| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
6-acylamino-2-[(ethylsulfonyl)oxy]-1H-isoindole-1,3-diones mechanism-based inhibitors of human leukocyte elastase and cathepsin G: effect of chirality in the 6-acylamino substituent on inhibitory potency and selectivity
|
Vagnoni, Lisa M.
|
|
2001
|
9 |
3 |
p. 637-645
9 p.
|
artikel
|
| 2 |
Anti-leukemia selectivity in actinomycin analogues
|
Takusagawa, Fusao
|
|
2001
|
9 |
3 |
p. 719-725
7 p.
|
artikel
|
| 3 |
Biotransformation of a 4(20),11(12)-taxadiene derivative
|
Sun, Di-An
|
|
2001
|
9 |
3 |
p. 793-800
8 p.
|
artikel
|
| 4 |
Carbonic anhydrase inhibitors: Sulfonamides as antitumor agents?
|
Supuran, Claudiu T
|
|
2001
|
9 |
3 |
p. 703-714
12 p.
|
artikel
|
| 5 |
Cytokine receptor dimerization and activation: prospects for small molecule agonists
|
Boger, Dale L.
|
|
2001
|
9 |
3 |
p. 557-562
6 p.
|
artikel
|
| 6 |
2,2-Dimethyl-2H-anthra[2,3-b]pyran-6,11-diones: a new class of cytotoxic compounds
|
Melliou, Eleni
|
|
2001
|
9 |
3 |
p. 607-612
6 p.
|
artikel
|
| 7 |
Discovery of a novel lead structure for anti-malarials
|
Wiesner, Jochen
|
|
2001
|
9 |
3 |
p. 785-792
8 p.
|
artikel
|
| 8 |
Effect of chemical modifications of cytosine and guanine in a cpg-motif of oligonucleotides: structure–immunostimulatory activity relationships
|
Kandimalla, Ekambar R
|
|
2001
|
9 |
3 |
p. 807-813
7 p.
|
artikel
|
| 9 |
Expanding the recognition of the minor groove of DNA by incorporation of β-alanine in hairpin polyamides
|
Wang, Clay C.C.
|
|
2001
|
9 |
3 |
p. 653-657
5 p.
|
artikel
|
| 10 |
Identification and structural determination of a potent p-selectin inhibitor
|
Kaila, Neelu
|
|
2001
|
9 |
3 |
p. 801-806
6 p.
|
artikel
|
| 11 |
Imidazoline-modified benzylimidazolines as h5-HT1D/1B serotonergic ligands
|
Prisinzano, Thomas
|
|
2001
|
9 |
3 |
p. 613-619
7 p.
|
artikel
|
| 12 |
Iminosugars: potential inhibitors of liver glycogen phosphorylase
|
Jakobsen, Palle
|
|
2001
|
9 |
3 |
p. 733-744
12 p.
|
artikel
|
| 13 |
New polycyclic pyrimidine derivatives with antiplatelet in vitro activity: synthesis and pharmacological screening
|
Bruno, Olga
|
|
2001
|
9 |
3 |
p. 629-636
8 p.
|
artikel
|
| 14 |
Polycyclic aromatic compounds as anticancer agents: structure–activity relationships of chrysene and pyrene derivatives
|
Banik, Bimal K
|
|
2001
|
9 |
3 |
p. 593-605
13 p.
|
artikel
|
| 15 |
Ring-deactivated hydroxymethylpyrroles as inhibitors of α-chymotrypsin
|
Abell, Andrew D.
|
|
2001
|
9 |
3 |
p. 621-628
8 p.
|
artikel
|
| 16 |
Selective inhibition of Trypanosoma brucei GAPDH by 1,3-bisphospho-d-glyceric acid (1,3-diPG) analogues
|
Ladame, Sylvain
|
|
2001
|
9 |
3 |
p. 773-783
11 p.
|
artikel
|
| 17 |
Short and efficient syntheses of analogues of way-100635: new and potent 5-HT1A receptor antagonists
|
Marchais, Sandrine
|
|
2001
|
9 |
3 |
p. 695-702
8 p.
|
artikel
|
| 18 |
Structure–activity relationships in a series of 8-substituted xanthines as A1-adenosine receptor antagonists
|
Strappaghetti, Giovannella
|
|
2001
|
9 |
3 |
p. 575-583
9 p.
|
artikel
|
| 19 |
Synthesis and acetylcholinesterase/butyrylcholinesterase inhibition activity of new tacrine-like analogues
|
Marco, José L
|
|
2001
|
9 |
3 |
p. 727-732
6 p.
|
artikel
|
| 20 |
Synthesis and anti-inflammatory activities of N 4,N 5-disubstituted-3-methyl-1H-pyrazolo[3,4-c]pyridazines
|
Tewari, Ashish Kumar
|
|
2001
|
9 |
3 |
p. 715-718
4 p.
|
artikel
|
| 21 |
Synthesis and pharmacological evaluation of imidazoline sites I 1 and I 2 selective ligands
|
Anastassiadou, Maria
|
|
2001
|
9 |
3 |
p. 585-592
8 p.
|
artikel
|
| 22 |
Synthesis, electrochemistry, and molluscicidal activity of nitroaromatic compounds: effects of substituents and the role of redox potential
|
de Abreu, Fabiane C.
|
|
2001
|
9 |
3 |
p. 659-664
6 p.
|
artikel
|
| 23 |
Synthesis of 2-amido-3-hydroxypyridin-4(1H)-ones: novel iron chelators with enhanced pFe3+ values
|
Liu, Zu D.
|
|
2001
|
9 |
3 |
p. 563-573
11 p.
|
artikel
|
| 24 |
Synthesis of [18F]-labeled EF3 [2-(2-nitroimidazol-1-yl)-N-(3,3,3-trifluoropropyl)-acetamide], a marker for PET detection of hypoxia
|
Josse, Olivier
|
|
2001
|
9 |
3 |
p. 665-675
11 p.
|
artikel
|
| 25 |
Synthesis of high-specific-radioactivity 4- and 6-[18F]fluorometaraminol- PET tracers for the adrenergic nervous system of the heart
|
Langer, Oliver
|
|
2001
|
9 |
3 |
p. 677-694
18 p.
|
artikel
|
| 26 |
Synthesis of indomethacin analogues for evaluation as modulators of MRP activity
|
Maguire, Anita R.
|
|
2001
|
9 |
3 |
p. 745-762
18 p.
|
artikel
|
| 27 |
Synthesis, receptor binding affinities and conformational properties of cyclic methylenedithioether analogues of angiotensin II
|
Lindman, Susanna
|
|
2001
|
9 |
3 |
p. 763-772
10 p.
|
artikel
|
| 28 |
The crystal structure of the complex of non-peptidic inhibitor of human neutrophil elastase ONO-6818 and porcine pancreatic elastase
|
Odagaki, Y
|
|
2001
|
9 |
3 |
p. 647-651
5 p.
|
artikel
|
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