nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Acylphloroglucinols with acetylcholinesterase inhibitory effects from the fruits of Eucalyptus robusta
|
Liu, Hui |
|
|
103 |
C |
p. |
artikel |
2 |
Annular oxygenation and rearrangement products of cryptotanshinone by biotransformation with marine-derived fungi Cochliobolus lunatus and Aspergillus terreus
|
Wu, Jing-Shuai |
|
|
103 |
C |
p. |
artikel |
3 |
Antioxidant activity of novel imidazo[2,1-b]thiazole derivatives: Design, synthesis, biological evaluation, molecular docking study and in silico ADME prediction
|
Dincel, Efe Doğukan |
|
|
103 |
C |
p. |
artikel |
4 |
2-Aryl benzazole derived new class of anti-tubercular compounds: Endowed to eradicate mycobacterium tuberculosis in replicating and non-replicating forms
|
Velappan, Anand Babu |
|
|
103 |
C |
p. |
artikel |
5 |
Attacking the mitochondria of colorectal carcinoma by novel 2-cyanoacrylamides linked to ethyl 1,3-diphenylpyrazole-4-carboxylates moiety as a new trend for chemotherapy
|
Mohamed, Magda F. |
|
|
103 |
C |
p. |
artikel |
6 |
Capsaicin: A “hot” KDM1A/LSD1 inhibitor from peppers
|
Jia, Gang |
|
|
103 |
C |
p. |
artikel |
7 |
Co-evolution of activity and thermostability of an aldo-keto reductase KmAKR for asymmetric synthesis of statin precursor dichiral diols
|
Qiu, Shuai |
|
|
103 |
C |
p. |
artikel |
8 |
Corrigendum to “The fatty acid amide hydrolase and cyclooxygenase-inhibitory properties of novel amide derivatives of carprofen” [Bioorg. Chem. 101 (2020) 104034]
|
Deplano, Alessandro |
|
|
103 |
C |
p. |
artikel |
9 |
Coumaric acid derivatives as tyrosinase inhibitors: Efficacy studies through in silico, in vitro and ex vivo approaches
|
Varela, Marina Themoteo |
|
|
103 |
C |
p. |
artikel |
10 |
Cytotoxic sesquiterpenoids against hepatic stellate cell line LX2 from Artemisia lavandulaefolia
|
Shen, Cheng |
|
|
103 |
C |
p. |
artikel |
11 |
Daphnanes diterpenes from the latex of Hura crepitans L. And activity against human colorectal cancer cells Caco-2
|
Trinel, Manon |
|
|
103 |
C |
p. |
artikel |
12 |
Derivatives of 1,2,4-triazole imines acting as dual iNOS and tumor cell growth inhibitors
|
Guillon, Christophe |
|
|
103 |
C |
p. |
artikel |
13 |
Design and synthesis of novel antimicrobial peptide scaffolds
|
Jakas, Andreja |
|
|
103 |
C |
p. |
artikel |
14 |
Design and synthesis of novel desfluoroquinolone-aminopyrimidine hybrids as potent anti-MRSA agents with low hERG activity
|
Song, Runzhe |
|
|
103 |
C |
p. |
artikel |
15 |
Design, synthesis and biological evaluation of dual-function inhibitors targeting NMDAR and HDAC for Alzheimer’s disease
|
He, Feng |
|
|
103 |
C |
p. |
artikel |
16 |
Design, synthesis and biological evaluation of imidazolidine-2,4-dione and 2-thioxothiazolidin-4-one derivatives as lymphoid-specific tyrosine phosphatase inhibitors
|
Liang, Xiao |
|
|
103 |
C |
p. |
artikel |
17 |
Design, synthesis and biological evaluation of novel (E)-N-phenyl-4-(pyridine-acylhydrazone) benzamide derivatives as potential antitumor agents for the treatment of multiple myeloma (MM)
|
Li, Xin-yang |
|
|
103 |
C |
p. |
artikel |
18 |
Design, synthesis and biological evaluation of triazole-oxadiazole conjugates for the management of cognitive dysfunction
