nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
6-Acetyl-5-hydroxy-4,7-dimethylcoumarin derivatives: Design, synthesis, modeling studies, 5-HT1A, 5-HT2A and D2 receptors affinity
|
Ostrowska, Kinga |
|
|
100 |
C |
p. |
artikel |
2 |
An acylhydroquinone derivative produces OXPHOS uncoupling and sensitization to BH3 mimetic ABT-199 (Venetoclax) in human promyelocytic leukemia cells
|
Donoso-Bustamante, Viviana |
|
|
100 |
C |
p. |
artikel |
3 |
An okadaic acid fragment analogue prevents nicotine-induced resistance to cisplatin by recovering PP2A activity in non-small cell lung cancer cells
|
Arribas, Raquel L. |
|
|
100 |
C |
p. |
artikel |
4 |
A novel fluorescent sensor for specific recognition of GSH based on the copper complex and its bioimaging in living cells
|
Li, Shengling |
|
|
100 |
C |
p. |
artikel |
5 |
Antibacterial activities and DNA-cleavage properties of novel fluorescent imidazo-phenanthroline derivatives
|
Obalı, Aslıhan Yılmaz |
|
|
100 |
C |
p. |
artikel |
6 |
Anti-inflammatory octahydroindolizine alkaloid enantiomers from Dendrobium crepidatum
|
Hu, Yang |
|
|
100 |
C |
p. |
artikel |
7 |
Antimalarial diterpenoids from Vitex rotundifolia: Isolation, structure elucidation, and in vitro antiplasmodial activity
|
Kim, You Ah |
|
|
100 |
C |
p. |
artikel |
8 |
Benzofuran-selenadiazole hybrids as novel α-glucosidase and cyclooxygenase-2 inhibitors with antioxidant and cytotoxic properties
|
Olomola, Temitope O. |
|
|
100 |
C |
p. |
artikel |
9 |
Bioinformatic and biochemical findings disclosed anti-hepatic steatosis mechanism of calycosin
|
Cheng, Xuebing |
|
|
100 |
C |
p. |
artikel |
10 |
Bioisosteric investigation of ebselen: Synthesis and in vitro characterization of 1,2-benzisothiazol-3(2H)-one derivatives as potent New Delhi metallo-β-lactamase inhibitors
|
Jin, Wen Bin |
|
|
100 |
C |
p. |
artikel |
11 |
Calix[6]arene diminishes receptor tyrosine kinase lifespan in pancreatic cancer cells and inhibits their migration and invasion efficiency
|
Rocha-Brito, Karin Juliane Pelizzaro |
|
|
100 |
C |
p. |
artikel |
12 |
Corrigendum to “Optimization of the benzamide fragment targeting the S2′ site leads to potent dipeptidyl Peptidase-IV inhibitors” [Bioorg. Chem. 94 (2020) 103366]
|
Deng, Xiaoyan |
|
|
100 |
C |
p. |
artikel |
13 |
Corrigendum to “Technetium-99 m-PEGylated dendrimer-G2-(Dabcyle-Lys6,Phe7)-pHBSP: A novel Nano-Radiotracer for molecular and early detecting of cardiac ischemic region” [Bioorg. Chem. 98 (2020) 103731]
|
Mohtavinejad, Naser |
|
|
100 |
C |
p. |
artikel |
14 |
Design, synthesis and anticancer/antiestrogenic activities of novel indole-benzimidazoles
|
Karadayi, Fikriye Zengin |
|
|
100 |
C |
p. |
artikel |
15 |
Design, synthesis and antitrypanosomal activity of heteroaryl-based 1,2,4-triazole and 1,3,4-oxadiazole derivatives
|
Shaykoon, Montaser Sh. |
|
|
100 |
C |
p. |
artikel |
16 |
Design, synthesis and biological evaluation of novel Pseudomonas aeruginosa DNA gyrase B inhibitors
|
Jogula, Sridhar |
|
|
100 |
C |
p. |
artikel |
17 |
Design, synthesis and biological evaluation of pyridine derivatives as selective SHP2 inhibitors
|
Liu, Wen-Shan |
|
|
100 |
C |
p. |
artikel |
18 |
Design, synthesis, and evaluation of a novel benzamidine-based inhibitor of VEGF-C binding to Neuropilin-2
|
Said, Ahmed M. |
|
|
100 |
C |
p. |
artikel |
19 |
Design, synthesis and evaluation of novel nonquaternary and 3 non-oxime reactivators for acetylcholinesterase inhibited by organophosphates
|
Bi, Huanglei |
|
|
100 |
C |
p. |
artikel |
20 |
Design, synthesis, and pharmacological evaluation of novel and selective COX-2 inhibitors based on bumetanide scaffold
|
Ibrahim, Tarek S. |
|
|
100 |
C |
p. |
artikel |
21 |
