nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
Chemical modification of β-glucocerebrosidase inhibitor N-octyl-β-valienamine: synthesis and biological evaluation of N-alkanoyl and N-alkyl derivatives
|
Ogawa, Seiichiro |
|
1998 |
6 |
10 |
p. 1955-1962 8 p. |
artikel |
2 |
Design, synthesis and evaluation of transition-state analogue inhibitors of Escherichia coli γ-glutamylcysteine synthetase
|
Tokutake, Nobuya |
|
1998 |
6 |
10 |
p. 1935-1953 19 p. |
artikel |
3 |
2,2′-dithiobisbenzamides derived from α-, β- and γ-amino acids possessing anti-HIV activities: synthesis and structure–activity relationship
|
Vara Prasad, J.V.N |
|
1998 |
6 |
10 |
p. 1707-1730 24 p. |
artikel |
4 |
Effect of 2′-OH acetylation on the bioactivity and conformation of 7-O-[N-(4′-fluoresceincarbonyl)-l-alanyl]taxol. A NMR-fluorescence microscopy study
|
Jiménez-Barbero, Jesús |
|
1998 |
6 |
10 |
p. 1857-1863 7 p. |
artikel |
5 |
Functional correlation of molecular electronic properties with potency of synthetic carbinolamine antimalarial agents
|
Bhattacharjee, Apurba K |
|
1998 |
6 |
10 |
p. 1927-1933 7 p. |
artikel |
6 |
Glycosyl-transferase catalyzed assemblage of sialyl-lewisx-saccharopeptides
|
Baisch, Gabi |
|
1998 |
6 |
10 |
p. 1673-1682 10 p. |
artikel |
7 |
Impact of mixed-backbone oligonucleotides on target binding affinity and target cleaving specificity and selectivity by Escherichia coli RNase H
|
Shen, Ling X |
|
1998 |
6 |
10 |
p. 1695-1705 11 p. |
artikel |
8 |
Inactivation of monoamine oxidase B by cis- and trans-5-aminomethyl-3-(4-methoxyphenyl)dihydrofuran-2(3H)-ones
|
Lu, Xingliang |
|
1998 |
6 |
10 |
p. 1851-1856 6 p. |
artikel |
9 |
Inhibition of myo-inositol monophosphatase isoforms by aromatic phosphonates
|
Ganzhorn, Axel J. |
|
1998 |
6 |
10 |
p. 1865-1874 10 p. |
artikel |
10 |
Mechanism of biochemical action of substituted 4-methylbenzopyran-2-ones. Part II: Mechanism-based inhibition of rat liver microsome-mediated aflatoxin B1–DNA binding by the candidate antimutagen 7,8-diacetoxy-4-methylcoumarin
|
Raj, Hanumantharao G |
|
1998 |
6 |
10 |
p. 1895-1904 10 p. |
artikel |
11 |
Molecular modeling studies of the binding modes of aldose reductase inhibitors at the active site of human aldose reductase
|
Lee, Yong S |
|
1998 |
6 |
10 |
p. 1811-1819 9 p. |
artikel |
12 |
Molecular structure and stereoelectronic properties of sarmazenil—a weak inverse agonist at the omega modulatory sites (benzodiazepine receptors): comparison with bretazenil and flumazenil
|
López-Romero, B |
|
1998 |
6 |
10 |
p. 1745-1757 13 p. |
artikel |
13 |
Novel rhenium complexes derived from α-tropanol as potential ligands for the dopamine transporter
|
Hoepping, Alexander |
|
1998 |
6 |
10 |
p. 1663-1672 10 p. |
artikel |
14 |
Potent acetylcholinesterase inhibitors: design, synthesis, and structure–Activity relationships of bis-interacting ligands in the galanthamine series
|
Mary, Aude |
|
1998 |
6 |
10 |
p. 1835-1850 16 p. |
artikel |
15 |
Rational design and synthesis of phenethyl-5-bromopyridyl thiourea derivatives as potent non-nucleoside inhibitors of HIV reverse transcriptase