|
Jain, Ankit |
|
|
103 |
C |
p. |
artikel |
19 |
Design, synthesis and molecular modeling of phenyl dihydropyridazinone derivatives as B-Raf inhibitors with anticancer activity
|
Thabit, Mohamed G. |
|
|
103 |
C |
p. |
artikel |
20 |
Design, synthesis, biological evaluation, and docking study of novel dual-acting thiazole-pyridiniums inhibiting acetylcholinesterase and β-amyloid aggregation for Alzheimer’s disease
|
Ghotbi, Golaleh |
|
|
103 |
C |
p. |
artikel |
21 |
Design, synthesis, molecular modeling, and biological evaluation of pyrazole-naphthalene derivatives as potential anticancer agents on MCF-7 breast cancer cells by inhibiting tubulin polymerization
|
Wang, Guangcheng |
|
|
103 |
C |
p. |
artikel |
22 |
Design, synthesis, molecular modeling, in vivo studies and anticancer activity evaluation of new phthalazine derivatives as potential DNA intercalators and topoisomerase II inhibitors
|
El-Helby, Abdel-Ghany A. |
|
|
103 |
C |
p. |
artikel |
23 |
Development of multitarget inhibitors for the treatment of pain: Design, synthesis, biological evaluation and molecular modeling studies
|
Wilt, Stephanie |
|
|
103 |
C |
p. |
artikel |
24 |
Diapolycopenedioic-acid-diglucosyl ester and keto-myxocoxanthin glucoside ester: Novel carotenoids derived from Exiguobacterium acetylicum S01 and evaluation of their anticancer and anti-inflammatory activities
|
Jinendiran, Sekar |
|
|
103 |
C |
p. |
artikel |
25 |
Diarylurea derivatives comprising 2,4-diarylpyrimidines: Discovery of novel potential anticancer agents via combined failed-ligands repurposing and molecular hybridization approaches
|
Farag, Ahmed Karam |
|
|
103 |
C |
p. |
artikel |
26 |
Direct inhibition of Keap1-Nrf2 Protein-Protein interaction as a potential therapeutic strategy for Alzheimer's disease
|
Sun, Yi |
|
|
103 |
C |
p. |
artikel |
27 |
Discovery of new benzhydrol biscarbonate esters as potent and selective apoptosis inducers of human melanomas bearing the activated ERK pathway: SAR studies on an ERK MAPK signaling modulator, ACA-28
|
Satoh, Ryosuke |
|
|
103 |
C |
p. |
artikel |
28 |
Diterpenoids from Cephalotaxus fortunei var. alpina and their cytotoxic activity
|
Li, Yanzhi |
|
|
103 |
C |
p. |
artikel |
29 |
Editorial Board
|
|
|
|
103 |
C |
p. |
artikel |
30 |
Evaluation of anti rheumatic activity of Piper betle L. (Betelvine) extract using in silico, in vitro and in vivo approaches
|
Murugesan, Selvakumar |
|
|
103 |
C |
p. |
artikel |
31 |
From orexin receptor agonist YNT-185 to novel antagonists with drug-like properties for the treatment of insomnia
|
Mezeiova, Eva |
|
|
103 |
C |
p. |
artikel |
32 |
Hydroxynaphthalenecarboxamides and substituted piperazinylpropandiols, two new series of BRAF inhibitors. A theoretical and experimental study
|
Campos, Ludmila E. |
|
|
103 |
C |
p. |
artikel |
33 |
Identification and structure–activity relationship (SAR) studies of carvacrol derivatives as potential anti-malarial against Plasmodium falciparum falcipain-2 protease
|
Uddin, Amad |
|
|
103 |
C |
p. |
artikel |
34 |
Indolizine-phenothiazine hybrids as the first dual inhibitors of tubulin polymerization and farnesyltransferase with synergistic antitumor activity
|
Moise, Iuliana-Monica |
|
|
