| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
Acyclic amides as estrogen receptor ligands: Synthesis, binding, activity and receptor interaction
|
Stauffer, Shaun R
|
|
2000
|
8 |
6 |
p. 1293-1316
24 p.
|
artikel
|
| 2 |
Alkyl and alkoxycarbonyl derivatives of ginkgolide B
|
Hu, Lihong
|
|
2000
|
8 |
6 |
p. 1515-1521
7 p.
|
artikel
|
| 3 |
Antimalarial sulfide, sulfone, and sulfonamide trioxanes
|
Posner, Gary H.
|
|
2000
|
8 |
6 |
p. 1361-1370
10 p.
|
artikel
|
| 4 |
Antimycobacterial pyrroles: synthesis, anti-Mycobacterium tuberculosis activity and QSAR studies
|
Ragno, Rino
|
|
2000
|
8 |
6 |
p. 1423-1432
10 p.
|
artikel
|
| 5 |
aziridinyl peptides as inhibitors of cysteine proteases: Effect of a free carboxylic acid function on inhibition
|
Schirmeister, T.
|
|
2000
|
8 |
6 |
p. 1281-1291
11 p.
|
artikel
|
| 6 |
Bioisosteric replacement strategy for the synthesis of 1-azacyclic compounds with high affinity for the central nicotinic cholinergic receptors
|
Olesen, Preben H.
|
|
2000
|
8 |
6 |
p. 1443-1450
8 p.
|
artikel
|
| 7 |
Bromal-derived tetrahydro-β-carbolines as neurotoxic agents: chemistry, impairment of the dopamine metabolism, and inhibitory effects on mitochondrial respiration
|
Bringmann, Gerhard
|
|
2000
|
8 |
6 |
p. 1467-1478
12 p.
|
artikel
|
| 8 |
Comparative molecular field analysis of colchicine inhibition and tubulin polymerization for combretastatins binding to the colchicine binding site on β-tubulin
|
Brown, Milton L
|
|
2000
|
8 |
6 |
p. 1433-1441
9 p.
|
artikel
|
| 9 |
Corrigendum to “Imidazole-containing amino acids as selective inhibitors of nitric oxide synthases”
|
Lee, Younghee
|
|
2000
|
8 |
6 |
p. 1523-
1 p.
|
artikel
|
| 10 |
Corrigendum to “Synthesis and anti-HIV evaluation of 2′,3′-dideoxy imidazo- and ν-triazolo[4,5-d]pyridazine nucleosides”
|
Bussolari, Jacqueline C
|
|
2000
|
8 |
6 |
p. 1525-
1 p.
|
artikel
|
| 11 |
Corticotropin releasing hormone: therapeutic implications and medicinal chemistry developments
|
Keller, Paul A
|
|
2000
|
8 |
6 |
p. 1213-1223
11 p.
|
artikel
|
| 12 |
Coumarinic derivatives as mechanism-based inhibitors of α-chymotrypsin and human leukocyte elastase
|
Pochet, Lionel
|
|
2000
|
8 |
6 |
p. 1489-1501
13 p.
|
artikel
|
| 13 |
2,3-Dihydro-dithiin and -dithiepine-1,1,4,4-tetroxides: small molecule non-peptide antagonists of the human galanin hGAL-1 receptor
|
Scott, Malcolm K
|
|
2000
|
8 |
6 |
p. 1383-1391
9 p.
|
artikel
|
| 14 |
Identification of new Cdc25 dual specificity phosphatase inhibitors in a targeted small molecule array
|
Ducruet, Alexander P
|
|
2000
|
8 |
6 |
p. 1451-1466
16 p.
|
artikel
|
| 15 |
Lincomycin and clindamycin conformations. A fragment shared by macrolides, ketolides and lincosamides determined from TRNOE ribosome-bound conformations
|
Verdier, Laurent
|
|
2000
|
8 |
6 |
p. 1225-1243
19 p.
|
artikel
|
| 16 |
Multicomponent synthesis of novel amino acid–nucleobase chimeras: a versatile approach to PNA-monomers
|
Maison, Wolfgang
|
|
2000
|
8 |
6 |
p. 1343-1360
18 p.
|
artikel
|
| 17 |
New anti-HIV derivatives: synthesis and antiviral evaluation
|
De Michelis, C.
|
|
2000
|
8 |
6 |
p. 1253-1262
10 p.
|
artikel
|
| 18 |
Novel imidazolyl and triazolyl substituted biphenyl compounds: synthesis and evaluation as nonsteroidal inhibitors of human 17α-hydroxylase-C17, 20-Lyase (P450 17)
|
Zhuang, Yan
|
|
2000
|
8 |
6 |
p. 1245-1252
8 p.
|
artikel
|
| 19 |
Observations on the covalent cross-linking of the binding domain (BD) of the high mobility group I/Y (HMG I/Y) proteins to DNA by FR66979
|
Rajski, Scott R
|
|
2000
|
8 |
6 |
p. 1331-1342
12 p.
|
artikel
|
| 20 |
Pyrrolo-quinoline derivatives as potential antineoplastic drugs
|
Ferlin, M.G
|
|
2000
|
8 |
6 |
p. 1415-1422
8 p.
|
artikel
|
| 21 |
6-Substituted 2,2-Bis(fluoromethyl)-benzopyran-4-carboxamide K+ channel openers
|
Taka, Naoki
|
|
2000
|
8 |
6 |
p. 1393-1405
13 p.
|
artikel
|
| 22 |
Substituted 1-phenyl-2-cyclopropylmethylamines with high affinity and selectivity for sigma sites
|
Ronsisvalle, Giuseppe
|
|
2000
|
8 |
6 |
p. 1503-1513
11 p.
|
artikel
|
| 23 |
2″-Substituted 5-phenylterbenzimidazoles as topoisomerase I poisons
|
Rangarajan, Meera
|
|
2000
|
8 |
6 |
p. 1371-1382
12 p.
|
artikel
|
| 24 |
Synthesis, incorporation efficiency, and stability of disulfide bridged functional groups at RNA 5′-ends
|
Sengle, Gerhard
|
|
2000
|
8 |
6 |
p. 1317-1329
13 p.
|
artikel
|
| 25 |
Synthesis of acyclic 6,7-dihaloquinolone nucleoside analogues as potential antibacterial and antiviral agents
|
Al-Masoudi, Najim A
|
|
2000
|
8 |
6 |
p. 1407-1413
7 p.
|
artikel
|
| 26 |
Synthesis of N-substituted piperidine-4-(benzylidene-4-carboxylic acids) and evaluation as inhibitors of steroid-5α-reductase type 1 and 2
|
Picard, Franck
|
|
2000
|
8 |
6 |
p. 1479-1487
9 p.
|
artikel
|
| 27 |
Taxus canadensis abundant taxane: conversion to paclitaxel and rearrangements
|
Nikolakakis, Anastasia
|
|
2000
|
8 |
6 |
p. 1269-1280
12 p.
|
artikel
|
| 28 |
The discovery of [1-(4-dimethylamino-benzyl)-piperidin-4-yl]-[4-(3,3-dimethylbutyl)-phenyl]-(3-methyl-but-2-enyl)-amine, an N-type Ca+2 channel blocker with oral activity for analgesia
|
Hu, Lain-Yen
|
|
2000
|
8 |
6 |
p. 1203-1212
10 p.
|
artikel
|
| 29 |
Tyrosine analogues as alternative substrates for protein tyrosine kinase Csk: Insights into substrate selectivity and catalytic mechanism
|
Kim, Kyonghee
|
|
2000
|
8 |
6 |
p. 1263-1268
6 p.
|
artikel
|
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