Design, synthesis, DNA binding studies and evaluation of anticancer potential of novel substituted biscarbazole derivatives against human glioma U87 MG cell line
|
Kumar, Nitin |
|
|
100 |
C |
p. |
artikel |
22 |
Development of a selective inhibitor for Kv1.1 channels prevalent in demyelinated nerves
|
Al-Sabi, Ahmed |
|
|
100 |
C |
p. |
artikel |
23 |
DFT calculations and POM analyses of cytotoxicity of some flavonoids from aerial parts of Cupressus sempervirens: Docking and identification of pharmacophore sites
|
Elsharkawy, Eman R. |
|
|
100 |
C |
p. |
artikel |
24 |
Dihydroartemisinin ameliorates dextran sulfate sodium induced inflammatory bowel diseases in mice
|
Lei, Zili |
|
|
100 |
C |
p. |
artikel |
25 |
Discovery of deoxylimonin δ-lactam derivative with favorable anti-inflammation and antinociception efficacy from chemical modified limonin/deoxylimonin analogs
|
Wang, Shaochi |
|
|
100 |
C |
p. |
artikel |
26 |
Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation
|
Upadhyay, Neha |
|
|
100 |
C |
p. |
artikel |
27 |
Discovery of 1,2,3-triazole based quinoxaline-1,4-di-N-oxide derivatives as potential anti-tubercular agents
|
Srinivasarao, Singireddi |
|
|
100 |
C |
p. |
artikel |
28 |
Discovery of triazoloquinoxaline as novel STING agonists via structure-based virtual screening
|
Hou, Hui |
|
|
100 |
C |
p. |
artikel |
29 |
Dispiropyrrolidine tethered piperidone heterocyclic hybrids with broad-spectrum antifungal activity against Candida albicans and Cryptococcus neoformans
|
Lawson, Sarah |
|
|
100 |
C |
p. |
artikel |
30 |
Editorial Board
|
|
|
|
100 |
C |
p. |
artikel |
31 |
Effectiveness of deferiprone-loaded nanocarrier in experimentally induced rhabdomyolysis: A dose-comparison study
|
Rashed, Rasha Refaat |
|
|
100 |
C |
p. |
artikel |
32 |
Evaluation radioprotective effect of curcumin conjugated albumin nanoparticles
|
Nosrati, Hamed |
|
|
100 |
C |
p. |
artikel |
33 |
Exhibiting the diagnostic face of selenium nanoparticles as a radio-platform for tumor imaging
|
Korany, Mohamed |
|
|
100 |
C |
p. |
artikel |
34 |
Exploring interaction dynamics of designed organic cocrystal charge transfer complex of 2-hydroxypyridine and oxalic acid with human serum albumin: Single crystal, spectrophotometric, theoretical and antimicrobial studies
|
Khan, Ishaat M. |
|
|
100 |
C |
p. |
artikel |
35 |
Functionalized aromatic esters of the Amaryllidaceae alkaloid haemanthamine and their in vitro and in silico biological activity connected to Alzheimer’s disease
|
Peřinová, Rozálie |
|
|
100 |
C |
p. |
artikel |
36 |
Furanasperterpenes A and B, two meroterpenoids with a novel 6/6/6/6/5 ring system from the marine-derived fungus Aspergillus terreus GZU-31-1
|
Tang, Yuqian |
|
|
100 |
C |
p. |
artikel |
37 |
Fusicoccane-derived diterpenoids with bridgehead double-bond-containing tricyclo[9.2.1.03,7]tetradecane ring systems from Alternaria brassicicola
|
Li, Fengli |
|
|
100 |
C |
p. |
artikel |
38 |
Hopane-type triterpenes from Cnidoscolus spinosus and their bioactivities
|
López-Huerta, Fabiola A. |
|
|
100 |
C |
p. |
artikel |
39 |
Identification and development of thiazole leads as COX-2/5-LOX inhibitors through in-vitro and in-vivo biological evaluation for anti-inflammatory activity
|
Jacob P, Jaismy |
|
|
100 |
C |
p. |
artikel |
40 |
Interaction of an abiraterone with calf thymus DNA: Investigation with spectroscopic technique and modelling studies
|
Wani, Tanveer A. |
|
|
100 |
C |
p. |
artikel |
41 |
In vitro cytotoxic activity of thiazole-indenoquinoxaline hybrids as apoptotic agents, design, synthesis, physicochemical and pharmacokinetic studies
|
Fayed, Eman A. |
|
|
100 |
C |
p. |
artikel |
42 |
Issue TOC
|
|
|
|
100 |
C |
p. |
artikel |
43 |
Limonoids and tricyclic diterpenoids from Azadirachta indica and their antitumor activities