103 |
C |
p. |
artikel |
35 |
Inhibition of colitis by ring-modified analogues of 6-acetamido-2,4,5-trimethylpyridin-3-ol
|
Chaudhary, Chhabi Lal |
|
|
103 |
C |
p. |
artikel |
36 |
Interactions of tolcapone analogues as stabilizers of the amyloidogenic protein transthyretin
|
Loconte, Valentina |
|
|
103 |
C |
p. |
artikel |
37 |
Issue TOC
|
|
|
|
103 |
C |
p. |
artikel |
38 |
Jasmonates from Chinese acorns (Quercus serrata var. brevipetiolata) exert pronounced anti-neuroinflammatory activities
|
Wang, Yihai |
|
|
103 |
C |
p. |
artikel |
39 |
Molecular modelling guided design, synthesis and QSAR analysis of new small molecule non-lipid autotaxin inhibitors
|
Banerjee, Souvik |
|
|
103 |
C |
p. |
artikel |
40 |
N-Cyclohexylimidazo[1,2-a]pyridine derivatives as multi-target-directed ligands for treatment of Alzheimer's disease
|
Haghighijoo, Zahra |
|
|
103 |
C |
p. |
artikel |
41 |
New antimicrobial terpenoids and phloroglucinol glucosides from Syzygium szemaoense
|
Xu, Wen |
|
|
103 |
C |
p. |
artikel |
42 |
New fused pyrimidine derivatives with anticancer activity: Synthesis, topoisomerase II inhibition, apoptotic inducing activity and molecular modeling study
|
Nemr, Mohamed T.M. |
|
|
103 |
C |
p. |
artikel |
43 |
Novel 2′-alkoxymethyl substituted klavuzon derivatives as inhibitors of Topo I and CRM1
|
Çetinkaya, Hakkı |
|
|
103 |
C |
p. |
artikel |
44 |
Novel CoFe2O4@ZnO-CeO2 ternary nanocomposite: Sonochemical green synthesis using Crataegus microphylla extract, characterization and their application in catalytic and antibacterial activities
|
Naghizadeh, Ali |
|
|
103 |
C |
p. |
artikel |
45 |
Novel HLA-A2 restricted antigenic peptide derivatives with high affinity for the treatment of breast cancer expressing NY-ESO-1
|
Shi, Wei |
|
|
103 |
C |
p. |
artikel |
46 |
Novel scaffold hopping of potent benzothiazole and isatin analogues linked to 1,2,3-triazole fragment that mimic quinazoline epidermal growth factor receptor inhibitors: Synthesis, antitumor and mechanistic analyses
|
Rezki, Nadjet |
|
|
103 |
C |
p. |
artikel |
47 |
Novel Schiff bases derived from N-aryl maleimide derivatives as an effective antimicrobial agent: Theoretical and experimental approach
|
Bhagare, Arun M. |
|
|
103 |
C |
p. |
artikel |
48 |
NQO1-selective activated prodrugs of combretastatin A-4: Synthesis and biological evaluation
|
Zhang, Chong |
|
|
103 |
C |
p. |
artikel |
49 |
Porcine pancreas lipase as a green catalyst for synthesis of bis-4-hydroxy coumarins
|
Bavandi, Hossein |
|
|
103 |
C |
p. |
artikel |
50 |
Preparation and optimization of ciprofloxacin encapsulated niosomes: A new approach for enhanced antibacterial activity, biofilm inhibition and reduced antibiotic resistance in ciprofloxacin-resistant methicillin-resistance Staphylococcus aureus
|
Mirzaie, Amir |
|
|
103 |
C |
p. |
artikel |
51 |
Pyridinium derivatives of 3-aminobenzenesulfonamide are nanomolar-potent inhibitors of tumor-expressed carbonic anhydrase isozymes CA IX and CA XII
|
Akocak, Suleyman |
|
|
103 |
C |
p. |
artikel |
52 |
Rare new bicyclic cembranoid ethers and a novel trihydroxy prenylated guaiane from the Xisha soft coral Lobophytum sp
|
Li, Song-Wei |
|
|
103 |
C |
p. |
artikel |
53 |
