimers from the fruits of Psoralea corylifolia L.
|
Gao, Hu-Tong-Yue |
|
|
112 |
C |
p. |
artikel |
8 |
Bioactive naphthoquinones and triterpenoids from the fruiting bodies of Taiwanofungus salmoneus
|
Cheng, Kun-Ching |
|
|
112 |
C |
p. |
artikel |
9 |
Bioconversion of antifungal viridin to phytotoxin viridiol by environmental non-viridin producing microorganisms
|
Pakora, Gilles-Alex |
|
|
112 |
C |
p. |
artikel |
10 |
Briarane-type diterpenoids suppress osteoclastogenisis by regulation of Nrf2 and MAPK/NF-kB signaling pathway
|
Meng, Junjun |
|
|
112 |
C |
p. |
artikel |
11 |
Chromene and chromone derivatives as liver X receptors modulators from a marine-derived Pestalotiopsis neglecta fungus
|
Liang, Zhi |
|
|
112 |
C |
p. |
artikel |
12 |
Co-delivery of hesperidin and clarithromycin in a nanostructured lipid carrier for the eradication of Helicobacter pylori in vitro
|
Sharaf, Mohamed |
|
|
112 |
C |
p. |
artikel |
13 |
Concise synthesis and biological evaluation of 2-Aryl-3-Anilinobenzo[b]thiophene derivatives as potent apoptosis-inducing agents
|
Romagnoli, Romeo |
|
|
112 |
C |
p. |
artikel |
14 |
Design and discovery of new antiproliferative 1,2,4-triazin-3(2H)-ones as tubulin polymerization inhibitors targeting colchicine binding site
|
Eissa, Ibrahim H. |
|
|
112 |
C |
p. |
artikel |
15 |
Design and synthesis of novel substituted benzyl pyrrolopyrimidine derivatives as selective BTK inhibitors for treating mantle cell lymphoma
|
Ran, Fansheng |
|
|
112 |
C |
p. |
artikel |
16 |
Design, microwave assisted synthesis, and molecular modeling study of some new 1,3,4-thiadiazole derivatives as potent anticancer agents and potential VEGFR-2 inhibitors
|
Atta-Allah, Saad R. |
|
|
112 |
C |
p. |
artikel |
17 |
Design, synthesis, and antibacterial evaluation of new quinoline-1,3,4-oxadiazole and quinoline-1,2,4-triazole hybrids as potential inhibitors of DNA gyrase and topoisomerase IV
|
Hofny, Heba A. |
|
|
112 |
C |
p. |
artikel |
18 |
Design, synthesis, and anticancer evaluation of novel andrographolide derivatives bearing an α,β-unsaturated ketone moiety
|
Cai, Wei |
|
|
112 |
C |
p. |
artikel |
19 |
Design, synthesis and anti-influenza virus activity of furan-substituted spirothiazolidinones
|
Apaydın, Çağla Begüm |
|
|
112 |
C |
p. |
artikel |
20 |
Design, synthesis, and biological evaluation of novel EGFR inhibitors containing 5-chloro-3-hydroxymethyl-indole-2-carboxamide scaffold with apoptotic antiproliferative activity
|
Mohamed, Fatma A.M. |
|
|
112 |
C |
p. |
artikel |
21 |
Design, synthesis and biological evaluation of novel estrone phosphonates as high affinity organic anion-transporting polypeptide 2B1 (OATP2B1) inhibitors
|
Jójárt, Rebeka |
|
|
112 |
C |
p. |
artikel |
22 |
Design, synthesis and biological evaluation of novel imidazole-chalcone derivatives as potential anticancer agents and tubulin polymerization inhibitors
|
Rahimzadeh Oskuei, Sara |
|
|
112 |
C |
p. |
artikel |
23 |
Design, synthesis and biological evaluation of 7–(5–((substituted – amino)-methyl)-thiophen–2–yl)-spiro-[chroman–2,4′–piperidin]–4–one hydrochloride analogues as anticancer agents
|
Chitti, Surendar |
|
|
112 |
C |
p. |
artikel |
24 |
Design, synthesis and evaluation of anti-proliferative activity of 2-aryl-4-aminoquinazoline derivatives as EGFR inhibitors
|
Zhou, Zhihui |
|
|
112 |
C |
p. |
artikel |
25 |
Design, synthesis and evaluation of cinnamic acid hybrids as multi-target-directed agents for the treatment of Alzheimer’s disease
|
Wang, Keren |
|
|
112 |
C |
p. |
artikel |
26 |
Design, synthesis, in vitro and in vivo evaluation against MRSA and molecular docking studies of novel pleuromutilin derivatives bearing 1, 3, 4-oxadiazole linker
|
Liu, Jie |
|
|
112 |
C |
p. |
artikel |
27 |
Development of biotinylated and magnetic bead-immobilized enzymes for efficient glyco-engineering and isolation of antibodies
|
Chuang, Hong-Yang |
|
|
112 |
C |
p. |
artikel |
28 |