|
Vig, Rakesh |
|
1998 |
6 |
10 |
p. 1789-1797 9 p. |
artikel |
16 |
Structure–activity relationship and conformational analysis of monoglycosylceramides on the syngeneic mixed leukocyte reaction
|
Iijima, Hiroshi |
|
1998 |
6 |
10 |
p. 1905-1910 6 p. |
artikel |
17 |
Structure-based design and synthesis of small molecule protein–tyrosine phosphatase 1B inhibitors 1 A preliminary account of this work have been reported: Burke, T. R., Jr.; Yao, Z. J.; Ye, B.; Wang, S.; Zhang, Z. Y. Structure-based design of protein–tyrosine phosphatase inhibitors. Presented at the 213th National ACS Meeting, San Francisco, CA, April 13–17, 1997; MEDI-313. 1
|
Yao, Zhu-Jun |
|
1998 |
6 |
10 |
p. 1799-1810 12 p. |
artikel |
18 |
Substituted pyrazoles as novel selective ligands for the human dopamine D4 receptor
|
Bourrain, Sylvie |
|
1998 |
6 |
10 |
p. 1731-1743 13 p. |
artikel |
19 |
Synthesis and antiallergic activity of pyridothienopyrimidines
|
Quintela, José M. |
|
1998 |
6 |
10 |
p. 1911-1925 15 p. |
artikel |
20 |
Synthesis and antiplatelet activity of phenyl quinolones
|
Huang, Li-Jiau |
|
1998 |
6 |
10 |
p. 1657-1662 6 p. |
artikel |
21 |
Synthesis and biological evaluation of 2-Hydroxy derivatives of digitoxigenin and 3-Epidigitoxigenin 1 A preliminary account of this work has been presented at the First International Electronic Conference on Synthetic Organic Chemistry (ECSOC-1), A0012, 1–30 September 1997; http://www.mdpi.org/escoc-1.htm 1
|
Gobbini, M |
|
1998 |
6 |
10 |
p. 1889-1894 6 p. |
artikel |
22 |
Synthesis and in vitro activity of some epimeric 20α-hydroxy, 20-oxime and aziridine pregnene derivatives as inhibitors of human 17α-hydroxylase/c17,20-lyase and 5α-reductase
|
Ling, Yang-zhi |
|
1998 |
6 |
10 |
p. 1683-1693 11 p. |
artikel |
23 |
Synthesis and kinetic studies of an amidine-containing phosphonofluoridate: a novel potent inhibitor of trypsin-like enzymes
|
Ni, Li-Ming |
|
1998 |
6 |
10 |
p. 1767-1773 7 p. |
artikel |
24 |
Synthesis and screening of conformationally restricted and conformationally free N-(tertiary aminoalkyl)dithiocarbamic acids and esters as inhibitors of neuronal nitric oxide synthase
|
Sassaman, Mark B. |
|
1998 |
6 |
10 |
p. 1759-1766 8 p. |
artikel |
25 |
Synthesis and structure–activity relationships of novel naphthalenic and bioisosteric related amidic derivatives as melatonin receptor ligands
|
Leclerc, Véronique |
|
1998 |
6 |
10 |
p. 1875-1887 13 p. |
artikel |
26 |
The design, synthesis, and initial evaluation of benzophenone-containing peptides as potential photoaffinity labels of oligosaccharyltransferase
|
Xu, Tong |
|
1998 |
6 |
10 |
p. 1821-1834 14 p. |
artikel |
27 |
The specificity of Prolyl Endopeptidase from Flavobacterium meningoseptum: mapping the S′ subsites by positional scanning via acyl transfer
|
Bordusa, Frank |
|
1998 |
6 |
10 |
p. 1775-1780 6 p. |
artikel |
28 |
18-Vinyldeoxycorticosterone: a potent inhibitor of the bovine cytochrome P-45011β
|
Davioud, Elisabeth |
|
1998 |
6 |
10 |
p. 1781-1788 8 p. |
artikel |