Rational design of a far-red fluorescent probe for endogenous biothiol imbalance induced by hydrogen peroxide in living cells and mice
|
Lu, Zhengliang |
|
|
103 |
C |
p. |
artikel |
54 |
Rational design, synthesis and biological evaluation of triphenylphosphonium-ginsenoside conjugates as mitochondria-targeting anti-cancer agents
|
Ma, Lu |
|
|
103 |
C |
p. |
artikel |
55 |
Recent advancements of coumarin-based anticancer agents: An up-to-date review
|
Al-Warhi, Tarfah |
|
|
103 |
C |
p. |
artikel |
56 |
Recent advances in the development of ligands specifically targeting telomeric multimeric G-quadruplexes
|
Zhao, Jingfang |
|
|
103 |
C |
p. |
artikel |
57 |
Selective VEGFR-2 inhibitors: Synthesis of pyridine derivatives, cytotoxicity and apoptosis induction profiling
|
AbdelHaleem, Amal |
|
|
103 |
C |
p. |
artikel |
58 |
Sesquineolignan and neolignan enantiomers from Triadica sebifera
|
Yu, Min |
|
|
103 |
C |
p. |
artikel |
59 |
Stomopneulactone D from long-spined sea urchin Stomopneustes variolaris: Anti-inflammatory macrocylic lactone attenuates cyclooxygenase-2 expression in lipopolysaccharide-activated macrophages
|
Chakraborty, Kajal |
|
|
103 |
C |
p. |
artikel |
60 |
Structurally diverse sesquiterpenoids from the aerial parts of Artemisia annua (Qinghao) and their striking systemically anti-inflammatory activities
|
Qin, Da-Peng |
|
|
103 |
C |
p. |
artikel |
61 |
Sunset yellow degradation product, as an efficient water-soluble inducer, accelerates 1N4R Tau amyloid oligomerization: In vitro preliminary evidence against the food colorant safety in terms of “Triggered Amyloid Aggregation”
|
Ojaghi, Sara |
|
|
103 |
C |
p. |
artikel |
62 |
Synthesis and antitumor effects of novel 18β-glycyrrhetinic acid derivatives featuring an exocyclic α,β-unsaturated carbonyl moiety in ring A
|
Huang, Min |
|
|
103 |
C |
p. |
artikel |
63 |
Synthesis and biological evaluation of 2′-Aminochalcone: A multi-target approach to find drug candidates to treat Alzheimer’s disease
|
Sakata, Renata P. |
|
|
103 |
C |
p. |
artikel |
64 |
Synthesis and biological evaluation of substituted N-(2-(1H-benzo[d]imidazol-2-yl)phenyl)cinnamides as tubulin polymerization inhibitors
|
Donthiboina, Kavitha |
|
|
103 |
C |
p. |
artikel |
65 |
Synthesis of 3,4-dihydroquinolin-2(1H)-one derivatives with anticonvulsant activity and their binding to the GABAA receptor
|
Wang, Shiben |
|
|
103 |
C |
p. |
artikel |
66 |
Synthesis of nitrogen, phosphorus, selenium and sulfur-containing heterocyclic compounds – Determination of their carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibition properties
|
Gülçin, İlhami |
|
|
103 |
C |
p. |
artikel |
67 |
Synthesis, optimization and characterization of silver nanoparticles using the catkin extract of Piper longum for bactericidal effect against food-borne pathogens via conventional and mathematical approaches
|
Huang, Hui |
|
|
103 |
C |
p. |
artikel |
68 |
Synthesis, trypanocidal and anti-leishmania activity of new triazole-lapachol and nor-lapachol hybrids
|
Pertino, Mariano Walter |
|
|
103 |
C |
p. |
artikel |
69 |
Unconventional amino acids in medicinal chemistry: First report on taurine merged within carbonic anhydrase inhibitors
|
Akgül, Özlem |
|
|
103 |
C |
p. |
artikel |