| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Acyloxymethyl as a drug protecting group. Part 7: Tertiary sulfonamidomethyl ester prodrugs of benzylpenicillin: chemical hydrolysis and anti-bacterial activity
|
Iley, Jim
|
|
2000
|
8 |
7 |
p. 1629-1636
8 p.
|
artikel
|
| 2 |
Analyses of insulin-potentiating fragments of human growth hormone by computative simulation; essential unit for insulin-Involved biological responses
|
Ohkura, Kazuto
|
|
2000
|
8 |
7 |
p. 1733-1740
8 p.
|
artikel
|
| 3 |
Analysis of stereoelectronic properties of camptothecin analogues in relation to biological activity
|
Werbovetz, Karl A.
|
|
2000
|
8 |
7 |
p. 1741-1747
7 p.
|
artikel
|
| 4 |
Anti-tumor promoting effects of sesquiterpenes from Maytenus cuzcoina (celastraceae)
|
González, Antonio G.
|
|
2000
|
8 |
7 |
p. 1773-1778
6 p.
|
artikel
|
| 5 |
Attempts to obtain more efficient GAC-cleaving hammerhead ribozymes by in vitro selection
|
Kore, Anilkumar R
|
|
2000
|
8 |
7 |
p. 1767-1771
5 p.
|
artikel
|
| 6 |
Aurine tricarboxylic acid, a potent metal-chelating inhibitor of NFκB–DNA binding
|
Kumar Sharma, Rakesh
|
|
2000
|
8 |
7 |
p. 1819-1823
5 p.
|
artikel
|
| 7 |
Comparative QSAR studies on substituted bis-(acridines) and bis-(phenazines)-carboxamides: a new class of anticancer agents
|
Garg, Rajni
|
|
2000
|
8 |
7 |
p. 1835-1839
5 p.
|
artikel
|
| 8 |
Conformations in solution and bound to bacterial ribosomes of ketolides, HMR 3647 (telithromycin) and RU 72366: A new class of highly potent antibacterials
|
Evrard-Todeschi, Nathalie
|
|
2000
|
8 |
7 |
p. 1579-1597
19 p.
|
artikel
|
| 9 |
Controlled site-selective protein glycosylation for precise glycan structure–catalytic activity relationships
|
Davis, Benjamin G
|
|
2000
|
8 |
7 |
p. 1527-1535
9 p.
|
artikel
|
| 10 |
Design, synthesis and binding at cloned muscarinic receptors of N-[5-(1′-substituted-acetoxymethyl)-3-oxadiazolyl] and N-[4-(1′-substituted-acetoxymethyl)-2-dioxolanyl] dialkyl amines
|
Manfredini, Stefano
|
|
2000
|
8 |
7 |
p. 1559-1566
8 p.
|
artikel
|
| 11 |
Design, synthesis and cytotoxicity evaluation of 1-chloromethyl-5-hydroxy-1,2-dihydro-3H-benz[e]indole (seco-CBI) dimers
|
Jia, Guofeng
|
|
2000
|
8 |
7 |
p. 1607-1617
11 p.
|
artikel
|
| 12 |
Development of a 3D pharmacophore for nonspecific ligand recognition of α1, α2, α3, α5, and α6 containing gabaA/benzodiazepine receptors
|
Filizola, Marta
|
|
2000
|
8 |
7 |
p. 1799-1807
9 p.
|
artikel
|
| 13 |
Flavonols from Heterotheca inuloides: Tyrosinase Inhibitory Activity and Structural Criteria
|
Kubo, Isao
|
|
2000
|
8 |
7 |
p. 1749-1755
7 p.
|
artikel
|
| 14 |
Hydrogen bonding isosteres: bimolecular carboxylic acid and amine-N-oxide interactions mediated via CH···O hydrogen bonds
|
Baures, P.W
|
|
2000
|
8 |
7 |
p. 1599-1605
7 p.
|
artikel
|
| 15 |
Mechanism of biochemical action of substituted 4-methylbenzopyran-2-ones. Part 7: assay and characterization of 7,8-diacetoxy-4-methylcoumarin:protein transacetylase from rat liver microsomes based on the irreversible inhibition of cytosolic glutathione S-Transferase
|
Raj, Hanumantharao G
|
|
2000
|
8 |
7 |
p. 1707-1712
6 p.