Dimeric clerodane diterpenoids and antiviral constituents of Dodonaea viscosa
|
Zhao, Xiao-Tong |
|
|
112 |
C |
p. |
artikel |
29 |
Disaccharide-polyethylenimine organic nanoparticles as non-toxic in vitro gene transporters and their anticancer potential
|
Singh, Reena |
|
|
112 |
C |
p. |
artikel |
30 |
Discovery and development of tumor glycolysis rate-limiting enzyme inhibitors
|
Sun, Xueyan |
|
|
112 |
C |
p. |
artikel |
31 |
Discovery of anti-infective adipostatins through bioactivity-guided isolation and heterologous expression of a type III polyketide synthase
|
Hou, Lukuan |
|
|
112 |
C |
p. |
artikel |
32 |
Discovery of 5-(or 6)-benzoxazoles and oxazolo[4,5-b]pyridines as novel candidate antitumor agents targeting hTopo IIα
|
Karatas, Esin |
|
|
112 |
C |
p. |
artikel |
33 |
Discovery of pseudolaric acid A as a new Hsp90 inhibitor uncovers its potential anticancer mechanism
|
Liu, Jiangxin |
|
|
112 |
C |
p. |
artikel |
34 |
Discovery of thieno[2,3-d]pyrimidine-based derivatives as potent VEGFR-2 kinase inhibitors and anti-cancer agents
|
El-Metwally, Souad A. |
|
|
112 |
C |
p. |
artikel |
35 |
Diterpenoids from the seeds of Euphorbia lathyris and their anti-inflammatory activity
|
Wang, Yali |
|
|
112 |
C |
p. |
artikel |
36 |
Diversity-oriented synthesis through gamma radiolysis: Preparation of unusual ecdysteroid derivatives activating Akt and AMPK in skeletal muscle cells
|
Issaadi, Halima Meriem |
|
|
112 |
C |
p. |
artikel |
37 |
Ebsulfur and Ebselen as highly potent scaffolds for the development of potential SARS-CoV-2 antivirals
|
Sun, Le-Yun |
|
|
112 |
C |
p. |
artikel |
38 |
Editorial Board
|
|
|
|
112 |
C |
p. |
artikel |
39 |
Exploration of benzofuran-based compounds as potent and selective Plasmodium falciparum glycogen synthase kinase-3 (PfGSK-3) inhibitors
|
Moolman, Chantalle |
|
|
112 |
C |
p. |
artikel |
40 |
Functional triterpenoids from medicinal fungi Ganoderma applanatum: A continuous search for antiadipogenic agents
|
Su, Hai-Guo |
|
|
112 |
C |
p. |
artikel |
41 |
(±)-Gancochlearols J − N, renoprotective meroterpenoids from Ganoderma cochlear
|
Meng, Xiao-Hui |
|
|
112 |
C |
p. |
artikel |
42 |
Hispidin, Harmaline, and Harmine as potent inhibitors of bovine xanthine oxidase: Gout treatment, in vitro, ADMET prediction, and SAR studies
|
Linani, Abderahmane |
|
|
112 |
C |
p. |
artikel |
43 |
8-Hydroxyquinoline derived p-halo N4-phenyl substituted thiosemicarbazones: Crystal structures, spectral characterization and in vitro cytotoxic studies of their Co(III), Ni(II) and Cu(II) complexes
|
Kotian, Avinash |
|
|
112 |
C |
p. |
artikel |
44 |
Identification of novel anti-inflammatory Nur77 modulators by virtual screening
|
Ding, Xiaoyu |
|
|
112 |
C |
p. |
artikel |
45 |
Identification of selective ligands targeting two GPCRs by receptor-affinity chromatography coupled with high-throughput sequencing techniques
|
Liang, Qi |
|
|
112 |
C |
p. |
artikel |
46 |
Insight on a new indolinone derivative as an orally bioavailable lead compound against renal cell carcinoma
|
Fouad, Marwa A. |
|
|
112 |
C |
p. |
artikel |
47 |
Issue TOC
|
|
|
|
112 |
C |
p. |
artikel |
48 |
Jatrophane diterpenoids as multidrug resistance modulators from Euphorbia sororia
|
Yang, Hequn |
|
|
112 |
C |
p. |
artikel |
49 |
Lepipyrrolins A-B, two new dimeric pyrrole 2-carbaldehyde alkaloids from the tubers of Lepidium meyenii
|
Liu, Jun-Hong |
|
|
112 |
C |
p. |
artikel |
50 |
Microwave assisted one-pot synthesis, photophysical and physicochemical studies of novel biologically active heterocyclic Donor (D)-π-Acceptor (A) chromophore
|
Khan, Salman A. |
|
|
112 |
C |
p. |
artikel |
51 |
Molecular characteristics supporting l-Type amino acid transporter 1 (LAT1)-mediated translocation
|
Kärkkäinen, Jussi |
|
|
112 |
C |
p. |
artikel |
52 |
Monoterpene-flavonoid conjugates from Sarcandra glabra and their autophagy modulating activities
|
Liu, Xin |
|
|
112 |
C |
p. |
artikel |
53 |
