nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Anti-tyrosinase, anti-cholinesterase and cytotoxic activities of extracts and phytochemicals from the Tunisian Citharexylum spinosum L.: Molecular docking and SAR analysis
|
Saidi, Ilyes |
|
|
102 |
C |
p. |
artikel |
2 |
Asymmetric trisalkylamine cyclopropenium derivatives with antimicrobial activity
|
Belay, Chen |
|
|
102 |
C |
p. |
artikel |
3 |
Cytotoxic bufadienolides from the leaves of a medicinal plant Melianthus comosus collected in South Africa
|
Bedane, Kibrom Gebreheiwot |
|
|
102 |
C |
p. |
artikel |
4 |
Design and synthesis of new 1,6-dihydropyrimidin-2-thio derivatives targeting VEGFR-2: Molecular docking and antiproliferative evaluation
|
Marzouk, Adel A. |
|
|
102 |
C |
p. |
artikel |
5 |
Design and synthesis of novel pyridazine N-aryl acetamides: In-vitro evaluation of α-glucosidase inhibition, docking, and kinetic studies
|
Moghimi, Setareh |
|
|
102 |
C |
p. |
artikel |
6 |
Design and synthesis of pinane oxime derivatives as novel anti-influenza agents
|
Dong, Jianghong |
|
|
102 |
C |
p. |
artikel |
7 |
Design of peptide-based inhibitor agent against amyloid-β aggregation: Molecular docking, synthesis and in vitro evaluation
|
Jokar, Safura |
|
|
102 |
C |
p. |
artikel |
8 |
Design, synthesis ADMET and molecular docking of new imidazo[4,5-b]pyridine-5-thione derivatives as potential tyrosyl-tRNA synthetase inhibitors
|
Othman, Ismail M.M. |
|
|
102 |
C |
p. |
artikel |
9 |
Design, synthesis and anti-HIV evaluation of 5-alkyl- 6-(benzo[d][1,3]dioxol-5-alkyl)-2-mercaptopyrimidin-4(3H)-ones as potent HIV-1 NNRTIs
|
Li, Yi-Ming |
|
|
102 |
C |
p. |
artikel |
10 |
Design, synthesis and antimycobacterial activity of new benzothiazinones inspired by rifampicin/rifapentine
|
Wang, Apeng |
|
|
102 |
C |
p. |
artikel |
11 |
Design, synthesis and biological evaluation of methylenehydrazine-1-carboxamide derivatives with (5-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)-1H-indole scaffold: Novel potential CDK9 inhibitors
|
Hu, Hongyu |
|
|
102 |
C |
p. |
artikel |
12 |
Design, synthesis and biological evaluation of novel triaryldimethylaminobutan-2-ol derivatives against Mycobacterium tuberculosis
|
Liu, Ping |
|
|
102 |
C |
p. |
artikel |
13 |
Design, synthesis and biological evaluation of some new 2-Pyrazoline derivatives as potential anticancer agents
|
Tok, Fatih |
|
|
102 |
C |
p. |
artikel |
14 |
Design, synthesis and SARs of novel telomerase inhibitors based on BIBR1532
|
Liu, Chao |
|
|
102 |
C |
p. |
artikel |
15 |
Design, synthesis, anti-tobacco mosaic viral and molecule docking simulations of urea/thiourea derivatives of 2-(piperazine-1-yl)-pyrimidine and 1-(4-Fluoro/4-Chloro phenyl)-piperazine and 1-(4-Chloro phenyl)-piperazine – A study
|
Nagalakshmamma, Vadabingi |
|
|
102 |
C |
p. |
artikel |
16 |
Design, synthesis, biological evaluation and in silico studies of novel pyrrolo[3,4-d]pyridazinone derivatives withpromising anti-inflammatory and antioxidant activity
|
Szczukowski, Łukasz |
|
|
102 |
C |
p. |
artikel |
17 |
Design, synthesis, in vitro and in silico investigation of aldose reductase inhibitory effects of new thiazole-based compounds
|
Sever, Belgin |
|
|
102 |
C |
p. |
artikel |
18 |
Design, synthesis, molecular docking and anticancer evaluations of 5-benzylidenethiazolidine-2,4-dione derivatives targeting VEGFR-2 enzyme