|
artikel
|
| 16 |
Monoamine oxidase-catalyzed oxidation of endo,endo-2-amino-6-[(Z)-2′-phenyl]ethenylbicyclo[2.2.1]heptane, a potential probe for a radical cation intermediate
|
Wang, Xueqing
|
|
2000
|
8 |
7 |
p. 1645-1651
7 p.
|
artikel
|
| 17 |
New aromatic iminoimidazolidine derivatives as α1-adrenoceptor antagonists: a novel synthetic approach and pharmacological activity
|
Dardonville, Christophe
|
|
2000
|
8 |
7 |
p. 1567-1577
11 p.
|
artikel
|
| 18 |
Nicorandil analogues containing NO-donor furoxans and related furazans
|
Boschi, Donatella
|
|
2000
|
8 |
7 |
p. 1727-1732
6 p.
|
artikel
|
| 19 |
Potent inhibition of serine proteases by heterocyclic sulfide derivatives of 1,2,5-thiadiazolidin-3-one 1,1 dioxide
|
He, Shu
|
|
2000
|
8 |
7 |
p. 1713-1717
5 p.
|
artikel
|
| 20 |
Site-selective glycosylation of subtilisin Bacillus lentus causes dramatic increases in esterase activity
|
Lloyd, Richard C
|
|
2000
|
8 |
7 |
p. 1537-1544
8 p.
|
artikel
|
| 21 |
Syntheses and biological activity of C-3′-difluoromethyl-taxoids
|
Ojima, Iwao
|
|
2000
|
8 |
7 |
p. 1619-1628
10 p.
|
artikel
|
| 22 |
Synthesis and antitumor activity of duocarmycin derivatives
|
Amishiro, Nobuyoshi
|
|
2000
|
8 |
7 |
p. 1637-1643
7 p.
|
artikel
|
| 23 |
Synthesis and biological activities of 2′-deoxy-2′-fluoro-4′-thioarabinofuranosylpyrimidine and -purine nucleosides
|
Yoshimura, Yuichi
|
|
2000
|
8 |
7 |
p. 1545-1558
14 p.
|
artikel
|
| 24 |
Synthesis and biological activities of the marine bryozoan alkaloids convolutamines A, C and F, and lutamides A and C
|
Hashima, Hirofumi
|
|
2000
|
8 |
7 |
p. 1757-1766
10 p.
|
artikel
|
| 25 |
Synthesis and biological evaluations of C-23-modified 26,26,26,27,27,27-F6-vitamin D3 analogues
|
Ikeda, Masahiko
|
|
2000
|
8 |
7 |
p. 1809-1817
9 p.
|
artikel
|
| 26 |
Synthesis and characterisation of polyamine–poly(ethylene glycol) constructs for DNA binding and gene delivery
|
Garrett, Shane W
|
|
2000
|
8 |
7 |
p. 1779-1797
19 p.
|
artikel
|
| 27 |
Synthesis and evaluation of fructose analogues as inhibitors of the d-fructose transporter GLUT5
|
Tatibouët, Arnaud
|
|
2000
|
8 |
7 |
p. 1825-1833
9 p.
|
artikel
|
| 28 |
The design and synthesis of a new tumor-selective fluoropyrimidine carbamate, Capecitabine
|
Shimma, Nobuo
|
|
2000
|
8 |
7 |
p. 1697-1706
10 p.
|
artikel
|
| 29 |
The synthesis and antibacterial activity of totarol derivatives. part 3: modification of ring-B
|
Evans, Gary B
|
|
2000
|
8 |
7 |
p. 1663-1675
13 p.
|
artikel
|
| 30 |
The synthesis and antibacterial activity of totarol derivatives. part 2: modifications at C-12 and O-13
|
Evans, Gary B
|
|
2000
|
8 |
7 |
p. 1653-1662
10 p.
|
artikel
|
| 31 |
Total synthesis and antifungal evaluation of cyclic aminohexapeptides
|
Klein, Larry L.
|
|
2000
|
8 |
7 |
p. 1677-1696
20 p.
|
artikel
|
| 32 |
Triazene drug metabolites. Part 17: synthesis and plasma hydrolysis of acyloxymethyl carbamate derivatives of antitumour triazenes
|
Carvalho *, Emı́lia
|
|
2000
|
8 |
7 |
p. 1719-1725
7 p.
|
artikel
|
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