|
Zhu, Wan-fang |
|
|
100 |
C |
p. |
artikel |
44 |
Linolenic fatty acid hydroperoxide acts as biocide on plant pathogenic bacteria: Biophysical investigation of the mode of action
|
Estelle, Deboever |
|
|
100 |
C |
p. |
artikel |
45 |
Mammea type coumarins isolated from Calophyllum brasiliense induced apoptotic cell death of Trypanosoma cruzi through mitochondrial dysfunction, ROS production and cell cycle alterations
|
Rodríguez-Hernández, Karla Daniela |
|
|
100 |
C |
p. |
artikel |
46 |
Melanogenesis-inhibitory activities of limonoids and tricyclic diterpenoids from Azadirachta indica
|
Su, Shengzhi |
|
|
100 |
C |
p. |
artikel |
47 |
Merulinic acid C overcomes gentamicin resistance in Enterococcus faecium
|
Rodrigues-Costa, Fernanda |
|
|
100 |
C |
p. |
artikel |
48 |
Modified pyrazole platinum(II) complex can circumvent albumin and glutathione: Synthesis, structure and cytotoxic activity
|
Querino, Ana Luiza de Andrade |
|
|
100 |
C |
p. |
artikel |
49 |
N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions
|
Poli, Giulio |
|
|
100 |
C |
p. |
artikel |
50 |
New insight into nucleo α-amino acids – Synthesis and SAR studies on cytotoxic activity of β-pyrimidine alanines
|
Ignatowska, Jolanta |
|
|
100 |
C |
p. |
artikel |
51 |
New lupane bidesmosides exhibiting strong cytotoxic activities in vitro
|
Korda, Anna |
|
|
100 |
C |
p. |
artikel |
52 |
New pyrazolopyrimidine derivatives with anticancer activity: Design, synthesis, PIM-1 inhibition, molecular docking study and molecular dynamics
|
Philoppes, John N. |
|
|
100 |
C |
p. |
artikel |
53 |
Novel coumarin-thiazolyl ester derivatives as potential DNA gyrase Inhibitors: Design, synthesis, and antibacterial activity
|
Liu, Hao |
|
|
100 |
C |
p. |
artikel |
54 |
Novel formyl peptide receptor (FPR) agonists with pyridinone and pyrimidindione scaffolds that are potentially useful for the treatment of rheumatoid arthritis
|
Crocetti, Letizia |
|
|
100 |
C |
p. |
artikel |
55 |
Novel pyranopyrazole derivatives comprising a benzoxazole core as antimicrobial inhibitors: Design, synthesis, microbial resistance and machine aided results
|
Reddy, Guda Mallikarjuna |
|
|
100 |
C |
p. |
artikel |
56 |
Novel triazolophthalazine-hydrazone hybrids as potential PCAF inhibitors: Design, synthesis, in vitro anticancer evaluation, apoptosis, and molecular docking studies
|
Abulkhair, Hamada S. |
|
|
100 |
C |
p. |
artikel |
57 |
N-Quinary heterocycle-4-sulphamoylbenzamides exert anti-hypoxic effects as dual inhibitors of carbonic anhydrases I/II
|
Yang, Chaofu |
|
|
100 |
C |
p. |
artikel |
58 |
Phthalocyanines for G-quadruplex aptamers binding
|
Lopes-Nunes, Jéssica |
|
|
100 |
C |
p. |
artikel |
59 |
Renoprotective ganodermaones A and B with rearranged meroterpenoid carbon skelotons from Ganoderma fungi
|
Zhang, Jiao-Jiao |
|
|
100 |
C |
p. |
artikel |
60 |
Semi-synthesis and biological evaluation of flavone hybrids as multifunctional agents for the potential treatment of Alzheimer's disease
|
Shi, Shaochun |
|
|
100 |
C |
p. |
artikel |
61 |
Structurally diverse lanostane triterpenoids from medicinal and edible mushroom Ganoderma resinaceum Boud
|
Shi, Qiang-Qiang |
|
|
100 |
C |
p. |
artikel |
62 |
Structural optimization of imidazothiazole derivatives affords a new promising series as B-Raf V600E inhibitors; synthesis, in vitro assay and in silico screening
|
Ammar, Usama M. |
|
|
100 |
C |
p. |
artikel |
63 |
Sulfonylhydrazones: Design, synthesis and investigation of ectonucleotidase (ALP & e5′NT) inhibition activities
|
Younus, Hafiza Amna |
|
|
100 |
C |
p. |
artikel |
64 |
Synthesis and anticancer evaluation of novel 1H-benzo[d]imidazole derivatives of dehydroabietic acid as PI3Kα inhibitors
|
Yang, Ya-Qun |
|
|
100 |
C |
