| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A class of 4-aza-lithocholic acid-derived haptens for the generation of catalytic antibodies with steroid synthase capabilities
|
Hasserodt, Jens
|
|
2000
|
8 |
5 |
p. 995-1003
9 p.
|
artikel
|
| 2 |
A new affinity ligand for the isolation of a single ‘feruloyl esterase’ (FAE-III) from Aspergillus niger
|
Zhao, Yongxin
|
|
2000
|
8 |
5 |
p. 917-924
8 p.
|
artikel
|
| 3 |
Bacterial diaminopimelate metabolism as a target for antibiotic design
|
Cox, Russell J.
|
|
2000
|
8 |
5 |
p. 843-871
29 p.
|
artikel
|
| 4 |
Biaryl diacid inhibitors of human s-PLA2 with anti-inflammatory activity
|
Springer, Dane M.
|
|
2000
|
8 |
5 |
p. 1087-1109
23 p.
|
artikel
|
| 5 |
Brain-targeted chemical delivery of [Leu2, Pip3]-TRH
|
Yoon, Sung-Hwa
|
|
2000
|
8 |
5 |
p. 1059-1063
5 p.
|
artikel
|
| 6 |
Chemoenzymatic synthesis of PSGL-1 glycopeptides: sulfation on tyrosine affects glycosyltransferase-catalyzed synthesis of the O-glycan
|
Koeller, Kathryn M
|
|
2000
|
8 |
5 |
p. 1017-1025
9 p.
|
artikel
|
| 7 |
Conformationally restricted analogues designed for selective inhibition of GAR Tfase versus thymidylate synthase or dihydrofolate reductase
|
Boger, Dale L.
|
|
2000
|
8 |
5 |
p. 1075-1086
12 p.
|
artikel
|
| 8 |
Cyclobutane carboxamide inhibitors of fungal melanin: biosynthesis and their evaluation as fungicides
|
Jennings, Lee D.
|
|
2000
|
8 |
5 |
p. 897-907
11 p.
|
artikel
|
| 9 |
Design, synthesis and structure–affinity relationships of 4-methylidenepiperidine and 4-aryl-1,2,3,6-tetrahydropyridine derivatives as corticotropin-releasing factor1 receptor antagonists
|
Nakazato, Atsuro
|
|
2000
|
8 |
5 |
p. 1183-1193
11 p.
|
artikel
|
| 10 |
2H-Thieno[3,2-e]- and [2,3-e]-1,2-thiazine-6-sulfonamide 1,1-dioxides as ocular hypotensive agents: synthesis, carbonic anhydrase inhibition and evaluation in the rabbit
|
Chen, Hwang-Hsing
|
|
2000
|
8 |
5 |
p. 957-975
19 p.
|
artikel
|
| 11 |
Interaction of pyrimethamine, cycloguanil, WR99210 and their analogues with Plasmodium falciparum dihydrofolate reductase: structural basis of antifolate resistance
|
Rastelli, Giulio
|
|
2000
|
8 |
5 |
p. 1117-1128
12 p.
|
artikel
|
| 12 |
Ionization behaviour and tautomerism-dependent lipophilicity of pyridine-2(1H)-one cardiotonic agents
|
Altomare, C.
|
|
2000
|
8 |
5 |
p. 909-916
8 p.
|
artikel
|
| 13 |
Microbial transformation of 2-hydroxy and 2-acetoxy ketones with Geotrichum sp.
|
Wei, Zhi-Liang
|
|
2000
|
8 |
5 |
p. 1129-1137
9 p.
|
artikel
|
| 14 |
New antineoplastic prenylhydroquinones. Synthesis and evaluation
|
Molinari, Aurora
|
|
2000
|
8 |
5 |
p. 1027-1032
6 p.
|
artikel
|
| 15 |
New aromatase inhibitors. Synthesis and biological activity of aryl-substituted pyrrolizine and indolizine derivatives
|
Sonnet, Pascal
|
|
2000
|
8 |
5 |
p. 945-955
11 p.
|
artikel
|
| 16 |
New carbamoylpiperidines as human platelet aggregation inhibitors
|
Guo, Zhengming
|
|
2000
|
8 |
5 |
p. 1041-1058
18 p.
