nr |
titel |
auteur |
tijdschrift |
jaar |
jaarg. |
afl. |
pagina('s) |
type |
1 |
A novel tricyclic β-lactam exhibiting potent antibacterial activities against carbapenem-resistant Enterobacterales: Synthesis and structure-activity-relationships
|
Sato, Jun |
|
|
46 |
C |
p. |
artikel |
2 |
Antiviral fungal metabolites and some insights into their contribution to the current COVID-19 pandemic
|
Takahashi, Jacqueline Aparecida |
|
|
46 |
C |
p. |
artikel |
3 |
Antiviral strategies targeting host factors and mechanisms obliging +ssRNA viral pathogens
|
Mahajan, Supreeti |
|
|
46 |
C |
p. |
artikel |
4 |
A review upon medicinal perspective and designing rationale of DPP-4 inhibitors
|
Kumar, Shubham |
|
|
46 |
C |
p. |
artikel |
5 |
Biofunctional supramolecular hydrogels fabricated from a short self-assembling peptide modified with bioactive sequences for the 3D culture of breast cancer MCF-7 cells
|
Chia, Jyh Yea |
|
|
46 |
C |
p. |
artikel |
6 |
CYPlebrity: Machine learning models for the prediction of inhibitors of cytochrome P450 enzymes
|
Plonka, Wojciech |
|
|
46 |
C |
p. |
artikel |
7 |
Cysteine proteases as potential targets for anti-trypanosomatid drug discovery
|
Judice, Wagner A.S. |
|
|
46 |
C |
p. |
artikel |
8 |
Design, synthesis and anti-fibrosis evaluation of imidazo[1,2–a]pyridine derivatives as potent ATX inhibitors
|
Chen, Yuxiang |
|
|
46 |
C |
p. |
artikel |
9 |
Design, synthesis, and antitumor activity evaluation of steroidal oximes
|
Gomes, Ana R. |
|
|
46 |
C |
p. |
artikel |
10 |
Design, synthesis and biological evaluation of novel acridine and quinoline derivatives as tubulin polymerization inhibitors with anticancer activities
|
Ren, Yichang |
|
|
46 |
C |
p. |
artikel |
11 |
Design, synthesis, and biological evaluation of novel 6-(pyridin-3-yl) quinazolin-4(3H)-one derivatives as potential anticancer agents via PI3K inhibition
|
Yang, Huarong |
|
|
46 |
C |
p. |
artikel |
12 |
Design, synthesis, and biological evaluation of potent 1,2,3,4-tetrahydroisoquinoline derivatives as anticancer agents targeting NF-κB signaling pathway
|
Sim, Seongrak |
|
|
46 |
C |
p. |
artikel |
13 |
Design, synthesis, and target identification of new hypoxia-inducible factor 1 (HIF-1) inhibitors containing 1-alkyl-1H-pyrazole-3-carboxamide moiety
|
Sakai, Marina |
|
|
46 |
C |
p. |
artikel |
14 |
Development of curcumin-based amyloid β aggregation inhibitors for Alzheimer's disease using the SAR matrix approach
|
Yudi Utomo, Rohmad |
|
|
46 |
C |
p. |
artikel |
15 |
Discovery of benzimidazole derivatives as potent and selective aldehyde dehydrogenase 1A1 (ALDH1A1) inhibitors with glucose consumption improving activity
|
Ma, Zonghui |
|
|
46 |
C |
p. |
artikel |
16 |
Discovery of 1,3,4-oxadiazole derivatives as potential antitumor agents inhibiting the programmed cell death-1/programmed cell death-ligand 1 interaction
|
Fang, Lincheng |
|
|
46 |
C |
p. |
artikel |
17 |
Discovery of pyrazole N-aryl sulfonate: A novel and highly potent cyclooxygenase-2 (COX-2) selective inhibitors
|
Yao, Haiyan |
|
|
46 |
C |
p. |
artikel |
18 |
Docking and mutagenesis studies lead to improved inhibitor development of ML355 for human platelet 12-lipoxygenase
|
Tsai, Wan-Chen |
|
|
46 |
C |
p. |
artikel |
19 |
Editorial Board
|
|
|
|
46 |
C |
p. |
artikel |
20 |
EGFR-targeted prodrug activation using bioorthogonal alkene-azide click-and-release chemistry
|
Fairhall, Jessica M. |
|
|
46 |
