| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Accelerating the identification of subtype selective inhibitors via Three-Dimensional Biologically Relevant Spectrum (BRS-3D): The monoamine oxidase subtypes as a case study
|
Wang, Dong
|
|
|
106 |
C |
p.
|
artikel
|
| 2 |
A novel amino cellulose derivative using ATRP method: Preparation, characterization, and investigation of its antibacterial activity
|
Shokri, Mastaneh
|
|
|
106 |
C |
p.
|
artikel
|
| 3 |
Antimicrobial and antitumor activity of peptidomimetics synthesized from amino acids
|
Li, Huan
|
|
|
106 |
C |
p.
|
artikel
|
| 4 |
5-Aryl-furan derivatives bearing a phenylalanine- or isoleucine-derived rhodanine moiety as potential PTP1B inhibitors
|
Niu, Tianwei
|
|
|
106 |
C |
p.
|
artikel
|
| 5 |
5-[Aryloxypyridyl (or nitrophenyl)]-4H-1,2,4-triazoles as novel flexible benzodiazepine analogues: Synthesis, receptor binding affinity and lipophilicity-dependent anti-seizure onset of action
|
Navidpour, Latifeh
|
|
|
106 |
C |
p.
|
artikel
|
| 6 |
Assessing the biological potential of new symmetrical ferrocene based bisthiourea analogues
|
Patujo, Jahangeer
|
|
|
106 |
C |
p.
|
artikel
|
| 7 |
BODIPY based red emitters: Synthesis, computational and biological studies
|
Pandey, Vijayalakshmi
|
|
|
106 |
C |
p.
|
artikel
|
| 8 |
Celebrex derivatives: Synthesis, α-glucosidase inhibition, crystal structures and molecular docking studies
|
Kausar, Nabeela
|
|
|
106 |
C |
p.
|
artikel
|
| 9 |
Chemoenzymatic synthesis of enantiomerically enriched diprophylline and xanthinol nicotinate
|
Borowiecki, Paweł
|
|
|
106 |
C |
p.
|
artikel
|
| 10 |
Computational drug discovery and repurposing for the treatment of COVID-19: A systematic review
|
Mohamed, Kawthar
|
|
|
106 |
C |
p.
|
artikel
|
| 11 |
Design and development of Tetrahydro-Quinoline derivatives as dual mTOR-C1/C2 inhibitors for the treatment of lung cancer
|
Chaube, Udit J.
|
|
|
106 |
C |
p.
|
artikel
|
| 12 |
Design and synthesis of novel quinoline/chalcone/1,2,4-triazole hybrids as potent antiproliferative agent targeting EGFR and BRAFV600E kinases
|
Mohassab, Aliaa M.
|
|
|
106 |
C |
p.
|
artikel
|
| 13 |
Design, synthesis and anticancer activity of 5-aryl-4-(4-arylpiperazine-1-carbonyl)-1,2,3-thiadiazoles as microtubule-destabilizing agents
|
Wang, Chao
|
|
|
106 |
C |
p.
|
artikel
|
| 14 |
Design, synthesis and antimycobacterial evaluation of novel adamantane and adamantanol analogues effective against drug-resistant tuberculosis
|
Alsayed, Shahinda S.R.
|
|
|
106 |
C |
p.
|
artikel
|
| 15 |
Design, synthesis and biological activity of 1,4-quinone moiety attached to betulin derivatives as potent DT-diaphorase substrate
|
Kadela-Tomanek, Monika
|
|
|
106 |
C |
p.
|
artikel
|
| 16 |
Design, synthesis, and biological evaluation of new raloxifene analogues of improved antagonist activity and endometrial safety
|
Lambrinidis, George
|
|
|
106 |
C |
p.
|
artikel
|
| 17 |
Design, synthesis, and biological evaluation of novel imidazole derivatives possessing terminal sulphonamides as potential BRAFV600E inhibitors
|
Ali, Eslam M.H.
|
|
|
106 |
C |
p.
|
artikel
|
| 18 |
Design, synthesis and drug resistance reversal potential of novel curcumin mimics Van D
|
Raj Dwivedi, Gaurav
|
|
|
106 |
C |
p.
|
artikel
|
| 19 |
Design, synthesis, and evaluation of new 2-oxoquinoline arylaminothiazole derivatives as potential anticancer agents
|
Fang, Yilin
|
|
|
106 |
C |
p.
|
artikel
|
| 20 |
Design, synthesis of Cinnamyl-paeonol derivatives with 1, 3-Dioxypropyl as link arm and screening of tyrosinase inhibition activity in vitro
|
Tang, Kai
|
|
|
106 |
C |
p.
|
artikel
|
| 21 |
Development of β-carboline-benzothiazole hybrids via carboxamide formation as cytotoxic agents: DNA intercalative topoisomerase IIα inhibition and apoptosis induction
|
Tokala, Ramya
|
|
|
106 |
C |
p.