New bis([1,2,4]triazolo)[4,3-a:3′,4′-c]quinoxaline derivatives as VEGFR-2 inhibitors and apoptosis inducers: Design, synthesis, in silico studies, and anticancer evaluation
|
Alanazi, Mohammed M. |
|
|
112 |
C |
p. |
artikel |
54 |
Novel chiral naphthalimide-cycloalkanediamine conjugates: Design, synthesis and antitumor activity
|
Costales, Paula |
|
|
112 |
C |
p. |
artikel |
55 |
Novel 2,5-disubstituted-1,3,4-oxadiazole derivatives as MAO-B inhibitors: Synthesis, biological evaluation and molecular modeling studies
|
Tok, Fatih |
|
|
112 |
C |
p. |
artikel |
56 |
Novel ginsenoside derivatives have shown their effects on PC-3 cells by inducing G1-phase arrest and reactive oxygen species-mediate cell apoptosis
|
Xiao, Shengnan |
|
|
112 |
C |
p. |
artikel |
57 |
Novel hypoglycemic compounds from wild mushroom Paxillus involutus
|
Lv, Jianhua |
|
|
112 |
C |
p. |
artikel |
58 |
On-cell saturation transfer difference NMR for the identification of FimH ligands and inhibitors
|
Palmioli, Alessandro |
|
|
112 |
C |
p. |
artikel |
59 |
Orientin and vitexin production by a one-pot enzymatic cascade of a glycosyltransferase and sucrose synthase
|
Qiu, Cong |
|
|
112 |
C |
p. |
artikel |
60 |
Potential new targets and drugs related to histone modifications in glioma treatment
|
Wei, Xiuhong |
|
|
112 |
C |
p. |
artikel |
61 |
Simple heteroaryl modifications in the 4,5-diarylisoxazol-3-carboxylic acid scaffold favorably modulates the activity as dual mPGES-1/5-LO inhibitors with in vivo efficacy
|
Gürses, Tuğba |
|
|
112 |
C |
p. |
artikel |
62 |
Steroidal alkaloids from the bulbs of Fritillaria pallidiflora Schrenk and their anti-inflammatory activity
|
Wang, Lun |
|
|
112 |
C |
p. |
artikel |
63 |
Structure-based modification of pyrazolone derivatives to inhibit mTORC1 by targeting the leucyl-tRNA synthetase-RagD interaction
|
Kim, Jae Hyun |
|
|
112 |
C |
p. |
artikel |
64 |
Synthesis and evaluation of disulfide-rich cyclic α-conotoxin [S9A]TxID analogues as novel α3β4 nAChR antagonists
|
Wang, Shuai |
|
|
112 |
C |
p. |
artikel |
65 |
Synthesis, antimicrobial, anti-cancer and in silico studies of new urea derivatives
|
Sroor, Farid M. |
|
|
112 |
C |
p. |
artikel |
66 |
Synthesis, DFT, and eco-friendly insecticidal activity of some N-heterocycles derived from 4-((2-oxo-1,2-dihydroquinolin-3-yl)methylene)-2-phenyloxazol-5(4H)-one
|
Ghareeb, Eman A. |
|
|
112 |
C |
p. |
artikel |
67 |
Synthesis, in silico, in vitro and in vivo evaluations of isatin aroylhydrazones as highly potent anticonvulsant agents
|
Emami, Saeed |
|
|
112 |
C |
p. |
artikel |
68 |
Synthesis, In-vitro evaluation and molecular docking studies of oxoindolin phenylhydrazine carboxamides as potent and selective inhibitors of ectonucleoside triphosphate diphosphohydrolase (NTPDase)
|
Afzal, Saira |
|
|
112 |
C |
p. |
artikel |
69 |
Synthesis, molecular docking, and in silico ADMET studies of 4-benzyl-1-(2,4,6-trimethyl-benzyl)-piperidine: Potential Inhibitor of SARS-CoV2
|
Nandini Asha, R. |
|
|
112 |
C |
p. |
artikel |
70 |
Synthesis, molecular modeling and biological evaluation of new benzo[4,5]thieno[3,2-b]pyran derivatives as topoisomerase I-DNA binary complex poisons
|
Ahmed, Eman M. |
|
|
112 |
C |
p. |
artikel |
71 |
Synthesis of sorafenib analogues incorporating a 1,2,3-triazole ring and cytotoxicity towards hepatocellular carcinoma cell lines
|
Palakhachane, Sarinya |
|
|
112 |
C |
p. |
artikel |
72 |
Tailoring the substitution pattern of Pyrrolidine-2,5-dione for discovery of new structural template for dual COX/LOX inhibition
|
Sadiq, Abdul |
|
|
112 |
C |
p. |
artikel |
73 |
The mode of antibacterial action of quaternary N-benzylimidazole salts against emerging opportunistic pathogens
|
Crnčević, Doris |
|
|
112 |
C |
p. |
artikel |
74 |
1,2,3-Triazole tethered 1,2,4‑trioxane trimer induces apoptosis in metastatic cancer cells and inhibits their proliferation, migration and invasion
|
Khongsti, Kitboklang |
|
|
112 |
C |
p. |
artikel |