C |
p. |
artikel |
21 |
Erratum to “De novo design with deep generative models based on 3D similarity scoring” [Bioorg. Med. Chem. 44 (2021) 116308]
|
Papadopoulos, Kostas |
|
|
46 |
C |
p. |
artikel |
22 |
Evaluation of γ-carboline-phenothiazine conjugates as simultaneous NMDA receptor blockers and cholinesterase inhibitors
|
Schwarthoff, Sigrid |
|
|
46 |
C |
p. |
artikel |
23 |
Further SAR studies on natural template based neuroprotective molecules for the treatment of Alzheimer’s disease
|
Singh, Yash Pal |
|
|
46 |
C |
p. |
artikel |
24 |
Graphical Abstract Contents Continued
|
|
|
|
46 |
C |
p. |
artikel |
25 |
Graphical abstract TOC
|
|
|
|
46 |
C |
p. |
artikel |
26 |
Graphical abstract TOC
|
|
|
|
46 |
C |
p. |
artikel |
27 |
Harmine-inspired design and synthesis of benzo[d]imidazo[2,1-b]thiazole derivatives bearing 1,3,4-oxadiazole moiety as potential tumor suppressors
|
Zhao, Tianming |
|
|
46 |
C |
p. |
artikel |
28 |
High allele discrimination in the typing of single nucleotide polymorphisms of miRNA
|
Takei, Fumie |
|
|
46 |
C |
p. |
artikel |
29 |
Identification of new [1,2,4]triazolo[4,3-a]quinoxalines as potent VEGFR-2 tyrosine kinase inhibitors: Design, synthesis, anticancer evaluation, and in silico studies
|
Alsaif, Nawaf A. |
|
|
46 |
C |
p. |
artikel |
30 |
Inhibition of amyloid formation of amyloid β (1–42), amylin and insulin by 1,5-diazacyclooctanes, a spermine-acrolein conjugate
|
Kunitomi, Risako |
|
|
46 |
C |
p. |
artikel |
31 |
In vivo organic synthesis by metal catalysts
|
Chang, Tsung-Che |
|
|
46 |
C |
p. |
artikel |
32 |
Kinetic and structural investigations of novel inhibitors of human epithelial 15-lipoxygenase-2
|
Tsai, Wan-Chen |
|
|
46 |
C |
p. |
artikel |
33 |
New FDA oncology small molecule drugs approvals in 2020: Mechanism of action and clinical applications
|
Cristina Mendonça Nogueira, Thais |
|
|
46 |
C |
p. |
artikel |
34 |
Potency and pharmacokinetics of GS-441524 derivatives against SARS-CoV-2
|
Wei, Daibao |
|
|
46 |
C |
p. |
artikel |
35 |
Preparation, biological & cheminformatics-based assessment of N 2,N 4-diphenylpyrimidine-2,4-diamine as potential Kinase-targeted antimalarials
|
Toviwek, Borvornwat |
|
|
46 |
C |
p. |
artikel |
36 |
Synthesis and duplex-forming ability of oligonucleotides modified with 4′-C,5′-C-methylene-bridged nucleic acid (4′,5′-BNA)
|
Yamaguchi, Takao |
|
|
46 |
C |
p. |
artikel |
37 |
Synthesis and evaluation of squaramide and thiosquaramide inhibitors of the DNA repair enzyme SNM1A
|
Berney, Mark |
|
|
46 |
C |
p. |
artikel |
38 |
Synthesis, in vitro cytotoxicity and biological evaluation of twenty novel 1,3-benzenedisulfonyl piperazines as antiplatelet agents
|
Liu, Xiu-jie |
|
|
46 |
C |
p. |
artikel |
39 |
Synthesis of acyclic nucleoside phosphonates targeting flavin-dependent thymidylate synthase in Mycobacterium tuberculosis
|
Biteau, Nicolas G. |
|
|
46 |
C |
p. |
artikel |
40 |
Synthetic and computational efforts towards the development of peptidomimetics and small-molecule SARS-CoV 3CLpro inhibitors
|
Paul, Abhik |
|
|
46 |
C |
p. |
artikel |
41 |
Virtual screening and biological evaluation of PPARγ antagonists as potential anti-prostate cancer agents
|
Almahmoud, Suliman |
|
|
46 |
C |
p. |
artikel |
42 |
Zinc ionophores isolated from Terminalia bellirica fruit rind extract protect against cardiomyocyte hypoxia/reoxygenation injury
|
Bodiga, Vijaya Lakshmi |
|
|
46 |
C |
p. |
artikel |