|
artikel
|
| 22 |
Development of pyridazine derivatives as potential EGFR inhibitors and apoptosis inducers: Design, synthesis, anticancer evaluation, and molecular modeling studies
|
Ahmed, Marwa F.
|
|
|
106 |
C |
p.
|
artikel
|
| 23 |
1,2-Diborolanes with strong donor substituents: Synthesis and high antimicrobial activity
|
Şahin, Yüksel
|
|
|
106 |
C |
p.
|
artikel
|
| 24 |
Discovery of a novel GLP-1/GIP dual receptor agonist CY-5 as long-acting hypoglycemic, anti-obesity agent
|
Liu, Chunxia
|
|
|
106 |
C |
p.
|
artikel
|
| 25 |
Discovery of 4-((4-(4-(3-(2-(2,6-difluorophenyl)-4-oxothiazolidin-3-yl)ureido)-2-fluorophenoxy)-6-methoxyquinolin-7-yl)oxy)-N,N-diethylpiperidine-1-carboxamide as kinase inhibitor for the treatment of colorectal cancer
|
Zhou, Yuting
|
|
|
106 |
C |
p.
|
artikel
|
| 26 |
Drug repurposing for the treatment of COVID-19: Pharmacological aspects and synthetic approaches
|
Batalha, Pedro N.
|
|
|
106 |
C |
p.
|
artikel
|
| 27 |
Editorial Board
|
|
|
|
106 |
C |
p.
|
artikel
|
| 28 |
Efficient biogenesis of Cu2O nanoparticles using extract of Camellia sinensis leaf: Evaluation of catalytic, cytotoxicity, antioxidant, and anti-human ovarian cancer properties
|
Dou, Lei
|
|
|
106 |
C |
p.
|
artikel
|
| 29 |
Evaluation of catacholase mimicking activity and apoptosis in human colorectal carcinoma cell line by activating mitochondrial pathway of copper(II) complex coupled with 2-(quinolin-8-yloxy)(methyl)benzonitrile and 8-hydroxyquinoline
|
Ali, Arif
|
|
|
106 |
C |
p.
|
artikel
|
| 30 |
5-HT1A targeting PARCEST agent DO3AM-MPP with potential for receptor imaging: Synthesis, physico-chemical and MR studies
|
Anju,
|
|
|
106 |
C |
p.
|
artikel
|
| 31 |
Identification of fusarielin M as a novel inhibitor of Mycobacterium tuberculosis protein tyrosine phosphatase B (MptpB)
|
Chen, Dongni
|
|
|
106 |
C |
p.
|
artikel
|
| 32 |
In silico designing, in vitro and in vivo evaluation of potential PPAR-γ agonists derived from aryl propionic acid scaffold
|
Kharbanda, Chetna
|
|
|
106 |
C |
p.
|
artikel
|
| 33 |
Investigation of the effect of different linker chemotypes on the inhibition of histone deacetylases (HDACs)
|
Linciano, Pasquale
|
|
|
106 |
C |
p.
|
artikel
|
| 34 |
In vitro adjuvant antitumor activity of various classes of semi-synthetic poststerone derivatives
|
Savchenko, Rimma G.
|
|
|
106 |
C |
p.
|
artikel
|
| 35 |
Issue TOC
|
|
|
|
106 |
C |
p.
|
artikel
|
| 36 |
Multifaceted activity of polyciclic MDR revertant agents in drug-resistant leukemic cells: Role of the spacer
|
Caciolla, Jessica
|
|
|
106 |
C |
p.
|
artikel
|
| 37 |
New flavonoids from the roots of Sophora davidii (Franch.) Skeels and their glucose transporter 4 translocation activities
|
Ma, Yuanren
|
|
|
106 |
C |
p.
|
artikel
|
| 38 |
Novel artemisinin derivatives with potent anticancer activities and the anti-colorectal cancer effect by the mitochondria-mediated pathway
|
Lin, Lan
|
|
|
106 |
C |
p.
|
artikel
|
| 39 |
Novel urea linked ciprofloxacin-chalcone hybrids having antiproliferative topoisomerases I/II inhibitory activities and caspases-mediated apoptosis
|
Mohammed, Hamada H.H.
|
|
|
106 |
C |
p.
|
artikel
|
| 40 |
Protective effects of four new saponins from Gynostemma pentaphyllum against hydrogen peroxide-induced neurotoxicity in SH-SY5Y cells
|
Zhai, Xin-Fang
|
|
|
106 |
C |
p.
|
artikel
|
| 41 |
Pyridylethanol(phenylethyl)amines are non-azole, highly selective Candida albicans sterol 14α-demethylase inhibitors
|
Ogris, Iza
|
|
|
106 |
C |
p.
|
artikel
|
| 42 |
Pyrrole-2,5-dione analogs as a promising antioxidant agents: microwave-assisted synthesis, bio-evaluation, SAR analysis and DFT studies/interpretation
|
Mallikarjuna Reddy, Guda
|
|
|
106 |
C |
p.