p. |
artikel |
65 |
Synthesis and antioxidant activities of phenol derivatives from 1,6-bis(dimethoxyphenyl)hexane-1,6-dione
|
Artunc, Tekin |
|
|
100 |
C |
p. |
artikel |
66 |
Synthesis and biological activity of 5-aryliden-2-thiohydantoin S-aryl derivatives
|
Finko, Alexander V. |
|
|
100 |
C |
p. |
artikel |
67 |
Synthesis and characterization of new 4H-chromene-3-carboxylates ensuring potent elastase inhibition activity along with their molecular docking and chemoinformatics properties
|
Dige, Nilam C. |
|
|
100 |
C |
p. |
artikel |
68 |
Synthesis and characterization of pyridine-based organic salts: Their antibacterial, antibiofilm and wound healing activities
|
Ali, Imdad |
|
|
100 |
C |
p. |
artikel |
69 |
Synthesis and evaluation of new 1,2,4-oxadiazole based trans- acrylic acid derivatives as potential PPAR-alpha/gamma dual agonist
|
Kaur, Paranjeet |
|
|
100 |
C |
p. |
artikel |
70 |
Synthesis and evaluation of resveratrol derivatives as fetal hemoglobin inducers
|
Bosquesi, Priscila Longhin |
|
|
100 |
C |
p. |
artikel |
71 |
Synthesis and nucleic acid binding evaluation of a thyminyl l-diaminobutanoic acid-based nucleopeptide
|
Musumeci, Domenica |
|
|
100 |
C |
p. |
artikel |
72 |
Synthesis, bioactivity and binding energy calculations of novel 3-ethoxysalicylaldehyde based thiosemicarbazone derivatives
|
Ishaq, Muhammad |
|
|
100 |
C |
p. |
artikel |
73 |
Synthesis, biological evaluation and modeling of hybrids from tetrahydro-1H-pyrazolo[3,4-b]quinolines as dual cholinestrase and COX-2 inhibitors
|
Mroueh, Mohamed |
|
|
100 |
C |
p. |
artikel |
74 |
Synthesis, characterization and evaluation of 68Ga labelled monomeric and dimeric quinazoline derivatives of the HBED-CC chelator targeting the epidermal growth factor receptor
|
Liolios, Christos |
|
|
100 |
C |
p. |
artikel |
75 |
Synthesis, characterization, and in vivo pharmacological evaluation of novel mannich bases derived from 1,2,4-triazole containing a naproxen moiety
|
Avci, Ahmet |
|
|
100 |
C |
p. |
artikel |
76 |
Synthesis, characterization, inhibition effects, and molecular docking studies as acetylcholinesterase, α-glycosidase, and carbonic anhydrase inhibitors of novel benzenesulfonamides incorporating 1,3,5-triazine structural motifs
|
Lolak, Nebih |
|
|
100 |
C |
p. |
artikel |
77 |
Synthesis, evaluation of thymidine phosphorylase and angiogenic inhibitory potential of ciprofloxacin analogues: Repositioning of ciprofloxacin from antibiotic to future anticancer drugs
|
Shahzad, Sohail Anjum |
|
|
100 |
C |
p. |
artikel |
78 |
Synthesis, in vitro and in silico screening of 2-amino-4-aryl-6-(phenylthio) pyridine-3,5-dicarbonitriles as novel α-glucosidase inhibitors
|
Ali, Muhammad |
|
|
100 |
C |
p. |
artikel |
79 |
Synthesis of Gemini analogs of 19-norcalcitriol and their platinum(II) complexes
|
Brzeminski, Pawel |
|
|
100 |
C |
p. |
artikel |
80 |
Targeted photoresponsive carbazole–coumarin and drug conjugates for efficient combination therapy in leukemia cancer cells
|
Wang, Bing-Yen |
|
|
100 |
C |
p. |
artikel |
81 |
The antidiabetic drug lobeglitazone has the potential to inhibit PTP1B activity
|
Rocha, Ruth F. |
|
|
100 |
C |
p. |
artikel |
82 |
The conjugation of targeted therapy and image-guided phototdynamic therapy of cancer in vitro and in vivo
|
Xu, Peng |
|
|
100 |
C |
p. |
artikel |
83 |
The N-terminus of MTRR plays a role in MTR reactivation cycle beyond electron transfer
|
Zhang, Jun |
|
|
100 |
C |
p. |
artikel |
84 |
Twenty-five limonoids from the Hainan mangrove, Xylocarpus granatum
|
Zhang, Jia-Cheng |
|
|
100 |
C |
p. |
artikel |
85 |
Unravelling the anticancer potential of functionalized chromeno[2,3-b]pyridines for breast cancer treatment
|
Oliveira-Pinto, Sofia |
|
|
100 |
C |
p. |
artikel |