|
El-Adl, Khaled |
|
|
102 |
C |
p. |
artikel |
19 |
Development of sulfonamide-based Schiff bases targeting urease inhibition: Synthesis, characterization, inhibitory activity assessment, molecular docking and ADME studies
|
Hamad, Asad |
|
|
102 |
C |
p. |
artikel |
20 |
Differential lethal action of C17:2 and C17:0 anacardic acid derivatives in Trypanosoma cruzi – A mechanistic study
|
Umehara, Eric |
|
|
102 |
C |
p. |
artikel |
21 |
Discovery of 7H-pyrrolo[2,3-d]pyridine derivatives as potent FAK inhibitors: Design, synthesis, biological evaluation and molecular docking study
|
Wang, Ruifeng |
|
|
102 |
C |
p. |
artikel |
22 |
Discovery of new ATP-competitive inhibitors of human DNA topoisomerase IIα through screening of bacterial topoisomerase inhibitors
|
Skok, Žiga |
|
|
102 |
C |
p. |
artikel |
23 |
Discovery of novel aminophosphonate derivatives containing pyrazole moiety as potential selective COX-2 inhibitors
|
Zhang, Bo |
|
|
102 |
C |
p. |
artikel |
24 |
1,3-Disubstituted urea derivatives: Synthesis, antimicrobial activity evaluation and in silico studies
|
Gündüz, Miyase Gözde |
|
|
102 |
C |
p. |
artikel |
25 |
Editorial Board
|
|
|
|
102 |
C |
p. |
artikel |
26 |
Exploiting the 4-hydrazinobenzoic acid moiety for the development of anticancer agents: Synthesis and biological profile
|
Abuelizz, Hatem A. |
|
|
102 |
C |
p. |
artikel |
27 |
Exploring the interaction between citrus flavonoids and phytopathogenic fungi through enzymatic activities
|
Costa, Jonas Henrique |
|
|
102 |
C |
p. |
artikel |
28 |
Flavone inspired discovery of benzylidenebenzofuran-3(2H)-ones (aurones) as potent inhibitors of human protein kinase CK2
|
Protopopov, M.V. |
|
|
102 |
C |
p. |
artikel |
29 |
Four new sucrose diesters of substituted truxinic acids from Trigonostemon honbaensis with their anoctamin-1 inhibitory activity
|
Ban, Ninh Khac |
|
|
102 |
C |
p. |
artikel |
30 |
Identification of novel scaffold using ligand and structure based approach targeting shikimate kinase
|
Rahul Reddy, M.B. |
|
|
102 |
C |
p. |
artikel |
31 |
Insight into antimicrobial activity of substituted phenylcarbamoyloxypiperazinylpropanols
|
Pospisilova, Sarka |
|
|
102 |
C |
p. |
artikel |
32 |
Inula japonica ameliorated bleomycin-induced pulmonary fibrosis via inhibiting soluble epoxide hydrolase
|
Zhao, Wen-Yu |
|
|
102 |
C |
p. |
artikel |
33 |
In vitro C132-dealkoxycarbonylations of zinc chlorophyll a derivatives including C132-substitutes by a BciC enzyme
|
Hirose, Mitsuaki |
|
|
102 |
C |
p. |
artikel |
34 |
Issue TOC
|
|
|
|
102 |
C |
p. |
artikel |
35 |
177Lu-labeled cyclic RGD peptide as an imaging and targeted radionuclide therapeutic agent in non-small cell lung cancer: Biological evaluation and preclinical study
|
Pirooznia, Nazanin |
|
|
102 |
C |
p. |
artikel |
36 |
Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists
|
Shahien, Mohamed |
|
|
102 |
C |
p. |
artikel |
37 |
Monoterpene indole alkaloids with acetylcholinesterase inhibitory activity from the leaves of Rauvolfia vomitoria
|
Zhan, Guanqun |
|
|
102 |
C |
p. |
artikel |
38 |
N-Acetyldopamine derivatives from Periostracum Cicadae and their regulatory activities on Th1 and Th17 cell differentiation
|
Thapa, Punam |
|
|
102 |
C |
p. |
artikel |
39 |
N-alkylated linear heptamethine polyenes as potent non-azole leads against Candida albicans fungal infections
