| nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
| 1 |
A comprehensive review of BET-targeting PROTACs for cancer therapy
|
Zhou, Xiao-Li
|
|
|
73 |
C |
p.
|
artikel
|
| 2 |
A concise synthesis of l-gulose and its C-6 derivatives
|
Teng, Kai-Ching
|
|
|
73 |
C |
p.
|
artikel
|
| 3 |
A simplified analog of debromoaplysiatoxin lacking the B-ring of spiroketal moiety retains protein kinase C-binding and antiproliferative activities
|
Sekido, Tomoki
|
|
|
73 |
C |
p.
|
artikel
|
| 4 |
Biphenyl-based small molecule inhibitors: Novel cancer immunotherapeutic agents targeting PD-1/PD-L1 interaction
|
Sasmal, Pujan
|
|
|
73 |
C |
p.
|
artikel
|
| 5 |
Design and evaluation of novel analogs of 2-amino-4-boronobutanoic acid (ABBA) as inhibitors of human gamma-glutamyl transpeptidase
|
Nguyen, Luong
|
|
|
73 |
C |
p.
|
artikel
|
| 6 |
Development of a penetratin-conjugated stapled peptide that inhibits Wnt/β-catenin signaling
|
Tsuchiya, Keisuke
|
|
|
73 |
C |
p.
|
artikel
|
| 7 |
Discovery and optimization of orally bioavailable and potent plasma Kallikrein inhibitors bearing a quaternary carbon
|
Zhang, Weihe
|
|
|
73 |
C |
p.
|
artikel
|
| 8 |
Discovery of biphenyls bearing thiobarbiturate fragment by structure-based strategy as Mycobacterium tuberculosis protein tyrosine phosphatase B inhibitors
|
Cheng, Shihao
|
|
|
73 |
C |
p.
|
artikel
|
| 9 |
Discovery of novel compounds as potent activators of Sirt3
|
Reverdy, Célina
|
|
|
73 |
C |
p.
|
artikel
|
| 10 |
Discovery of polymethoxyphenyl-pyridines bearing amino side chains as tubulin colchicine-binding site inhibitors
|
Li, XiaoYang
|
|
|
73 |
C |
p.
|
artikel
|
| 11 |
Dual MVK cleavable linkers effectively reduce renal retention of 111In-fibronectin-binding peptides
|
Valpreda, Giulia
|
|
|
73 |
C |
p.
|
artikel
|
| 12 |
Editorial Board
|
|
|
|
73 |
C |
p.
|
artikel
|
| 13 |
Evaluation of acute toxicity of cancer-targeting albumin-based artificial metalloenzymes
|
Chang, Tsung-Che
|
|
|
73 |
C |
p.
|
artikel
|
| 14 |
Expanding the scope of stereoselective α-galactosylation using glycosyl chlorides
|
Shadrick, Melanie
|
|
|
73 |
C |
p.
|
artikel
|
| 15 |
Graphical Abstract Contents Continued
|
|
|
|
73 |
C |
p.
|
artikel
|
| 16 |
Graphical abstract TOC
|
|
|
|
73 |
C |
p.
|
artikel
|
| 17 |
Graphical abstract TOC
|
|
|
|
73 |
C |
p.
|
artikel
|
| 18 |
Hetero-aryl bromide precursor fluorine-18 radiosynthesis and preclinical evaluation of a novel positron emission tomography (PET) tracer [18F]GSK1482160
|
Huang, Guolong
|
|
|
73 |
C |
p.
|
artikel
|
| 19 |
Identification of PI3K/HDAC Dual-targeted inhibitors with subtype selectivity as potential therapeutic agents against solid Tumors: Building HDAC6 potency in a Quinazolinone-based PI3Kδ-selective template
|
Li, Zhi
|
|
|
73 |
C |
p.
|
artikel
|
| 20 |
Identification of small-molecule inhibitors of the DNA repair proteins RuvAB from Pseudomonas aeruginosa
|
Dai, Lin
|
|
|
73 |
C |
p.
|
artikel
|
| 21 |
Improving lipophilicity of 5-(1-acetyl-5-phenylpyrazolidin-3-ylidene)-1,3-dimethylbarbituric acid increases its efficacy to activate hypoxia-inducible factors
|
Sonoda, Kento
|
|
|
73 |
C |
p.
|
artikel
|
| 22 |
Isatoic anhydrides as novel inhibitors of monoamine oxidase
|
Hitge, Rialette
|
|
|
73 |
C |
p.
|
artikel
|
| 23 |
Multiple approaches to repurposing drugs for neuroblastoma
|
Rank, Laura
|
|
|
73 |
C |
p.
|
artikel
|
| 24 |
New potent ciprofloxacin-uracil conjugates as DNA gyrase and topoisomerase IV inhibitors against methicillin-resistant Staphylococcus aureus
|
Samir, Mohamed
|
|
|
73 |
C |
p.
|
artikel
|
| 25 |
Nucleic acid extraction from complex biofluid using toothpick-actuated over-the-counter medical-grade cotton
|
Kumar, Shrawan
|
|
|
73 |
C |
p.
|
artikel
|
| 26 |
Practical syntheses of DOTAGA-DBCO and DFO-DBCO, strained alkyne pre-cursors to radioimmunoconjugates for targeted alpha therapy
|
Sales, Zachary S.
|
|
|
73 |
C |
p.
|
artikel
|
| 27 |
Structure-activity relationships of mixed σ1R/σ2R ligands with antiproliferative and anticancer effects
|
Fallica, Antonino N.
|
|
|
73 |
C |
p.
|
artikel
|
| 28 |
Structure-activity-relationship study of semi-synthetically modified fusicoccins on their stabilization effect for 14-3-3-phospholigand interactions
|
Ogino, Nanami
|
|
|
73 |
C |
p.
|
artikel
|
| 29 |
Synthesis and evaluation of 2,9-disubstituted-1,10-phenanthroline derivatives as G-quadruplex binders
|
Figueiredo, Joana
|
|
|
73 |
C |
p.
|
artikel
|
| 30 |
Synthesis and evaluation of glycosylated quercetin to enhance neuroprotective effects on cerebral ischemia-reperfusion
|
Wang, Siqi
|
|
|
73 |
C |
p.
|
artikel
|
| 31 |
Synthesis and preclinical evaluation of rhenium and technetium-99m “4 + 1” mixed-ligand complexes bearing quinazoline derivatives as potential EGFR imaging agents
|
Kiritsis, Christos
|
|
|
73 |
C |
p.
|
artikel
|
| 32 |
Synthesis of capuramycin and its analogues via a Ferrier-type I reaction and their biological evaluation
|
Kusaka, Shintaro
|
|
|
73 |
C |
p.
|
artikel
|
| 33 |
Synthesis of 2′-O-[3-(N-methylsulfamoyl)propan-1-yl]ribothymidine as a potentially applicable 2′-modified nucleoside for antisense oligonucleotides
|
Tomori, Takahito
|
|
|
73 |
C |
p.
|
artikel
|
| 34 |
The 2022 Monkeypox outbreak: How the medicinal chemistry could help us?
|
Silva-Júnior, Edeildo Ferreira da
|
|
|
73 |
C |
p.
|
artikel
|
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