|
artikel
|
| 17 |
Orally active cephalosporins. Part 2: Synthesis, structure–activity relationships and oral absorption of cephalosporins having a C-3 pyridyl side chain
|
Yamamoto, Hirofumi
|
|
2000
|
8 |
5 |
p. 1159-1170
12 p.
|
artikel
|
| 18 |
(Partial) agonist/antagonist properties of novel diarylalkyl carbamates on histamine H3 receptors
|
Sasse, Astrid
|
|
2000
|
8 |
5 |
p. 1139-1149
11 p.
|
artikel
|
| 19 |
Preparation of dopaminergic N-alkyl-benzyltetrahydro-isoquinolines using a ‘one-pot’ procedure in acid medium
|
Andreu, Inmaculada
|
|
2000
|
8 |
5 |
p. 889-895
7 p.
|
artikel
|
| 20 |
Sequence-selectivity of 5,11-dimethyl-5H-indolo[2,3-b]quinoline binding to DNA. Footprinting and molecular modeling studies
|
Osiadacz, Jarosław
|
|
2000
|
8 |
5 |
p. 937-943
7 p.
|
artikel
|
| 21 |
Sterol C-methyl transferase from Prototheca wickerhamii mechanism, sterol specificity and inhibition
|
Mangla, Anil T
|
|
2000
|
8 |
5 |
p. 925-936
12 p.
|
artikel
|
| 22 |
Structural bases for the inhibition of aldose reductase by phenolic compounds
|
Rastelli, Giulio
|
|
2000
|
8 |
5 |
p. 1151-1158
8 p.
|
artikel
|
| 23 |
Structure–activity relationship at α-adrenergic receptors within a series of imidazoline analogues of cirazoline
|
Pigini, Maria
|
|
2000
|
8 |
5 |
p. 883-888
6 p.
|
artikel
|
| 24 |
Substituted benz[a]acridines and benz[c]acridines as mammalian topoisomerase poisons
|
Makhey, Darshan
|
|
2000
|
8 |
5 |
p. 1171-1182
12 p.
|
artikel
|
| 25 |
1-Substituted-4-[3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl]piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and α1 receptors. Part 6
|
Perrone, Roberto
|
|
2000
|
8 |
5 |
p. 873-881
9 p.
|
artikel
|
| 26 |
Synthesis and antimalarial activities of base-catalyzed adducts of 11-azaartemisinin
|
Mekonnen, Belew
|
|
2000
|
8 |
5 |
p. 1111-1116
6 p.
|
artikel
|
| 27 |
Synthesis and antitumor activity of duocarmycin derivatives: modification at the C-7 position of segment-A of A-ring pyrrole compounds
|
Amishiro, Nobuyoshi
|
|
2000
|
8 |
5 |
p. 1195-1201
7 p.
|
artikel
|
| 28 |
Synthesis and antitumor activity of selected 7-alkylidene substituted cephems
|
Veinberg, G.
|
|
2000
|
8 |
5 |
p. 1033-1040
8 p.
|
artikel
|
| 29 |
Synthesis and antitumor activity of some indeno[1,2-b]quinoline-based bis carboxamides
|
Deady, Leslie W
|
|
2000
|
8 |
5 |
p. 977-984
8 p.
|
artikel
|
| 30 |
Synthesis and evaluation of oligo-1,3-thiazolecarboxamide derivatives as HIV-1 reverse transcriptase inhibitors
|
Ryabinin, Vladimir A.
|
|
2000
|
8 |
5 |
p. 985-993
9 p.
|
artikel
|
| 31 |
Synthesis, hydroxyl radical production and cytotoxicity of analogues of bleomycin
|
Highfield, Jackie A.
|
|
2000
|
8 |
5 |
p. 1065-1073
9 p.
|
artikel
|
| 32 |
Utilization of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold in the design of potent inhibitors of serine proteases: SAR studies using carboxylates
|
Kuang, Rongze
|
|
2000
|
8 |
5 |
p. 1005-1016
12 p.
|
artikel
|
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