|
Lawrence, Clare L. |
|
|
102 |
C |
p. |
artikel |
40 |
Novel antiproliferative agents bearing morpholinopyrimidine scaffold as PI3K inhibitors and apoptosis inducers; design, synthesis and molecular docking
|
Helwa, Amira A. |
|
|
102 |
C |
p. |
artikel |
41 |
Novel benzimidazole-triazole hybrids as apoptosis inducing agents in lung cancer: Design, synthesis, 18F-radiolabeling & galectin-1 inhibition studies
|
Sridhar Goud, Nerella |
|
|
102 |
C |
p. |
artikel |
42 |
Novel bis(pyrazole-benzofuran) hybrids possessing piperazine linker: Synthesis of potent bacterial biofilm and MurB inhibitors
|
Mekky, Ahmed E.M. |
|
|
102 |
C |
p. |
artikel |
43 |
Novel N-substituted 5-phosphate-d-arabinonamide derivatives as strong inhibitors of phosphoglucose isomerases: Synthesis, structure-activity relationship and crystallographic studies
|
Ahmad, Lama |
|
|
102 |
C |
p. |
artikel |
44 |
Novel panaxadiol triazole derivatives induce apoptosis in HepG-2 cells through the mitochondrial pathway
|
Xiao, Shengnan |
|
|
102 |
C |
p. |
artikel |
45 |
Phytosterols demonstrate selective inhibition of COX-2: In-vivo and in-silico studies of Nicotiana tabacum
|
Akinloye, O. Adeboye |
|
|
102 |
C |
p. |
artikel |
46 |
Poncirin, an orally active flavonoid exerts antidiabetic complications and improves glucose uptake activating PI3K/Akt signaling pathway in insulin resistant C2C12 cells with anti-glycation capacities
|
Yousof Ali, Md |
|
|
102 |
C |
p. |
artikel |
47 |
Probing 2-acetylbenzofuran hydrazones and their metal complexes as α-glucosidase inhibitors
|
Khan, Samra |
|
|
102 |
C |
p. |
artikel |
48 |
p-TSA.H2O mediated one-pot, multi-component synthesis of isatin derived imidazoles as dual-purpose drugs against inflammation and cancer
|
Rajesh Kumar, M. |
|
|
102 |
C |
p. |
artikel |
49 |
(+)-(R)- and (−)-(S)-Perhexiline maleate: Enantioselective synthesis and functional studies on Schistosoma mansoni larval and adult stages
|
Guidi, Alessandra |
|
|
102 |
C |
p. |
artikel |
50 |
Rare benzonaphthoxanthenones from Chinese folk herbal medicine Polytrichum commune and their anti-neuroinflammatory activities in vitro
|
Guo, Zi-feng |
|
|
102 |
C |
p. |
artikel |
51 |
Self assembly and hydrogelation of N-terminal modified tetrapeptide for sustained release and synergistic action of antibacterial drugs against methicillin resistant S. aureus
|
Prasad Dewangan, Rikeshwer |
|
|
102 |
C |
p. |
artikel |
52 |
Structural characterization, antiproliferative and anti-inflammatory activities of alkaloids from the roots of Zanthoxylum austrosinense
|
Fu, Yan-Hui |
|
|
102 |
C |
p. |
artikel |
53 |
Structural determination and in vitro tumor cytotoxicity evaluation of five new cycloartane glycosides from Asplenium ruprechtii Sa. Kurata
|
Wang, Fang |
|
|
102 |
C |
p. |
artikel |
54 |
Sulfur and nitrogen-containing compounds from the whole bodies of Blaps japanensis
|
Yan, Yong-Ming |
|
|
102 |
C |
p. |
artikel |
55 |
Symmetric benzidine derivatives as anti-HCV agents: Insight into the nature, stereochemistry of the capping amino acid and the size of the terminal capping carbamates
|
Abdel Karim, Shereen E. |
|
|
102 |
C |
p. |
artikel |
56 |
Syntheses, quantum mechanical modeling, biomolecular interaction and in vitro anticancer – Tubulin activity of thiosemicarbazones
|
Xavier, Janet Sabina |
|
|
102 |