|
artikel
|
| 43 |
Selective stabilization of multiple promoter G-quadruplex DNA by using 2-phenyl-1H-imidazole-based tanshinone IIA derivatives and their potential suppressing function in the metastatic breast cancer
|
Zeng, Liang
|
|
|
106 |
C |
p.
|
artikel
|
| 44 |
Separation and configurational assignment of stereoisomeric phenalenones from the marine mangrove-derived fungus Penicillium herquei MA-370
|
Yang, Sui-Qun
|
|
|
106 |
C |
p.
|
artikel
|
| 45 |
Structurally homologous sialidases exhibit a commonality in reactivity: Glycoside hydrolase-catalyzed hydrolysis of Kdn-thioglycosides
|
Nejatie, Ali
|
|
|
106 |
C |
p.
|
artikel
|
| 46 |
Structure-based design of glycyrrhetinic acid derivatives as potent anti-sepsis agents targeting high-mobility group box-1
|
Wang, Yuanyuan
|
|
|
106 |
C |
p.
|
artikel
|
| 47 |
Suntamide A, a neuroprotective cyclic peptide from Cicadidae Periostracum
|
Thapa, Punam
|
|
|
106 |
C |
p.
|
artikel
|
| 48 |
Supramolecular self-assemblies of engineered polyethylenimines as multifunctional nanostructures for DNA transportation with excellent antimicrobial activity
|
Singh, Reena
|
|
|
106 |
C |
p.
|
artikel
|
| 49 |
Synthesis and antimicrobial activity of (−)-cleistenolide and analogues
|
Benedeković, Goran
|
|
|
106 |
C |
p.
|
artikel
|
| 50 |
Synthesis and biological activity of imidazole group-substituted arylaminopyrimidines (IAAPs) as potent BTK inhibitors against B-cell lymphoma and AML
|
Li, Si
|
|
|
106 |
C |
p.
|
artikel
|
| 51 |
Synthesis and biological evaluation as well as in silico studies of arylpiperazine-1,2-benzothiazine derivatives as novel anti-inflammatory agents
|
Szczęśniak-Sięga, Berenika M.
|
|
|
106 |
C |
p.
|
artikel
|
| 52 |
Synthesis, antidiabetic activity and molecular docking study of rhodanine-substitued spirooxindole pyrrolidine derivatives as novel α-amylase inhibitors
|
Toumi, Amani
|
|
|
106 |
C |
p.
|
artikel
|
| 53 |
Synthesis, biological activity and POM/DFT/docking analyses of annulated pyrano[2,3-d]pyrimidine derivatives: Identification of antibacterial and antitumor pharmacophore sites
|
Bhat, Ajmal R.
|
|
|
106 |
C |
p.
|
artikel
|
| 54 |
Synthesis, biological evaluation and QSAR studies of new thieno[2,3-d]pyrimidin-4(3H)-one derivatives as antimicrobial and antifungal agents
|
Magoulas, George E.
|
|
|
106 |
C |
p.
|
artikel
|
| 55 |
Synthesis, biological properties and structural study of new halogenated azolo[4,5-b]pyridines as inhibitors of CK2 kinase
|
Chojnacki, K.
|
|
|
106 |
C |
p.
|
artikel
|
| 56 |
Synthesis, characterization and anti-inflammatory properties of karanjin (Pongamia pinnata seed) and its derivatives
|
Rekha, M.J.
|
|
|
106 |
C |
p.
|
artikel
|
| 57 |
Synthesis, molecular docking, and in silico ADME/Tox profiling studies of new 1-aryl-5-(3-azidopropyl)indol-4-ones: Potential inhibitors of SARS CoV-2 main protease
|
Domínguez-Villa, Francisco Xavier
|
|
|
106 |
C |
p.
|
artikel
|
| 58 |
Synthesis of azachalcones, their α-amylase, α-glucosidase inhibitory activities, kinetics, and molecular docking studies
|
Saleem, Faiza
|
|
|
106 |
C |
p.
|
artikel
|
| 59 |
Synthesis of ring-opened derivatives of triazole-containing quinolinones and their antidepressant and anticonvulsant activities
|
Song, Ming-Xia
|
|
|
106 |
C |
p.
|
artikel
|
| 60 |
Targeting and imaging of HER2 overexpression tumor with a new peptide-based 68Ga-PET radiotracer
|
Biabani Ardakani, Javad
|
|
|
106 |
C |
p.
|
artikel
|
| 61 |
The relationship between stereochemical and both, pharmacological and ADME-Tox, properties of the potent hydantoin 5-HT7R antagonist MF-8
|
Kucwaj-Brysz, Katarzyna
|
|
|
106 |
C |
p.
|
artikel
|
| 62 |
Vibsane-type diterpenoids from Viburnum odoratissimum and their cytotoxic activities
|
Li, Shi-Fang
|
|
|
106 |
C |
p.
|
artikel
|
Tijdschrift beschrijving