C |
p. |
artikel |
57 |
Synthesis and biological evaluation of benzofuran-based 3,4,5-trimethoxybenzamide derivatives as novel tubulin polymerization inhibitors
|
Li, Qiu |
|
|
102 |
C |
p. |
artikel |
58 |
Synthesis and DNA binding of novel bioactive thiazole derivatives pendent to N-phenylmorpholine moiety
|
Farghaly, Thoraya A. |
|
|
102 |
C |
p. |
artikel |
59 |
Synthesis and evaluation of sulfonyl piperazine LpxH inhibitors
|
Kwak, Seung-Hwa |
|
|
102 |
C |
p. |
artikel |
60 |
Synthesis and in vitro antitubercular activity of pyridine analouges against the resistant Mycobacterium tuberculosis
|
Patel, Harun |
|
|
102 |
C |
p. |
artikel |
61 |
Synthesis, biological evaluation and docking studies of a novel class of sulfur-bridged diazabicyclo[3.3.1]nonanes
|
Murineddu, Gabriele |
|
|
102 |
C |
p. |
artikel |
62 |
Synthesis, characterization and SAR studies of bis(imino)pyridines as antioxidants, acetylcholinesterase inhibitors and antimicrobial agents
|
Milošević, Milena D. |
|
|
102 |
C |
p. |
artikel |
63 |
Synthesis, characterization, in vitro tissue-nonspecific alkaline phosphatase (TNAP) and intestinal alkaline phosphatase (IAP) inhibition studies and computational evaluation of novel thiazole derivatives
|
Aziz, Hamid |
|
|
102 |
C |
p. |
artikel |
64 |
Synthesis, cytotoxicity of some pyrazoles and pyrazolo[1,5-a]pyrimidines bearing benzothiazole moiety and investigation of their mechanism of action
|
Husseiny, Ebtehal M. |
|
|
102 |
C |
p. |
artikel |
65 |
Synthesis, docking and evaluation of in vitro anti-inflammatory activity of novel morpholine capped β-lactam derivatives
|
Heiran, Roghayeh |
|
|
102 |
C |
p. |
artikel |
66 |
Synthesis, docking studies and antitumor activity of phenanthroimidazole derivatives as promising c-myc G-quadruplex DNA stabilizers
|
Wu, Qiong |
|
|
102 |
C |
p. |
artikel |
67 |
Synthesis, docking study and inhibitory activity of 2,6-diketopiperazines derived from α-amino acids on HDAC8
|
Garrido González, Flor Paulina |
|
|
102 |
C |
p. |
artikel |
68 |
Synthesis, in vivo anti-inflammatory, COX-1/COX-2 and 5-LOX inhibitory activities of new 2,3,4-trisubstituted thiophene derivatives
|
Qandeel, Nermeen A. |
|
|
102 |
C |
p. |
artikel |
69 |
Synthesis of a far-red emitting flavonoid-based lysosome marker for live cell imaging applications
|
Bertman, Keti Assor |
|
|
102 |
C |
p. |
artikel |
70 |
Synthesis of 2,3-dihydrobenzo[b][1,4]dioxine-5-carboxamide and 3-oxo-3,4-dihydrobenzo[b][1,4]oxazine-8-carboxamide derivatives as PARP1 inhibitors
|
Shao, Xuwei |
|
|
102 |
C |
p. |
artikel |
71 |
Synthetic flavonoid derivatives targeting the glycogen phosphorylase inhibitor site: QM/MM-PBSA motivated synthesis of substituted 5,7-dihydroxyflavones, crystallography, in vitro kinetics and ex-vivo cellular experiments reveal novel potent inhibitors
|
Chetter, Ben A. |
|
|
102 |
C |
p. |
artikel |
72 |
Ten new glycosides, carissaedulosides A–J from the root barks of Carissa edulis and their cytotoxicities
|
Kaunda, Joseph Sakah |
|
|
102 |
C |
p. |
artikel |
73 |
Terpenoids from stigma maydis (Zea mays L.) alleviate hydrogen peroxide-induced SH-SY5Y cell injury by activating Nrf2
|
Song, Xiao-Yu |
|
|
102 |
C |
p. |
artikel |
74 |
Tolnaftate inhibits ergosterol production and impacts cell viability of Leishmania sp.
|
Yamamoto, Eduardo Seiji |
|
|
102 |
C |
p. |
artikel |